One of a class of drugs that acts by selective inhibition of calcium influx through cell membranes or on the release and binding of calcium in intracellular pools.
| Member | Definition | Class |
|---|
| 2-aminoethoxydiphenyl borate | An organoboron compound that is diphenylborane in which the borane hydrogen is replaced by a 2-aminoethoxy group. | 2-aminoethoxydiphenylborane |
| amlodipine | A fully substituted dialkyl 1,4-dihydropyridine-3,5-dicarboxylate derivative, which is used for the treatment of hypertension, chronic stable angina and confirmed or suspected vasospastic angina. | amlodipine |
| amlodipine besylate | The benzenesulfonate salt of amlodipine. | amlodipine benzenesulfonate |
| bepridil | A tertiary amine in which the substituents on nitrogen are benzyl, phenyl and 3-(2-methylpropoxy)-2-(pyrrolidin-1-yl)propyl. | bepridil |
| bevantolol | A propanolamine that is 3-aminopropane-1,2-diol in which the hydrogen of the primary hydroxy group is substituted by 3-methylphenyl and one of the hydrogens attached to the nitrogen is substituted by 2-(3,4-dimethoxyphenyl)ethyl. A beta1 adrenoceptor antagonist, it has been shown to be as effective as other beta-blockers for the treatment of angina pectoris and hypertension. | bevantolol |
| cilnidipine | A diesterified 1,4-dihydropyridine-3,5-dicarboxylic acid. A calcium channel blocker, it is used as an antihypertensive. | cilnidipine |
| cinnarizine | | cinnarizine |
| cobaltous chloride | A cobalt salt in which the cobalt metal is in the +2 oxidation state and the counter-anion is chloride. It is used as an indicator for water in desiccants. | cobalt dichloride |
| cromolyn | A dicarboxylic acid that is the bis-chromone derivative of glycerol. It is effective as a mast cell stabilizer. | cromoglycic acid |
| d 888 | A nitrile that acts as an L-type calcium channel blocker. | devapamil |
| diethylstilbestrol | An olefinic compound that is trans-hex-3-ene in which the hydrogens at positions 3 and 4 have been replaced by p-hydroxyphenyl groups. | diethylstilbestrol |
| diltiazem | A 5-[2-(dimethylamino)ethyl]-2-(4-methoxyphenyl)-4-oxo-2,3,4,5-tetrahydro-1,5-benzothiazepin-3-yl acetate in which both stereocentres have S configuration. A calcium-channel blocker and vasodilator, it is used as the hydrochloride in the management of angina pectoris and hypertension. | diltiazem |
| diltiazem hydrochloride | A hydrochloride salt resulting from the reaction of equimolar amounts of diltiazem and hydrogen chloride. A calcium-channel blocker and vasodilator, it is used in the management of angina pectoris and hypertension. | diltiazem hydrochloride |
| dotarizine | An N-alkylpiperazine in which the two amino hydrogens of piperazine have been replaced by diphenylmethyl and 3-(2-phenyl-1,3-dioxolan-2-yl)propyl groups. A calcium channel blocker and serotonin (5-HT2) receptor antagonist used in the treatment of migraine. | dotarizine |
| eupatorin | A trimethoxyflavone that is 6-hydroxyluteolin in which the phenolic hydogens at positions 4', 6 and 7 have been replaced by methyl groups. | eupatorin |
| fasudil | An isoquinoline substituted by a (1,4-diazepan-1-yl)sulfonyl group at position 5. It is a Rho-kinase inhibitor and its hydrochloride hydrate form is approved for the treatment of cerebral vasospasm and cerebral ischemia. | fasudil |
| fasudil hydrochloride | A hydrochloride obtained by reaction of fasudil with one equivalent of hydrochloric acid. | fasudil hydrochloride |
| felodipine | The mixed (methyl, ethyl) diester of 4-(2,3-dichlorophenyl)-2,6-dimethyl-1,4-dihydropyridine-3,5-dicarboxylic acid. A calcium-channel blocker, it lowers blood pressure by reducing peripheral vascular resistance through a highly selective action on smooth muscle in arteriolar resistance vessels. It is used in the management of hypertension and angina pectoris. | felodipine |
| gabapentin | A gamma-amino acid that is cyclohexane substituted at position 1 by aminomethyl and carboxymethyl groups. Used for treatment of neuropathic pain and restless legs syndrome. | gabapentin |
| gsk-5498a | A member of the class of pyrazoles that is 1H-pyrazole substituted by 2-fluoro-6-(trifluoromethyl)benzyl and (2,6-difluorobenzoyl)amino groups at positions 1 and 3, respectively. It is a inhibitor of Ca(2+) release-activated Ca(2+) (CRAC) channel and inhibits the release of mast cell mediators and T-cell cytokines in human and rat preparations. | GSK-5498A |
| lamotrigine | A member of the class of 1,2,4-triazines in which the triazene skeleton is substituted by amino groups at positions 3 and 5, and by a 2,3-dichlorophenyl group at position 6. | lamotrigine |
| lanperisone | A 2-methyl-3-(pyrrolidin-1-yl)-1-[4-(trifluoromethyl)phenyl]propan-1-one in which the methyl group at position 2 adopts R-configuration. It is a muscle relaxant and induces ferroptosis in cancer cells. | lanperisone |
| magnesium sulfate | A magnesium salt having sulfate as the counterion. | magnesium sulfate |
| nemadipine-a | A dihydropyridine that is that is 1,4-dihydropyridine which is substituted at positions 2 and 6 by methyl groups, at positions 3 and 5 by ethoxycarbonyl groups, and at position 4 by a pentafluorophenyl group. An L-type calcium channel alpha1-subunit antagonist. When exposed to the microscopic soil nematode Caenorhabditis elegans, nemadipine-A induces a variety of defects including those affecting morphology and egg laying. | nemadipine-A |
| nickel chloride | A compound of nickel and chloride in which the ratio of nickel (in the +2 oxidation state) to chloride is 1:2. | nickel dichloride |
| nifedipine | | nifedipine |
| nimodipine | A dihydropyridine that is 1,4-dihydropyridine which is substituted by methyl groups at positions 2 and 6, a (2-methoxyethoxy)carbonyl group at position 3, a m-nitrophenyl group at position 4, and an isopropoxycarbonyl group at position 5. An L-type calcium channel blocker, it acts particularly on cerebral circulation, and is used both orally and intravenously for the prevention and treatment of subarachnoid hemorrhage from ruptured intracranial aneurysm. | nimodipine |
| nitrendipine | A dihydropyridine that is 1,4-dihydropyridine substituted by methyl groups at positions 2 and 6, a 3-nitrophenyl group at position 4, a ethoxycarbonyl group at position 3 and a methoxycarbonyl group at position 5. It is a calcium-channel blocker used in the treatment of hypertension. | nitrendipine |
| ochratoxin a | A phenylalanine derivative resulting from the formal condensation of the amino group of L-phenylalanine with the carboxy group of (3R)-5-chloro-8-hydroxy-3-methyl-1-oxo-3,4-dihydro-1H-2-benzopyran-7-carboxylic acid (ochratoxin alpha). It is among the most widely occurring food-contaminating mycotoxins, produced by Aspergillus ochraceus, Aspergillus carbonarius and Penicillium verrucosum. | ochratoxin A |
| ochratoxin b | A phenylalanine derivative resulting from the formal condensation of the amino group of L-phenylalanine with the carboxy group of (3R)-8-hydroxy-3-methyl-1-oxo-3,4-dihydro-1H-2-benzopyran-7-carboxylic acid. Ochratoxin B differs from the more naturally abundant ochratoxin A in the absence of the dihydroisocoumarin chlorine atom. It has cytotoxic effects on kidney and liver cells in vitro but only minor effects in vivo, due to its rapid metabolism and excretion. It inhibits cell proliferation of human liver HepG2 cells at doses as low as 1 mug/ ml but lacks the genotoxic activity of ochratoxin A, even at higher concentrations. | ochratoxin B |
| oxybutynin | A racemate comprising equimolar amounts of (R)-oxybutynin and esoxybutynin. An antispasmodic used for the treatment of overactive bladder. | 4-(diethylamino)but-2-yn-1-ol; oxybutynin |
| pregabalin | A gamma-amino acid that is gamma-aminobutyric acid (GABA) carrying an isobutyl substitutent at the beta-position (the S-enantiomer). Binds with high affinity to the alpha2-delta site (an auxiliary subunit of voltage-gated calcium channels) in central nervous system tissues. | pregabalin |
| thapsigargin | An organic heterotricyclic compound that is a hexa-oxygenated 6,7-guaianolide isolated fron the roots of Thapsia garganica L., Apiaceae. A potent skin irritant, it is used in traditional medicine as a counter-irritant. Thapsigargin inhibits Ca(2+)-transporting ATPase mediated uptake of calcium ions into sarcoplasmic reticulum and is used in experimentation examining the impacts of increasing cytosolic calcium concentrations. | thapsigargin |
| tilmicosin | A macrolide antibiotic with formula C46H80N2O13. It is used for the treatment of respiratory disease in cattle at high risk of developing bovine respiratory disease associated with Mannheimia haemolytica. | tilmicosin |
| tranilast | An amidobenzoic acid that is anthranilic acid in which one of the anilino hydrogens is replaced by a 3,4-dimethoxycinnamoyl group. | tranilast |
| u-50488 | A monocarboxylic acid amide obtained by formal condensation between the carboxy group of 3,4-dichlorophenylacetic acid and the secondary amino group of (1R,2R)-N-methyl-2-(pyrrolidin-1-yl)cyclohexanamine | U50488 |
| Protein | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Drugs |
|---|
| 15-hydroxyprostaglandin dehydrogenase [NAD(+)] isoform 1 | Homo sapiens (human) | Potency | 22.8955 | 1 | 6 |
| 15-lipoxygenase, partial | Homo sapiens (human) | Potency | 6.6102 | 1 | 2 |
| 67.9K protein | Vaccinia virus | Potency | 12.5070 | 2 | 11 |
| acetylcholinesterase | Homo sapiens (human) | Potency | 17.7238 | 1 | 2 |
| acid sphingomyelinase | Homo sapiens (human) | Potency | 26.7449 | 1 | 4 |
| activating transcription factor 6 | Homo sapiens (human) | Potency | 35.0860 | 1 | 3 |
| aldehyde dehydrogenase 1 family, member A1 | Homo sapiens (human) | Potency | 26.5854 | 1 | 16 |
| alpha-galactosidase | Homo sapiens (human) | Potency | 27.7170 | 2 | 2 |
| Alpha-synuclein | Homo sapiens (human) | Potency | 31.2224 | 1 | 3 |
| AR protein | Homo sapiens (human) | Potency | 26.9987 | 11 | 73 |
| aryl hydrocarbon receptor | Homo sapiens (human) | Potency | 6.0008 | 2 | 14 |
| arylsulfatase A | Homo sapiens (human) | Potency | 11.2257 | 1 | 6 |
