Proteins > high affinity choline transporter 1 isoform a
Page last updated: 2024-08-07 22:57:48

high affinity choline transporter 1 isoform a

[no definition available]

Synonyms

Research

Bioassay Publications (0)

TimeframeStudies on this Protein(%)All Drugs %
pre-19900 (0)18.7374
1990's0 (0)18.2507
2000's0 (0)29.6817
2010's0 (0)24.3611
2020's0 (0)2.80

Compounds (66)

Drugs with Inhibition Measurements

DrugTaxonomyMeasurementAverage (mM)Bioassay(s)Publication(s)
9-xylosyladenineHomo sapiens (human)IC500.551120
acetylcholine chlorideHomo sapiens (human)IC503.415220
2-chloroadenosineHomo sapiens (human)IC500.537720
2-(alpha-thenoylamino)-2-nitro-5-thiazoleHomo sapiens (human)IC501.669620
alosetron hydrochlorideHomo sapiens (human)IC501.762520
adenosineHomo sapiens (human)IC500.385120
dobutamine hydrochlorideHomo sapiens (human)IC500.164520
ondansetron hydrochlorideHomo sapiens (human)IC501.513820
magnololHomo sapiens (human)IC502.295220
honokiolHomo sapiens (human)IC5012.022610
lobaric acidHomo sapiens (human)IC5010.964810
phenylisopropyladenosineHomo sapiens (human)IC501.861320
n(6)-(3-iodobenzyl)-5'-n-methylcarboxamidoadenosineHomo sapiens (human)IC502.100220
2-(1-adamantyl)imidazoleHomo sapiens (human)IC505.501220
(R)-norlaudanosolineHomo sapiens (human)IC500.470310
diethylstilbestrolHomo sapiens (human)IC5012.589310
6-methyl-2-oxo-5-[oxo-(1-phenylethylamino)methyl]-1H-pyridine-3-carboxylic acid ethyl esterHomo sapiens (human)IC501.110520
N,N-bis(but-2-ynyl)-3-methoxy-4-(1-tetrazolyl)benzenesulfonamideHomo sapiens (human)IC503.162310
methamilane methiodideHomo sapiens (human)IC500.899520
N-[5-(ethylthio)-1,3,4-thiadiazol-2-yl]-3,3,3-trifluoro-2-methyl-2-(trifluoromethyl)propanamideHomo sapiens (human)IC503.142920
3-[(3aR,6aS)-6'-chloro-5-(4-chlorophenyl)-7'-methyl-2',4,6-trioxo-1-spiro[1,2,3a,6a-tetrahydropyrrolo[3,4-c]pyrrole-3,3'-1H-indole]yl]propanamideHomo sapiens (human)IC504.276020
7-butyl-8-[[4-(3-chlorophenyl)-1-piperazinyl]methyl]-1,3-dimethylpurine-2,6-dioneHomo sapiens (human)IC5015.135610
3-(4-methylbenzoyl)acrylic acidHomo sapiens (human)IC5010.471310
ondansetron, (s)-isomerHomo sapiens (human)IC500.571720
N-(3-phenyl-1,3-benzothiazol-2-ylidene)-2-propenamideHomo sapiens (human)IC503.071720
N-[(2,3-dimethoxyphenyl)methyl]-4-(4-methyl-1-piperidinyl)anilineHomo sapiens (human)IC5013.182610
6-(2-phenylethyl)-3-(phenylmethyl)-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazoleHomo sapiens (human)IC5027.542310
4-(3,4-dihydro-1H-isoquinolin-2-ylmethyl)-N-(2,6-dimethylphenyl)benzamideHomo sapiens (human)IC5018.197010
2,4-dichloro-5-(diethylsulfamoyl)-N-(1,3,4-thiadiazol-2-yl)benzamideHomo sapiens (human)IC506.920520
5-[3-[(2,4-dichlorophenyl)methoxy]-2-thiophenyl]-1,2-dihydro-1,2,4-triazole-3-thioneHomo sapiens (human)IC5011.481510
epalrestatHomo sapiens (human)IC507.963520
5-bromo-N-[[[oxo(thiophen-2-yl)methyl]hydrazo]-sulfanylidenemethyl]-2-furancarboxamideHomo sapiens (human)IC5028.840310
N-[[[(2-methylphenyl)-oxomethyl]hydrazo]-sulfanylidenemethyl]benzamideHomo sapiens (human)IC5012.589310
N-[(tert-butylamino)-oxomethyl]-2-[4-(3-chlorophenyl)-1-piperazinyl]acetamideHomo sapiens (human)IC505.899720
