anti-inflammatory drug

A substance that reduces or suppresses inflammation.

ChEBI ID: 35472

Members (50)

Member	Definition	Class
amcinonide		amcinonide
andrographolide	A labdane diterpenoid isolated from the leaves and roots of Andrographis paniculata that exhibits anti-HIV, anti-inflammatory and antineoplastic properties.	andrographolide
beclomethasone	A 17alpha-hydroxy steroid that is prednisolone in which the hydrogens at the 9alpha and 16beta positions are substituted by a chlorine and a methyl group, respectively.	beclomethasone
beclomethasone dipropionate	A steroid ester comprising beclomethasone having propionyl groups at the 17- and 21-positions.	beclomethasone dipropionate
betamethasone		betamethasone
betamethasone valerate	A steroid ester that is betamethasone in which the hydroxy group at the 17alpha position has been converted to the corresponding pentanoate ester.	betamethasone valerate
celastrol	A pentacyclic triterpenoid that is 24,25,26-trinoroleana-1(10),3,5,7-tetraen-29-oic acid bearing an oxo substituent at position 2, a hydroxy substituent at position 3 and two methyl groups at positions 9 and 13. An antioxidant and anti-inflammatory agent. Potently inhibits lipid peroxidation in mitochondria and inhibits TNF-alpha-induced NFkappaB activation. Also shown to inhibit topoisomerase II activity in vitro (IC50 = 7.41 muM).	celastrol
clobetasol	A 3-oxo-Delta(1),Delta(4)-steroid that is 16beta-methylpregna-1,4-diene-3,20-dione bearing hydroxy groups at the 11beta and 17alpha positions, fluorine at position 9, and a chlorine substituent at position 21. It is used as its 17alpha-propionate ester to treat various skin disorders, including exzema and psoriasis.	clobetasol
clobetasol propionate	The 17-O-propionate ester of clobetasol. A potent corticosteroid, it is used to treat various skin disorders, including exzema and psoriasis.	clobetasol propionate
clocortolone pivalate	The 21-O-pivalate ester of clocortolone. It is used for the relief of inflammatory and pruritic (itching) skin disorders.	clocortolone pivalate
dapsone	A sulfone that is diphenylsulfone in which the hydrogen atom at the 4 position of each of the phenyl groups is substituted by an amino group. It is active against a wide range of bacteria, but is mainly employed for its actions against Mycobacterium leprae, being used as part of multidrug regimens in the treatment of all forms of leprosy.	dapsone
delgocitinib	A pyrrolopyrimidine that is 7H-pyrrolo[2,3-d]pyrimidine substituted by a (3S,4R)-1-(cyanoacetyl)-3-methyl-1,6-diazaspiro[3.4]octan-6-yl group at position 4. It is a pan-Janus kinase (JAK) inhibitor and is approved for treatment of atopic dermatitis (AD) in Japan.	delgocitinib
desonide	Triamcinolone acetonide with hydrogen instead of the fluorine substituent at position 9. A corticosteroid anti-inflammatory, it is used topically as a cream, ointment or lotion for the treatment of various skin disorders.	desonide
desoximetasone	Dexamethasone in which the hydroxy group at the 17alpha position is substituted by hydrogen. A synthetic corticosteroid with glucocorticoid activity, it is used as an anti-inflammatory and anti-pruritic in the treatment of various skin disorders, including skin allergies and psoriasis.	desoximetasone
diflorasone	The 16beta-analogue of flumethasone. It is used as the 17,21-diacetate as a topical anti-inflammatory and antipruritic in the treatment of various skin disorders.	diflorasone
diflorasone diacetate	The 17,21-diacetate derivative of diflorasone. It is used topically for its anti-inflammatory and antipruritic properties in the treatment of various skin disorders.	diflorasone diacetate
e 3040	A member of the class of benzothiazoles that is 1,3-benzothiazole substituted by a methylnitrilo group, (pyridin-3-yl)methyl group, methyl group, hydroxy group and methyl group at position 2,4,5,6 and 7, respectively. It is a dual inhibitor of 5-lipoxygenase and thromboxane A2 synthetase and exhibits anti-inflammatory properties. The drug was being developed by Eisai (Tokyo, Japan) for the treatment of bowel disease.	E3040
ebselen	A benzoselenazole that is 1,2-benzoselenazol-3-one carrying an additional phenyl substituent at position 2. Acts as a mimic of glutathione peroxidase.	ebselen
fludrocortisone		fludrocortisone
flumethasone		flumethasone
flumethasone pivalate		flumethasone pivalate
flunisolide		flunisolide
fluocinolone acetonide	A fluorinated steroid that is flunisolide in which the hydrogen at position 9 is replaced by fluorine. A corticosteroid with glucocorticoid activity, it is used (both as the anhydrous form and as the dihydrate) in creams, gels and ointments for the treatment of various skin disorders.	fluocinolone acetonide
fluorometholone	A member of the class of glucocorticoids that is Delta(1)-progesterone substituted at positions 11beta and 17 by hydroxy groups, at position 6alpha by a methyl group and at position 9 by a fluoro group. Used for the treatment of corticosteroid-responsive inflammation of the palpebral and bulbar conjunctiva, cornea and anterior segment of the globe.	fluorometholone
fluticasone propionate	A trifluorinated corticosteroid that consists of 6alpha,9-difluoro-11beta,17alpha-dihydroxy-17beta-{[(fluoromethyl)sulfanyl]carbonyl}-16-methyl-3-oxoandrosta-1,4-diene bearing a propionyl substituent at position 17; has anti-inflammatory, anti-asthmatic and anti-allergic activity.	fluticasone propionate
friedelin	A pentacyclic triterpenoid that is perhydropicene which is substituted by an oxo group at position 3 and by methyl groups at the 4, 4a, 6b, 8a, 11, 11, 12b, and 14a-positions (the 4R,4aS,6aS,6bR,8aR,12aR,12bS,14aS,14bS-enantiomer). It is the major triterpenoid constituent of cork.	friedelin
ginsenoside rb1	A ginsenoside found in Panax ginseng and Panax japonicus var. major that is ginsenoside Rd in which the beta-D-glucopyranoside group at position 20 is replaced by a beta-D-glucopyranosyl-beta-D-glucopyranoside group.	ginsenoside Rb1
ginsenoside rd	A ginsenoside found in Panax ginseng and Panax japonicus var. major that is (20S)-ginsenoside Rg3 in which the hydroxy group at position 20 has been converted to its beta-D-glucopyranoside.	ginsenoside Rd
hydrocortamate		hydrocortamate
loteprednol etabonate		loteprednol etabonate
lupeol	A pentacyclic triterpenoid that is lupane in which the hydrogen at the 3beta position is substituted by a hydroxy group. It occurs in the skin of lupin seeds, as well as in the latex of fig trees and of rubber plants. It is also found in many edible fruits and vegetables.	lupeol
methylprednisolone	The 6alpha-stereoisomer of 6-methylprednisolone.	6alpha-methylprednisolone
methylprednisolone acetate	An acetate ester resulting from the formal condensation of the 21-hydroxy function of 6alpha-methylprednisolone compound with acetic acid.	methylprednisolone acetate
mometasone furoate		mometasone furoate
palmidrol	An N-(long-chain-acyl)ethanolamine that is the ethanolamide of palmitic (hexadecanoic) acid.	palmitoyl ethanolamide
prednisolone	A glucocorticoid that is prednisone in which the oxo group at position 11 has been reduced to the corresponding beta-hydroxy group. It is a drug metabolite of prednisone.	prednisolone
prednisolone hemisuccinate	A hemisuccinate resulting from the formal condensation of the 21-hydroxy group prednisolone with one of the carboxy groups of succinic acid. It is used to treat mild to moderate non-infectious eye allergies and inflammation, including damage caused by chemical and thermal burns.	prednisolone succinate
prednisolone sodium succinate	The organic sodium salt of prednisolone succinate.	prednisolone sodium succinate
prednisone	A synthetic glucocorticoid drug that is particularly effective as an immunosuppressant, and affects virtually all of the immune system. Prednisone is a prodrug that is converted by the liver into prednisolone (a beta-hydroxy group instead of the oxo group at position 11), which is the active drug and also a steroid.	prednisone
probucol	A dithioketal that is propane-2,2-dithiol in which the hydrogens attached to both sulfur atoms are replaced by 3,5-di-tert-butyl-4-hydroxyphenyl groups. An anticholesteremic drug with antioxidant and anti-inflammatory properties, it is used to treat high levels of cholesterol in blood.	probucol
pulmicort	A glucocorticoid steroid having a highly oxygenated pregna-1,4-diene structure. It is used mainly in the treatment of asthma and non-infectious rhinitis and for treatment and prevention of nasal polyposis.	budesonide
rizatriptan		rizatriptan
sar 1118	An N-acyl-L-alpha-amino acid obtained by formal condensation of the carboxy group of N-[2-(1-benzofuran-6-carbonyl)]-5,7-dichloro-1,2,3,4-tetrahydroisoquinoline-6-carboxylic acid with the amino group of 3-(methanesulfonyl)-L-phenylalanine. Used for treatment of keratoconjunctivitis sicca (dry eye syndrome).	lifitegrast
sch 22219	A prednisolone compound having an alpha-chloro substituent at the 7-position, an alpha-methyl substituent at the 16-position and O-propanoyl groups at the 17- and 21-positions.	alclometasone dipropionate
triamcinolone	A C21-steroid hormone that is 1,4-pregnadiene-3,20-dione carrying four hydroxy substituents at positions 11beta, 16alpha, 17alpha and 21 as well as a fluoro substituent at position 9. Used in the form of its 16,17-acetonide to treat various skin infections.	triamcinolone
triamcinolone acetonide	A synthetic glucocorticoid that is the 16,17-acetonide of triamcinolone. Used to treat various skin infections.	triamcinolone acetonide
varespladib	A member of the class of indoles that is 1H-indole substituted by benzyl, ethyl, oxamoyl, and carboxymethoxy groups at positions 1, 2, 3, and 4, respectively. It is an oral secretory phospholipase A2 inhibitor and exhibits anti-inflammatory effects.	varespladib
varespladib methyl	A methyl ester resulting from the formal condensation of the carboxy group of varespladib with methanol. It is a potential therapy for the treatment of snakebite envenomings in which toxicity depends on the action of PLA2s.	varespladib methyl
vx-745	A member of the class of pyrimidopyridazines that is 6H-pyrimido[1,6-b]pyridazin-6-one substituted at positions 2 and 5 by (2,4-difluorophenyl)sulfanyl and 2,6-dichlorophenyl groups respectively	VX-745
zolmitriptan	A member of the class of tryptamines that is N,N-dimethyltryptamine in which the hydrogen at position 5 of the indole ring has been replaced by a [(4S)-2-oxo-1,3-oxazolidin-4-yl]methyl group. A serotonin 5-HT1 B and D receptor agonist, it is used for the treatment of migraine.	zolmitriptan

Research

Studies (117,700)

Timeframe	Studies, Drugs with This Role(%)	All Drugs %
pre-1990	40,194 (34.15)	18.7374
1990's	19,125 (16.25)	18.2507
2000's	24,300 (20.65)	29.6817
2010's	26,224 (22.28)	24.3611
2020's	7,857 (6.68)	2.80

Study Types

Publication Type	Studies, Drugs with this Role (%)	All Drugs (%)
Trials	18,390 (13.28%)	5.53%
Reviews	9,778 (7.06%)	6.00%
Case Studies	38,386 (27.71%)	4.05%
Observational	553 (0.40%)	0.25%
Other	71,421 (51.56%)	84.16%

Protein Targets (787)