| ATAD5 protein, partial | Homo sapiens (human) | Potency | 16.3662 | 4 | 21 |
| Ataxin-2 | Homo sapiens (human) | Potency | 18.1751 | 2 | 10 |
| ATP-dependent phosphofructokinase | Trypanosoma brucei brucei TREU927 | Potency | 20.8752 | 3 | 11 |
| ATPase family AAA domain-containing protein 5 | Homo sapiens (human) | Potency | 15.1681 | 2 | 7 |
| atrial natriuretic peptide receptor 1 precursor | Homo sapiens (human) | Potency | 9.3392 | 1 | 4 |
| atrial natriuretic peptide receptor 2 precursor | Homo sapiens (human) | Potency | 14.3981 | 1 | 4 |
| beta-2 adrenergic receptor | Homo sapiens (human) | Potency | 28.1838 | 1 | 1 |
| Bloom syndrome protein isoform 1 | Homo sapiens (human) | Potency | 249.9047 | 2 | 14 |
| bromodomain adjacent to zinc finger domain 2B | Homo sapiens (human) | Potency | 62.0468 | 1 | 6 |
| C-terminal-binding protein 1 | Homo sapiens (human) | Potency | 10.6928 | 1 | 1 |
| caspase 7, apoptosis-related cysteine protease | Homo sapiens (human) | Potency | 33.4915 | 1 | 1 |
| caspase-3 | Cricetulus griseus (Chinese hamster) | Potency | 33.4915 | 1 | 1 |
| caspase-3 | Homo sapiens (human) | Potency | 33.4915 | 1 | 1 |
| Caspase-7 | Cricetulus griseus (Chinese hamster) | Potency | 33.4915 | 1 | 1 |
| Cellular tumor antigen p53 | Homo sapiens (human) | Potency | 23.6021 | 3 | 19 |
| cellular tumor antigen p53 isoform a | Homo sapiens (human) | Potency | 18.4921 | 2 | 9 |
| Chain A, 2-oxoglutarate Oxygenase | Homo sapiens (human) | Potency | 24.4458 | 1 | 11 |
| Chain A, Beta-lactamase | Escherichia coli K-12 | Potency | 80.1249 | 2 | 10 |
| Chain A, Cruzipain | Trypanosoma cruzi | Potency | 39.8107 | 1 | 5 |
| Chain A, Ferritin light chain | Equus caballus (horse) | Potency | 32.9390 | 2 | 10 |
| Chain A, HADH2 protein | Homo sapiens (human) | Potency | 19.8357 | 2 | 7 |
| Chain A, JmjC domain-containing histone demethylation protein 3A | Homo sapiens (human) | Potency | 61.3991 | 1 | 4 |
| Chain A, MAJOR APURINIC/APYRIMIDINIC ENDONUCLEASE | Homo sapiens (human) | Potency | 15.4078 | 2 | 9 |
| Chain A, Putative fructose-1,6-bisphosphate aldolase | Giardia intestinalis | Potency | 12.7415 | 1 | 3 |
| Chain A, TYROSYL-DNA PHOSPHODIESTERASE | Homo sapiens (human) | Potency | 31.2292 | 1 | 9 |
| Chain B, HADH2 protein | Homo sapiens (human) | Potency | 19.8357 | 2 | 7 |
| chaperonin-containing TCP-1 beta subunit homolog | Homo sapiens (human) | Potency | 15.8489 | 1 | 1 |
| chromobox protein homolog 1 | Homo sapiens (human) | Potency | 29.2547 | 2 | 15 |
| ClpP | Bacillus subtilis | Potency | 11.2202 | 1 | 1 |
| cytochrome P450 2C19 precursor | Homo sapiens (human) | Potency | 11.8961 | 1 | 2 |
| cytochrome P450 2C9 precursor | Homo sapiens (human) | Potency | 23.7358 | 1 | 2 |
| cytochrome P450 2C9, partial | Homo sapiens (human) | Potency | 9.6487 | 1 | 10 |
| cytochrome P450 2D6 | Homo sapiens (human) | Potency | 17.2448 | 1 | 15 |
| cytochrome P450 2D6 isoform 1 | Homo sapiens (human) | Potency | 10.3120 | 1 | 5 |
| cytochrome P450 3A4 isoform 1 | Homo sapiens (human) | Potency | 9.2320 | 2 | 24 |
| cytochrome P450 family 3 subfamily A polypeptide 4 | Homo sapiens (human) | Potency | 6.0070 | 2 | 15 |
| cytochrome P450, family 19, subfamily A, polypeptide 1, isoform CRA_a | Homo sapiens (human) | Potency | 29.7400 | 1 | 11 |
| D(1A) dopamine receptor | Homo sapiens (human) | Potency | 8.3011 | 3 | 11 |
| D(1A) dopamine receptor | Sus scrofa (pig) | Potency | 11.2815 | 1 | 3 |
| Disintegrin and metalloproteinase domain-containing protein 17 | Homo sapiens (human) | Potency | 25.1189 | 1 | 1 |
| DNA dC->dU-editing enzyme APOBEC-3G isoform 1 | Homo sapiens (human) | Potency | 19.9526 | 1 | 1 |
| DNA polymerase beta | Homo sapiens (human) | Potency | 79.4328 | 1 | 1 |
| DNA polymerase III, partial | Bacillus subtilis | Potency | 21.1923 | 1 | 1 |
| DNA polymerase iota isoform a (long) | Homo sapiens (human) | Potency | 29.9897 | 1 | 3 |
| DNA polymerase kappa isoform 1 | Homo sapiens (human) | Potency | 25.3525 | 1 | 3 |
| dopamine D1 receptor | Homo sapiens (human) | Potency | 14.5580 | 1 | 2 |
| endonuclease IV | Escherichia coli | Potency | 10.9837 | 1 | 3 |
| estrogen nuclear receptor alpha | Homo sapiens (human) | Potency | 24.4724 | 12 | 77 |
| estrogen receptor 2 (ER beta) | Homo sapiens (human) | Potency | 24.3338 | 3 | 13 |
| estrogen-related nuclear receptor alpha | Homo sapiens (human) | Potency | 24.0881 | 9 | 85 |
| euchromatic histone-lysine N-methyltransferase 2 | Homo sapiens (human) | Potency | 17.5880 | 2 | 26 |
| EWS/FLI fusion protein | Homo sapiens (human) | Potency | 28.8101 | 4 | 11 |
| eyes absent homolog 2 isoform a | Homo sapiens (human) | Potency | 10.6928 | 1 | 1 |
| farnesoid X nuclear receptor | Homo sapiens (human) | Potency | 28.6709 | 5 | 20 |
| flap endonuclease 1 | Homo sapiens (human) | Potency | 8.1310 | 1 | 3 |
| Fumarate hydratase | Homo sapiens (human) | Potency | 29.1362 | 1 | 8 |
| G | Vesicular stomatitis virus | Potency | 9.6487 | 1 | 10 |
| GABA theta subunit | Rattus norvegicus (Norway rat) | Potency | 9.2320 | 1 | 12 |
| GALC protein | Homo sapiens (human) | Potency | 0.7079 | 1 | 3 |
| Gamma-aminobutyric acid receptor subunit alpha-1 | Rattus norvegicus (Norway rat) | Potency | 9.2320 | 1 | 12 |
| Gamma-aminobutyric acid receptor subunit alpha-2 | Rattus norvegicus (Norway rat) | Potency | 9.2320 | 1 | 12 |
| Gamma-aminobutyric acid receptor subunit alpha-3 | Rattus norvegicus (Norway rat) | Potency | 9.2320 | 1 | 12 |
| Gamma-aminobutyric acid receptor subunit alpha-4 | Rattus norvegicus (Norway rat) | Potency | 9.2320 | 1 | 12 |
| Gamma-aminobutyric acid receptor subunit alpha-5 | Rattus norvegicus (Norway rat) | Potency | 9.2320 | 1 | 12 |
| Gamma-aminobutyric acid receptor subunit alpha-6 | Rattus norvegicus (Norway rat) | Potency | 9.2320 | 1 | 12 |
| Gamma-aminobutyric acid receptor subunit beta-1 | Rattus norvegicus (Norway rat) | Potency | 9.2320 | 1 | 12 |
| Gamma-aminobutyric acid receptor subunit beta-2 | Rattus norvegicus (Norway rat) | Potency | 9.2320 | 1 | 12 |
| Gamma-aminobutyric acid receptor subunit beta-3 | Rattus norvegicus (Norway rat) | Potency | 9.2320 | 1 | 12 |
| Gamma-aminobutyric acid receptor subunit delta | Rattus norvegicus (Norway rat) | Potency | 9.2320 | 1 | 12 |
| Gamma-aminobutyric acid receptor subunit epsilon | Rattus norvegicus (Norway rat) | Potency | 9.2320 | 1 | 12 |
| Gamma-aminobutyric acid receptor subunit gamma-1 | Rattus norvegicus (Norway rat) | Potency | 9.2320 | 1 | 12 |
| Gamma-aminobutyric acid receptor subunit gamma-2 | Rattus norvegicus (Norway rat) | Potency | 9.2320 | 1 | 12 |
| Gamma-aminobutyric acid receptor subunit gamma-3 | Rattus norvegicus (Norway rat) | Potency | 9.2320 | 1 | 12 |
| Gamma-aminobutyric acid receptor subunit pi | Rattus norvegicus (Norway rat) | Potency | 9.2320 | 1 | 12 |
| geminin | Homo sapiens (human) | Potency | 19.7511 | 3 | 35 |
| GLI family zinc finger 3 | Homo sapiens (human) | Potency | 19.9107 | 3 | 23 |
| glp-1 receptor, partial | Homo sapiens (human) | Potency | 12.7142 | 3 | 8 |
| GLS protein | Homo sapiens (human) | Potency | 12.8120 | 2 | 11 |
| glucocerebrosidase | Homo sapiens (human) | Potency | 37.0814 | 1 | 3 |
| glucocorticoid receptor [Homo sapiens] | Homo sapiens (human) | Potency | 19.0675 | 5 | 29 |
| Glutamate receptor 2 | Rattus norvegicus (Norway rat) | Potency | 30.4688 | 1 | 7 |
| GTP-binding nuclear protein Ran isoform 1 | Homo sapiens (human) | Potency | 3.6626 | 1 | 1 |
| Guanine nucleotide-binding protein G | Homo sapiens (human) | Potency | 28.1838 | 1 | 1 |
| heat shock 70kDa protein 5 (glucose-regulated protein, 78kDa) | Homo sapiens (human) | Potency | 17.6022 | 2 | 7 |
| heat shock protein beta-1 | Homo sapiens (human) | Potency | 35.4333 | 2 | 8 |
| Histamine H2 receptor | Cavia porcellus (domestic guinea pig) | Potency | 18.5140 | 2 | 14 |
| histone acetyltransferase KAT2A isoform 1 | Homo sapiens (human) | Potency | 37.0814 | 1 | 3 |
| Histone H2A.x | Cricetulus griseus (Chinese hamster) | Potency | 71.5271 | 2 | 4 |
| histone-lysine N-methyltransferase 2A isoform 2 precursor | Homo sapiens (human) | Potency | 30.7879 | 1 | 5 |
| HLA class I histocompatibility antigen, B alpha chain | Homo sapiens (human) | Potency | 9.6487 | 1 | 10 |
| huntingtin isoform 2 | Homo sapiens (human) | Potency | 27.9339 | 1 | 4 |
| hypothetical protein, conserved | Trypanosoma brucei | Potency | 16.7058 | 2 | 2 |
| hypoxia-inducible factor 1 alpha subunit | Homo sapiens (human) | Potency | 36.9184 | 2 | 9 |
| hypoxia-inducible factor 1, alpha subunit (basic helix-loop-helix transcription factor) | Homo sapiens (human) | Potency | 9.8589 | 3 | 13 |
| IDH1 | Homo sapiens (human) | Potency | 18.4664 | 1 | 7 |
| importin subunit beta-1 isoform 1 | Homo sapiens (human) | Potency | 3.6626 | 1 | 1 |
| Inositol hexakisphosphate kinase 1 | Homo sapiens (human) | Potency | 9.6487 | 1 | 20 |
| Inositol monophosphatase 1 | Rattus norvegicus (Norway rat) | Potency | 8.1724 | 2 | 11 |
| Integrin alpha-IIb | Homo sapiens (human) | Potency | 16.5301 | 1 | 5 |
| Integrin beta-3 | Homo sapiens (human) | Potency | 16.5301 | 1 | 5 |
| Interferon beta | Homo sapiens (human) | Potency | 13.6783 | 3 | 20 |
| interleukin 8 | Homo sapiens (human) | Potency | 74.9780 | 1 | 1 |
| lamin isoform A-delta10 | Homo sapiens (human) | Potency | 15.0198 | 2 | 18 |
| lethal factor (plasmid) | Bacillus anthracis str. A2012 | Potency | 20.0203 | 1 | 3 |
| Luciferase | Photinus pyralis (common eastern firefly) | Potency | 18.0830 | 4 | 8 |
| lysosomal alpha-glucosidase preproprotein | Homo sapiens (human) | Potency | 23.3507 | 4 | 4 |
| M-phase phosphoprotein 8 | Homo sapiens (human) | Potency | 27.7326 | 1 | 10 |
| Microtubule-associated protein tau | Homo sapiens (human) | Potency | 15.6440 | 2 | 15 |
| mitogen-activated protein kinase 1 | Homo sapiens (human) | Potency | 22.3902 | 2 | 11 |
| muscarinic acetylcholine receptor M1 | Rattus norvegicus (Norway rat) | Potency | 11.6856 | 2 | 10 |
| muscleblind-like protein 1 isoform 1 | Homo sapiens (human) | Potency | 33.9745 | 1 | 4 |
| Neuronal acetylcholine receptor subunit alpha-4 | Rattus norvegicus (Norway rat) | Potency | 11.2202 | 1 | 1 |
