Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
etilefrine | Homo sapiens (human) | IC50 | 1.3310 | 1 | 0 |
3,5,14-trihydroxy-13-methyl-17-(5-oxo-2H-furan-3-yl)-2,3,4,6,7,8,9,11,12,15,16,17-dodecahydro-1H-cyclopenta[a]phenanthrene-10-carboxaldehyde | Homo sapiens (human) | IC50 | 29.8880 | 1 | 0 |
methacholine chloride | Homo sapiens (human) | IC50 | 7.3650 | 1 | 0 |
betamethasone | Homo sapiens (human) | IC50 | 29.9000 | 1 | 0 |
dibromsalicil | Homo sapiens (human) | IC50 | 1.1020 | 1 | 0 |
mitomycin | Homo sapiens (human) | IC50 | 0.9320 | 1 | 0 |
salmeterol xinafoate | Homo sapiens (human) | IC50 | 29.9160 | 1 | 0 |
acetylcholine bromide | Homo sapiens (human) | IC50 | 1.6580 | 1 | 0 |
2,6-di-tert-butyl-4-nitrophenol | Homo sapiens (human) | IC50 | 2.0020 | 1 | 0 |
chlormidazole | Homo sapiens (human) | IC50 | 0.7331 | 2 | 0 |
pyridaben | Homo sapiens (human) | IC50 | 0.0146 | 2 | 0 |
acetylcholine perchlorate | Homo sapiens (human) | IC50 | 0.6178 | 1 | 0 |
carboxyamido-triazole | Homo sapiens (human) | IC50 | 1.8696 | 2 | 0 |
1',2'-dihydrorotenone | Homo sapiens (human) | IC50 | 0.0139 | 2 | 0 |
N-benzylquinazolin-4-amine | Homo sapiens (human) | IC50 | 2.4190 | 1 | 0 |
6-ethyl-N-[2-(4-methoxyphenyl)ethyl]-5-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-7-amine | Homo sapiens (human) | IC50 | 3.2020 | 1 | 0 |
2-[[5-(1-benzotriazolylmethyl)-1,3,4-oxadiazol-2-yl]thio]-N-[(4-fluorophenyl)methyl]-N-phenylacetamide | Homo sapiens (human) | IC50 | 1.2375 | 2 | 0 |
N-[4-(4-fluorophenyl)-2-thiazolyl]-2-[(4-methylphenyl)sulfonylamino]benzamide | Homo sapiens (human) | IC50 | 1.4430 | 1 | 0 |
2-[(3-oxo-5-phenyl-1,2-dihydropyrazol-4-yl)-(3-thiophenyl)methyl]propanedinitrile | Homo sapiens (human) | IC50 | 29.9130 | 1 | 0 |
1-[5-(trifluoromethyl)-1,3,4-thiadiazol-2-yl]-3-[1,1,1-trifluoro-2-(trifluoromethyl)butan-2-yl]urea | Homo sapiens (human) | IC50 | 3.3250 | 1 | 0 |
4-(cyclohexylamino)-2-(3,5-dimethyl-1-pyrazolyl)-5-pyrimidinecarboxylic acid ethyl ester | Homo sapiens (human) | IC50 | 29.9030 | 1 | 0 |
4-cyano-3-methyl-5-(4-methylphenyl)-2-thiophenecarbohydrazide | Homo sapiens (human) | IC50 | 29.9430 | 1 | 0 |
5-bromo-N-(pyridin-4-ylmethyl)-2-thiophenesulfonamide | Homo sapiens (human) | IC50 | 1.9260 | 2 | 0 |
4-(2,4-dichlorophenyl)-2-[(1-oxo-2-phenylethyl)amino]-3-thiophenecarboxamide | Homo sapiens (human) | IC50 | 1.4400 | 2 | 0 |
N-[[[(2,4-dichlorophenyl)-oxomethyl]hydrazo]-sulfanylidenemethyl]-2,2-dimethylpropanamide | Homo sapiens (human) | IC50 | 29.9030 | 1 | 0 |
1-(5-isoquinolinyl)-3-(2-phenylethyl)thiourea | Homo sapiens (human) | IC50 | 2.1440 | 2 | 0 |
2-(1-benzimidazolyl)acetic acid [2-[1-(4-methoxyphenyl)-2,5-dimethyl-3-pyrrolyl]-2-oxoethyl] ester | Homo sapiens (human) | IC50 | 15.3360 | 2 | 0 |
nsc 105827 | Homo sapiens (human) | IC50 | 1.0100 | 1 | 0 |
3-[4-(2-hydroxyethylamino)-3-nitrophenyl]-4-methyl-4,5-dihydro-1H-pyridazin-6-one | Homo sapiens (human) | IC50 | 0.3672 | 1 | 0 |