Potency Measurements

Protein	Taxonomy	Measurement	Average (mM)	Bioassay(s)	Drugs
15-hydroxyprostaglandin dehydrogenase [NAD(+)] isoform 1	Homo sapiens (human)	Potency	0.5646	1	3
15-lipoxygenase, partial	Homo sapiens (human)	Potency	0.2306	1	2
2,3-bisphosphoglycerate-independent phosphoglycerate mutase	Leishmania major strain Friedlin	Potency	7.5686	1	1
67.9K protein	Vaccinia virus	Potency	13.8894	2	6
acetylcholinesterase	Homo sapiens (human)	Potency	31.3416	2	3
activating transcription factor 6	Homo sapiens (human)	Potency	22.0840	2	4
aldehyde dehydrogenase 1 family, member A1	Homo sapiens (human)	Potency	3.0003	1	6
alpha-galactosidase	Homo sapiens (human)	Potency	32.4648	2	2
Alpha-synuclein	Homo sapiens (human)	Potency	4.4780	1	3
Amyloid-beta precursor protein	Homo sapiens (human)	Potency	16.3601	1	1
AR protein	Homo sapiens (human)	Potency	3.6503	12	329
aryl hydrocarbon receptor	Homo sapiens (human)	Potency	11.3109	2	20
arylsulfatase A	Homo sapiens (human)	Potency	1.0691	1	1
ATAD5 protein, partial	Homo sapiens (human)	Potency	8.1758	3	5
Ataxin-2	Homo sapiens (human)	Potency	0.0250	1	11
ATP-dependent phosphofructokinase	Trypanosoma brucei brucei TREU927	Potency	12.1337	3	5
ATPase family AAA domain-containing protein 5	Homo sapiens (human)	Potency	0.6481	2	13
atrial natriuretic peptide receptor 1 precursor	Homo sapiens (human)	Potency	6.7456	1	1
atrial natriuretic peptide receptor 2 precursor	Homo sapiens (human)	Potency	26.1216	1	1
Bloom syndrome protein isoform 1	Homo sapiens (human)	Potency	0.0045	2	2
bromodomain adjacent to zinc finger domain 2B	Homo sapiens (human)	Potency	42.6696	1	4
caspase 7, apoptosis-related cysteine protease	Homo sapiens (human)	Potency	29.8493	1	1
caspase-3	Cricetulus griseus (Chinese hamster)	Potency	33.4915	1	1
caspase-3	Homo sapiens (human)	Potency	29.8493	1	1
Caspase-7	Cricetulus griseus (Chinese hamster)	Potency	33.4915	1	1
Cellular tumor antigen p53	Homo sapiens (human)	Potency	26.7616	2	9
cellular tumor antigen p53 isoform a	Homo sapiens (human)	Potency	7.9433	1	1
Chain A, 2-oxoglutarate Oxygenase	Homo sapiens (human)	Potency	11.9443	1	4
Chain A, Beta-lactamase	Escherichia coli K-12	Potency	33.9898	2	12
Chain A, Cruzipain	Trypanosoma cruzi	Potency	28.2665	2	4
Chain A, Ferritin light chain	Equus caballus (horse)	Potency	12.5893	1	1
Chain A, HADH2 protein	Homo sapiens (human)	Potency	10.4195	2	8
Chain A, JmjC domain-containing histone demethylation protein 3A	Homo sapiens (human)	Potency	8.9125	1	1
Chain A, MAJOR APURINIC/APYRIMIDINIC ENDONUCLEASE	Homo sapiens (human)	Potency	15.4412	1	6
Chain A, Putative fructose-1,6-bisphosphate aldolase	Giardia intestinalis	Potency	22.6655	3	5
Chain A, TYROSYL-DNA PHOSPHODIESTERASE	Homo sapiens (human)	Potency	9.0630	1	7
Chain B, HADH2 protein	Homo sapiens (human)	Potency	10.4195	2	8
chromobox protein homolog 1	Homo sapiens (human)	Potency	60.2754	2	8
cytochrome P450 2C19 precursor	Homo sapiens (human)	Potency	0.8554	1	2
cytochrome P450 2C9 precursor	Homo sapiens (human)	Potency	0.6246	1	3
cytochrome P450 2C9, partial	Homo sapiens (human)	Potency	15.1833	1	17
cytochrome P450 2D6	Homo sapiens (human)	Potency	17.4934	1	9
cytochrome P450 2D6 isoform 1	Homo sapiens (human)	Potency	5.5000	1	2
cytochrome P450 3A4 isoform 1	Homo sapiens (human)	Potency	12.9878	2	10
cytochrome P450 family 3 subfamily A polypeptide 4	Homo sapiens (human)	Potency	11.9628	2	30
cytochrome P450, family 19, subfamily A, polypeptide 1, isoform CRA_a	Homo sapiens (human)	Potency	2.2244	1	40
D(1A) dopamine receptor	Homo sapiens (human)	Potency	22.3872	1	1
DNA dC->dU-editing enzyme APOBEC-3F isoform a	Homo sapiens (human)	Potency	30.3001	1	2
DNA dC->dU-editing enzyme APOBEC-3G isoform 1	Homo sapiens (human)	Potency	35.4813	1	1
DNA polymerase beta	Homo sapiens (human)	Potency	3.1623	1	1
DNA polymerase III, partial	Bacillus subtilis	Potency	4.7444	1	1
DNA polymerase iota isoform a (long)	Homo sapiens (human)	Potency	39.2615	1	3
DNA polymerase kappa isoform 1	Homo sapiens (human)	Potency	89.1251	1	1
Endothelin receptor type B	Rattus norvegicus (Norway rat)	Potency	22.3872	1	1
Endothelin-1 receptor	Rattus norvegicus (Norway rat)	Potency	22.3872	1	1
estrogen nuclear receptor alpha	Homo sapiens (human)	Potency	10.1812	10	151
estrogen receptor 2 (ER beta)	Homo sapiens (human)	Potency	46.3997	2	6
estrogen-related nuclear receptor alpha	Homo sapiens (human)	Potency	26.5874	8	75
euchromatic histone-lysine N-methyltransferase 2	Homo sapiens (human)	Potency	29.5917	1	15
EWS/FLI fusion protein	Homo sapiens (human)	Potency	12.9170	4	19
farnesoid X nuclear receptor	Homo sapiens (human)	Potency	26.3808	2	4
flap endonuclease 1	Homo sapiens (human)	Potency	64.2145	1	5
fructose-bisphosphate aldolase A	Oryctolagus cuniculus (rabbit)	Potency	22.3872	1	1
Fumarate hydratase	Homo sapiens (human)	Potency	14.6536	1	2
G	Vesicular stomatitis virus	Potency	15.1833	1	17
GABA theta subunit	Rattus norvegicus (Norway rat)	Potency	12.9878	1	5
GALC protein	Homo sapiens (human)	Potency	2.5873	1	2
Gamma-aminobutyric acid receptor subunit alpha-1	Rattus norvegicus (Norway rat)	Potency	12.9878	1	5
Gamma-aminobutyric acid receptor subunit alpha-2	Rattus norvegicus (Norway rat)	Potency	12.9878	1	5
Gamma-aminobutyric acid receptor subunit alpha-3	Rattus norvegicus (Norway rat)	Potency	12.9878	1	5
Gamma-aminobutyric acid receptor subunit alpha-4	Rattus norvegicus (Norway rat)	Potency	12.9878	1	5
Gamma-aminobutyric acid receptor subunit alpha-5	Rattus norvegicus (Norway rat)	Potency	12.9878	1	5
Gamma-aminobutyric acid receptor subunit alpha-6	Rattus norvegicus (Norway rat)	Potency	12.9878	1	5
Gamma-aminobutyric acid receptor subunit beta-1	Rattus norvegicus (Norway rat)	Potency	12.9878	1	5
Gamma-aminobutyric acid receptor subunit beta-2	Rattus norvegicus (Norway rat)	Potency	12.9878	1	5
Gamma-aminobutyric acid receptor subunit beta-3	Rattus norvegicus (Norway rat)	Potency	12.9878	1	5
Gamma-aminobutyric acid receptor subunit delta	Rattus norvegicus (Norway rat)	Potency	12.9878	1	5
Gamma-aminobutyric acid receptor subunit epsilon	Rattus norvegicus (Norway rat)	Potency	12.9878	1	5
Gamma-aminobutyric acid receptor subunit gamma-1	Rattus norvegicus (Norway rat)	Potency	12.9878	1	5
Gamma-aminobutyric acid receptor subunit gamma-2	Rattus norvegicus (Norway rat)	Potency	12.9878	1	5
Gamma-aminobutyric acid receptor subunit gamma-3	Rattus norvegicus (Norway rat)	Potency	12.9878	1	5
Gamma-aminobutyric acid receptor subunit pi	Rattus norvegicus (Norway rat)	Potency	12.9878	1	5
geminin	Homo sapiens (human)	Potency	11.4367	4	30
GLI family zinc finger 3	Homo sapiens (human)	Potency	16.4994	3	36
glp-1 receptor, partial	Homo sapiens (human)	Potency	14.3918	1	8
GLS protein	Homo sapiens (human)	Potency	8.0141	2	4
glucocerebrosidase	Homo sapiens (human)	Potency	34.3725	1	4
glucocorticoid receptor [Homo sapiens]	Homo sapiens (human)	Potency	0.3578	5	123
glucokinase regulatory protein	Homo sapiens (human)	Potency	14.1254	1	1
Glutamate receptor 2	Rattus norvegicus (Norway rat)	Potency	8.9329	1	7
Glutamate receptor ionotropic, NMDA 1	Rattus norvegicus (Norway rat)	Potency	5.7988	1	1
Glutamate receptor ionotropic, NMDA 2A	Rattus norvegicus (Norway rat)	Potency	5.7988	1	1
Glutamate receptor ionotropic, NMDA 2B	Rattus norvegicus (Norway rat)	Potency	5.7988	1	1
Glutamate receptor ionotropic, NMDA 2C	Rattus norvegicus (Norway rat)	Potency	5.7988	1	1
Glutamate receptor ionotropic, NMDA 2D	Rattus norvegicus (Norway rat)	Potency	5.7988	1	1
Glutamate receptor ionotropic, NMDA 3A	Rattus norvegicus (Norway rat)	Potency	5.7988	1	1
Glutamate receptor ionotropic, NMDA 3B	Rattus norvegicus (Norway rat)	Potency	5.7988	1	1
GTP-binding nuclear protein Ran isoform 1	Homo sapiens (human)	Potency	11.3852	1	3
Guanine nucleotide-binding protein G	Homo sapiens (human)	Potency	22.7496	1	3
guanine nucleotide-binding protein G(i) subunit alpha-1 isoform 1	Homo sapiens (human)	Potency	12.5893	1	1
heat shock protein beta-1	Homo sapiens (human)	Potency	21.8892	2	5
hexokinase-4 isoform 1	Homo sapiens (human)	Potency	14.1254	1	1
Histamine H2 receptor	Cavia porcellus (domestic guinea pig)	Potency	0.6066	2	13
histone acetyltransferase KAT2A isoform 1	Homo sapiens (human)	Potency	0.4496	1	4
Histone H2A.x	Cricetulus griseus (Chinese hamster)	Potency	111.5860	2	3
histone-lysine N-methyltransferase 2A isoform 2 precursor	Homo sapiens (human)	Potency	44.6684	1	1
HLA class I histocompatibility antigen, B alpha chain	Homo sapiens (human)	Potency	15.1833	1	17
huntingtin isoform 2	Homo sapiens (human)	Potency	20.8954	1	2
hypothetical protein, conserved	Trypanosoma brucei	Potency	11.1471	4	5
hypoxia-inducible factor 1 alpha subunit	Homo sapiens (human)	Potency	9.0485	2	8
hypoxia-inducible factor 1, alpha subunit (basic helix-loop-helix transcription factor)	Homo sapiens (human)	Potency	3.5236	3	31
IDH1	Homo sapiens (human)	Potency	10.3508	1	12
importin subunit beta-1 isoform 1	Homo sapiens (human)	Potency	11.3852	1	3
Inositol hexakisphosphate kinase 1	Homo sapiens (human)	Potency	15.1833	1	34
Inositol monophosphatase 1	Rattus norvegicus (Norway rat)	Potency	10.0000	1	2
Interferon beta	Homo sapiens (human)	Potency	8.0036	3	38
interleukin 8	Homo sapiens (human)	Potency	66.8242	1	1
isocitrate dehydrogenase 1, partial	Homo sapiens (human)	Potency	25.1998	2	6
lamin isoform A-delta10	Homo sapiens (human)	Potency	9.9073	1	10
lethal factor (plasmid)	Bacillus anthracis str. A2012	Potency	10.6530	1	3
Luciferase	Photinus pyralis (common eastern firefly)	Potency	21.0236	3	6
luciferase	Photuris pensylvanica (Pennsylania firefly)	Potency	18.0789	3	5
lysosomal alpha-glucosidase preproprotein	Homo sapiens (human)	Potency	2.9006	2	4
M-phase phosphoprotein 8	Homo sapiens (human)	Potency	4.0027	1	2
Microtubule-associated protein tau	Homo sapiens (human)	Potency	10.3260	2	10
mitogen-activated protein kinase 1	Homo sapiens (human)	Potency	3.1623	1	1
muscarinic acetylcholine receptor M1	Rattus norvegicus (Norway rat)	Potency	0.0891	1	1
muscleblind-like protein 1 isoform 1	Homo sapiens (human)	Potency	40.3582	1	3
Neuronal acetylcholine receptor subunit alpha-4	Rattus norvegicus (Norway rat)	Potency	2.9006	1	2
Neuronal acetylcholine receptor subunit beta-2	Rattus norvegicus (Norway rat)	Potency	2.9006	1	2
neuropeptide S receptor isoform A	Homo sapiens (human)	Potency	5.7738	5	7
NFKB1 protein, partial	Homo sapiens (human)	Potency	4.0554	2	8
nonstructural protein 1	Influenza A virus (A/WSN/1933(H1N1))	Potency	3.8263	1	5
Nrf2	Homo sapiens (human)	Potency	29.2953	2	2
nuclear factor erythroid 2-related factor 2 isoform 1	Homo sapiens (human)	Potency	32.1519	3	21
nuclear factor erythroid 2-related factor 2 isoform 2	Homo sapiens (human)	Potency	0.0579	2	24
nuclear factor of kappa light polypeptide gene enhancer in B-cells 1 (p105), isoform CRA_a	Homo sapiens (human)	Potency	14.9300	1	5
Nuclear receptor ROR-gamma	Homo sapiens (human)	Potency	20.4946	1	2
nuclear receptor ROR-gamma isoform 1	Mus musculus (house mouse)	Potency	18.3093	4	18
nuclear receptor subfamily 1, group I, member 2	Rattus norvegicus (Norway rat)	Potency	7.5570	1	21
nuclear receptor subfamily 1, group I, member 3	Homo sapiens (human)	Potency	27.0964	3	11
Ornithine decarboxylase	Rattus norvegicus (Norway rat)	Potency	10.0000	1	1
parathyroid hormone/parathyroid hormone-related peptide receptor precursor	Homo sapiens (human)	Potency	85.0323	1	4
peptidyl-prolyl cis-trans isomerase NIMA-interacting 1	Homo sapiens (human)	Potency	68.0131	1	3
peripheral myelin protein 22	Rattus norvegicus (Norway rat)	Potency	28.6954	1	1
peripheral myelin protein 22 isoform 1	Homo sapiens (human)	Potency	54.7470	1	2
peroxisome proliferator activated receptor gamma	Homo sapiens (human)	Potency	30.1033	3	11
peroxisome proliferator-activated receptor delta	Homo sapiens (human)	Potency	27.7547	4	8
phosphopantetheinyl transferase	Bacillus subtilis	Potency	2.6383	1	4
plasminogen precursor	Mus musculus (house mouse)	Potency	6.5629	1	6
polyprotein	Zika virus	Potency	14.6536	1	2
polyunsaturated fatty acid lipoxygenase ALOX12	Homo sapiens (human)	Potency	2.8371	1	2
Polyunsaturated fatty acid lipoxygenase ALOX15B	Homo sapiens (human)	Potency	0.5661	1	2
potassium voltage-gated channel subfamily H member 2 isoform d	Homo sapiens (human)	Potency	24.0387	1	3
PPM1D protein	Homo sapiens (human)	Potency	3.1481	1	8
pregnane X nuclear receptor	Homo sapiens (human)	Potency	21.2835	3	37
pregnane X receptor	Rattus norvegicus (Norway rat)	Potency	23.8165	1	3
progesterone receptor	Homo sapiens (human)	Potency	8.3267	3	63
pyruvate kinase	Leishmania mexicana mexicana	Potency	15.5513	5	5
pyruvate kinase PKM isoform a	Homo sapiens (human)	Potency	5.1189	4	4
pyruvate kinase PKM isoform b	Homo sapiens (human)	Potency	10.0000	2	2
RAR-related orphan receptor gamma	Mus musculus (house mouse)	Potency	22.4535	2	25
ras-related protein Rab-9A	Homo sapiens (human)	Potency	1.0000	1	1
regulator of G-protein signaling 4	Homo sapiens (human)	Potency	14.4270	1	2
retinoic acid nuclear receptor alpha variant 1	Homo sapiens (human)	Potency	36.2145	3	37
retinoid X nuclear receptor alpha	Homo sapiens (human)	Potency	29.3017	3	16
RGS12	Homo sapiens (human)	Potency	12.5893	1	1
serine/threonine-protein kinase mTOR isoform 1	Homo sapiens (human)	Potency	20.4054	2	2
serine/threonine-protein kinase PLK1	Homo sapiens (human)	Potency	14.8365	1	2
Sigma non-opioid intracellular receptor 1	Homo sapiens (human)	Potency	5.7988	1	1
SMAD family member 2	Homo sapiens (human)	Potency	19.9912	2	15
SMAD family member 3	Homo sapiens (human)	Potency	19.9912	2	15
Smad3	Homo sapiens (human)	Potency	10.2756	1	5
snurportin-1	Homo sapiens (human)	Potency	11.3852	1	3
Sodium channel protein type 1 subunit alpha	Rattus norvegicus (Norway rat)	Potency	5.7988	1	1
Sodium channel protein type 2 subunit alpha	Rattus norvegicus (Norway rat)	Potency	5.7988	1	1
Sodium channel protein type 3 subunit alpha	Rattus norvegicus (Norway rat)	Potency	5.7988	1	1
Spike glycoprotein	Severe acute respiratory syndrome-related coronavirus	Potency	28.9003	1	3
survival motor neuron protein isoform d	Homo sapiens (human)	Potency	1.4846	1	6
TAR DNA-binding protein 43	Homo sapiens (human)	Potency	17.5727	1	4
TDP1 protein	Homo sapiens (human)	Potency	15.9524	2	50
thioredoxin glutathione reductase	Schistosoma mansoni	Potency	33.0846	1	3
thioredoxin reductase	Rattus norvegicus (Norway rat)	Potency	39.1287	3	8
Thrombopoietin	Homo sapiens (human)	Potency	1.5862	2	4
thyroid hormone receptor beta isoform 2	Rattus norvegicus (Norway rat)	Potency	34.0554	2	19
thyroid hormone receptor beta isoform a	Homo sapiens (human)	Potency	5.0119	1	1
thyroid stimulating hormone receptor	Homo sapiens (human)	Potency	23.0397	5	9
transient receptor potential cation channel subfamily V member 1	Homo sapiens (human)	Potency	31.6228	1	1
urokinase plasminogen activator surface receptor precursor	Mus musculus (house mouse)	Potency	6.5629	1	6
urokinase-type plasminogen activator precursor	Mus musculus (house mouse)	Potency	6.5629	1	6
USP1 protein, partial	Homo sapiens (human)	Potency	21.3018	2	4
v-jun sarcoma virus 17 oncogene homolog (avian)	Homo sapiens (human)	Potency	36.9669	2	11
vitamin D (1,25- dihydroxyvitamin D3) receptor	Homo sapiens (human)	Potency	18.6997	4	14
vitamin D3 receptor isoform VDRA	Homo sapiens (human)	Potency	37.8765	1	6
Voltage-dependent calcium channel gamma-2 subunit	Mus musculus (house mouse)	Potency	8.9329	1	7