| Neuronal acetylcholine receptor subunit beta-2 | Rattus norvegicus (Norway rat) | Potency | 11.2202 | 1 | 1 |
| neuropeptide S receptor isoform A | Homo sapiens (human) | Potency | 15.6485 | 3 | 8 |
| NFKB1 protein, partial | Homo sapiens (human) | Potency | 19.7020 | 2 | 4 |
| nonstructural protein 1 | Influenza A virus (A/WSN/1933(H1N1)) | Potency | 27.2150 | 1 | 9 |
| NPC intracellular cholesterol transporter 1 precursor | Homo sapiens (human) | Potency | 36.8537 | 1 | 4 |
| nuclear factor erythroid 2-related factor 2 isoform 1 | Homo sapiens (human) | Potency | 30.2193 | 4 | 27 |
| nuclear factor erythroid 2-related factor 2 isoform 2 | Homo sapiens (human) | Potency | 29.0929 | 1 | 2 |
| nuclear factor NF-kappa-B p105 subunit isoform 1 | Homo sapiens (human) | Potency | 44.6684 | 1 | 1 |
| nuclear factor of kappa light polypeptide gene enhancer in B-cells 1 (p105), isoform CRA_a | Homo sapiens (human) | Potency | 31.3193 | 1 | 3 |
| Nuclear receptor ROR-gamma | Homo sapiens (human) | Potency | 50.1579 | 1 | 2 |
| nuclear receptor ROR-gamma isoform 1 | Mus musculus (house mouse) | Potency | 15.1395 | 2 | 29 |
| nuclear receptor subfamily 1, group I, member 2 | Rattus norvegicus (Norway rat) | Potency | 10.0000 | 1 | 1 |
| nuclear receptor subfamily 1, group I, member 3 | Homo sapiens (human) | Potency | 17.4663 | 3 | 23 |
| Ornithine decarboxylase | Rattus norvegicus (Norway rat) | Potency | 19.9526 | 1 | 1 |
| parathyroid hormone/parathyroid hormone-related peptide receptor precursor | Homo sapiens (human) | Potency | 35.4813 | 1 | 1 |
| Parkin | Homo sapiens (human) | Potency | 13.8115 | 3 | 11 |
| peptidyl-prolyl cis-trans isomerase NIMA-interacting 1 | Homo sapiens (human) | Potency | 57.9898 | 2 | 2 |
| peripheral myelin protein 22 | Rattus norvegicus (Norway rat) | Potency | 14.5627 | 1 | 7 |
| peripheral myelin protein 22 isoform 1 | Homo sapiens (human) | Potency | 58.7864 | 1 | 6 |
| peroxisome proliferator activated receptor gamma | Homo sapiens (human) | Potency | 23.0457 | 5 | 16 |
| peroxisome proliferator-activated receptor delta | Homo sapiens (human) | Potency | 37.1680 | 5 | 15 |
| phosphopantetheinyl transferase | Bacillus subtilis | Potency | 41.9124 | 2 | 10 |
| PINK1 | Homo sapiens (human) | Potency | 39.8107 | 1 | 1 |
| plasminogen precursor | Mus musculus (house mouse) | Potency | 4.1692 | 1 | 2 |
| polyprotein | Zika virus | Potency | 29.1362 | 1 | 8 |
| polyunsaturated fatty acid lipoxygenase ALOX12 | Homo sapiens (human) | Potency | 16.2676 | 1 | 4 |
| Polyunsaturated fatty acid lipoxygenase ALOX15B | Homo sapiens (human) | Potency | 14.5977 | 1 | 4 |
| potassium voltage-gated channel subfamily H member 2 isoform d | Homo sapiens (human) | Potency | 16.5608 | 1 | 7 |
| PPM1D protein | Homo sapiens (human) | Potency | 14.7136 | 1 | 4 |
| pregnane X nuclear receptor | Homo sapiens (human) | Potency | 25.3387 | 3 | 17 |
| pregnane X receptor | Rattus norvegicus (Norway rat) | Potency | 70.7946 | 1 | 1 |
| progesterone receptor | Homo sapiens (human) | Potency | 20.8600 | 2 | 14 |
| pyruvate kinase | Leishmania mexicana mexicana | Potency | 12.5893 | 2 | 2 |
| pyruvate kinase PKM isoform b | Homo sapiens (human) | Potency | 19.9526 | 2 | 2 |
| Rap guanine nucleotide exchange factor 4 | Homo sapiens (human) | Potency | 48.5236 | 1 | 3 |
| RAR-related orphan receptor gamma | Mus musculus (house mouse) | Potency | 28.2631 | 2 | 19 |
| ras-related protein Rab-9A | Homo sapiens (human) | Potency | 21.0481 | 1 | 5 |
| regulator of G-protein signaling 4 | Homo sapiens (human) | Potency | 18.3216 | 1 | 12 |
| retinoic acid nuclear receptor alpha variant 1 | Homo sapiens (human) | Potency | 29.9903 | 3 | 21 |
| retinoid X nuclear receptor alpha | Homo sapiens (human) | Potency | 30.7044 | 4 | 17 |
| serine/threonine-protein kinase mTOR isoform 1 | Homo sapiens (human) | Potency | 15.3707 | 4 | 12 |
| serine/threonine-protein kinase PLK1 | Homo sapiens (human) | Potency | 17.3396 | 1 | 2 |
| Single-stranded DNA cytosine deaminase | Homo sapiens (human) | Potency | 50.1187 | 1 | 3 |
| SMAD family member 2 | Homo sapiens (human) | Potency | 5.1298 | 2 | 2 |
| SMAD family member 3 | Homo sapiens (human) | Potency | 5.1298 | 2 | 2 |
| Smad3 | Homo sapiens (human) | Potency | 23.5754 | 1 | 8 |
| snurportin-1 | Homo sapiens (human) | Potency | 3.6626 | 1 | 1 |
| Spike glycoprotein | Severe acute respiratory syndrome-related coronavirus | Potency | 21.8525 | 1 | 11 |
| survival motor neuron protein isoform d | Homo sapiens (human) | Potency | 11.1840 | 1 | 9 |
| TAR DNA-binding protein 43 | Homo sapiens (human) | Potency | 32.3756 | 1 | 5 |
| TDP1 protein | Homo sapiens (human) | Potency | 18.7610 | 2 | 71 |
| thioredoxin glutathione reductase | Schistosoma mansoni | Potency | 89.1251 | 1 | 1 |
| thioredoxin reductase | Rattus norvegicus (Norway rat) | Potency | 21.4361 | 4 | 23 |
| Thrombopoietin | Homo sapiens (human) | Potency | 5.7925 | 2 | 4 |
| thyroid hormone receptor beta isoform 2 | Rattus norvegicus (Norway rat) | Potency | 18.1584 | 3 | 32 |
| thyroid hormone receptor beta isoform a | Homo sapiens (human) | Potency | 446.5231 | 4 | 6 |
| thyroid stimulating hormone receptor | Homo sapiens (human) | Potency | 32.8082 | 5 | 20 |
| tumor necrosis factor | Homo sapiens (human) | Potency | 10.5909 | 1 | 1 |
| ubiquitin carboxyl-terminal hydrolase 2 isoform a | Homo sapiens (human) | Potency | 19.9040 | 2 | 2 |
| urokinase plasminogen activator surface receptor precursor | Mus musculus (house mouse) | Potency | 4.1692 | 1 | 2 |
| urokinase-type plasminogen activator precursor | Mus musculus (house mouse) | Potency | 4.1692 | 1 | 2 |
| USP1 protein, partial | Homo sapiens (human) | Potency | 44.6401 | 1 | 16 |
| v-jun sarcoma virus 17 oncogene homolog (avian) | Homo sapiens (human) | Potency | 24.0742 | 2 | 7 |
| vitamin D (1,25- dihydroxyvitamin D3) receptor | Homo sapiens (human) | Potency | 30.1923 | 5 | 12 |
| vitamin D3 receptor isoform VDRA | Homo sapiens (human) | Potency | 21.9800 | 5 | 32 |
| Voltage-dependent calcium channel gamma-2 subunit | Mus musculus (house mouse) | Potency | 30.4688 | 1 | 7 |
| Protein | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Drugs |
|---|
| 1-acylglycerol-3-phosphate O-acyltransferase ABHD5 isoform a | Homo sapiens (human) | IC50 | 8.3760 | 2 | 2 |
| 3-oxo-5-alpha-steroid 4-dehydrogenase 1 | Rattus norvegicus (Norway rat) | IC50 | 1.1200 | 1 | 1 |
| 3-oxo-5-alpha-steroid 4-dehydrogenase 2 | Rattus norvegicus (Norway rat) | IC50 | 1.1200 | 1 | 1 |
| 5-hydroxytryptamine receptor 1A | Rattus norvegicus (Norway rat) | IC50 | 1.0830 | 1 | 1 |
| 5-hydroxytryptamine receptor 1A | Rattus norvegicus (Norway rat) | Ki | 0.6190 | 1 | 1 |
| 5-hydroxytryptamine receptor 1B | Rattus norvegicus (Norway rat) | IC50 | 1.0830 | 1 | 1 |
| 5-hydroxytryptamine receptor 1B | Rattus norvegicus (Norway rat) | Ki | 0.6190 | 1 | 1 |
| 5-hydroxytryptamine receptor 2A | Homo sapiens (human) | IC50 | 2.5750 | 1 | 2 |
| 5-hydroxytryptamine receptor 2A | Rattus norvegicus (Norway rat) | IC50 | 10.0000 | 1 | 1 |
| 5-hydroxytryptamine receptor 2A | Homo sapiens (human) | Ki | 0.7360 | 1 | 2 |
| 5-hydroxytryptamine receptor 2A | Rattus norvegicus (Norway rat) | Ki | 0.0006 | 1 | 2 |
| 5-hydroxytryptamine receptor 2B | Homo sapiens (human) | IC50 | 1.5543 | 1 | 3 |
| 5-hydroxytryptamine receptor 2B | Homo sapiens (human) | Ki | 0.9890 | 1 | 3 |
| 5-hydroxytryptamine receptor 2C | Homo sapiens (human) | IC50 | 34.5460 | 1 | 2 |
| 5-hydroxytryptamine receptor 2C | Homo sapiens (human) | Ki | 18.0955 | 1 | 2 |
| 5-hydroxytryptamine receptor 4 | Cavia porcellus (domestic guinea pig) | IC50 | 34.5460 | 1 | 2 |
| 5-hydroxytryptamine receptor 4 | Cavia porcellus (domestic guinea pig) | Ki | 18.0955 | 1 | 2 |
| 5-hydroxytryptamine receptor 6 | Homo sapiens (human) | IC50 | 7.8950 | 1 | 2 |
| 5-hydroxytryptamine receptor 6 | Homo sapiens (human) | Ki | 3.6660 | 1 | 2 |
| 5-hydroxytryptamine receptor 7 | Cavia porcellus (domestic guinea pig) | IC50 | 12.4000 | 1 | 2 |
| Acetylcholinesterase | Homo sapiens (human) | IC50 | 25.5500 | 1 | 1 |
| Adenosine receptor A1 | Homo sapiens (human) | IC50 | 5.2785 | 1 | 2 |
| Adenosine receptor A1 | Homo sapiens (human) | Ki | 3.0790 | 1 | 2 |
| Adenosine receptor A2a | Homo sapiens (human) | IC50 | 9.0130 | 1 | 1 |
| Adenosine receptor A2a | Homo sapiens (human) | Ki | 73.3650 | 4 | 4 |
| Adenosine receptor A2a | Rattus norvegicus (Norway rat) | Ki | 23.8750 | 1 | 4 |
| Adenosine receptor A3 | Homo sapiens (human) | IC50 | 3.4930 | 1 | 3 |
| Adenosine receptor A3 | Homo sapiens (human) | Ki | 6.1591 | 3 | 8 |
| Aldehyde oxidase | Homo sapiens (human) | IC50 | 0.4600 | 1 | 1 |
| Aldo-keto reductase family 1 member B1 | Rattus norvegicus (Norway rat) | IC50 | 3.0324 | 1 | 3 |
| Aldo-keto reductase family 1 member B1 | Rattus norvegicus (Norway rat) | Ki | 1.9203 | 2 | 5 |
| Alpha-1A adrenergic receptor | Rattus norvegicus (Norway rat) | IC50 | 3.4930 | 1 | 3 |
| Alpha-1A adrenergic receptor | Homo sapiens (human) | Ki | 2.3440 | 1 | 1 |
| Alpha-1A adrenergic receptor | Rattus norvegicus (Norway rat) | Ki | 1.9743 | 1 | 3 |
| Alpha-1B adrenergic receptor | Rattus norvegicus (Norway rat) | IC50 | 3.4930 | 1 | 3 |
| Alpha-1B adrenergic receptor | Homo sapiens (human) | Ki | 7.9430 | 1 | 1 |
| Alpha-1B adrenergic receptor | Rattus norvegicus (Norway rat) | Ki | 1.9743 | 1 | 3 |
| Alpha-1D adrenergic receptor | Homo sapiens (human) | IC50 | 5.9965 | 1 | 2 |
| Alpha-1D adrenergic receptor | Homo sapiens (human) | Ki | 3.7547 | 2 | 3 |
| Alpha-2A adrenergic receptor | Homo sapiens (human) | IC50 | 5.0577 | 1 | 3 |
| Alpha-2A adrenergic receptor | Homo sapiens (human) | Ki | 1.8967 | 1 | 3 |
| Alpha-2A adrenergic receptor | Rattus norvegicus (Norway rat) | Ki | 5.3700 | 1 | 1 |
| Alpha-2B adrenergic receptor | Homo sapiens (human) | IC50 | 6.9700 | 1 | 2 |
| Alpha-2B adrenergic receptor | Homo sapiens (human) | Ki | 3.1815 | 1 | 2 |
| Alpha-2B adrenergic receptor | Rattus norvegicus (Norway rat) | Ki | 5.3700 | 1 | 1 |
| Alpha-2C adrenergic receptor | Homo sapiens (human) | IC50 | 5.8677 | 1 | 3 |
| Alpha-2C adrenergic receptor | Homo sapiens (human) | Ki | 0.8523 | 1 | 3 |
