Page last updated: 2024-08-07 22:55:26

galanin receptor type 3

[no definition available]

Synonyms

Research

Bioassay Publications (0)

TimeframeStudies on this Protein(%)All Drugs %
pre-19900 (0)18.7374
1990's0 (0)18.2507
2000's0 (0)29.6817
2010's0 (0)24.3611
2020's0 (0)2.80

Compounds (29)

Drugs with Inhibition Measurements

DrugTaxonomyMeasurementAverage (mM)Bioassay(s)Publication(s)
etilefrineHomo sapiens (human)IC501.331010
3,5,14-trihydroxy-13-methyl-17-(5-oxo-2H-furan-3-yl)-2,3,4,6,7,8,9,11,12,15,16,17-dodecahydro-1H-cyclopenta[a]phenanthrene-10-carboxaldehydeHomo sapiens (human)IC5029.888010
methacholine chlorideHomo sapiens (human)IC507.365010
betamethasoneHomo sapiens (human)IC5029.900010
dibromsalicilHomo sapiens (human)IC501.102010
mitomycinHomo sapiens (human)IC500.932010
salmeterol xinafoateHomo sapiens (human)IC5029.916010
acetylcholine bromideHomo sapiens (human)IC501.658010
2,6-di-tert-butyl-4-nitrophenolHomo sapiens (human)IC502.002010
chlormidazoleHomo sapiens (human)IC500.733120
pyridabenHomo sapiens (human)IC500.014620
acetylcholine perchlorateHomo sapiens (human)IC500.617810
carboxyamido-triazoleHomo sapiens (human)IC501.869620
1',2'-dihydrorotenoneHomo sapiens (human)IC500.013920
N-benzylquinazolin-4-amineHomo sapiens (human)IC502.419010
6-ethyl-N-[2-(4-methoxyphenyl)ethyl]-5-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-7-amineHomo sapiens (human)IC503.202010
2-[[5-(1-benzotriazolylmethyl)-1,3,4-oxadiazol-2-yl]thio]-N-[(4-fluorophenyl)methyl]-N-phenylacetamideHomo sapiens (human)IC501.237520
N-[4-(4-fluorophenyl)-2-thiazolyl]-2-[(4-methylphenyl)sulfonylamino]benzamideHomo sapiens (human)IC501.443010
2-[(3-oxo-5-phenyl-1,2-dihydropyrazol-4-yl)-(3-thiophenyl)methyl]propanedinitrileHomo sapiens (human)IC5029.913010
1-[5-(trifluoromethyl)-1,3,4-thiadiazol-2-yl]-3-[1,1,1-trifluoro-2-(trifluoromethyl)butan-2-yl]ureaHomo sapiens (human)IC503.325010
4-(cyclohexylamino)-2-(3,5-dimethyl-1-pyrazolyl)-5-pyrimidinecarboxylic acid ethyl esterHomo sapiens (human)IC5029.903010
4-cyano-3-methyl-5-(4-methylphenyl)-2-thiophenecarbohydrazideHomo sapiens (human)IC5029.943010
5-bromo-N-(pyridin-4-ylmethyl)-2-thiophenesulfonamideHomo sapiens (human)IC501.926020
4-(2,4-dichlorophenyl)-2-[(1-oxo-2-phenylethyl)amino]-3-thiophenecarboxamideHomo sapiens (human)IC501.440020
N-[[[(2,4-dichlorophenyl)-oxomethyl]hydrazo]-sulfanylidenemethyl]-2,2-dimethylpropanamideHomo sapiens (human)IC5029.903010
1-(5-isoquinolinyl)-3-(2-phenylethyl)thioureaHomo sapiens (human)IC502.144020
2-(1-benzimidazolyl)acetic acid [2-[1-(4-methoxyphenyl)-2,5-dimethyl-3-pyrrolyl]-2-oxoethyl] esterHomo sapiens (human)IC5015.336020
nsc 105827Homo sapiens (human)IC501.010010
3-[4-(2-hydroxyethylamino)-3-nitrophenyl]-4-methyl-4,5-dihydro-1H-pyridazin-6-oneHomo sapiens (human)IC500.367210