Inhibition Measurements

Protein	Taxonomy	Measurement	Average (mM)	Bioassay(s)	Drugs
1-acylglycerol-3-phosphate O-acyltransferase ABHD5 isoform a	Homo sapiens (human)	IC50	2.2555	2	2
5-hydroxytryptamine receptor 1A	Homo sapiens (human)	IC50	0.3572	2	2
5-hydroxytryptamine receptor 1A	Homo sapiens (human)	Ki	0.1589	3	4
5-hydroxytryptamine receptor 1B	Homo sapiens (human)	IC50	0.0236	2	2
5-hydroxytryptamine receptor 1B	Homo sapiens (human)	Ki	0.0072	2	2
5-hydroxytryptamine receptor 1D	Homo sapiens (human)	IC50	0.0311	3	3
5-hydroxytryptamine receptor 1D	Sus scrofa (pig)	IC50	0.0501	1	1
5-hydroxytryptamine receptor 1D	Homo sapiens (human)	Ki	0.0106	4	6
5-hydroxytryptamine receptor 2A	Homo sapiens (human)	IC50	7.9433	1	1
5-hydroxytryptamine receptor 2A	Rattus norvegicus (Norway rat)	IC50	6.3096	1	1
5-hydroxytryptamine receptor 2C	Homo sapiens (human)	IC50	8.9716	2	2
5-hydroxytryptamine receptor 3A	Homo sapiens (human)	IC50	10.0000	1	1
5-hydroxytryptamine receptor 3A	Mus musculus (house mouse)	IC50	10.0000	1	1
5-hydroxytryptamine receptor 3A	Rattus norvegicus (Norway rat)	IC50	3.9811	1	1
5-hydroxytryptamine receptor 3B	Homo sapiens (human)	IC50	10.0000	1	1
5-hydroxytryptamine receptor 3B	Mus musculus (house mouse)	IC50	10.0000	1	1
5-hydroxytryptamine receptor 3B	Rattus norvegicus (Norway rat)	IC50	3.9811	1	1
5-hydroxytryptamine receptor 3C	Homo sapiens (human)	IC50	10.0000	1	1
5-hydroxytryptamine receptor 3D	Homo sapiens (human)	IC50	10.0000	1	1
5-hydroxytryptamine receptor 3E	Homo sapiens (human)	IC50	10.0000	1	1
5-hydroxytryptamine receptor 6	Homo sapiens (human)	Ki	0.1830	1	1
6-hydroxymethyl-7,8-dihydropterin pyrophosphokinase	Plasmodium berghei	IC50	12.4100	1	1
85/88 kDa calcium-independent phospholipase A2	Homo sapiens (human)	IC50	3.0076	8	8
Acetylcholinesterase	Electrophorus electricus (electric eel)	IC50	28.0050	2	2
Acetylcholinesterase	Homo sapiens (human)	IC50	15.0000	1	1
Adenosine receptor A3	Homo sapiens (human)	IC50	8.5470	1	1
Adenosine receptor A3	Homo sapiens (human)	Ki	4.8310	1	1
Aldo-keto reductase family 1 member B1	Rattus norvegicus (Norway rat)	IC50	20.4040	1	1
Aldo-keto reductase family 1 member B1	Rattus norvegicus (Norway rat)	Ki	20.2360	1	1
Alpha-1A adrenergic receptor	Homo sapiens (human)	IC50	10.0000	1	1
Alpha-1A adrenergic receptor	Rattus norvegicus (Norway rat)	IC50	8.5470	1	1
Alpha-1A adrenergic receptor	Rattus norvegicus (Norway rat)	Ki	4.8310	1	1
Alpha-1B adrenergic receptor	Rattus norvegicus (Norway rat)	IC50	8.5470	1	1
Alpha-1B adrenergic receptor	Rattus norvegicus (Norway rat)	Ki	4.8310	1	1
Alpha-2A adrenergic receptor	Homo sapiens (human)	IC50	34.1670	1	1
Alpha-2A adrenergic receptor	Homo sapiens (human)	Ki	12.8130	1	1
Alpha-2B adrenergic receptor	Homo sapiens (human)	IC50	31.8860	1	1
Alpha-2B adrenergic receptor	Homo sapiens (human)	Ki	14.5570	1	1
Amine oxidase [flavin-containing] B	Rattus norvegicus (Norway rat)	IC50	0.0290	1	1
Androgen receptor	Homo sapiens (human)	IC50	18.0000	2	2
Androgen receptor	Rattus norvegicus (Norway rat)	IC50	12.3918	3	7
Androgen receptor	Homo sapiens (human)	Ki	2.6807	3	3
Androgen receptor	Rattus norvegicus (Norway rat)	Ki	5.5625	1	4
Angiotensin-converting enzyme 2	Homo sapiens (human)	IC50	0.6700	1	1
Arrestin, beta 1	Homo sapiens (human)	IC50	1.5240	1	1
ATP-binding cassette sub-family C member 3	Homo sapiens (human)	IC50	113.4020	1	10
Bifunctional epoxide hydrolase 2	Homo sapiens (human)	IC50	0.7575	4	4
Bile acid receptor	Homo sapiens (human)	IC50	9.7000	2	2
Bile salt export pump	Homo sapiens (human)	IC50	181.1304	6	28
Bile salt export pump	Rattus norvegicus (Norway rat)	IC50	517.5000	1	2
Canalicular multispecific organic anion transporter 1	Homo sapiens (human)	IC50	133.0000	1	10
Cannabinoid receptor 1	Homo sapiens (human)	Ki	5.0000	2	3
Cannabinoid receptor 2	Homo sapiens (human)	Ki	5.0000	2	3
Caspase-1	Homo sapiens (human)	IC50	4.0400	1	1
Cholinesterase	Equus caballus (horse)	IC50	10.4740	2	2
Cocaine esterase	Homo sapiens (human)	IC50	1.9000	1	1
Corticosteroid-binding globulin	Homo sapiens (human)	Ki	0.0309	1	1
Corticotropin-releasing factor receptor 2	Homo sapiens (human)	Ki	5.0000	1	1
Cyclin-dependent kinase 2	Homo sapiens (human)	IC50	5.0000	1	1
Cytochrome P450 1A2	Homo sapiens (human)	IC50	40.0000	1	1
Cytochrome P450 2C19	Homo sapiens (human)	IC50	40.0000	1	1
Cytochrome P450 2C9	Homo sapiens (human)	IC50	30.4940	3	5
Cytochrome P450 2D6	Homo sapiens (human)	IC50	40.0000	1	1
Cytochrome P450 2J2	Homo sapiens (human)	IC50	36.4900	1	3
Cytochrome P450 3A4	Homo sapiens (human)	IC50	15.0517	4	4
Cytochrome P450 3A5	Homo sapiens (human)	IC50	3.1692	5	5
Dihydrofolate reductase	Pneumocystis carinii	IC50	1.5000	1	1
DNA topoisomerase 1	Homo sapiens (human)	IC50	250.0000	1	2
DNA topoisomerase 2-alpha	Homo sapiens (human)	IC50	190.1000	2	4
dual specificity protein phosphatase 6	Rattus norvegicus (Norway rat)	IC50	100.0000	1	1
Estrogen receptor	Homo sapiens (human)	IC50	32.5000	3	4
Estrogen receptor	Homo sapiens (human)	Ki	3.6667	3	3
Estrogen receptor beta	Homo sapiens (human)	IC50	32.5000	3	4
Estrogen receptor beta	Homo sapiens (human)	Ki	1.0000	1	1
eukaryotic translation initiation factor 4 gamma 1 isoform 4	Homo sapiens (human)	IC50	1.1500	1	1
eukaryotic translation initiation factor 4E isoform 1	Mus musculus (house mouse)	IC50	1.1500	1	1
Fatty acid-binding protein, liver	Rattus norvegicus (Norway rat)	Ki	51.8300	2	2
Fatty-acid amide hydrolase 1	Rattus norvegicus (Norway rat)	IC50	5.0119	1	1
galanin receptor type 3	Homo sapiens (human)	IC50	29.9000	1	1
Gamma-butyrobetaine dioxygenase	Homo sapiens (human)	IC50	0.7420	5	5
Glucocorticoid receptor	Homo sapiens (human)	IC50	0.0541	46	62
Glucocorticoid receptor	Rattus norvegicus (Norway rat)	IC50	0.0258	6	7
Glucocorticoid receptor	Homo sapiens (human)	Ki	0.0210	17	30
Glucose-6-phosphate 1-dehydrogenase	Homo sapiens (human)	Ki	540.5000	1	1
glucose-6-phosphate 1-dehydrogenase isoform b	Homo sapiens (human)	IC50	13.2000	1	1
glucose-6-phosphate dehydrogenase-6-phosphogluconolactonase	Plasmodium berghei	IC50	15.0867	3	3
Glycine receptor subunit alpha-1	Rattus norvegicus (Norway rat)	IC50	0.0913	1	14
Glycine receptor subunit alpha-1	Rattus norvegicus (Norway rat)	Ki	0.0415	1	14
Glycine receptor subunit alpha-2	Rattus norvegicus (Norway rat)	IC50	0.0913	1	14
Glycine receptor subunit alpha-2	Rattus norvegicus (Norway rat)	Ki	0.0415	1	14
Glycine receptor subunit alpha-3	Rattus norvegicus (Norway rat)	IC50	0.0913	1	14
Glycine receptor subunit alpha-3	Rattus norvegicus (Norway rat)	Ki	0.0415	1	14
Glycine receptor subunit beta	Rattus norvegicus (Norway rat)	IC50	0.0913	1	14
Glycine receptor subunit beta	Rattus norvegicus (Norway rat)	Ki	0.0415	1	14
Group 10 secretory phospholipase A2	Homo sapiens (human)	IC50	0.0918	8	8
Group 10 secretory phospholipase A2	Mus musculus (house mouse)	IC50	0.0750	2	2
Group 3 secretory phospholipase A2	Homo sapiens (human)	IC50	0.1225	2	2
Group IID secretory phospholipase A2	Homo sapiens (human)	IC50	0.1017	3	3
Group IID secretory phospholipase A2	Mus musculus (house mouse)	IC50	0.4300	1	1
Group IIE secretory phospholipase A2	Homo sapiens (human)	IC50	0.0862	4	4
Group IIE secretory phospholipase A2	Mus musculus (house mouse)	IC50	0.0750	2	2
Group IIF secretory phospholipase A2	Homo sapiens (human)	IC50	0.1250	3	3
Group IIF secretory phospholipase A2	Mus musculus (house mouse)	IC50	1.6000	1	1
Group XIIA secretory phospholipase A2	Homo sapiens (human)	IC50	0.1225	2	2
Group XIIB secretory phospholipase A2-like protein	Homo sapiens (human)	IC50	0.1225	2	2
hexokinase	Trypanosoma brucei brucei TREU927	IC50	0.9009	1	1
Hexokinase-2	Homo sapiens (human)	IC50	50.0000	1	1
Histone deacetylase 5	Homo sapiens (human)	IC50	3.4000	1	1
Histone deacetylase 6	Homo sapiens (human)	IC50	6.5333	3	3
Histone deacetylase 9	Homo sapiens (human)	IC50	3.7000	1	1
Histone-lysine N-methyltransferase EHMT1	Homo sapiens (human)	IC50	0.7300	1	1
Histone-lysine N-methyltransferase EHMT2	Homo sapiens (human)	IC50	0.4000	1	1
Hypoxia-inducible factor 1-alpha	Homo sapiens (human)	IC50	0.2500	1	1
Indoleamine 2,3-dioxygenase 1	Homo sapiens (human)	IC50	8.4100	1	1
Indoleamine 2,3-dioxygenase 1	Homo sapiens (human)	Ki	0.0940	3	3
Insulin-degrading enzyme	Homo sapiens (human)	IC50	33.3520	3	3
Insulin-like growth factor 1 receptor	Homo sapiens (human)	IC50	5.0000	1	1
Integrin alpha-L	Homo sapiens (human)	IC50	0.0415	2	2
Integrin beta-2	Homo sapiens (human)	IC50	0.0415	2	2
Intercellular adhesion molecule 1	Homo sapiens (human)	IC50	0.0287	3	3
Interleukin-5	Homo sapiens (human)	IC50	26.8000	1	1
Interleukin-5	Mus musculus (house mouse)	IC50	26.5375	8	8
Interleukin-5 receptor subunit alpha	Mus musculus (house mouse)	IC50	26.2000	1	1
Kappa-type opioid receptor	Cavia porcellus (domestic guinea pig)	IC50	250.0000	1	2
L-ornithine N(5)-monooxygenase	Aspergillus fumigatus Af293	IC50	11.0000	2	2
large T antigen	Betapolyomavirus macacae	IC50	13.9100	1	1
Leukotriene B4 receptor 1	Homo sapiens (human)	IC50	0.2100	1	1