| Alpha-2C adrenergic receptor | Rattus norvegicus (Norway rat) | Ki | 5.3700 | 1 | 1 |
| Amyloid-beta precursor protein | Homo sapiens (human) | Ki | 0.0059 | 1 | 1 |
| Androgen receptor | Rattus norvegicus (Norway rat) | IC50 | 14.1254 | 1 | 1 |
| ATP-binding cassette sub-family C member 3 | Homo sapiens (human) | IC50 | 133.0000 | 1 | 10 |
| ATP-dependent translocase ABCB1 | Homo sapiens (human) | IC50 | 88.9563 | 10 | 12 |
| Beta-1 adrenergic receptor | Homo sapiens (human) | IC50 | 22.0880 | 1 | 1 |
| Beta-1 adrenergic receptor | Homo sapiens (human) | Ki | 12.7550 | 1 | 1 |
| Bile acid receptor | Homo sapiens (human) | IC50 | 6.9600 | 1 | 2 |
| Bile salt export pump | Homo sapiens (human) | IC50 | 170.4696 | 6 | 26 |
| Bile salt export pump | Rattus norvegicus (Norway rat) | IC50 | 522.7000 | 1 | 2 |
| Broad substrate specificity ATP-binding cassette transporter ABCG2 | Homo sapiens (human) | IC50 | 156.2397 | 6 | 6 |
| C-C chemokine receptor type 2 | Homo sapiens (human) | IC50 | 24.0637 | 3 | 3 |
| C-C chemokine receptor type 2 | Homo sapiens (human) | Ki | 0.8470 | 1 | 1 |
| C-C motif chemokine 2 | Homo sapiens (human) | IC50 | 6.9183 | 1 | 1 |
| Calcium release-activated calcium channel protein 1 | Homo sapiens (human) | IC50 | 1.0000 | 1 | 1 |
| Calcium/calmodulin-dependent 3',5'-cyclic nucleotide phosphodiesterase 1C | Homo sapiens (human) | IC50 | 4.3643 | 1 | 3 |
| cAMP-dependent protein kinase catalytic subunit alpha | Bos taurus (cattle) | IC50 | 1.8043 | 1 | 12 |
| cAMP-dependent protein kinase catalytic subunit alpha | Homo sapiens (human) | IC50 | 4.5800 | 1 | 1 |
| cAMP-dependent protein kinase catalytic subunit alpha | Homo sapiens (human) | Ki | 0.4600 | 1 | 1 |
| cAMP-dependent protein kinase catalytic subunit alpha | Mus musculus (house mouse) | Ki | 0.4950 | 1 | 2 |
| cAMP-dependent protein kinase catalytic subunit beta | Homo sapiens (human) | IC50 | 4.5800 | 1 | 1 |
| cAMP-dependent protein kinase catalytic subunit beta | Homo sapiens (human) | Ki | 0.4600 | 1 | 1 |
| cAMP-dependent protein kinase catalytic subunit gamma | Homo sapiens (human) | IC50 | 4.5800 | 1 | 1 |
| cAMP-dependent protein kinase catalytic subunit gamma | Homo sapiens (human) | Ki | 0.4600 | 1 | 1 |
| cAMP-specific 3',5'-cyclic phosphodiesterase 4D | Homo sapiens (human) | IC50 | 7.1500 | 1 | 1 |
| Canalicular multispecific organic anion transporter 1 | Homo sapiens (human) | IC50 | 125.5000 | 2 | 10 |
| Cannabinoid receptor 1 | Homo sapiens (human) | IC50 | 1.7360 | 1 | 1 |
| Cannabinoid receptor 1 | Homo sapiens (human) | Ki | 1.3710 | 1 | 1 |
| Carbonic anhydrase 1 | Homo sapiens (human) | IC50 | 91.5000 | 1 | 2 |
| Carbonic anhydrase 2 | Homo sapiens (human) | IC50 | 91.5000 | 1 | 2 |
| Cathepsin B | Homo sapiens (human) | IC50 | 50.0000 | 1 | 1 |
| Cell division control protein 42 homolog | Homo sapiens (human) | IC50 | 6.5000 | 2 | 2 |
| Chain A, cAMP-dependent protein kinase, alpha-catalytic subunit | Bos taurus (cattle) | IC50 | 2.2800 | 1 | 5 |
| Chain A, Rho-associated protein kinase 1 | Homo sapiens (human) | Ki | 0.5300 | 1 | 3 |
| Chain B, Rho-associated protein kinase 1 | Homo sapiens (human) | Ki | 0.5300 | 1 | 1 |
| Chain E, cAMP-dependent protein kinase, alpha-catalytic subunit | Mus musculus (house mouse) | Ki | 0.5300 | 1 | 1 |
| Chain I, cAMP-dependent protein kinase inhibitor alpha | synthetic construct | IC50 | 2.2800 | 1 | 2 |
| Chain I, cAMP-dependent protein kinase inhibitor, alpha form | synthetic construct | Ki | 0.5300 | 1 | 1 |
| Cruzipain | Trypanosoma cruzi | IC50 | 212.0000 | 2 | 2 |
| Cysteinyl leukotriene receptor 1 | Homo sapiens (human) | IC50 | 17.7450 | 1 | 1 |
| Cysteinyl leukotriene receptor 1 | Homo sapiens (human) | Ki | 8.8720 | 1 | 1 |
| Cytochrome P450 1A1 | Homo sapiens (human) | Ki | 0.2100 | 1 | 1 |
| Cytochrome P450 1A2 | Homo sapiens (human) | IC50 | 0.3000 | 1 | 1 |
| Cytochrome P450 1B1 | Homo sapiens (human) | Ki | 0.0350 | 2 | 2 |
| Cytochrome P450 2C19 | Homo sapiens (human) | IC50 | 2.5333 | 1 | 3 |
| Cytochrome P450 2C9 | Homo sapiens (human) | IC50 | 10.5456 | 2 | 7 |
| Cytochrome P450 2J2 | Homo sapiens (human) | IC50 | 16.9850 | 1 | 4 |
| Cytochrome P450 3A4 | Homo sapiens (human) | IC50 | 69.0240 | 3 | 4 |
| Cytochrome P450 3A4 | Homo sapiens (human) | Ki | 1.3500 | 2 | 2 |
| D(1A) dopamine receptor | Homo sapiens (human) | IC50 | 7.7630 | 1 | 1 |
| D(1A) dopamine receptor | Homo sapiens (human) | Ki | 3.8820 | 1 | 1 |
| D(2) dopamine receptor | Homo sapiens (human) | IC50 | 7.0485 | 1 | 2 |
| D(2) dopamine receptor | Homo sapiens (human) | Ki | 2.3495 | 1 | 2 |
| D(3) dopamine receptor | Homo sapiens (human) | IC50 | 3.1589 | 1 | 3 |
| D(3) dopamine receptor | Homo sapiens (human) | Ki | 1.0729 | 1 | 3 |
| Delta-type opioid receptor | Homo sapiens (human) | IC50 | 2.7180 | 1 | 1 |
| Delta-type opioid receptor | Rattus norvegicus (Norway rat) | IC50 | 8.7167 | 2 | 3 |
| Delta-type opioid receptor | Homo sapiens (human) | Ki | 5.9553 | 6 | 9 |
| Delta-type opioid receptor | Mus musculus (house mouse) | Ki | 3.2500 | 4 | 4 |
| Delta-type opioid receptor | Rattus norvegicus (Norway rat) | Ki | 5.0000 | 1 | 1 |
| Dihydrofolate reductase | Escherichia coli K-12 | IC50 | 348.9000 | 1 | 1 |
| Dihydrofolate reductase | Escherichia coli K-12 | Ki | 15.2400 | 1 | 1 |
| Estrogen receptor | Homo sapiens (human) | IC50 | 0.1312 | 6 | 6 |
| Estrogen receptor | Homo sapiens (human) | Ki | 0.0002 | 5 | 5 |
| Estrogen receptor 1 | Homo sapiens (human) | IC50 | 50.0000 | 1 | 1 |
| Estrogen receptor beta | Homo sapiens (human) | IC50 | 0.1588 | 4 | 4 |
| Estrogen receptor beta | Homo sapiens (human) | Ki | 0.0003 | 3 | 3 |
| estrogen receptor beta isoform 1 | Homo sapiens (human) | IC50 | 50.0000 | 1 | 1 |
| fructose-bisphosphate aldolase | Mycobacterium tuberculosis H37Rv | IC50 | 9.9910 | 1 | 1 |
| G-protein coupled receptor 35 | Homo sapiens (human) | Ki | 2.3400 | 1 | 1 |
| G-protein coupled receptor 55 | Homo sapiens (human) | IC50 | 1.4652 | 1 | 1 |
| Glucocorticoid receptor | Homo sapiens (human) | IC50 | 10.6000 | 1 | 1 |
| Glucocorticoid receptor | Homo sapiens (human) | Ki | 4.8180 | 1 | 1 |
| Glutathione reductase, mitochondrial | Homo sapiens (human) | IC50 | 23.4000 | 1 | 1 |
| Glutathione reductase, mitochondrial | Homo sapiens (human) | Ki | 17.4000 | 1 | 1 |
| Glycine receptor subunit alpha-1 | Rattus norvegicus (Norway rat) | IC50 | 10.6000 | 1 | 1 |
| Glycine receptor subunit alpha-1 | Rattus norvegicus (Norway rat) | Ki | 4.8180 | 1 | 1 |
| Glycine receptor subunit alpha-2 | Rattus norvegicus (Norway rat) | IC50 | 10.6000 | 1 | 1 |
| Glycine receptor subunit alpha-2 | Rattus norvegicus (Norway rat) | Ki | 4.8180 | 1 | 1 |
| Glycine receptor subunit alpha-3 | Rattus norvegicus (Norway rat) | IC50 | 10.6000 | 1 | 1 |
| Glycine receptor subunit alpha-3 | Rattus norvegicus (Norway rat) | Ki | 4.8180 | 1 | 1 |
| Glycine receptor subunit beta | Rattus norvegicus (Norway rat) | IC50 | 10.6000 | 1 | 1 |
| Glycine receptor subunit beta | Rattus norvegicus (Norway rat) | Ki | 4.8180 | 1 | 1 |
| Hematopoietic prostaglandin D synthase | Homo sapiens (human) | IC50 | 11.6000 | 2 | 2 |
| high affinity choline transporter 1 isoform a | Homo sapiens (human) | IC50 | 12.5893 | 1 | 1 |
| Histamine H1 receptor | Homo sapiens (human) | IC50 | 0.0740 | 1 | 1 |
| Histamine H1 receptor | Homo sapiens (human) | Ki | 0.0086 | 1 | 1 |
| Indoleamine 2,3-dioxygenase 1 | Mus musculus (house mouse) | IC50 | 46.0000 | 1 | 1 |
| Indoleamine 2,3-dioxygenase 2 | Mus musculus (house mouse) | IC50 | 1.5000 | 1 | 1 |
| Kappa-type opioid receptor | Cavia porcellus (domestic guinea pig) | IC50 | 0.0958 | 2 | 2 |
| Kappa-type opioid receptor | Homo sapiens (human) | IC50 | 0.3543 | 14 | 15 |
| Kappa-type opioid receptor | Mus musculus (house mouse) | IC50 | 0.0027 | 2 | 3 |
| Kappa-type opioid receptor | Rattus norvegicus (Norway rat) | IC50 | 5.2303 | 4 | 5 |
| Kappa-type opioid receptor | Cavia porcellus (domestic guinea pig) | Ki | 0.0191 | 13 | 16 |
| Kappa-type opioid receptor | Homo sapiens (human) | Ki | 0.0756 | 26 | 27 |
| Kappa-type opioid receptor | Mus musculus (house mouse) | Ki | 0.0081 | 1 | 1 |
| Kappa-type opioid receptor | Rattus norvegicus (Norway rat) | Ki | 0.0005 | 2 | 2 |
| L-cysteine:1D-myo-inositol 2-amino-2-deoxy-alpha-D-glucopyranoside ligase | Mycobacterium tuberculosis H37Rv | IC50 | 2,500.0000 | 1 | 1 |
| Lethal factor | Bacillus anthracis | IC50 | 4.8000 | 1 | 1 |
| Lethal(3)malignant brain tumor-like protein 1 | Homo sapiens (human) | IC50 | 100.0000 | 1 | 1 |
| Lethal(3)malignant brain tumor-like protein 3 | Homo sapiens (human) | IC50 | 54.0000 | 1 | 1 |
| Lethal(3)malignant brain tumor-like protein 4 | Homo sapiens (human) | IC50 | 100.0000 | 1 | 1 |
| MBT domain-containing protein 1 | Homo sapiens (human) | IC50 | 100.0000 | 1 | 1 |
| Mitogen-activated protein kinase 14 | Homo sapiens (human) | IC50 | 32.9030 | 1 | 1 |
| MO15-related protein kinase Pfmrk | Plasmodium falciparum (malaria parasite P. falciparum) | IC50 | 500.0000 | 1 | 1 |
| Mu-type opioid receptor | Homo sapiens (human) | IC50 | 4.0250 | 1 | 2 |
| Mu-type opioid receptor | Rattus norvegicus (Norway rat) | IC50 | 8.7167 | 2 | 3 |
| Mu-type opioid receptor | Cavia porcellus (domestic guinea pig) | Ki | 0.5226 | 6 | 13 |
| Mu-type opioid receptor | Homo sapiens (human) | Ki | 1.1857 | 2 | 3 |
| Mu-type opioid receptor | Mus musculus (house mouse) | Ki | 0.5050 | 3 | 4 |
| Mu-type opioid receptor | Rattus norvegicus (Norway rat) | Ki | 1.3345 | 5 | 6 |
| Multidrug resistance-associated protein 4 | Homo sapiens (human) | IC50 | 108.1600 | 1 | 10 |
| Muscarinic acetylcholine receptor M1 | Homo sapiens (human) | IC50 | 5.8958 | 1 | 3 |
| Muscarinic acetylcholine receptor M1 | Homo sapiens (human) | Ki | 0.8526 | 3 | 5 |
| Muscarinic acetylcholine receptor M1 | Rattus norvegicus (Norway rat) | Ki | 0.0059 | 1 | 1 |
| Muscarinic acetylcholine receptor M2 | Homo sapiens (human) | IC50 | 0.0270 | 1 | 1 |
| Muscarinic acetylcholine receptor M2 | Homo sapiens (human) | Ki | 0.0114 | 4 | 4 |
| Muscarinic acetylcholine receptor M2 | Rattus norvegicus (Norway rat) | Ki | 0.0105 | 2 | 2 |