2-[(5-chloro-2-thiophenyl)sulfonylamino]-N-(2-furanylmethyl)benzamideHomo sapiens (human)IC506.037420
2-[(5-chloro-2-thiophenyl)sulfonylamino]-N-(2-methoxy-5-methylphenyl)benzamideHomo sapiens (human)IC503.784220
3-hydroxybenzoic acid [2-(1H-indol-3-yl)-2-oxoethyl] esterHomo sapiens (human)IC5015.848910
4,5-dichloro-2-[2-[2,5-dimethyl-1-(2,2,2-trifluoroethyl)-3-pyrrolyl]-2-oxoethyl]-3-pyridazinoneHomo sapiens (human)IC5020.893010
Betaine Aldehyde ChlorideHomo sapiens (human)IC5015.135610
2-[(3-methoxyphenyl)-oxomethyl]-3,3-bis(methylthio)-2-propenenitrileHomo sapiens (human)IC5011.247010
2,2'-[3-(2-methoxyphenyl)-1,2-propanediyl]bis(1H-benzimidazole)Homo sapiens (human)IC5013.803810
1-[1-(4-methoxyphenyl)-2,5-dimethyl-3-pyrrolyl]-2-[[4-methyl-5-(2-methyl-3-furanyl)-1,2,4-triazol-3-yl]thio]ethanoneHomo sapiens (human)IC5013.803810
3-(4-fluorophenyl)-N-[3-(1-imidazolyl)propyl]-1-phenyl-4-pyrazolecarboxamideHomo sapiens (human)IC5011.481510
2-[[5-(dimethylsulfamoyl)-1H-indol-3-yl]methylidene]propanedioic acid diethyl esterHomo sapiens (human)IC5015.848910
5-methyl-2-[[(4-nitrophenyl)-oxomethyl]hydrazo]-4-thiazolecarboxylic acid ethyl esterHomo sapiens (human)IC509.914710
N-[3-[3-(1-piperidinylsulfonyl)anilino]-2-quinoxalinyl]benzenesulfonamideHomo sapiens (human)IC5012.022610
2,5-dichloro-N-[5-(4-fluorophenyl)-1,3,4-oxadiazol-2-yl]-3-thiophenecarboxamideHomo sapiens (human)IC5014.454410
dinoprost tromethamineHomo sapiens (human)IC502.858120
bicyclo-PGE2Homo sapiens (human)IC502.253820
4-[[[1-[[2-(3-chlorophenyl)-5-methyl-4-oxazolyl]methyl]-3-piperidinyl]-oxomethyl]amino]-1-piperidinecarboxylic acid ethyl esterHomo sapiens (human)IC506.918310
erbstatinHomo sapiens (human)IC502.462120
serratinHomo sapiens (human)IC5013.665210
7-hydroxy-2-methyl-6-propyl-3-(2-pyridinyl)-1-benzopyran-4-oneHomo sapiens (human)IC5012.305910
fenoterolHomo sapiens (human)IC500.000720
nab-365Homo sapiens (human)IC500.014820
N-[2-(2-fluorophenyl)ethyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[5,1-b]quinazolin-9-amineHomo sapiens (human)IC5013.803810
8-(n,n-diethylamino)octyl-3,4,5-trimethoxybenzoate hydrochlorideHomo sapiens (human)IC5015.135610
cgs 21680aHomo sapiens (human)IC500.860920
4-iodoclonidineHomo sapiens (human)IC500.979020
2-[4-[1-[(2-fluorophenyl)methyl]-2,4-dioxo-3-quinazolinyl]phenyl]-N-(2-oxolanylmethyl)acetamideHomo sapiens (human)IC505.558820
(3E,9E)-5,6-Dihydroxy-9,13,14-trimethyl-16-(2-methylpropyl)-17-azatricyclo[9.7.0.01,15]octadeca-3,9,12-triene-2,18-dioneHomo sapiens (human)IC503.773020
5-chloro-2-[(4-methylphenyl)methylsulfonyl]-N-(5-propan-2-yl-1,3,4-thiadiazol-2-yl)-4-pyrimidinecarboxamideHomo sapiens (human)IC504.448020
2-(2,4-dimethoxyphenyl)-5-methyl-4-[[4-(4-quinazolinyl)-1-piperazinyl]methyl]oxazoleHomo sapiens (human)IC5016.754510
1-[[3-(4-fluorophenyl)-1-(4-methylphenyl)-4-pyrazolyl]methyl]-4-[(1-methyl-2-imidazolyl)methyl]piperazineHomo sapiens (human)IC5010.087510
2-[(6-chloro-3-pyridinyl)sulfonylamino]-N-[(4-methylphenyl)methyl]benzamideHomo sapiens (human)IC505.768820

Drugs with Activation Measurements

DrugTaxonomyMeasurementAverage (mM)Bioassay(s)Publication(s)
2-[2-(2-chlorophenyl)-1-benzimidazolyl]-N-(2-propan-2-ylphenyl)acetamideHomo sapiens (human)EC5018.320010