Liver carboxylesterase 1	Homo sapiens (human)	IC50	0.1000	1	1
Macrophage migration inhibitory factor	Homo sapiens (human)	IC50	2.4000	1	1
Macrophage migration inhibitory factor	Homo sapiens (human)	Ki	0.5700	2	2
MAP kinase-activated protein kinase 2	Homo sapiens (human)	IC50	5.0000	1	1
Matrix metalloproteinase-9	Homo sapiens (human)	IC50	1.9890	1	1
Methionine aminopeptidase 2	Homo sapiens (human)	IC50	2.4300	1	1
Mineralocorticoid receptor	Homo sapiens (human)	IC50	0.0463	6	7
Mineralocorticoid receptor	Homo sapiens (human)	Ki	0.0186	2	2
Mitogen-activated protein kinase 1	Homo sapiens (human)	IC50	5.0000	1	1
Mitogen-activated protein kinase 10	Homo sapiens (human)	IC50	5.0000	1	1
Mitogen-activated protein kinase 11	Homo sapiens (human)	IC50	0.2462	5	5
Mitogen-activated protein kinase 11	Homo sapiens (human)	Ki	0.1104	2	2
Mitogen-activated protein kinase 12	Homo sapiens (human)	IC50	0.0577	4	4
Mitogen-activated protein kinase 12	Homo sapiens (human)	Ki	0.0008	1	1
Mitogen-activated protein kinase 13	Homo sapiens (human)	IC50	0.0577	4	4
Mitogen-activated protein kinase 13	Homo sapiens (human)	Ki	0.0008	1	1
Mitogen-activated protein kinase 14	Homo sapiens (human)	IC50	1.8567	15	17
Mitogen-activated protein kinase 14	Homo sapiens (human)	Ki	0.0008	1	1
Mitogen-activated protein kinase 14	Mus musculus (house mouse)	IC50	0.0442	2	4
Mitogen-activated protein kinase 9	Homo sapiens (human)	IC50	200.0000	1	1
MPI protein	Homo sapiens (human)	IC50	0.2905	2	2
Mu-type opioid receptor	Rattus norvegicus (Norway rat)	IC50	0.0008	1	1
Multidrug resistance-associated protein 4	Homo sapiens (human)	IC50	114.1970	1	10
Myeloperoxidase	Homo sapiens (human)	IC50	0.4200	1	1
NAD-dependent protein deacylase sirtuin-5, mitochondrial	Homo sapiens (human)	IC50	1.6000	1	1
neutrophil cytosol factor 1	Homo sapiens (human)	IC50	0.3900	1	1
Neutrophil cytosol factor 1	Homo sapiens (human)	Ki	125.0000	3	3
Nitric oxide synthase, inducible	Mus musculus (house mouse)	IC50	50.0000	1	1
Non-receptor tyrosine-protein kinase TYK2	Homo sapiens (human)	IC50	0.0533	3	3
Nuclear factor NF-kappa-B p105 subunit	Homo sapiens (human)	IC50	49.6000	1	1
perilipin-1	Homo sapiens (human)	IC50	3.4100	1	1
perilipin-5	Homo sapiens (human)	IC50	1.1010	1	1
Phosphatidylinositol 3,4,5-trisphosphate 3-phosphatase and dual-specificity protein phosphatase PTEN	Homo sapiens (human)	IC50	13.3000	1	1
phosphoethanolamine/phosphocholine phosphatase isoform 1	Homo sapiens (human)	IC50	0.1110	1	1
Phospholipase A2	Homo sapiens (human)	IC50	0.3668	6	6
Phospholipase A2	Mus musculus (house mouse)	IC50	0.1400	2	2
Phospholipase A2 group V	Homo sapiens (human)	IC50	0.2738	5	5
Phospholipase A2 group V	Mus musculus (house mouse)	IC50	0.7500	2	2
Phospholipase A2, major isoenzyme	Sus scrofa (pig)	IC50	0.0480	2	2
Phospholipase A2, membrane associated	Homo sapiens (human)	IC50	0.0527	11	11
Phospholipase A2, membrane associated	Mus musculus (house mouse)	IC50	0.0700	2	2
phosphomannomutase 2	Homo sapiens (human)	IC50	0.6720	1	1
Platelet-derived growth factor receptor beta	Homo sapiens (human)	IC50	1.0000	1	1
Polyunsaturated fatty acid 5-lipoxygenase	Homo sapiens (human)	IC50	0.1000	1	1
Polyunsaturated fatty acid 5-lipoxygenase	Rattus norvegicus (Norway rat)	IC50	0.1650	2	2
Polyunsaturated fatty acid lipoxygenase ALOX15	Homo sapiens (human)	IC50	14.0000	1	1
Potassium voltage-gated channel subfamily H member 2	Homo sapiens (human)	IC50	20.0000	1	1
Procathepsin L	Homo sapiens (human)	IC50	0.6700	1	1
procathepsin L isoform 1 preproprotein	Homo sapiens (human)	IC50	50.0000	2	2
Progesterone receptor	Homo sapiens (human)	IC50	4.5161	7	8
Progesterone receptor	Homo sapiens (human)	Ki	5.4286	7	7
Prostaglandin G/H synthase 1	Homo sapiens (human)	IC50	100.0000	1	1
Prostaglandin G/H synthase 1	Bos taurus (cattle)	IC50	2.1000	1	1
Prostaglandin G/H synthase 2	Homo sapiens (human)	IC50	100.0000	1	1
Prostaglandin G/H synthase 2	Homo sapiens (human)	Ki	5.0000	1	2
Proto-oncogene tyrosine-protein kinase Src	Homo sapiens (human)	IC50	3.0000	2	2
Putative inactive group IIC secretory phospholipase A2	Homo sapiens (human)	IC50	0.1225	2	2
RAC-gamma serine/threonine-protein kinase	Homo sapiens (human)	IC50	5.0000	1	1
Receptor-type tyrosine-protein phosphatase epsilon	Homo sapiens (human)	IC50	500.0000	1	1
Receptor-type tyrosine-protein phosphatase eta	Homo sapiens (human)	IC50	111.5000	1	1
Regulator of G-protein signaling 17	Homo sapiens (human)	IC50	27.9338	5	5
Replicase polyprotein 1a	Severe acute respiratory syndrome-related coronavirus	IC50	0.6700	1	1
Replicase polyprotein 1ab	Betacoronavirus England 1	IC50	5.3350	2	2
Replicase polyprotein 1ab	Human coronavirus 229E	IC50	0.6700	1	1
Replicase polyprotein 1ab	Severe acute respiratory syndrome coronavirus 2	IC50	2.2750	14	16
Replicase polyprotein 1ab	Severe acute respiratory syndrome-related coronavirus	IC50	4.4920	3	5
Replicase polyprotein 1ab	Severe acute respiratory syndrome coronavirus 2	Ki	4.2000	1	1
Replicase polyprotein 1ab	Severe acute respiratory syndrome-related coronavirus	Ki	4.2000	2	2
Rho-associated protein kinase 1	Homo sapiens (human)	IC50	5.0000	1	1
RNA polymerase beta subunit (EC 2.7.7.6), partial	Escherichia coli	IC50	11.6872	1	1
Serine/threonine-protein kinase pim-1	Homo sapiens (human)	IC50	5.0000	1	1
Sodium-dependent dopamine transporter	Homo sapiens (human)	IC50	8.0980	1	1
Sodium-dependent dopamine transporter	Homo sapiens (human)	Ki	6.4340	1	1
Sodium-dependent noradrenaline transporter	Homo sapiens (human)	IC50	20.4040	1	1
Sodium-dependent noradrenaline transporter	Homo sapiens (human)	Ki	20.2360	1	1
Sodium-dependent serotonin transporter	Rattus norvegicus (Norway rat)	IC50	27.1000	1	1
Solute carrier organic anion transporter family member 1B1	Homo sapiens (human)	IC50	2.9512	1	1
Solute carrier organic anion transporter family member 1B1	Homo sapiens (human)	Ki	1.6200	1	1
Solute carrier organic anion transporter family member 1B3	Homo sapiens (human)	IC50	1.1482	1	1
Solute carrier organic anion transporter family member 1B3	Homo sapiens (human)	Ki	0.8700	1	1
Spike glycoprotein	Betacoronavirus England 1	IC50	0.6700	1	1
Spike glycoprotein	Severe acute respiratory syndrome-related coronavirus	IC50	0.6700	1	1
Structural capsid protein	Human immunodeficiency virus 1	IC50	0.0467	1	1
Sulfhydryl oxidase 1	Homo sapiens (human)	IC50	5.4000	1	1
Telomerase reverse transcriptase	Homo sapiens (human)	IC50	0.7800	1	1
Thromboxane-A synthase	Rattus norvegicus (Norway rat)	IC50	0.0900	1	1
Thromboxane-A synthase	Homo sapiens (human)	IC50	0.0495	2	2
Toxin B	Clostridioides difficile	IC50	0.0172	1	1
TPA: protein transporter TIM10	Saccharomyces cerevisiae S288C	IC50	5.2900	2	2
TPA: protein transporter TIM23	Saccharomyces cerevisiae S288C	IC50	7.8900	2	2
Transient receptor potential cation channel subfamily V member 2	Rattus norvegicus (Norway rat)	IC50	10.0000	2	2
Transmembrane protease serine 2	Homo sapiens (human)	IC50	0.6700	1	1
Tryptophan 2,3-dioxygenase	Homo sapiens (human)	IC50	100.0000	1	1
Tyrosine-protein kinase ABL1	Homo sapiens (human)	IC50	1.0000	1	1
Tyrosine-protein kinase ABL2	Homo sapiens (human)	IC50	1.0000	1	1
Tyrosine-protein kinase ITK/TSK	Homo sapiens (human)	IC50	10.0000	1	1
Tyrosine-protein kinase JAK1	Homo sapiens (human)	IC50	0.0203	6	6
Tyrosine-protein kinase JAK2	Homo sapiens (human)	IC50	0.0745	6	6
Tyrosine-protein kinase JAK3	Homo sapiens (human)	IC50	0.0220	3	3
Tyrosine-protein kinase Lck	Homo sapiens (human)	IC50	5.8000	1	1
Tyrosine-protein kinase SYK	Homo sapiens (human)	IC50	5.0000	1	1
Tyrosine-protein kinase ZAP-70	Homo sapiens (human)	IC50	5.0000	1	1
Tyrosine-protein phosphatase non-receptor type 1	Homo sapiens (human)	IC50	4.8680	5	5
Tyrosine-protein phosphatase non-receptor type 11	Homo sapiens (human)	IC50	3.5667	3	3
Tyrosine-protein phosphatase non-receptor type 2	Homo sapiens (human)	IC50	20.9000	2	2
Tyrosine-protein phosphatase non-receptor type 6	Homo sapiens (human)	IC50	15.4500	2	2
Tyrosine-protein phosphatase non-receptor type 7	Homo sapiens (human)	IC50	75.7000	1	1
Ubiquitin carboxyl-terminal hydrolase 15	Homo sapiens (human)	IC50	31.4000	1	5
Ubiquitin carboxyl-terminal hydrolase 2	Homo sapiens (human)	IC50	31.4000	1	5
Ubiquitin carboxyl-terminal hydrolase isozyme L1	Homo sapiens (human)	IC50	31.4000	1	5
Ubiquitin carboxyl-terminal hydrolase isozyme L3	Homo sapiens (human)	IC50	31.4000	1	5
Ubiquitin carboxyl-terminal hydrolase isozyme L5	Homo sapiens (human)	IC50	31.4000	1	5
UDP-glucose 4-epimerase	Homo sapiens (human)	IC50	0.0140	1	1
Uracil nucleotide/cysteinyl leukotriene receptor	Homo sapiens (human)	IC50	30.0000	1	1
Urease subunit alpha	Helicobacter pylori 26695	IC50	30.4725	4	4
Urease subunit alpha	Helicobacter pylori 26695	Ki	0.2260	1	1
Urease subunit beta	Helicobacter pylori 26695	IC50	30.4725	4	4
Urease subunit beta	Helicobacter pylori 26695	Ki	0.2260	1	1
Vascular cell adhesion protein 1	Homo sapiens (human)	IC50	50.0000	1	1
Vascular endothelial growth factor receptor 2	Homo sapiens (human)	IC50	5.0000	1	1

Activation Measurements

Protein	Taxonomy	Measurement	Average (mM)	Bioassay(s)	Drugs
3-phosphoinositide-dependent protein kinase 1	Homo sapiens (human)	Kd	10.0000	2	2
5-hydroxytryptamine receptor 1B	Homo sapiens (human)	EC50	0.0157	1	1
5-hydroxytryptamine receptor 1D	Homo sapiens (human)	EC50	0.0057	2	2
5'-AMP-activated protein kinase catalytic subunit alpha-1	Homo sapiens (human)	Kd	10.0000	2	2
5'-AMP-activated protein kinase catalytic subunit alpha-2	Homo sapiens (human)	EC50	0.0168	1	2
5'-AMP-activated protein kinase catalytic subunit alpha-2	Homo sapiens (human)	Kd	10.0000	2	2
5'-AMP-activated protein kinase subunit beta-1	Homo sapiens (human)	EC50	0.0168	1	2
5'-AMP-activated protein kinase subunit gamma-1	Homo sapiens (human)	EC50	0.0168	1	2
Activated CDC42 kinase 1	Homo sapiens (human)	Kd	10.0000	2	2
Activin receptor type-1	Homo sapiens (human)	Kd	10.0000	2	2
Activin receptor type-1B	Homo sapiens (human)	Kd	10.0000	2	2
Activin receptor type-2A	Homo sapiens (human)	Kd	10.0000	2	2
Activin receptor type-2B	Homo sapiens (human)	Kd	10.0000	2	2
ALK tyrosine kinase receptor	Homo sapiens (human)	Kd	10.0000	2	2
Alpha-2A adrenergic receptor	Rattus norvegicus (Norway rat)	Kd	0.0070	1	2
Alpha-2B adrenergic receptor	Rattus norvegicus (Norway rat)	Kd	0.0070	1	2
Alpha-2C adrenergic receptor	Rattus norvegicus (Norway rat)	Kd	0.0070	1	2
Angiopoietin-1 receptor	Homo sapiens (human)	Kd	10.0000	2	2
Angiotensin-converting enzyme 2	Homo sapiens (human)	EC50	4.6700	1	1
Ankyrin repeat and protein kinase domain-containing protein 1	Homo sapiens (human)	Kd	10.0000	2	2
AP2-associated protein kinase 1	Homo sapiens (human)	Kd	10.0000	2	2
Atypical kinase COQ8A, mitochondrial	Homo sapiens (human)	Kd	10.0000	2	2
Atypical kinase COQ8B, mitochondrial	Homo sapiens (human)	Kd	10.0000	2	2
Aurora kinase A	Homo sapiens (human)	Kd	10.0000	2	2
Aurora kinase B	Homo sapiens (human)	Kd	10.0000	2	2
Aurora kinase C	Homo sapiens (human)	Kd	10.0000	2	2
BDNF/NT-3 growth factors receptor	Homo sapiens (human)	Kd	10.0000	2	2
BMP-2-inducible protein kinase	Homo sapiens (human)	Kd	10.0000	2	2
Bone morphogenetic protein receptor type-1A	Homo sapiens (human)	Kd	10.0000	2	2
Bone morphogenetic protein receptor type-1B	Homo sapiens (human)	Kd	10.0000	1	1
Bone morphogenetic protein receptor type-2	Homo sapiens (human)	Kd	10.0000	2	2
Calcium-dependent protein kinase 1	Plasmodium falciparum 3D7	Kd	10.0000	1	1
Calcium/calmodulin-dependent protein kinase kinase 1	Homo sapiens (human)	Kd	10.0000	2	2
Calcium/calmodulin-dependent protein kinase kinase 2	Homo sapiens (human)	Kd	10.0000	2	2
Calcium/calmodulin-dependent protein kinase type 1	Homo sapiens (human)	Kd	10.0000	2	2
Calcium/calmodulin-dependent protein kinase type 1D	Homo sapiens (human)	Kd	10.0000	2	2
Calcium/calmodulin-dependent protein kinase type 1G	Homo sapiens (human)	Kd	10.0000	2	2
Calcium/calmodulin-dependent protein kinase type II subunit alpha	Homo sapiens (human)	Kd	10.0000	2	2
Calcium/calmodulin-dependent protein kinase type II subunit beta	Homo sapiens (human)	Kd	10.0000	2	2
Calcium/calmodulin-dependent protein kinase type II subunit delta	Homo sapiens (human)	Kd	10.0000	2	2
Calcium/calmodulin-dependent protein kinase type II subunit gamma	Homo sapiens (human)	Kd	10.0000	2	2
Calcium/calmodulin-dependent protein kinase type IV	Homo sapiens (human)	Kd	10.0000	2	2
cAMP-dependent protein kinase catalytic subunit alpha	Homo sapiens (human)	Kd	10.0000	2	2
cAMP-dependent protein kinase catalytic subunit beta	Homo sapiens (human)	Kd	10.0000	2	2
cAMP-dependent protein kinase catalytic subunit PRKX	Homo sapiens (human)	Kd	10.0000	2	2
Casein kinase I isoform alpha	Homo sapiens (human)	Kd	10.0000	1	1
Casein kinase I isoform alpha-like	Homo sapiens (human)	Kd	10.0000	2	2
Casein kinase I isoform delta	Homo sapiens (human)	Kd	10.0000	2	2
Casein kinase I isoform epsilon	Homo sapiens (human)	Kd	10.0000	2	2
Casein kinase I isoform gamma-1	Homo sapiens (human)	Kd	10.0000	2	2
Casein kinase I isoform gamma-2	Homo sapiens (human)	Kd	10.0000	2	2
Casein kinase I isoform gamma-3	Homo sapiens (human)	Kd	10.0000	2	2
Casein kinase II subunit alpha	Homo sapiens (human)	Kd	10.0000	2	2
Casein kinase II subunit alpha'	Homo sapiens (human)	Kd	10.0000	2	2
Cell division control protein 2 homolog	Plasmodium falciparum 3D7	Kd	10.0000	1	1
cGMP-dependent protein kinase 1	Homo sapiens (human)	Kd	10.0000	2	2
cGMP-dependent protein kinase 2	Homo sapiens (human)	Kd	10.0000	2	2
Citron Rho-interacting kinase	Homo sapiens (human)	Kd	10.0000	2	2
Cyclin-dependent kinase 11A	Homo sapiens (human)	Kd	10.0000	2	2
Cyclin-dependent kinase 11B	Homo sapiens (human)	Kd	10.0000	2	2
Cyclin-dependent kinase 13	Homo sapiens (human)	Kd	10.0000	1	1
Cyclin-dependent kinase 14	Homo sapiens (human)	Kd	10.0000	2	2
Cyclin-dependent kinase 15	Homo sapiens (human)	Kd	10.0000	1	1
Cyclin-dependent kinase 16	Homo sapiens (human)	Kd	10.0000	2	2
Cyclin-dependent kinase 17	Homo sapiens (human)	Kd	10.0000	2	2
Cyclin-dependent kinase 18	Homo sapiens (human)	Kd	10.0000	2	2
Cyclin-dependent kinase 19	Homo sapiens (human)	Kd	10.0000	2	2
Cyclin-dependent kinase 2	Homo sapiens (human)	Kd	10.0000	2	2
Cyclin-dependent kinase 3	Homo sapiens (human)	Kd	10.0000	2	2
Cyclin-dependent kinase 4	Homo sapiens (human)	Kd	10.0000	2	2
Cyclin-dependent kinase 7	Homo sapiens (human)	Kd	10.0000	2	2
Cyclin-dependent kinase 8	Homo sapiens (human)	Kd	10.0000	2	2
Cyclin-dependent kinase 9	Homo sapiens (human)	Kd	10.0000	2	2
Cyclin-dependent kinase-like 1	Homo sapiens (human)	Kd	10.0000	1	1
Cyclin-dependent kinase-like 2	Homo sapiens (human)	Kd	10.0000	1	1
Cyclin-dependent kinase-like 3	Homo sapiens (human)	Kd	10.0000	1	1
Cyclin-dependent kinase-like 5	Homo sapiens (human)	Kd	10.0000	1	1
Cyclin-dependent-like kinase 5	Homo sapiens (human)	Kd	10.0000	2	2
Cyclin-G-associated kinase	Homo sapiens (human)	Kd	10.0000	2	2
Cytochrome P450 3A5	Homo sapiens (human)	Kd	0.1000	1	1
Cytoplasmic tyrosine-protein kinase BMX	Homo sapiens (human)	Kd	10.0000	2	2
Death-associated protein kinase 1	Homo sapiens (human)	Kd	10.0000	2	2
Death-associated protein kinase 2	Homo sapiens (human)	Kd	10.0000	2	2
Death-associated protein kinase 3	Homo sapiens (human)	Kd	10.0000	3	3
Discoidin domain-containing receptor 2	Homo sapiens (human)	Kd	10.0000	2	2
Dual serine/threonine and tyrosine protein kinase	Homo sapiens (human)	Kd	10.0000	1	1
Dual specificity mitogen-activated protein kinase kinase 1	Homo sapiens (human)	Kd	10.0000	2	2
Dual specificity mitogen-activated protein kinase kinase 2	Homo sapiens (human)	Kd	10.0000	2	2
Dual specificity mitogen-activated protein kinase kinase 3	Homo sapiens (human)	Kd	10.0000	2	2
Dual specificity mitogen-activated protein kinase kinase 4	Homo sapiens (human)	Kd	10.0000	2	2
Dual specificity mitogen-activated protein kinase kinase 5	Homo sapiens (human)	Kd	10.0000	1	1
Dual specificity mitogen-activated protein kinase kinase 6	Homo sapiens (human)	Kd	10.0000	2	2
Dual specificity mitogen-activated protein kinase kinase 7	Homo sapiens (human)	Kd	10.0000	1	1
Dual specificity protein kinase CLK1	Homo sapiens (human)	Kd	10.0000	2	2
Dual specificity protein kinase CLK2	Homo sapiens (human)	Kd	10.0000	2	2
Dual specificity protein kinase CLK3	Homo sapiens (human)	Kd	10.0000	2	2
Dual specificity protein kinase CLK4	Homo sapiens (human)	Kd	10.0000	2	2
Dual specificity protein kinase TTK	Homo sapiens (human)	Kd	10.0000	2	2
Dual specificity testis-specific protein kinase 1	Homo sapiens (human)	Kd	10.0000	2	2
Dual specificity tyrosine-phosphorylation-regulated kinase 1A	Homo sapiens (human)	Kd	10.0000	1	1
Dual specificity tyrosine-phosphorylation-regulated kinase 1B	Homo sapiens (human)	Kd	10.0000	2	2
Dual specificity tyrosine-phosphorylation-regulated kinase 2	Homo sapiens (human)	Kd	10.0000	1	1
eIF-2-alpha kinase GCN2	Homo sapiens (human)	Kd	10.0000	2	2
Ephrin type-A receptor 1	Homo sapiens (human)	Kd	7.3500	2	2
Ephrin type-A receptor 2	Homo sapiens (human)	Kd	7.3667	3	3
Ephrin type-A receptor 3	Homo sapiens (human)	Kd	10.0000	2	2
Ephrin type-A receptor 4	Homo sapiens (human)	Kd	10.0000	3	3
Ephrin type-A receptor 5	Homo sapiens (human)	Kd	7.3000	3	3
Ephrin type-A receptor 6	Homo sapiens (human)	Kd	10.0000	2	2
Ephrin type-A receptor 7	Homo sapiens (human)	Kd	10.0000	2	2
Ephrin type-A receptor 8	Homo sapiens (human)	Kd	7.7000	3	3
Ephrin type-B receptor 1	Homo sapiens (human)	Kd	5.9333	3	3
Ephrin type-B receptor 2	Homo sapiens (human)	Kd	10.0000	2	2
Ephrin type-B receptor 3	Homo sapiens (human)	Kd	10.0000	2	2
Ephrin type-B receptor 4	Homo sapiens (human)	Kd	7.0000	3	3
Ephrin type-B receptor 6	Homo sapiens (human)	Kd	10.0000	1	1
Epidermal growth factor receptor	Homo sapiens (human)	Kd	10.0000	22	22
Epithelial discoidin domain-containing receptor 1	Homo sapiens (human)	Kd	1.1000	2	2
Eukaryotic translation initiation factor 2-alpha kinase 1	Homo sapiens (human)	Kd	10.0000	1	1
Fibroblast growth factor receptor 1	Homo sapiens (human)	Kd	10.0000	2	2
Fibroblast growth factor receptor 2	Homo sapiens (human)	Kd	10.0000	2	2
Fibroblast growth factor receptor 3	Homo sapiens (human)	Kd	10.0000	4	4
Fibroblast growth factor receptor 4	Homo sapiens (human)	Kd	10.0000	2	2
Focal adhesion kinase 1	Homo sapiens (human)	Kd	10.0000	2	2
G protein-coupled receptor kinase 4	Homo sapiens (human)	Kd	10.0000	1	1
G-protein coupled bile acid receptor 1	Homo sapiens (human)	EC50	10.0000	1	1
Gamma-butyrobetaine dioxygenase	Homo sapiens (human)	Kd	4.1000	2	2
Glucocorticoid receptor	Homo sapiens (human)	EC50	0.0259	46	47
Glucocorticoid receptor	Mus musculus (house mouse)	EC50	0.0046	2	2
Glucocorticoid receptor	Rattus norvegicus (Norway rat)	EC50	0.0102	2	2
Glucocorticoid receptor	Homo sapiens (human)	Kd	0.0290	1	1
Glutamine synthetase	Homo sapiens (human)	EC50	0.0320	1	1
Glycogen synthase kinase-3 alpha	Homo sapiens (human)	Kd	10.0000	2	2
Glycogen synthase kinase-3 beta	Homo sapiens (human)	Kd	10.0000	2	2
Heat shock factor protein 1	Homo sapiens (human)	EC50	1.8500	2	2
Hepatocyte growth factor receptor	Homo sapiens (human)	Kd	10.0000	4	4
hexokinase HKDC1	Homo sapiens (human)	EC50	38.8000	1	1
hexokinase-1 isoform HKI	Homo sapiens (human)	EC50	41.9000	1	1
High affinity nerve growth factor receptor	Homo sapiens (human)	Kd	10.0000	2	2
Histamine H1 receptor	Cavia porcellus (domestic guinea pig)	EC50	0.0026	1	1
Homeodomain-interacting protein kinase 1	Homo sapiens (human)	Kd	10.0000	1	1
Homeodomain-interacting protein kinase 2	Homo sapiens (human)	Kd	10.0000	1	1
Homeodomain-interacting protein kinase 3	Homo sapiens (human)	Kd	10.0000	1	1
Homeodomain-interacting protein kinase 4	Homo sapiens (human)	Kd	10.0000	1	1
Hormonally up-regulated neu tumor-associated kinase	Homo sapiens (human)	Kd	10.0000	1	1
Inhibitor of nuclear factor kappa-B kinase subunit alpha	Homo sapiens (human)	Kd	10.0000	1	1
Inhibitor of nuclear factor kappa-B kinase subunit beta	Homo sapiens (human)	Kd	10.0000	1	1
Inhibitor of nuclear factor kappa-B kinase subunit epsilon	Homo sapiens (human)	Kd	10.0000	2	2
Insulin receptor	Homo sapiens (human)	Kd	10.0000	2	2
Insulin receptor-related protein	Homo sapiens (human)	Kd	10.0000	2	2
Insulin-like growth factor 1 receptor	Homo sapiens (human)	Kd	10.0000	2	2
Interferon-induced, double-stranded RNA-activated protein kinase	Homo sapiens (human)	Kd	10.0000	2	2
Interleukin-1 receptor-associated kinase 1	Homo sapiens (human)	Kd	10.0000	1	1
Interleukin-1 receptor-associated kinase 3	Homo sapiens (human)	Kd	10.0000	2	2
Interleukin-1 receptor-associated kinase 4	Homo sapiens (human)	Kd	10.0000	1	1
L-ornithine N(5)-monooxygenase	Aspergillus fumigatus Af293	Kd	1.4000	2	2
Leucine-rich repeat serine/threonine-protein kinase 2	Homo sapiens (human)	Kd	10.0000	2	2
Leukocyte tyrosine kinase receptor	Homo sapiens (human)	Kd	10.0000	2	2
Leukotriene C4 synthase	Cavia porcellus (domestic guinea pig)	Kd	10.0000	1	1
LIM domain kinase 1	Homo sapiens (human)	Kd	10.0000	2	2
LIM domain kinase 2	Homo sapiens (human)	Kd	10.0000	2	2
Macrophage colony-stimulating factor 1 receptor	Homo sapiens (human)	Kd	2.6000	2	2
Macrophage-stimulating protein receptor	Homo sapiens (human)	Kd	10.0000	1	1
MAP kinase-activated protein kinase 2	Homo sapiens (human)	Kd	10.0000	2	2
MAP kinase-activated protein kinase 5	Homo sapiens (human)	Kd	10.0000	2	2
MAP kinase-interacting serine/threonine-protein kinase 1	Homo sapiens (human)	Kd	10.0000	2	2
MAP kinase-interacting serine/threonine-protein kinase 2	Homo sapiens (human)	Kd	10.0000	2	2
MAP/microtubule affinity-regulating kinase 3	Homo sapiens (human)	Kd	10.0000	2	2
MAP/microtubule affinity-regulating kinase 4	Homo sapiens (human)	Kd	10.0000	2	2
Mast/stem cell growth factor receptor Kit	Homo sapiens (human)	Kd	10.0000	15	15
Maternal embryonic leucine zipper kinase	Homo sapiens (human)	Kd	10.0000	2	2
Megakaryocyte-associated tyrosine-protein kinase	Homo sapiens (human)	Kd	10.0000	1	1
Membrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinase	Homo sapiens (human)	Kd	10.0000	2	2
Microtubule-associated serine/threonine-protein kinase 1	Homo sapiens (human)	Kd	10.0000	1	1
Mineralocorticoid receptor	Homo sapiens (human)	EC50	0.0023	3	3
Misshapen-like kinase 1	Homo sapiens (human)	Kd	10.0000	1	1
Mitogen-activated protein kinase 1	Homo sapiens (human)	Kd	10.0000	2	2
Mitogen-activated protein kinase 10	Homo sapiens (human)	Kd	10.0000	2	2
Mitogen-activated protein kinase 11	Homo sapiens (human)	Kd	0.1027	3	3
Mitogen-activated protein kinase 12	Homo sapiens (human)	Kd	10.0000	3	3
Mitogen-activated protein kinase 13	Homo sapiens (human)	Kd	10.0000	1	1
Mitogen-activated protein kinase 14	Homo sapiens (human)	Kd	0.0029	4	4
Mitogen-activated protein kinase 15	Homo sapiens (human)	Kd	10.0000	2	2
Mitogen-activated protein kinase 3	Homo sapiens (human)	Kd	10.0000	2	2
Mitogen-activated protein kinase 4	Homo sapiens (human)	Kd	10.0000	2	2
Mitogen-activated protein kinase 6	Homo sapiens (human)	Kd	10.0000	2	2
Mitogen-activated protein kinase 7	Homo sapiens (human)	Kd	10.0000	2	2
Mitogen-activated protein kinase 8	Homo sapiens (human)	Kd	10.0000	2	2
Mitogen-activated protein kinase 9	Homo sapiens (human)	Kd	10.0000	2	2
Mitogen-activated protein kinase kinase kinase 1	Homo sapiens (human)	Kd	10.0000	1	1
Mitogen-activated protein kinase kinase kinase 10	Homo sapiens (human)	Kd	10.0000	2	2
Mitogen-activated protein kinase kinase kinase 11	Homo sapiens (human)	Kd	10.0000	2	2
Mitogen-activated protein kinase kinase kinase 12	Homo sapiens (human)	Kd	10.0000	1	1
Mitogen-activated protein kinase kinase kinase 13	Homo sapiens (human)	Kd	10.0000	1	1
Mitogen-activated protein kinase kinase kinase 15	Homo sapiens (human)	Kd	10.0000	1	1
Mitogen-activated protein kinase kinase kinase 19	Homo sapiens (human)	Kd	10.0000	1	1
Mitogen-activated protein kinase kinase kinase 2	Homo sapiens (human)	Kd	10.0000	1	1
Mitogen-activated protein kinase kinase kinase 20	Homo sapiens (human)	Kd	10.0000	2	2
Mitogen-activated protein kinase kinase kinase 3	Homo sapiens (human)	Kd	10.0000	1	1
Mitogen-activated protein kinase kinase kinase 4	Homo sapiens (human)	Kd	10.0000	2	2
Mitogen-activated protein kinase kinase kinase 5	Homo sapiens (human)	Kd	10.0000	2	2
Mitogen-activated protein kinase kinase kinase 6	Homo sapiens (human)	Kd	10.0000	1	1
Mitogen-activated protein kinase kinase kinase 7	Homo sapiens (human)	Kd	10.0000	1	1
Mitogen-activated protein kinase kinase kinase 9	Homo sapiens (human)	Kd	10.0000	2	2
Mitogen-activated protein kinase kinase kinase kinase 1	Homo sapiens (human)	Kd	10.0000	2	2
Mitogen-activated protein kinase kinase kinase kinase 2	Homo sapiens (human)	Kd	10.0000	1	1
Mitogen-activated protein kinase kinase kinase kinase 3	Homo sapiens (human)	Kd	10.0000	2	2
Mitogen-activated protein kinase kinase kinase kinase 4	Homo sapiens (human)	Kd	10.0000	2	2
Mitogen-activated protein kinase kinase kinase kinase 5	Homo sapiens (human)	Kd	10.0000	2	2
Muscle, skeletal receptor tyrosine-protein kinase	Homo sapiens (human)	Kd	10.0000	2	2
Myosin light chain kinase 2, skeletal/cardiac muscle	Homo sapiens (human)	Kd	10.0000	2	2
Myosin light chain kinase 3	Homo sapiens (human)	Kd	10.0000	1	1
Myosin light chain kinase family member 4	Homo sapiens (human)	Kd	10.0000	2	2
Myosin light chain kinase, smooth muscle	Gallus gallus (chicken)	Kd	10.0000	1	1
Myosin light chain kinase, smooth muscle	Homo sapiens (human)	Kd	10.0000	2	2
Myosin-IIIa	Homo sapiens (human)	Kd	10.0000	2	2
Myosin-IIIb	Homo sapiens (human)	Kd	10.0000	2	2
Myotonin-protein kinase	Homo sapiens (human)	Kd	10.0000	2	2
Nociceptin receptor	Rattus norvegicus (Norway rat)	EC50	0.0034	1	1
Non-receptor tyrosine-protein kinase TNK1	Homo sapiens (human)	Kd	10.0000	2	2
Non-receptor tyrosine-protein kinase TYK2	Homo sapiens (human)	Kd	10.0000	3	3
NT-3 growth factor receptor	Homo sapiens (human)	Kd	10.0000	2	2
NUAK family SNF1-like kinase 1	Homo sapiens (human)	Kd	10.0000	2	2
NUAK family SNF1-like kinase 2	Homo sapiens (human)	Kd	10.0000	2	2
Nuclear receptor subfamily 1 group I member 2	Homo sapiens (human)	EC50	12.2600	3	5
Nuclear receptor subfamily 1 group I member 2	Rattus norvegicus (Norway rat)	EC50	4.8000	1	3
Nuclear receptor subfamily 4 group A member 1	Homo sapiens (human)	Kd	0.3000	3	3
ORF73	Human gammaherpesvirus 8	EC50	75.0000	1	1
Peripheral plasma membrane protein CASK	Homo sapiens (human)	Kd	10.0000	1	1
Phosphatidylinositol 4-kinase beta	Homo sapiens (human)	Kd	10.0000	1	1
Phosphatidylinositol 4-phosphate 3-kinase C2 domain-containing subunit beta	Homo sapiens (human)	Kd	10.0000	1	1
Phosphatidylinositol 4-phosphate 3-kinase C2 domain-containing subunit gamma	Homo sapiens (human)	Kd	10.0000	1	1
Phosphatidylinositol 4-phosphate 5-kinase type-1 alpha	Homo sapiens (human)	Kd	10.0000	2	2
Phosphatidylinositol 4-phosphate 5-kinase type-1 gamma	Homo sapiens (human)	Kd	10.0000	1	1
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform	Homo sapiens (human)	Kd	10.0000	12	12
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform	Homo sapiens (human)	Kd	10.0000	1	1
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform	Homo sapiens (human)	Kd	10.0000	1	1
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform	Homo sapiens (human)	Kd	10.0000	1	1
Phosphatidylinositol 5-phosphate 4-kinase type-2 beta	Homo sapiens (human)	Kd	10.0000	2	2
Phosphatidylinositol 5-phosphate 4-kinase type-2 gamma	Homo sapiens (human)	Kd	10.0000	1	1
Phosphorylase b kinase gamma catalytic chain, liver/testis isoform	Homo sapiens (human)	Kd	10.0000	2	2
Phosphorylase b kinase gamma catalytic chain, skeletal muscle/heart isoform	Homo sapiens (human)	Kd	10.0000	2	2
Platelet-derived growth factor receptor alpha	Homo sapiens (human)	Kd	9.4000	2	2
Platelet-derived growth factor receptor beta	Homo sapiens (human)	Kd	5.8900	3	3
Procathepsin L	Homo sapiens (human)	EC50	4.6700	1	1
Progesterone receptor	Homo sapiens (human)	Kd	0.0001	1	1
Prostaglandin G/H synthase 2	Homo sapiens (human)	Kd	10.0000	1	1
Protein kinase C delta type	Homo sapiens (human)	Kd	10.0000	2	2
Protein kinase C epsilon type	Homo sapiens (human)	Kd	10.0000	2	2
Protein kinase C eta type	Homo sapiens (human)	Kd	10.0000	2	2
Protein kinase C iota type	Homo sapiens (human)	Kd	10.0000	1	1
Protein kinase C theta type	Homo sapiens (human)	Kd	10.0000	2	2
Protein-tyrosine kinase 2-beta	Homo sapiens (human)	Kd	10.0000	2	2
Protein-tyrosine kinase 6	Homo sapiens (human)	Kd	10.0000	2	2
Proto-oncogene tyrosine-protein kinase receptor Ret	Homo sapiens (human)	Kd	10.0000	6	6
Proto-oncogene tyrosine-protein kinase ROS	Homo sapiens (human)	Kd	10.0000	2	2
Proto-oncogene tyrosine-protein kinase Src	Homo sapiens (human)	Kd	3.9933	3	3
RAC-alpha serine/threonine-protein kinase	Homo sapiens (human)	Kd	10.0000	2	2
RAC-beta serine/threonine-protein kinase	Homo sapiens (human)	Kd	10.0000	2	2
RAC-gamma serine/threonine-protein kinase	Homo sapiens (human)	Kd	10.0000	2	2
RAF proto-oncogene serine/threonine-protein kinase	Homo sapiens (human)	Kd	10.0000	2	2
Receptor tyrosine-protein kinase erbB-2	Homo sapiens (human)	Kd	10.0000	2	2
Receptor tyrosine-protein kinase erbB-3	Homo sapiens (human)	Kd	10.0000	1	1
Receptor tyrosine-protein kinase erbB-4	Homo sapiens (human)	Kd	10.0000	1	1
Receptor-interacting serine/threonine-protein kinase 1	Homo sapiens (human)	Kd	10.0000	2	2
Receptor-interacting serine/threonine-protein kinase 2	Homo sapiens (human)	Kd	10.0000	2	2
Receptor-interacting serine/threonine-protein kinase 4	Homo sapiens (human)	Kd	10.0000	1	1
Receptor-type tyrosine-protein kinase FLT3	Homo sapiens (human)	Kd	10.0000	12	12
Replicase polyprotein 1a	Severe acute respiratory syndrome-related coronavirus	EC50	4.6700	1	1
Replicase polyprotein 1ab	Betacoronavirus England 1	EC50	4.6700	1	1
Replicase polyprotein 1ab	Human coronavirus 229E	EC50	4.6700	1	1
Replicase polyprotein 1ab	Severe acute respiratory syndrome coronavirus 2	EC50	4.6700	2	2
Replicase polyprotein 1ab	Severe acute respiratory syndrome-related coronavirus	EC50	4.6700	2	2
Rho-associated protein kinase 1	Homo sapiens (human)	Kd	10.0000	1	1
Rho-associated protein kinase 2	Homo sapiens (human)	Kd	10.0000	1	1
Rhodopsin kinase GRK1	Homo sapiens (human)	Kd	10.0000	1	1
Rhodopsin kinase GRK7	Homo sapiens (human)	Kd	10.0000	1	1
Ribosomal protein S6 kinase alpha-1	Homo sapiens (human)	Kd	10.0000	4	4
Ribosomal protein S6 kinase alpha-2	Homo sapiens (human)	Kd	10.0000	4	4
Ribosomal protein S6 kinase alpha-3	Homo sapiens (human)	Kd	10.0000	2	2
Ribosomal protein S6 kinase alpha-4	Homo sapiens (human)	Kd	10.0000	4	4
Ribosomal protein S6 kinase alpha-5	Homo sapiens (human)	Kd	10.0000	4	4
Ribosomal protein S6 kinase alpha-6	Homo sapiens (human)	Kd	10.0000	4	4
Ribosomal protein S6 kinase beta-1	Homo sapiens (human)	Kd	10.0000	1	1
Serine/threonine-protein kinase 10	Homo sapiens (human)	Kd	10.0000	2	2
Serine/threonine-protein kinase 16	Homo sapiens (human)	Kd	10.0000	2	2
Serine/threonine-protein kinase 17A	Homo sapiens (human)	Kd	10.0000	2	2
Serine/threonine-protein kinase 17B	Homo sapiens (human)	Kd	10.0000	2	2
Serine/threonine-protein kinase 24	Homo sapiens (human)	Kd	10.0000	2	2
Serine/threonine-protein kinase 25	Homo sapiens (human)	Kd	10.0000	2	2
Serine/threonine-protein kinase 26	Homo sapiens (human)	Kd	10.0000	2	2
Serine/threonine-protein kinase 3	Homo sapiens (human)	Kd	10.0000	2	2
Serine/threonine-protein kinase 32A	Homo sapiens (human)	Kd	10.0000	1	1
Serine/threonine-protein kinase 32B	Homo sapiens (human)	Kd	10.0000	2	2
Serine/threonine-protein kinase 32C	Homo sapiens (human)	Kd	10.0000	2	2
Serine/threonine-protein kinase 33	Homo sapiens (human)	Kd	10.0000	2	2
Serine/threonine-protein kinase 35	Homo sapiens (human)	Kd	10.0000	1	1
Serine/threonine-protein kinase 36	Homo sapiens (human)	Kd	10.0000	2	2
Serine/threonine-protein kinase 38	Homo sapiens (human)	Kd	10.0000	1	1
Serine/threonine-protein kinase 38-like	Homo sapiens (human)	Kd	10.0000	2	2
Serine/threonine-protein kinase 4	Homo sapiens (human)	Kd	10.0000	2	2
Serine/threonine-protein kinase B-raf	Homo sapiens (human)	Kd	10.0000	4	4
Serine/threonine-protein kinase BRSK1	Homo sapiens (human)	Kd	10.0000	2	2
Serine/threonine-protein kinase BRSK2	Homo sapiens (human)	Kd	10.0000	2	2
Serine/threonine-protein kinase Chk1	Homo sapiens (human)	Kd	10.0000	2	2
Serine/threonine-protein kinase Chk2	Homo sapiens (human)	Kd	10.0000	1	1
Serine/threonine-protein kinase D1	Homo sapiens (human)	Kd	10.0000	2	2
Serine/threonine-protein kinase D2	Homo sapiens (human)	Kd	10.0000	2	2
Serine/threonine-protein kinase D3	Homo sapiens (human)	Kd	10.0000	2	2
Serine/threonine-protein kinase DCLK1	Homo sapiens (human)	Kd	10.0000	2	2
Serine/threonine-protein kinase DCLK2	Homo sapiens (human)	Kd	10.0000	2	2
Serine/threonine-protein kinase DCLK3	Homo sapiens (human)	Kd	10.0000	2	2
Serine/threonine-protein kinase ICK	Homo sapiens (human)	Kd	10.0000	1	1
Serine/threonine-protein kinase LATS1	Homo sapiens (human)	Kd	10.0000	2	2
Serine/threonine-protein kinase LATS2	Homo sapiens (human)	Kd	10.0000	2	2
Serine/threonine-protein kinase MAK	Homo sapiens (human)	Kd	10.0000	1	1
Serine/threonine-protein kinase MARK1	Homo sapiens (human)	Kd	10.0000	2	2
Serine/threonine-protein kinase MARK2	Homo sapiens (human)	Kd	10.0000	2	2
Serine/threonine-protein kinase MRCK alpha	Homo sapiens (human)	Kd	10.0000	2	2
Serine/threonine-protein kinase MRCK beta	Homo sapiens (human)	Kd	10.0000	2	2
Serine/threonine-protein kinase MRCK gamma	Homo sapiens (human)	Kd	10.0000	2	2
Serine/threonine-protein kinase mTOR	Homo sapiens (human)	Kd	10.0000	1	1
Serine/threonine-protein kinase N1	Homo sapiens (human)	Kd	10.0000	2	2
Serine/threonine-protein kinase N2	Homo sapiens (human)	Kd	10.0000	2	2
Serine/threonine-protein kinase Nek1	Homo sapiens (human)	Kd	10.0000	2	2
Serine/threonine-protein kinase Nek11	Homo sapiens (human)	Kd	10.0000	1	1
Serine/threonine-protein kinase Nek2	Homo sapiens (human)	Kd	10.0000	2	2
Serine/threonine-protein kinase Nek3	Homo sapiens (human)	Kd	10.0000	1	1
Serine/threonine-protein kinase Nek4	Homo sapiens (human)	Kd	10.0000	1	1
Serine/threonine-protein kinase Nek5	Homo sapiens (human)	Kd	10.0000	2	2
Serine/threonine-protein kinase Nek6	Homo sapiens (human)	Kd	10.0000	2	2
Serine/threonine-protein kinase Nek7	Homo sapiens (human)	Kd	10.0000	2	2
Serine/threonine-protein kinase Nek9	Homo sapiens (human)	Kd	10.0000	2	2
Serine/threonine-protein kinase NIM1	Homo sapiens (human)	Kd	10.0000	1	1
Serine/threonine-protein kinase NLK	Homo sapiens (human)	Kd	10.0000	2	2
Serine/threonine-protein kinase OSR1	Homo sapiens (human)	Kd	10.0000	1	1
Serine/threonine-protein kinase PAK 1	Homo sapiens (human)	Kd	10.0000	2	2
Serine/threonine-protein kinase PAK 2	Homo sapiens (human)	Kd	10.0000	2	2
Serine/threonine-protein kinase PAK 3	Homo sapiens (human)	Kd	10.0000	2	2
Serine/threonine-protein kinase PAK 4	Homo sapiens (human)	Kd	10.0000	2	2
Serine/threonine-protein kinase PAK 5	Homo sapiens (human)	Kd	10.0000	2	2
Serine/threonine-protein kinase PAK 6	Homo sapiens (human)	Kd	10.0000	2	2
Serine/threonine-protein kinase pim-1	Homo sapiens (human)	Kd	10.0000	2	2
Serine/threonine-protein kinase pim-2	Homo sapiens (human)	Kd	10.0000	2	2
Serine/threonine-protein kinase pim-3	Homo sapiens (human)	Kd	10.0000	2	2
Serine/threonine-protein kinase PknB	Mycobacterium tuberculosis H37Rv	Kd	10.0000	1	1
Serine/threonine-protein kinase PLK1	Homo sapiens (human)	Kd	10.0000	2	2
Serine/threonine-protein kinase PLK2	Homo sapiens (human)	Kd	10.0000	1	1
Serine/threonine-protein kinase PLK3	Homo sapiens (human)	Kd	10.0000	2	2
Serine/threonine-protein kinase PLK4	Homo sapiens (human)	Kd	10.0000	2	2
Serine/threonine-protein kinase PRP4 homolog	Homo sapiens (human)	Kd	10.0000	1	1
Serine/threonine-protein kinase receptor R3	Homo sapiens (human)	Kd	10.0000	2	2
Serine/threonine-protein kinase RIO1	Homo sapiens (human)	Kd	10.0000	2	2
Serine/threonine-protein kinase RIO2	Homo sapiens (human)	Kd	10.0000	1	1
Serine/threonine-protein kinase RIO3	Homo sapiens (human)	Kd	10.0000	2	2
Serine/threonine-protein kinase SBK1	Homo sapiens (human)	Kd	10.0000	1	1
Serine/threonine-protein kinase Sgk3	Homo sapiens (human)	Kd	10.0000	1	1
Serine/threonine-protein kinase SIK1	Homo sapiens (human)	Kd	10.0000	2	2
Serine/threonine-protein kinase SIK2	Homo sapiens (human)	Kd	10.0000	2	2
Serine/threonine-protein kinase SIK3	Homo sapiens (human)	Kd	10.0000	1	1
Serine/threonine-protein kinase STK11	Homo sapiens (human)	Kd	10.0000	2	2
Serine/threonine-protein kinase TAO1	Homo sapiens (human)	Kd	10.0000	1	1
Serine/threonine-protein kinase TAO2	Homo sapiens (human)	Kd	10.0000	1	1
Serine/threonine-protein kinase TAO3	Homo sapiens (human)	Kd	10.0000	1	1
Serine/threonine-protein kinase TBK1	Homo sapiens (human)	Kd	10.0000	1	1
Serine/threonine-protein kinase TNNI3K	Homo sapiens (human)	Kd	10.0000	2	2
Serine/threonine-protein kinase tousled-like 1	Homo sapiens (human)	Kd	10.0000	2	2
Serine/threonine-protein kinase tousled-like 2	Homo sapiens (human)	Kd	10.0000	2	2
Serine/threonine-protein kinase ULK1	Homo sapiens (human)	Kd	10.0000	1	1
Serine/threonine-protein kinase ULK2	Homo sapiens (human)	Kd	10.0000	1	1
Serine/threonine-protein kinase ULK3	Homo sapiens (human)	Kd	10.0000	1	1
Serine/threonine-protein kinase VRK2	Homo sapiens (human)	Kd	10.0000	1	1
Serine/threonine-protein kinase/endoribonuclease IRE1	Homo sapiens (human)	Kd	10.0000	1	1
Signal transducer and activator of transcription 3	Homo sapiens (human)	EC50	10.0000	5	5
SNF-related serine/threonine-protein kinase	Homo sapiens (human)	Kd	10.0000	1	1
Spike glycoprotein	Betacoronavirus England 1	EC50	4.6700	1	1
Spike glycoprotein	Severe acute respiratory syndrome-related coronavirus	EC50	4.6700	1	1
SRSF protein kinase 1	Homo sapiens (human)	Kd	10.0000	2	2
SRSF protein kinase 2	Homo sapiens (human)	Kd	10.0000	2	2
SRSF protein kinase 3	Homo sapiens (human)	Kd	10.0000	1	1
STE20-like serine/threonine-protein kinase	Homo sapiens (human)	Kd	10.0000	2	2
STE20/SPS1-related proline-alanine-rich protein kinase	Homo sapiens (human)	Kd	10.0000	1	1
streptokinase A precursor	Streptococcus pyogenes M1 GAS	EC50	1.5190	1	1
Testis-specific serine/threonine-protein kinase 1	Homo sapiens (human)	Kd	10.0000	2	2
TGF-beta receptor type-1	Homo sapiens (human)	Kd	10.0000	2	2
TGF-beta receptor type-2	Homo sapiens (human)	Kd	10.0000	2	2
TRAF2 and NCK-interacting protein kinase	Homo sapiens (human)	Kd	10.0000	2	2
Transient receptor potential cation channel subfamily M member 6	Homo sapiens (human)	Kd	10.0000	1	1
Transient receptor potential cation channel subfamily V member 1	Homo sapiens (human)	EC50	10.0000	2	2
Transmembrane protease serine 2	Homo sapiens (human)	EC50	4.6700	1	1
Tubulin alpha-1A chain	Rattus norvegicus (Norway rat)	Kd	10.0000	1	1
Tyrosine-protein kinase ABL1	Homo sapiens (human)	Kd	6.8361	28	28
Tyrosine-protein kinase ABL2	Homo sapiens (human)	Kd	1.3400	3	3
Tyrosine-protein kinase Blk	Homo sapiens (human)	Kd	3.1000	2	2
Tyrosine-protein kinase BTK	Homo sapiens (human)	Kd	10.0000	2	2
Tyrosine-protein kinase CSK	Homo sapiens (human)	Kd	10.0000	2	2
Tyrosine-protein kinase Fer	Homo sapiens (human)	Kd	10.0000	2	2
Tyrosine-protein kinase Fes/Fps	Homo sapiens (human)	Kd	10.0000	2	2
Tyrosine-protein kinase Fgr	Homo sapiens (human)	Kd	1.2667	3	3
Tyrosine-protein kinase FRK	Homo sapiens (human)	Kd	7.7667	3	3
Tyrosine-protein kinase Fyn	Homo sapiens (human)	Kd	2.1000	2	2
Tyrosine-protein kinase HCK	Homo sapiens (human)	Kd	10.0000	3	3
Tyrosine-protein kinase ITK/TSK	Homo sapiens (human)	Kd	10.0000	2	2
Tyrosine-protein kinase JAK1	Homo sapiens (human)	Kd	10.0000	3	3
Tyrosine-protein kinase JAK2	Homo sapiens (human)	Kd	10.0000	2	2
Tyrosine-protein kinase JAK3	Homo sapiens (human)	Kd	10.0000	2	2
Tyrosine-protein kinase Lck	Homo sapiens (human)	Kd	3.6667	3	3
Tyrosine-protein kinase Lyn	Homo sapiens (human)	Kd	1.7000	2	2
Tyrosine-protein kinase Mer	Homo sapiens (human)	Kd	10.0000	2	2
Tyrosine-protein kinase receptor Tie-1	Homo sapiens (human)	Kd	10.0000	2	2
Tyrosine-protein kinase receptor TYRO3	Homo sapiens (human)	Kd	10.0000	2	2
Tyrosine-protein kinase receptor UFO	Homo sapiens (human)	Kd	10.0000	2	2
Tyrosine-protein kinase Srms	Homo sapiens (human)	Kd	10.0000	2	2
Tyrosine-protein kinase SYK	Homo sapiens (human)	Kd	10.0000	2	2
Tyrosine-protein kinase Tec	Homo sapiens (human)	Kd	10.0000	2	2
Tyrosine-protein kinase TXK	Homo sapiens (human)	Kd	10.0000	2	2
Tyrosine-protein kinase Yes	Homo sapiens (human)	Kd	1.9333	3	3
Tyrosine-protein kinase ZAP-70	Homo sapiens (human)	Kd	10.0000	2	2
Tyrosine-protein phosphatase non-receptor type 1	Homo sapiens (human)	Kd	6.0800	1	1
Uncharacterized serine/threonine-protein kinase SBK3	Homo sapiens (human)	Kd	10.0000	1	1
Vascular endothelial growth factor receptor 1	Homo sapiens (human)	Kd	10.0000	2	2
Vascular endothelial growth factor receptor 2	Homo sapiens (human)	Kd	10.0000	2	2
Vascular endothelial growth factor receptor 3	Homo sapiens (human)	Kd	10.0000	2	2
Wee1-like protein kinase	Homo sapiens (human)	Kd	10.0000	2	2
Wee1-like protein kinase 2	Homo sapiens (human)	Kd	10.0000	1	1

Other Measurements

Protein	Taxonomy	Measurement	Average (mM)	Bioassay(s)	Drugs
85/88 kDa calcium-independent phospholipase A2	Homo sapiens (human)	XI50	0.0047	8	8
bioA	Mycobacterium tuberculosis UT205	AC50	9.0600	1	1
Cytochrome P450 3A5	Homo sapiens (human)	IC90	1.8000	1	1
Glucocorticoid receptor	Homo sapiens (human)	Activity	0.0024	1	1
Glucocorticoid receptor	Homo sapiens (human)	ED50	0.0040	1	1
Glucocorticoid receptor	Homo sapiens (human)	fEC50	0.0240	1	1
Glucocorticoid receptor	Homo sapiens (human)	fIC20	0.0009	1	1
Glucocorticoid receptor	Homo sapiens (human)	fIC30	0.0200	1	1
Group 10 secretory phospholipase A2	Homo sapiens (human)	XI50	0.0010	7	7
Group 3 secretory phospholipase A2	Homo sapiens (human)	XI50	0.0010	7	7
Group IID secretory phospholipase A2	Homo sapiens (human)	XI50	0.0010	7	7
Group IIE secretory phospholipase A2	Homo sapiens (human)	XI50	0.0010	7	7
Group IIF secretory phospholipase A2	Homo sapiens (human)	XI50	0.0010	7	7
Group XIIA secretory phospholipase A2	Homo sapiens (human)	XI50	0.0010	7	7
Group XIIB secretory phospholipase A2-like protein	Homo sapiens (human)	XI50	0.0010	7	7
H3 histone acetyltransferase	Candida albicans SC5314	AC50	1.5500	1	1
hypothetical protein CAALFM_CR05890CA	Candida albicans SC5314	AC50	1.5500	1	1
luciferase	Photuris pensylvanica (Pennsylania firefly)	AC50	52.0000	1	2
Phospholipase A2	Homo sapiens (human)	XI50	0.0010	7	7
Phospholipase A2 group V	Homo sapiens (human)	XI50	0.0010	7	7
Phospholipase A2, membrane associated	Homo sapiens (human)	XI50	0.0010	7	7
Progesterone receptor	Homo sapiens (human)	Activity	5.0000	1	1
Putative inactive group IIC secretory phospholipase A2	Homo sapiens (human)	XI50	0.0010	7	7

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