| Muscarinic acetylcholine receptor M3 | Homo sapiens (human) | IC50 | 6.3989 | 1 | 3 |
| Muscarinic acetylcholine receptor M3 | Homo sapiens (human) | Ki | 0.6789 | 4 | 6 |
| Muscarinic acetylcholine receptor M3 | Rattus norvegicus (Norway rat) | Ki | 0.0031 | 2 | 2 |
| Muscarinic acetylcholine receptor M4 | Homo sapiens (human) | IC50 | 1.8310 | 1 | 2 |
| Muscarinic acetylcholine receptor M4 | Homo sapiens (human) | Ki | 0.1713 | 2 | 3 |
| Muscarinic acetylcholine receptor M5 | Homo sapiens (human) | IC50 | 0.3811 | 1 | 2 |
| Muscarinic acetylcholine receptor M5 | Homo sapiens (human) | Ki | 0.1871 | 2 | 3 |
| Myosin light chain kinase, smooth muscle | Homo sapiens (human) | IC50 | 9.0733 | 3 | 3 |
| Myosin light chain kinase, smooth muscle | Homo sapiens (human) | Ki | 36.0000 | 1 | 1 |
| Myotonin-protein kinase | Homo sapiens (human) | IC50 | 8.0000 | 1 | 1 |
| NACHT, LRR and PYD domains-containing protein 3 | Mus musculus (house mouse) | IC50 | 25.0000 | 1 | 1 |
| NEDD8-activating enzyme E1 regulatory subunit isoform a | Homo sapiens (human) | IC50 | 34.7000 | 1 | 1 |
| NEDD8-conjugating enzyme Ubc12 | Homo sapiens (human) | IC50 | 34.7000 | 1 | 1 |
| Nuclear receptor subfamily 1 group I member 2 | Homo sapiens (human) | IC50 | 14.6000 | 1 | 1 |
| perilipin-1 | Homo sapiens (human) | IC50 | 9.6190 | 1 | 1 |
| perilipin-5 | Homo sapiens (human) | IC50 | 7.1330 | 1 | 1 |
| Platelet-activating factor receptor | Cavia porcellus (domestic guinea pig) | Ki | 73.3100 | 1 | 1 |
| Polyunsaturated fatty acid 5-lipoxygenase | Homo sapiens (human) | Ki | 0.0001 | 1 | 1 |
| Polyunsaturated fatty acid lipoxygenase ALOX15 | Oryctolagus cuniculus (rabbit) | IC50 | 9.0320 | 1 | 2 |
| Potassium channel subfamily K member 2 | Homo sapiens (human) | IC50 | 0.4000 | 1 | 1 |
| Potassium channel subfamily K member 2 | Bos taurus (cattle) | IC50 | 4.3150 | 1 | 2 |
| Potassium voltage-gated channel subfamily A member 1 | Homo sapiens (human) | IC50 | 120.0000 | 1 | 2 |
| Potassium voltage-gated channel subfamily A member 5 | Homo sapiens (human) | IC50 | 6.1000 | 1 | 1 |
| Potassium voltage-gated channel subfamily E member 1 | Homo sapiens (human) | IC50 | 158.4890 | 1 | 1 |
| Potassium voltage-gated channel subfamily H member 2 | Homo sapiens (human) | IC50 | 64.4288 | 18 | 32 |
| Potassium voltage-gated channel subfamily H member 2 | Homo sapiens (human) | Ki | 6.5095 | 4 | 4 |
| Potassium voltage-gated channel subfamily KQT member 1 | Homo sapiens (human) | IC50 | 158.4890 | 1 | 1 |
| procathepsin L isoform 1 preproprotein | Homo sapiens (human) | IC50 | 50.0000 | 1 | 1 |
| Prostaglandin G/H synthase 1 | Homo sapiens (human) | IC50 | 5.6000 | 1 | 1 |
| Protein kinase C epsilon type | Homo sapiens (human) | IC50 | 3.0000 | 2 | 2 |
| Receptor-type tyrosine-protein kinase FLT3 | Homo sapiens (human) | IC50 | 1.1000 | 1 | 1 |
| Rho-associated protein kinase 1 | Homo sapiens (human) | IC50 | 1.0502 | 10 | 10 |
| Rho-associated protein kinase 1 | Homo sapiens (human) | Ki | 0.4300 | 6 | 7 |
| Rho-associated protein kinase 2 | Bos taurus (cattle) | IC50 | 1.8042 | 1 | 12 |
| Rho-associated protein kinase 2 | Homo sapiens (human) | IC50 | 1.3060 | 14 | 14 |
| Rho-associated protein kinase 2 | Rattus norvegicus (Norway rat) | IC50 | 1.9000 | 1 | 1 |
| Rho-associated protein kinase 2 | Homo sapiens (human) | Ki | 0.3300 | 1 | 1 |
| Ribosomal protein S6 kinase alpha-5 | Homo sapiens (human) | IC50 | 5.0000 | 1 | 1 |
| Sarcoplasmic/endoplasmic reticulum calcium ATPase 1 | Oryctolagus cuniculus (rabbit) | IC50 | 21.0010 | 4 | 4 |
| Sarcoplasmic/endoplasmic reticulum calcium ATPase 1 | Homo sapiens (human) | Ki | 0.0001 | 1 | 1 |
| Serine/threonine-protein kinase N1 | Homo sapiens (human) | IC50 | 1.7000 | 1 | 1 |
| Serine/threonine-protein kinase N2 | Homo sapiens (human) | IC50 | 1.8533 | 3 | 3 |
| Sigma non-opioid intracellular receptor 1 | Homo sapiens (human) | IC50 | 0.0321 | 1 | 2 |
| Sigma non-opioid intracellular receptor 1 | Rattus norvegicus (Norway rat) | IC50 | 10.0000 | 1 | 1 |
| Sigma non-opioid intracellular receptor 1 | Homo sapiens (human) | Ki | 0.0136 | 1 | 2 |
| Sodium channel protein type 1 subunit alpha | Homo sapiens (human) | IC50 | 27.3333 | 3 | 3 |
| Sodium channel protein type 1 subunit alpha | Rattus norvegicus (Norway rat) | IC50 | 82.6333 | 2 | 3 |
| Sodium channel protein type 10 subunit alpha | Homo sapiens (human) | IC50 | 55.2000 | 5 | 5 |
| Sodium channel protein type 11 subunit alpha | Homo sapiens (human) | IC50 | 27.3333 | 3 | 3 |
| Sodium channel protein type 2 subunit alpha | Homo sapiens (human) | IC50 | 34.8333 | 6 | 6 |
| Sodium channel protein type 2 subunit alpha | Rattus norvegicus (Norway rat) | IC50 | 63.5800 | 4 | 5 |
| Sodium channel protein type 3 subunit alpha | Homo sapiens (human) | IC50 | 24.7500 | 4 | 4 |
| Sodium channel protein type 3 subunit alpha | Rattus norvegicus (Norway rat) | IC50 | 82.6333 | 2 | 3 |
| Sodium channel protein type 4 subunit alpha | Homo sapiens (human) | IC50 | 27.3333 | 3 | 3 |
| Sodium channel protein type 4 subunit alpha | Homo sapiens (human) | Ki | 17.0000 | 1 | 1 |
| Sodium channel protein type 5 subunit alpha | Homo sapiens (human) | IC50 | 41.0730 | 7 | 7 |
| Sodium channel protein type 7 subunit alpha | Homo sapiens (human) | IC50 | 27.3333 | 3 | 3 |
| Sodium channel protein type 8 subunit alpha | Homo sapiens (human) | IC50 | 27.3333 | 3 | 3 |
| Sodium channel protein type 9 subunit alpha | Homo sapiens (human) | IC50 | 24.7500 | 4 | 4 |
| Sodium-dependent dopamine transporter | Homo sapiens (human) | IC50 | 2.0796 | 1 | 4 |
| Sodium-dependent dopamine transporter | Homo sapiens (human) | Ki | 1.6525 | 1 | 4 |
| Sodium-dependent noradrenaline transporter | Homo sapiens (human) | IC50 | 4.7743 | 2 | 4 |
| Sodium-dependent noradrenaline transporter | Homo sapiens (human) | Ki | 4.7554 | 2 | 4 |
| Sodium-dependent serotonin transporter | Homo sapiens (human) | IC50 | 6.7910 | 1 | 2 |
| Sodium-dependent serotonin transporter | Homo sapiens (human) | Ki | 3.6080 | 1 | 2 |
| Solute carrier family 22 member 1 | Homo sapiens (human) | IC50 | 12.4000 | 1 | 1 |
| Solute carrier family 22 member 20 | Mus musculus (house mouse) | Ki | 48.9890 | 1 | 2 |
| Solute carrier family 22 member 6 | Mus musculus (house mouse) | Ki | 6.2548 | 1 | 2 |
| Stromal interaction molecule 1 | Homo sapiens (human) | IC50 | 1.0000 | 1 | 1 |
| Substance-K receptor | Homo sapiens (human) | IC50 | 9.5530 | 1 | 1 |
| Substance-K receptor | Homo sapiens (human) | Ki | 3.1840 | 1 | 1 |
| Thromboxane-A synthase | Homo sapiens (human) | IC50 | 340.9843 | 2 | 3 |
| Transient receptor potential cation channel subfamily A member 1 | Homo sapiens (human) | IC50 | 125.9465 | 1 | 2 |
| Transient receptor potential cation channel subfamily M member 2 | Homo sapiens (human) | IC50 | 1.8800 | 5 | 5 |
| Transient receptor potential cation channel subfamily V member 2 | Homo sapiens (human) | IC50 | 10.0000 | 1 | 1 |
| Tyrosine-protein kinase Fyn | Homo sapiens (human) | IC50 | 14.2330 | 1 | 1 |
| ubiquitin-conjugating enzyme E2 N | Homo sapiens (human) | IC50 | 20.0000 | 1 | 1 |
| UDP-glucose 4-epimerase | Homo sapiens (human) | IC50 | 75.0000 | 1 | 1 |
| Vasopressin V1a receptor | Homo sapiens (human) | IC50 | 25.9250 | 1 | 1 |
| Vasopressin V1a receptor | Homo sapiens (human) | Ki | 10.4010 | 1 | 1 |
| Voltage-dependent calcium channel gamma-1 subunit | Homo sapiens (human) | IC50 | 14.0000 | 1 | 1 |
| Voltage-dependent calcium channel gamma-2 subunit | Homo sapiens (human) | IC50 | 14.0000 | 1 | 1 |
| Voltage-dependent calcium channel gamma-3 subunit | Homo sapiens (human) | IC50 | 14.0000 | 1 | 1 |
| Voltage-dependent calcium channel gamma-4 subunit | Homo sapiens (human) | IC50 | 14.0000 | 1 | 1 |
| Voltage-dependent calcium channel gamma-5 subunit | Homo sapiens (human) | IC50 | 14.0000 | 1 | 1 |
| Voltage-dependent calcium channel gamma-6 subunit | Homo sapiens (human) | IC50 | 14.0000 | 1 | 1 |
| Voltage-dependent calcium channel gamma-7 subunit | Homo sapiens (human) | IC50 | 14.0000 | 1 | 1 |
| Voltage-dependent calcium channel gamma-8 subunit | Homo sapiens (human) | IC50 | 14.0000 | 1 | 1 |
| Voltage-dependent calcium channel subunit alpha-2/delta-1 | Homo sapiens (human) | IC50 | 7.0149 | 2 | 2 |
| Voltage-dependent calcium channel subunit alpha-2/delta-1 | Homo sapiens (human) | Ki | 0.0190 | 2 | 2 |
| Voltage-dependent calcium channel subunit alpha-2/delta-1 | Mus musculus (house mouse) | Ki | 0.1201 | 1 | 2 |
| Voltage-dependent calcium channel subunit alpha-2/delta-2 | Homo sapiens (human) | IC50 | 14.0000 | 1 | 1 |
| Voltage-dependent calcium channel subunit alpha-2/delta-2 | Homo sapiens (human) | Ki | 0.0990 | 1 | 1 |
| Voltage-dependent calcium channel subunit alpha-2/delta-3 | Homo sapiens (human) | IC50 | 14.0000 | 1 | 1 |
| Voltage-dependent calcium channel subunit alpha-2/delta-4 | Homo sapiens (human) | IC50 | 14.0000 | 1 | 1 |
| Voltage-dependent L-type calcium channel subunit alpha-1C | Cavia porcellus (domestic guinea pig) | IC50 | 2.5340 | 9 | 19 |
| Voltage-dependent L-type calcium channel subunit alpha-1C | Homo sapiens (human) | IC50 | 134.1453 | 22 | 22 |
| Voltage-dependent L-type calcium channel subunit alpha-1C | Mus musculus (house mouse) | IC50 | 1.2000 | 1 | 1 |
| Voltage-dependent L-type calcium channel subunit alpha-1C | Rattus norvegicus (Norway rat) | IC50 | 9.6969 | 8 | 11 |
| Voltage-dependent L-type calcium channel subunit alpha-1C | Homo sapiens (human) | Ki | 0.0077 | 2 | 4 |
| Voltage-dependent L-type calcium channel subunit alpha-1C | Rattus norvegicus (Norway rat) | Ki | 0.0518 | 6 | 8 |
| Voltage-dependent L-type calcium channel subunit alpha-1D | Mus musculus (house mouse) | IC50 | 1.2000 | 1 | 1 |
| Voltage-dependent L-type calcium channel subunit alpha-1D | Rattus norvegicus (Norway rat) | IC50 | 0.6723 | 4 | 4 |
| Voltage-dependent L-type calcium channel subunit alpha-1D | Rattus norvegicus (Norway rat) | Ki | 0.0257 | 4 | 5 |
| Voltage-dependent L-type calcium channel subunit alpha-1D | Homo sapiens (human) | IC50 | 3.9660 | 10 | 10 |
| Voltage-dependent L-type calcium channel subunit alpha-1D | Homo sapiens (human) | Ki | 0.0147 | 1 | 2 |
| Voltage-dependent L-type calcium channel subunit alpha-1F | Homo sapiens (human) | IC50 | 4.2567 | 9 | 9 |
| Voltage-dependent L-type calcium channel subunit alpha-1F | Mus musculus (house mouse) | IC50 | 1.2000 | 1 | 1 |
| Voltage-dependent L-type calcium channel subunit alpha-1F | Homo sapiens (human) | Ki | 0.0147 | 1 | 2 |
| Voltage-dependent L-type calcium channel subunit alpha-1S | Homo sapiens (human) | IC50 | 4.2567 | 9 | 9 |
| Voltage-dependent L-type calcium channel subunit alpha-1S | Mus musculus (house mouse) | IC50 | 1.2000 | 1 | 1 |
| Voltage-dependent L-type calcium channel subunit alpha-1S | Rattus norvegicus (Norway rat) | IC50 | 0.6723 | 4 | 4 |
| Voltage-dependent L-type calcium channel subunit alpha-1S | Homo sapiens (human) | Ki | 0.0147 | 1 | 2 |
| Voltage-dependent L-type calcium channel subunit alpha-1S | Rattus norvegicus (Norway rat) | Ki | 0.0220 | 4 | 6 |
| Voltage-dependent L-type calcium channel subunit beta-1 | Homo sapiens (human) | IC50 | 14.0000 | 1 | 1 |
| Voltage-dependent L-type calcium channel subunit beta-2 | Homo sapiens (human) | IC50 | 7.0149 | 2 | 2 |
| Voltage-dependent L-type calcium channel subunit beta-3 | Homo sapiens (human) | IC50 | 14.0000 | 1 | 1 |
| Voltage-dependent L-type calcium channel subunit beta-4 | Homo sapiens (human) | IC50 | 14.0000 | 1 | 1 |
| Voltage-dependent N-type calcium channel subunit alpha-1B | Homo sapiens (human) | IC50 | 16.9000 | 4 | 4 |
| Voltage-dependent P/Q-type calcium channel subunit alpha-1A | Homo sapiens (human) | IC50 | 14.0000 | 1 | 1 |
| Voltage-dependent R-type calcium channel subunit alpha-1E | Homo sapiens (human) | IC50 | 14.0000 | 1 | 1 |
| Voltage-dependent T-type calcium channel subunit alpha-1G | Homo sapiens (human) | IC50 | 14.0000 | 1 | 1 |
| Voltage-dependent T-type calcium channel subunit alpha-1H | Homo sapiens (human) | IC50 | 19.0000 | 2 | 2 |
| Voltage-dependent T-type calcium channel subunit alpha-1I | Homo sapiens (human) | IC50 | 14.0000 | 1 | 1 |
| Protein | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Drugs |
|---|
| 26S proteasome regulatory subunit 6B | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| 5'-AMP-activated protein kinase catalytic subunit alpha-1 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| 5'-AMP-activated protein kinase subunit gamma-1 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| 5'-AMP-activated protein kinase subunit gamma-2 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| AarF domain-containing protein kinase 1 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Actin-related protein 2 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Actin-related protein 3 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Activated CDC42 kinase 1 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Activin receptor type-1 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Activin receptor type-1B | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Activin receptor type-2B | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Acyl-CoA dehydrogenase family member 10 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Acyl-CoA dehydrogenase family member 11 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Adenine phosphoribosyltransferase | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Adenosine kinase | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Adenylate kinase 2, mitochondrial | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| ADP/ATP translocase 2 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| ADP/ATP translocase 3 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| AP2-associated protein kinase 1 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| ATP-dependent 6-phosphofructokinase, platelet type | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| ATP-dependent RNA helicase DDX1 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| ATP-dependent RNA helicase DDX3X | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| ATP-dependent RNA helicase DDX42 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| ATP-dependent RNA helicase DHX30 | Homo sapiens (human) | Kd | 30.0000 | 1 | 2 |
| Atypical kinase COQ8A, mitochondrial | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Aurora kinase A | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Aurora kinase B | Homo sapiens (human) | Kd | 15.5700 | 2 | 2 |
| Beta-adrenergic receptor kinase 1 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| BMP-2-inducible protein kinase | Homo sapiens (human) | Kd | 33.7880 | 1 | 1 |
| Bone morphogenetic protein receptor type-1A | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Bone morphogenetic protein receptor type-1B | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Bone morphogenetic protein receptor type-2 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Breakpoint cluster region protein | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Calcium/calmodulin-dependent protein kinase kinase 2 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Calcium/calmodulin-dependent protein kinase type II subunit delta | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Calcium/calmodulin-dependent protein kinase type II subunit gamma | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Calcium/calmodulin-dependent protein kinase type IV | Homo sapiens (human) | Kd | 30.0000 | 1 | 2 |
| cAMP-dependent protein kinase catalytic subunit alpha | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| cAMP-dependent protein kinase catalytic subunit beta | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| cAMP-dependent protein kinase catalytic subunit gamma | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| cAMP-dependent protein kinase type II-alpha regulatory subunit | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Casein kinase I isoform alpha | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Casein kinase I isoform delta | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Casein kinase I isoform epsilon | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Casein kinase I isoform gamma-1 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Casein kinase I isoform gamma-2 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Casein kinase I isoform gamma-3 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Casein kinase II subunit alpha' | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Cell division cycle 7-related protein kinase | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| cGMP-dependent protein kinase 1 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Choline-phosphate cytidylyltransferase A | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Chromodomain-helicase-DNA-binding protein 4 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Citron Rho-interacting kinase | Homo sapiens (human) | Kd | 48.8760 | 1 | 1 |
| Cyclin-dependent kinase 1 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Cyclin-dependent kinase 12 | Homo sapiens (human) | Kd | 3.4800 | 1 | 1 |
| Cyclin-dependent kinase 13 | Homo sapiens (human) | Kd | 4.5180 | 1 | 1 |
| Cyclin-dependent kinase 16 | Homo sapiens (human) | Kd | 30.0000 | 1 | 2 |
| Cyclin-dependent kinase 17 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Cyclin-dependent kinase 2 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Cyclin-dependent kinase 3 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Cyclin-dependent kinase 4 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Cyclin-dependent kinase 6 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Cyclin-dependent kinase 7 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Cyclin-dependent kinase 9 | Homo sapiens (human) | Kd | 4.2510 | 1 | 1 |
| Cyclin-dependent-like kinase 5 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Cyclin-G-associated kinase | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Cysteine--tRNA ligase, cytoplasmic | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Cytochrome c1, heme protein, mitochondrial | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| dCTP pyrophosphatase 1 | Homo sapiens (human) | Kd | 30.0000 | 1 | 2 |
| Delta(24)-sterol reductase | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Deoxycytidine kinase | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Discoidin domain-containing receptor 2 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| DNA replication licensing factor MCM4 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| DNA topoisomerase 2-alpha | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| DNA topoisomerase 2-beta | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| DnaJ homolog subfamily A member 1 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Dual specificity mitogen-activated protein kinase kinase 1 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Dual specificity mitogen-activated protein kinase kinase 2 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Dual specificity mitogen-activated protein kinase kinase 3 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Dual specificity mitogen-activated protein kinase kinase 5 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Dual specificity mitogen-activated protein kinase kinase 6 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Dual specificity protein kinase CLK1 | Homo sapiens (human) | Kd | 0.1520 | 1 | 1 |
| Dual specificity protein kinase CLK2 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Dual specificity protein kinase CLK3 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Dual specificity protein kinase CLK4 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Dual specificity protein kinase TTK | Homo sapiens (human) | Kd | 30.0000 | 1 | 2 |
| Dual specificity testis-specific protein kinase 1 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Dual specificity testis-specific protein kinase 2 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Dual specificity tyrosine-phosphorylation-regulated kinase 1A | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Dynamin-like 120 kDa protein, mitochondrial | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| EKC/KEOPS complex subunit TP53RK | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Electron transfer flavoprotein subunit beta | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Elongation factor Tu, mitochondrial | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Envelope glycoprotein | Ebola virus - Mayinga, Zaire, 1976 | Kd | 290.0000 | 1 | 1 |
| Ephrin type-A receptor 1 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Ephrin type-A receptor 2 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Ephrin type-A receptor 4 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Ephrin type-A receptor 5 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Ephrin type-A receptor 7 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Ephrin type-B receptor 2 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Ephrin type-B receptor 3 | Homo sapiens (human) | Kd | 30.0000 | 1 | 2 |
| Ephrin type-B receptor 4 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Ephrin type-B receptor 6 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Epidermal growth factor receptor | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Epithelial discoidin domain-containing receptor 1 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Estrogen receptor | Homo sapiens (human) | EC50 | 0.0025 | 5 | 5 |
| Estrogen receptor beta | Homo sapiens (human) | EC50 | 0.0045 | 2 | 2 |
| Estrogen-related receptor gamma | Homo sapiens (human) | EC50 | 0.6300 | 2 | 2 |
| Eukaryotic peptide chain release factor GTP-binding subunit ERF3B | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Eukaryotic translation initiation factor 2-alpha kinase 1 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Eukaryotic translation initiation factor 5B | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Exosome RNA helicase MTR4 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Ferrochelatase, mitochondrial | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Fibroblast growth factor receptor 1 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Focal adhesion kinase 1 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| G protein-coupled receptor kinase 6 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| G-protein coupled receptor 35 | Homo sapiens (human) | EC50 | 1.9455 | 4 | 4 |
| General transcription and DNA repair factor IIH helicase subunit XPD | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Glycine--tRNA ligase | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Glycogen phosphorylase, brain form | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Glycogen phosphorylase, liver form | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Glycogen synthase kinase-3 alpha | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Glycogen synthase kinase-3 beta | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| GTP-binding nuclear protein Ran | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Guanine nucleotide-binding protein G(i) subunit alpha-2 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Heme oxygenase 2 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Hepatocyte growth factor receptor | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| High affinity nerve growth factor receptor | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Inhibitor of nuclear factor kappa-B kinase subunit epsilon | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Inosine-5'-monophosphate dehydrogenase 2 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Insulin receptor | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Insulin-like growth factor 1 receptor | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Integrin-linked protein kinase | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Interleukin-1 receptor-associated kinase 1 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Interleukin-1 receptor-associated kinase 3 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Interleukin-1 receptor-associated kinase 4 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Kappa-type opioid receptor | Homo sapiens (human) | EC50 | 0.0416 | 32 | 32 |
| Kappa-type opioid receptor | Mus musculus (house mouse) | EC50 | 1.6365 | 3 | 3 |
| LIM domain kinase 1 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| LIM domain kinase 2 | Homo sapiens (human) | Kd | 30.0000 | 1 | 2 |
| Long-chain-fatty-acid--CoA ligase 5 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Macrophage-stimulating protein receptor | Homo sapiens (human) | Kd | 30.0000 | 1 | 2 |
| MAP kinase-activated protein kinase 2 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| MAP kinase-activated protein kinase 5 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| MAP/microtubule affinity-regulating kinase 3 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| MAP/microtubule affinity-regulating kinase 4 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Maternal embryonic leucine zipper kinase | Homo sapiens (human) | Kd | 1.9220 | 1 | 1 |
| Membrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinase | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Midasin | Homo sapiens (human) | Kd | 30.0000 | 1 | 2 |
| Mitogen-activated protein kinase 1 | Homo sapiens (human) | Kd | 30.0000 | 1 | 2 |
| Mitogen-activated protein kinase 10 | Homo sapiens (human) | EC50 | 1.2400 | 1 | 1 |
| Mitogen-activated protein kinase 10 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Mitogen-activated protein kinase 11 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Mitogen-activated protein kinase 14 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Mitogen-activated protein kinase 15 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Mitogen-activated protein kinase 3 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Mitogen-activated protein kinase 7 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Mitogen-activated protein kinase 8 | Homo sapiens (human) | EC50 | 1.2400 | 1 | 1 |
| Mitogen-activated protein kinase 8 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Mitogen-activated protein kinase 9 | Homo sapiens (human) | EC50 | 1.2400 | 1 | 1 |
| Mitogen-activated protein kinase 9 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Mitogen-activated protein kinase kinase kinase 1 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Mitogen-activated protein kinase kinase kinase 11 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Mitogen-activated protein kinase kinase kinase 2 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Mitogen-activated protein kinase kinase kinase 20 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Mitogen-activated protein kinase kinase kinase 3 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Mitogen-activated protein kinase kinase kinase 4 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Mitogen-activated protein kinase kinase kinase 5 | Homo sapiens (human) | Kd | 30.0000 | 1 | 2 |
| Mitogen-activated protein kinase kinase kinase 6 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Mitogen-activated protein kinase kinase kinase kinase 1 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Mitogen-activated protein kinase kinase kinase kinase 2 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Mitogen-activated protein kinase kinase kinase kinase 3 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Mitogen-activated protein kinase kinase kinase kinase 4 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Mitogen-activated protein kinase kinase kinase kinase 5 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Mitotic checkpoint serine/threonine-protein kinase BUB1 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Mu-type opioid receptor | Cavia porcellus (domestic guinea pig) | EC50 | 0.0460 | 1 | 2 |
| Mu-type opioid receptor | Homo sapiens (human) | EC50 | 4.8400 | 1 | 1 |
| Multifunctional protein ADE2 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Muscarinic acetylcholine receptor | Cavia porcellus (domestic guinea pig) | Kd | 0.0794 | 1 | 1 |
| Muscarinic acetylcholine receptor M2 | Homo sapiens (human) | Kd | 0.0398 | 1 | 1 |
| Myosin light chain kinase 3 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Myosin light chain kinase, smooth muscle | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Myosin-10 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Myosin-14 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| NADH dehydrogenase [ubiquinone] 1 alpha subcomplex subunit 13 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Non-receptor tyrosine-protein kinase TNK1 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Non-receptor tyrosine-protein kinase TYK2 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| NUAK family SNF1-like kinase 2 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Nuclear receptor subfamily 1 group I member 2 | Homo sapiens (human) | EC50 | 14.9557 | 4 | 7 |
| Nuclear receptor subfamily 1 group I member 2 | Rattus norvegicus (Norway rat) | EC50 | 23.4000 | 1 | 1 |
| Nucleolar GTP-binding protein 1 | Homo sapiens (human) | Kd | 30.0000 | 1 | 2 |
| Obg-like ATPase 1 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| PAS domain-containing serine/threonine-protein kinase | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Peroxisomal acyl-coenzyme A oxidase 1 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Peroxisomal acyl-coenzyme A oxidase 3 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Phenylalanine--tRNA ligase beta subunit | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Phosphatidylethanolamine-binding protein 1 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Phosphatidylinositol 5-phosphate 4-kinase type-2 alpha | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Phosphatidylinositol 5-phosphate 4-kinase type-2 gamma | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Phosphorylase b kinase gamma catalytic chain, liver/testis isoform | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Platelet-derived growth factor receptor beta | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Potassium channel subfamily K member 2 | Homo sapiens (human) | EC50 | 4.3050 | 1 | 2 |
| Probable ATP-dependent RNA helicase DDX6 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Protein kinase C alpha type | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Protein kinase C beta type | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Protein kinase C delta type | Homo sapiens (human) | Kd | 4.7890 | 1 | 1 |
| Protein kinase C iota type | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Protein kinase C theta type | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Protein kinase C zeta type | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Protein-tyrosine kinase 2-beta | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Protein-tyrosine kinase 6 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Proto-oncogene tyrosine-protein kinase receptor Ret | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Proto-oncogene tyrosine-protein kinase Src | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Putative heat shock protein HSP 90-beta 2 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Pyridoxal kinase | Homo sapiens (human) | Kd | 30.0000 | 1 | 2 |
| RAC-alpha serine/threonine-protein kinase | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| RAC-beta serine/threonine-protein kinase | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| RAC-gamma serine/threonine-protein kinase | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Ras-related C3 botulinum toxin substrate 1 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Ras-related protein Rab-10 | Homo sapiens (human) | Kd | 30.0000 | 1 | 2 |
| Ras-related protein Rab-27A | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Ras-related protein Rab-6A | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Receptor-interacting serine/threonine-protein kinase 2 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Receptor-interacting serine/threonine-protein kinase 3 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Receptor-type tyrosine-protein kinase FLT3 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Rho-associated protein kinase 1 | Homo sapiens (human) | Kd | 0.9060 | 1 | 1 |
| Rho-associated protein kinase 2 | Homo sapiens (human) | Kd | 0.5105 | 2 | 2 |
| Ribosomal protein S6 kinase alpha-1 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Ribosomal protein S6 kinase alpha-3 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Ribosomal protein S6 kinase alpha-4 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Ribosomal protein S6 kinase alpha-5 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Ribosomal protein S6 kinase alpha-6 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Ribosomal protein S6 kinase beta-1 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Ribosyldihydronicotinamide dehydrogenase [quinone] | Homo sapiens (human) | Kd | 2.4510 | 1 | 1 |
| RNA cytidine acetyltransferase | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| S-adenosylmethionine synthase isoform type-2 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Sarcoplasmic/endoplasmic reticulum calcium ATPase 1 | Oryctolagus cuniculus (rabbit) | Kd | 0.0002 | 1 | 1 |
| Septin-9 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Serine/threonine-protein kinase 10 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Serine/threonine-protein kinase 16 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Serine/threonine-protein kinase 26 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Serine/threonine-protein kinase 3 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| serine/threonine-protein kinase 33 isoform a | Homo sapiens (human) | EC50 | 9.5830 | 1 | 1 |
| Serine/threonine-protein kinase 4 | Homo sapiens (human) | Kd | 30.0000 | 1 | 2 |
| Serine/threonine-protein kinase A-Raf | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Serine/threonine-protein kinase B-raf | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Serine/threonine-protein kinase Chk1 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Serine/threonine-protein kinase D2 | Homo sapiens (human) | Kd | 6.4160 | 1 | 1 |
| Serine/threonine-protein kinase D3 | Homo sapiens (human) | Kd | 23.3410 | 1 | 1 |
| Serine/threonine-protein kinase LATS1 | Homo sapiens (human) | Kd | 4.1700 | 1 | 1 |
| Serine/threonine-protein kinase MARK2 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Serine/threonine-protein kinase MRCK alpha | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Serine/threonine-protein kinase MRCK beta | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Serine/threonine-protein kinase MRCK gamma | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Serine/threonine-protein kinase N1 | Homo sapiens (human) | Kd | 0.8410 | 1 | 1 |
| Serine/threonine-protein kinase N2 | Homo sapiens (human) | Kd | 2.5990 | 1 | 1 |
| Serine/threonine-protein kinase N3 | Homo sapiens (human) | Kd | 0.0990 | 1 | 1 |
| Serine/threonine-protein kinase Nek1 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Serine/threonine-protein kinase Nek2 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Serine/threonine-protein kinase Nek3 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Serine/threonine-protein kinase Nek7 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Serine/threonine-protein kinase Nek9 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Serine/threonine-protein kinase NLK | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Serine/threonine-protein kinase PAK 2 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Serine/threonine-protein kinase PAK 4 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Serine/threonine-protein kinase pim-1 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Serine/threonine-protein kinase PLK1 | Homo sapiens (human) | Kd | 30.0000 | 1 | 2 |
| Serine/threonine-protein kinase PLK4 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Serine/threonine-protein kinase SIK2 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Serine/threonine-protein kinase SIK3 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Serine/threonine-protein kinase STK11 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Serine/threonine-protein kinase TAO1 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Serine/threonine-protein kinase TAO2 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Serine/threonine-protein kinase TAO3 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Serine/threonine-protein kinase TBK1 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Serine/threonine-protein kinase ULK1 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Serine/threonine-protein kinase ULK3 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Serine/threonine-protein kinase/endoribonuclease IRE1 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Serine/threonine-protein kinase/endoribonuclease IRE2 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Signal recognition particle receptor subunit alpha | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| STE20-like serine/threonine-protein kinase | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| STE20-related kinase adapter protein alpha | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Structural maintenance of chromosomes protein 1A | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Structural maintenance of chromosomes protein 2 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Succinate--CoA ligase [ADP-forming] subunit beta, mitochondrial | Homo sapiens (human) | Kd | 30.0000 | 1 | 2 |
| TGF-beta receptor type-1 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| TGF-beta receptor type-2 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Thyroid hormone receptor-associated protein 3 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| TRAF2 and NCK-interacting protein kinase | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Transient receptor potential cation channel subfamily A member 1 | Mus musculus (house mouse) | EC50 | 1.6667 | 1 | 3 |
| Transient receptor potential cation channel subfamily V member 1 | Homo sapiens (human) | EC50 | 129.0000 | 1 | 1 |
| Tyrosine--tRNA ligase, cytoplasmic | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Tyrosine-protein kinase ABL1 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Tyrosine-protein kinase ABL2 | Homo sapiens (human) | Kd | 30.0000 | 1 | 2 |
| Tyrosine-protein kinase BTK | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Tyrosine-protein kinase CSK | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Tyrosine-protein kinase Fer | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Tyrosine-protein kinase Fes/Fps | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Tyrosine-protein kinase Fgr | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Tyrosine-protein kinase FRK | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Tyrosine-protein kinase Fyn | Homo sapiens (human) | Kd | 30.0000 | 1 | 2 |
| Tyrosine-protein kinase HCK | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Tyrosine-protein kinase JAK1 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Tyrosine-protein kinase Lck | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Tyrosine-protein kinase Lyn | Homo sapiens (human) | Kd | 30.0000 | 1 | 2 |
| Tyrosine-protein kinase SYK | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Tyrosine-protein kinase Tec | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Tyrosine-protein kinase Yes | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| U5 small nuclear ribonucleoprotein 200 kDa helicase | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| UMP-CMP kinase | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Uncharacterized aarF domain-containing protein kinase 5 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Uncharacterized protein FLJ45252 | Homo sapiens (human) | Kd | 30.0000 | 1 | 2 |
| Very long-chain specific acyl-CoA dehydrogenase, mitochondrial | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Wee1-like protein kinase | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |