Assay ID | Title | Year | Journal | Article |
AID504749 | qHTS profiling for inhibitors of Plasmodium falciparum proliferation | 2011 | Science (New York, N.Y.), Aug-05, Volume: 333, Issue:6043
| Chemical genomic profiling for antimalarial therapies, response signatures, and molecular targets. |
AID1347092 | qHTS of pediatric cancer cell lines to identify multiple opportunities for drug repurposing: Primary screen for A673 cells | 2018 | Oncotarget, Jan-12, Volume: 9, Issue:4
| Quantitative high-throughput phenotypic screening of pediatric cancer cell lines identifies multiple opportunities for drug repurposing. |
AID1347094 | qHTS of pediatric cancer cell lines to identify multiple opportunities for drug repurposing: Primary screen for BT-37 cells | 2018 | Oncotarget, Jan-12, Volume: 9, Issue:4
| Quantitative high-throughput phenotypic screening of pediatric cancer cell lines identifies multiple opportunities for drug repurposing. |
AID1296008 | Cytotoxic Profiling of Annotated Libraries Using Quantitative High-Throughput Screening | 2020 | SLAS discovery : advancing life sciences R & D, 01, Volume: 25, Issue:1
| Cytotoxic Profiling of Annotated and Diverse Chemical Libraries Using Quantitative High-Throughput Screening. |
AID1347407 | qHTS to identify inhibitors of the type 1 interferon - major histocompatibility complex class I in skeletal muscle: primary screen against the NCATS Pharmaceutical Collection | 2020 | ACS chemical biology, 07-17, Volume: 15, Issue:7
| High-Throughput Screening to Identify Inhibitors of the Type I Interferon-Major Histocompatibility Complex Class I Pathway in Skeletal Muscle. |
AID1347425 | Rhodamine-PBP qHTS Assay for Modulators of WT P53-Induced Phosphatase 1 (WIP1) | 2019 | The Journal of biological chemistry, 11-15, Volume: 294, Issue:46
| Physiologically relevant orthogonal assays for the discovery of small-molecule modulators of WIP1 phosphatase in high-throughput screens. |
AID1347424 | RapidFire Mass Spectrometry qHTS Assay for Modulators of WT P53-Induced Phosphatase 1 (WIP1) | 2019 | The Journal of biological chemistry, 11-15, Volume: 294, Issue:46
| Physiologically relevant orthogonal assays for the discovery of small-molecule modulators of WIP1 phosphatase in high-throughput screens. |
AID1745845 | Primary qHTS for Inhibitors of ATXN expression | | | |
AID1347086 | qHTS for Inhibitors of the Functional Ribonucleoprotein Complex (vRNP) of Lymphocytic Choriomeningitis Arenaviruses (LCMV): LCMV Primary Screen - GLuc reporter signal | 2020 | Antiviral research, 01, Volume: 173 | A cell-based, infectious-free, platform to identify inhibitors of lassa virus ribonucleoprotein (vRNP) activity. |
AID1347082 | qHTS for Inhibitors of the Functional Ribonucleoprotein Complex (vRNP) of Lassa (LASV) Arenavirus: LASV Primary Screen - GLuc reporter signal | 2020 | Antiviral research, 01, Volume: 173 | A cell-based, infectious-free, platform to identify inhibitors of lassa virus ribonucleoprotein (vRNP) activity. |
AID1347091 | qHTS of pediatric cancer cell lines to identify multiple opportunities for drug repurposing: Primary screen for SJ-GBM2 cells | 2018 | Oncotarget, Jan-12, Volume: 9, Issue:4
| Quantitative high-throughput phenotypic screening of pediatric cancer cell lines identifies multiple opportunities for drug repurposing. |
AID1347101 | qHTS of pediatric cancer cell lines to identify multiple opportunities for drug repurposing: Primary screen for BT-12 cells | 2018 | Oncotarget, Jan-12, Volume: 9, Issue:4
| Quantitative high-throughput phenotypic screening of pediatric cancer cell lines identifies multiple opportunities for drug repurposing. |
AID1347089 | qHTS of pediatric cancer cell lines to identify multiple opportunities for drug repurposing: Primary screen for TC32 cells | 2018 | Oncotarget, Jan-12, Volume: 9, Issue:4
| Quantitative high-throughput phenotypic screening of pediatric cancer cell lines identifies multiple opportunities for drug repurposing. |
AID1347103 | qHTS of pediatric cancer cell lines to identify multiple opportunities for drug repurposing: Primary screen for OHS-50 cells | 2018 | Oncotarget, Jan-12, Volume: 9, Issue:4
| Quantitative high-throughput phenotypic screening of pediatric cancer cell lines identifies multiple opportunities for drug repurposing. |
AID1347096 | qHTS of pediatric cancer cell lines to identify multiple opportunities for drug repurposing: Primary screen for U-2 OS cells | 2018 | Oncotarget, Jan-12, Volume: 9, Issue:4
| Quantitative high-throughput phenotypic screening of pediatric cancer cell lines identifies multiple opportunities for drug repurposing. |
AID1347100 | qHTS of pediatric cancer cell lines to identify multiple opportunities for drug repurposing: Primary screen for LAN-5 cells | 2018 | Oncotarget, Jan-12, Volume: 9, Issue:4
| Quantitative high-throughput phenotypic screening of pediatric cancer cell lines identifies multiple opportunities for drug repurposing. |
AID1347090 | qHTS of pediatric cancer cell lines to identify multiple opportunities for drug repurposing: Primary screen for DAOY cells | 2018 | Oncotarget, Jan-12, Volume: 9, Issue:4
| Quantitative high-throughput phenotypic screening of pediatric cancer cell lines identifies multiple opportunities for drug repurposing. |
AID1347083 | qHTS for Inhibitors of the Functional Ribonucleoprotein Complex (vRNP) of Lassa (LASV) Arenavirus: Viability assay - alamar blue signal for LASV Primary Screen | 2020 | Antiviral research, 01, Volume: 173 | A cell-based, infectious-free, platform to identify inhibitors of lassa virus ribonucleoprotein (vRNP) activity. |
AID1347104 | qHTS of pediatric cancer cell lines to identify multiple opportunities for drug repurposing: Primary screen for RD cells | 2018 | Oncotarget, Jan-12, Volume: 9, Issue:4
| Quantitative high-throughput phenotypic screening of pediatric cancer cell lines identifies multiple opportunities for drug repurposing. |
AID1347098 | qHTS of pediatric cancer cell lines to identify multiple opportunities for drug repurposing: Primary screen for SK-N-SH cells | 2018 | Oncotarget, Jan-12, Volume: 9, Issue:4
| Quantitative high-throughput phenotypic screening of pediatric cancer cell lines identifies multiple opportunities for drug repurposing. |
AID1347099 | qHTS of pediatric cancer cell lines to identify multiple opportunities for drug repurposing: Primary screen for NB1643 cells | 2018 | Oncotarget, Jan-12, Volume: 9, Issue:4
| Quantitative high-throughput phenotypic screening of pediatric cancer cell lines identifies multiple opportunities for drug repurposing. |
AID1508630 | Primary qHTS for small molecule stabilizers of the endoplasmic reticulum resident proteome: Secreted ER Calcium Modulated Protein (SERCaMP) assay | 2021 | Cell reports, 04-27, Volume: 35, Issue:4
| A target-agnostic screen identifies approved drugs to stabilize the endoplasmic reticulum-resident proteome. |
AID1347108 | qHTS of pediatric cancer cell lines to identify multiple opportunities for drug repurposing: Primary screen for Rh41 cells | 2018 | Oncotarget, Jan-12, Volume: 9, Issue:4
| Quantitative high-throughput phenotypic screening of pediatric cancer cell lines identifies multiple opportunities for drug repurposing. |
AID1347095 | qHTS of pediatric cancer cell lines to identify multiple opportunities for drug repurposing: Primary screen for NB-EBc1 cells | 2018 | Oncotarget, Jan-12, Volume: 9, Issue:4
| Quantitative high-throughput phenotypic screening of pediatric cancer cell lines identifies multiple opportunities for drug repurposing. |
AID1347154 | Primary screen GU AMC qHTS for Zika virus inhibitors | 2020 | Proceedings of the National Academy of Sciences of the United States of America, 12-08, Volume: 117, Issue:49
| Therapeutic candidates for the Zika virus identified by a high-throughput screen for Zika protease inhibitors. |
AID651635 | Viability Counterscreen for Primary qHTS for Inhibitors of ATXN expression | | | |
AID1347107 | qHTS of pediatric cancer cell lines to identify multiple opportunities for drug repurposing: Primary screen for Rh30 cells | 2018 | Oncotarget, Jan-12, Volume: 9, Issue:4
| Quantitative high-throughput phenotypic screening of pediatric cancer cell lines identifies multiple opportunities for drug repurposing. |
AID1347102 | qHTS of pediatric cancer cell lines to identify multiple opportunities for drug repurposing: Primary screen for Rh18 cells | 2018 | Oncotarget, Jan-12, Volume: 9, Issue:4
| Quantitative high-throughput phenotypic screening of pediatric cancer cell lines identifies multiple opportunities for drug repurposing. |
AID1347093 | qHTS of pediatric cancer cell lines to identify multiple opportunities for drug repurposing: Primary screen for SK-N-MC cells | 2018 | Oncotarget, Jan-12, Volume: 9, Issue:4
| Quantitative high-throughput phenotypic screening of pediatric cancer cell lines identifies multiple opportunities for drug repurposing. |
AID1347105 | qHTS of pediatric cancer cell lines to identify multiple opportunities for drug repurposing: Primary screen for MG 63 (6-TG R) cells | 2018 | Oncotarget, Jan-12, Volume: 9, Issue:4
| Quantitative high-throughput phenotypic screening of pediatric cancer cell lines identifies multiple opportunities for drug repurposing. |
AID1347097 | qHTS of pediatric cancer cell lines to identify multiple opportunities for drug repurposing: Primary screen for Saos-2 cells | 2018 | Oncotarget, Jan-12, Volume: 9, Issue:4
| Quantitative high-throughput phenotypic screening of pediatric cancer cell lines identifies multiple opportunities for drug repurposing. |
AID1347106 | qHTS of pediatric cancer cell lines to identify multiple opportunities for drug repurposing: Primary screen for control Hh wild type fibroblast cells | 2018 | Oncotarget, Jan-12, Volume: 9, Issue:4
| Quantitative high-throughput phenotypic screening of pediatric cancer cell lines identifies multiple opportunities for drug repurposing. |
AID1346987 | P-glycoprotein substrates identified in KB-8-5-11 adenocarcinoma cell line, qHTS therapeutic library screen | 2019 | Molecular pharmacology, 11, Volume: 96, Issue:5
| A High-Throughput Screen of a Library of Therapeutics Identifies Cytotoxic Substrates of P-glycoprotein. |
AID1346986 | P-glycoprotein substrates identified in KB-3-1 adenocarcinoma cell line, qHTS therapeutic library screen | 2019 | Molecular pharmacology, 11, Volume: 96, Issue:5
| A High-Throughput Screen of a Library of Therapeutics Identifies Cytotoxic Substrates of P-glycoprotein. |
AID1286505 | Cytotoxicity against human HepG2 cells after 24 hrs by WST-1 based colorimetric assay | 2016 | Journal of medicinal chemistry, Mar-10, Volume: 59, Issue:5
| Robenidine Analogues as Gram-Positive Antibacterial Agents. |
AID1286456 | Bactericidal activity against Methicillin-sensitive Staphylococcus aureus clinical isolate USA300 assessed as log reduction in bacterial cell number at 4 times MIC after 8 hrs by time-kill curve analysis | 2016 | Journal of medicinal chemistry, Mar-10, Volume: 59, Issue:5
| Robenidine Analogues as Gram-Positive Antibacterial Agents. |
AID1286500 | Bactericidal activity against methicillin-sensitive Staphylococcus aureus ATCC 29213 after 24 and 48 hrs | 2016 | Journal of medicinal chemistry, Mar-10, Volume: 59, Issue:5
| Robenidine Analogues as Gram-Positive Antibacterial Agents. |
AID51255 | The compound was tested for anti-coccidial activity in chicken against E. maxima(DP-776) measured at dose 33(ppm in diet) | 1991 | Journal of medicinal chemistry, Sep, Volume: 34, Issue:9
| Benzylated 1,2,3-triazoles as anticoccidiostats. |
AID1286501 | Ratio of MBC for methicillin-sensitive Staphylococcus aureus ATCC 25923 to MIC90 for methicillin-sensitive Staphylococcus aureus ATCC 25923 | 2016 | Journal of medicinal chemistry, Mar-10, Volume: 59, Issue:5
| Robenidine Analogues as Gram-Positive Antibacterial Agents. |
AID1286487 | Selectivity index, ratio of GI50 for human HepG2 cells to MIC50 for methicillin-sensitive Staphylococcus aureus clinical isolate | 2016 | Journal of medicinal chemistry, Mar-10, Volume: 59, Issue:5
| Robenidine Analogues as Gram-Positive Antibacterial Agents. |
AID1286465 | Bactericidal activity against Methicillin-sensitive Staphylococcus aureus clinical isolate USA300 assessed as log reduction in bacterial cell number at 8 times MIC after 24 hrs by time-kill curve analysis | 2016 | Journal of medicinal chemistry, Mar-10, Volume: 59, Issue:5
| Robenidine Analogues as Gram-Positive Antibacterial Agents. |
AID1286504 | Ratio of MBC for methicillin-sensitive Staphylococcus aureus ATCC 29213 to MIC90 for methicillin-sensitive Staphylococcus aureus ATCC 29213 | 2016 | Journal of medicinal chemistry, Mar-10, Volume: 59, Issue:5
| Robenidine Analogues as Gram-Positive Antibacterial Agents. |
AID1286479 | Metabolic stability in human liver microsomes assessed as compound loss after 60 mins | 2016 | Journal of medicinal chemistry, Mar-10, Volume: 59, Issue:5
| Robenidine Analogues as Gram-Positive Antibacterial Agents. |
AID1286525 | Bactericidal activity against Methicillin-sensitive Staphylococcus aureus clinical isolate USA300 assessed as log reduction in bacterial cell number at 2 times MIC after 8 hrs by time-kill curve analysis | 2016 | Journal of medicinal chemistry, Mar-10, Volume: 59, Issue:5
| Robenidine Analogues as Gram-Positive Antibacterial Agents. |
AID1286483 | Toxicity in po dosed male rabbit | 2016 | Journal of medicinal chemistry, Mar-10, Volume: 59, Issue:5
| Robenidine Analogues as Gram-Positive Antibacterial Agents. |
AID1286486 | Selectivity index, ratio of GI50 for human HEL299 cells to MIC50 for methicillin-resistant Staphylococcus aureus clinical isolate | 2016 | Journal of medicinal chemistry, Mar-10, Volume: 59, Issue:5
| Robenidine Analogues as Gram-Positive Antibacterial Agents. |
AID1286496 | Antibacterial activity against methicillin-sensitive Staphylococcus aureus ATCC 29213 after 20 to 24 hrs in presence of 50% heat inactivated bovine serum | 2016 | Journal of medicinal chemistry, Mar-10, Volume: 59, Issue:5
| Robenidine Analogues as Gram-Positive Antibacterial Agents. |
AID1286467 | Inhibition of biofilm formation in methicillin-resistant Staphylococcus aureus assessed as log reduction at > 43.2 uM after 24 hrs by MBEC assay relative to control | 2016 | Journal of medicinal chemistry, Mar-10, Volume: 59, Issue:5
| Robenidine Analogues as Gram-Positive Antibacterial Agents. |
AID1286488 | Selectivity index, ratio of GI50 for human HepG2 cells to MIC50 for methicillin-resistant Staphylococcus aureus clinical isolate | 2016 | Journal of medicinal chemistry, Mar-10, Volume: 59, Issue:5
| Robenidine Analogues as Gram-Positive Antibacterial Agents. |
AID1286515 | Ratio of MBC for methicillin-resistant Staphylococcus aureus clinical isolate to MIC90 for methicillin-resistant Staphylococcus aureus clinical isolate | 2016 | Journal of medicinal chemistry, Mar-10, Volume: 59, Issue:5
| Robenidine Analogues as Gram-Positive Antibacterial Agents. |
AID1286521 | Bactericidal activity against methicillin-sensitive Staphylococcus aureus ATCC 29213 assessed as log reduction in bacterial cell number at 2 times MIC after 8 hrs by time-kill curve analysis | 2016 | Journal of medicinal chemistry, Mar-10, Volume: 59, Issue:5
| Robenidine Analogues as Gram-Positive Antibacterial Agents. |
AID1286499 | Bactericidal activity against methicillin-sensitive Staphylococcus aureus ATCC 49775 after 24 and 48 hrs | 2016 | Journal of medicinal chemistry, Mar-10, Volume: 59, Issue:5
| Robenidine Analogues as Gram-Positive Antibacterial Agents. |
AID1286477 | Intrinsic clearance in human liver microsomes assessed per mg of protein | 2016 | Journal of medicinal chemistry, Mar-10, Volume: 59, Issue:5
| Robenidine Analogues as Gram-Positive Antibacterial Agents. |
AID1286461 | Bactericidal activity against Methicillin-sensitive Staphylococcus aureus ATCC 29213 assessed as log reduction in bacterial cell number at 8 times MIC after 24 hrs by time-kill curve analysis | 2016 | Journal of medicinal chemistry, Mar-10, Volume: 59, Issue:5
| Robenidine Analogues as Gram-Positive Antibacterial Agents. |
AID1286508 | Antibacterial activity against vancomycin-resistant Enterococcus after 20 to 24 hrs | 2016 | Journal of medicinal chemistry, Mar-10, Volume: 59, Issue:5
| Robenidine Analogues as Gram-Positive Antibacterial Agents. |
AID1286523 | Bactericidal activity against methicillin-sensitive Staphylococcus aureus ATCC 29213 assessed as log reduction in bacterial cell number at 8 times MIC after 8 hrs by time-kill curve analysis | 2016 | Journal of medicinal chemistry, Mar-10, Volume: 59, Issue:5
| Robenidine Analogues as Gram-Positive Antibacterial Agents. |
AID1286516 | Antibacterial activity against Escherichia coli ATCC 25922 after 20 to 24 hrs in presence of polymyxin B nonapeptide | 2016 | Journal of medicinal chemistry, Mar-10, Volume: 59, Issue:5
| Robenidine Analogues as Gram-Positive Antibacterial Agents. |
AID51241 | The compound was tested for anti-coccidial activity in chicken against E. brunetti (FS-103) measured at dose 33(ppm in diet) | 1991 | Journal of medicinal chemistry, Sep, Volume: 34, Issue:9
| Benzylated 1,2,3-triazoles as anticoccidiostats. |
AID1286476 | Half life of compound in mouse liver microsomes | 2016 | Journal of medicinal chemistry, Mar-10, Volume: 59, Issue:5
| Robenidine Analogues as Gram-Positive Antibacterial Agents. |
AID1286495 | Antibacterial activity against methicillin-sensitive Staphylococcus aureus ATCC 49775 after 20 to 24 hrs in presence of 50% heat inactivated bovine serum | 2016 | Journal of medicinal chemistry, Mar-10, Volume: 59, Issue:5
| Robenidine Analogues as Gram-Positive Antibacterial Agents. |
AID1286462 | Bactericidal activity against Methicillin-sensitive Staphylococcus aureus clinical isolate USA300 assessed as log reduction in bacterial cell number at MIC after 24 hrs by time-kill curve analysis | 2016 | Journal of medicinal chemistry, Mar-10, Volume: 59, Issue:5
| Robenidine Analogues as Gram-Positive Antibacterial Agents. |
AID1286513 | Antibacterial activity against methicillin-resistant Staphylococcus aureus clinical isolate after 20 to 24 hrs in presence of 50% heat inactivated bovine serum | 2016 | Journal of medicinal chemistry, Mar-10, Volume: 59, Issue:5
| Robenidine Analogues as Gram-Positive Antibacterial Agents. |
AID1286519 | Ratio of MIC90 for Pseudomonas aeruginosa ATCC 27853 to MIC90 for Pseudomonas aeruginosa ATCC 27853 in presence of polymyxin B nonapeptide | 2016 | Journal of medicinal chemistry, Mar-10, Volume: 59, Issue:5
| Robenidine Analogues as Gram-Positive Antibacterial Agents. |
AID1286468 | Toxicity in sheep erythrocytes assessed as hemolysis after 30 mins | 2016 | Journal of medicinal chemistry, Mar-10, Volume: 59, Issue:5
| Robenidine Analogues as Gram-Positive Antibacterial Agents. |
AID1286497 | Bactericidal activity against methicillin-sensitive Staphylococcus aureus ATCC 25923 after 24 and 48 hrs | 2016 | Journal of medicinal chemistry, Mar-10, Volume: 59, Issue:5
| Robenidine Analogues as Gram-Positive Antibacterial Agents. |
AID1286471 | Lipophilicity, logD of the compound at pH 3 | 2016 | Journal of medicinal chemistry, Mar-10, Volume: 59, Issue:5
| Robenidine Analogues as Gram-Positive Antibacterial Agents. |
AID1286510 | Antibacterial activity against Pseudomonas aeruginosa ATCC 27853 after 20 to 24 hrs | 2016 | Journal of medicinal chemistry, Mar-10, Volume: 59, Issue:5
| Robenidine Analogues as Gram-Positive Antibacterial Agents. |
AID51261 | The compound was tested for anti-coccidial activity in chicken against E. mitis(LS-84) measured at dose 33(ppm in diet) | 1991 | Journal of medicinal chemistry, Sep, Volume: 34, Issue:9
| Benzylated 1,2,3-triazoles as anticoccidiostats. |
AID1286484 | Toxicity in po dosed female rabbit | 2016 | Journal of medicinal chemistry, Mar-10, Volume: 59, Issue:5
| Robenidine Analogues as Gram-Positive Antibacterial Agents. |
AID1286466 | Inhibition of biofilm formation in methicillin-resistant Staphylococcus aureus after 24 hrs by MBEC assay | 2016 | Journal of medicinal chemistry, Mar-10, Volume: 59, Issue:5
| Robenidine Analogues as Gram-Positive Antibacterial Agents. |
AID1286506 | Antiprotozoal activity against Babesia microti ATCC PRA-99 infected in BALB/c mouse assessed as suppression of parasitemia at 25 and 50 mg/kg, administered 4 times daily | 2016 | Journal of medicinal chemistry, Mar-10, Volume: 59, Issue:5
| Robenidine Analogues as Gram-Positive Antibacterial Agents. |
AID1286459 | Bactericidal activity against Methicillin-sensitive Staphylococcus aureus ATCC 29213 assessed as log reduction in bacterial cell number at 2 times MIC after 24 hrs by time kill curve analysis | 2016 | Journal of medicinal chemistry, Mar-10, Volume: 59, Issue:5
| Robenidine Analogues as Gram-Positive Antibacterial Agents. |
AID51092 | Anticoccidial activity in chicken against Eimeria acervulina. | 1991 | Journal of medicinal chemistry, Sep, Volume: 34, Issue:9
| Benzylated 1,2,3-triazoles as anticoccidiostats. |
AID1286457 | Bactericidal activity against Methicillin-sensitive Staphylococcus aureus clinical isolate USA300 assessed as log reduction in bacterial cell number at 8 times MIC after 8 hrs by time-kill curve analysis | 2016 | Journal of medicinal chemistry, Mar-10, Volume: 59, Issue:5
| Robenidine Analogues as Gram-Positive Antibacterial Agents. |
AID1286460 | Bactericidal activity against Methicillin-sensitive Staphylococcus aureus ATCC 29213 assessed as log reduction in bacterial cell number at 4 times MIC after 24 hrs by time kill curve analysis | 2016 | Journal of medicinal chemistry, Mar-10, Volume: 59, Issue:5
| Robenidine Analogues as Gram-Positive Antibacterial Agents. |
AID1286492 | Antibacterial activity against methicillin-sensitive Staphylococcus aureus ATCC 29213 after 20 to 24 hrs | 2016 | Journal of medicinal chemistry, Mar-10, Volume: 59, Issue:5
| Robenidine Analogues as Gram-Positive Antibacterial Agents. |
AID1286524 | Bactericidal activity against methicillin-sensitive Staphylococcus aureus clinical isolate USA300 assessed as log reduction in bacterial cell number at MIC after 8 hrs by time-kill curve analysis | 2016 | Journal of medicinal chemistry, Mar-10, Volume: 59, Issue:5
| Robenidine Analogues as Gram-Positive Antibacterial Agents. |
AID51411 | The compound was tested for anti-coccidial activity in chicken against E. praecox(DP-785) measured at dose 33(ppm in diet) | 1991 | Journal of medicinal chemistry, Sep, Volume: 34, Issue:9
| Benzylated 1,2,3-triazoles as anticoccidiostats. |
AID1286491 | Antibacterial activity against methicillin-sensitive Staphylococcus aureus ATCC 49775 after 20 to 24 hrs | 2016 | Journal of medicinal chemistry, Mar-10, Volume: 59, Issue:5
| Robenidine Analogues as Gram-Positive Antibacterial Agents. |
AID1286485 | Selectivity index, ratio of GI50 for human HEL299 cells to MIC50 for methicillin-sensitive Staphylococcus aureus clinical isolate | 2016 | Journal of medicinal chemistry, Mar-10, Volume: 59, Issue:5
| Robenidine Analogues as Gram-Positive Antibacterial Agents. |
AID51422 | The compound was tested for anti-coccidial activity in chicken against E. tenella(DP-761) measured at dose 33(ppm in diet) | 1991 | Journal of medicinal chemistry, Sep, Volume: 34, Issue:9
| Benzylated 1,2,3-triazoles as anticoccidiostats. |
AID1286512 | Antibacterial activity against Staphylococcus aureus ATCC 29213 after 20 to 24 hrs in presence of 2% heat inactivated bovine serum | 2016 | Journal of medicinal chemistry, Mar-10, Volume: 59, Issue:5
| Robenidine Analogues as Gram-Positive Antibacterial Agents. |
AID1286482 | Toxicity in po dosed rat | 2016 | Journal of medicinal chemistry, Mar-10, Volume: 59, Issue:5
| Robenidine Analogues as Gram-Positive Antibacterial Agents. |
AID1286503 | Ratio of MBC for methicillin-sensitive Staphylococcus aureus ATCC 49775 to MIC90 for methicillin-sensitive Staphylococcus aureus ATCC 49775 | 2016 | Journal of medicinal chemistry, Mar-10, Volume: 59, Issue:5
| Robenidine Analogues as Gram-Positive Antibacterial Agents. |
AID1286478 | Intrinsic clearance in mouse liver microsomes assessed per mg of protein | 2016 | Journal of medicinal chemistry, Mar-10, Volume: 59, Issue:5
| Robenidine Analogues as Gram-Positive Antibacterial Agents. |
AID1286493 | Antibacterial activity against methicillin-sensitive Staphylococcus aureus ATCC 25923 after 20 to 24 hrs in presence of 50% heat inactivated bovine serum | 2016 | Journal of medicinal chemistry, Mar-10, Volume: 59, Issue:5
| Robenidine Analogues as Gram-Positive Antibacterial Agents. |
AID1286502 | Ratio of MBC for methicillin-sensitive Staphylococcus aureus ATCC 6538 to MIC90 for methicillin-sensitive Staphylococcus aureus ATCC 6538 | 2016 | Journal of medicinal chemistry, Mar-10, Volume: 59, Issue:5
| Robenidine Analogues as Gram-Positive Antibacterial Agents. |
AID1286474 | Solubility of the compound at pH 6.5 | 2016 | Journal of medicinal chemistry, Mar-10, Volume: 59, Issue:5
| Robenidine Analogues as Gram-Positive Antibacterial Agents. |
AID1286464 | Bactericidal activity against Methicillin-sensitive Staphylococcus aureus clinical isolate USA300 assessed as log reduction in bacterial cell number at 4 times MIC after 24 hrs by time-kill curve analysis | 2016 | Journal of medicinal chemistry, Mar-10, Volume: 59, Issue:5
| Robenidine Analogues as Gram-Positive Antibacterial Agents. |
AID1286522 | Bactericidal activity against methicillin-sensitive Staphylococcus aureus ATCC 29213 assessed as log reduction in bacterial cell number at 4 times MIC after 8 hrs by time-kill curve analysis | 2016 | Journal of medicinal chemistry, Mar-10, Volume: 59, Issue:5
| Robenidine Analogues as Gram-Positive Antibacterial Agents. |
AID1286509 | Antibacterial activity against Escherichia coli ATCC 25922 after 20 to 24 hrs | 2016 | Journal of medicinal chemistry, Mar-10, Volume: 59, Issue:5
| Robenidine Analogues as Gram-Positive Antibacterial Agents. |
AID1286494 | Antibacterial activity against methicillin-sensitive Staphylococcus aureus ATCC 6538 after 20 to 24 hrs in presence of 50% heat inactivated bovine serum | 2016 | Journal of medicinal chemistry, Mar-10, Volume: 59, Issue:5
| Robenidine Analogues as Gram-Positive Antibacterial Agents. |
AID1286520 | Bactericidal activity against methicillin-sensitive Staphylococcus aureus ATCC 29213 assessed as log reduction in bacterial cell number at MIC after 8 hrs by time-kill curve analysis | 2016 | Journal of medicinal chemistry, Mar-10, Volume: 59, Issue:5
| Robenidine Analogues as Gram-Positive Antibacterial Agents. |
AID1286480 | Metabolic stability in mouse liver microsomes assessed as compound loss after 60 mins | 2016 | Journal of medicinal chemistry, Mar-10, Volume: 59, Issue:5
| Robenidine Analogues as Gram-Positive Antibacterial Agents. |
AID1286507 | Antibacterial activity against methicillin-resistant Staphylococcus aureus after 20 to 24 hrs | 2016 | Journal of medicinal chemistry, Mar-10, Volume: 59, Issue:5
| Robenidine Analogues as Gram-Positive Antibacterial Agents. |
AID1286514 | Bactericidal activity against methicillin-resistant Staphylococcus aureus clinical isolate after 24 and 48 hrs | 2016 | Journal of medicinal chemistry, Mar-10, Volume: 59, Issue:5
| Robenidine Analogues as Gram-Positive Antibacterial Agents. |
AID1286473 | Solubility of the compound at pH 2 | 2016 | Journal of medicinal chemistry, Mar-10, Volume: 59, Issue:5
| Robenidine Analogues as Gram-Positive Antibacterial Agents. |
AID1286463 | Bactericidal activity against Methicillin-sensitive Staphylococcus aureus clinical isolate USA300 assessed as log reduction in bacterial cell number at 2 times MIC after 24 hrs by time-kill curve analysis | 2016 | Journal of medicinal chemistry, Mar-10, Volume: 59, Issue:5
| Robenidine Analogues as Gram-Positive Antibacterial Agents. |
AID1286470 | Cytotoxicity against human HEL299 cells after 24 hrs by WST-1 based colorimetric assay | 2016 | Journal of medicinal chemistry, Mar-10, Volume: 59, Issue:5
| Robenidine Analogues as Gram-Positive Antibacterial Agents. |
AID1286490 | Antibacterial activity against methicillin-sensitive Staphylococcus aureus ATCC 6538 after 20 to 24 hrs | 2016 | Journal of medicinal chemistry, Mar-10, Volume: 59, Issue:5
| Robenidine Analogues as Gram-Positive Antibacterial Agents. |
AID51412 | Anticoccidial activity in chicken against E. tenella | 1991 | Journal of medicinal chemistry, Sep, Volume: 34, Issue:9
| Benzylated 1,2,3-triazoles as anticoccidiostats. |
AID1286472 | Lipophilicity, logD of the compound at pH 7.4 | 2016 | Journal of medicinal chemistry, Mar-10, Volume: 59, Issue:5
| Robenidine Analogues as Gram-Positive Antibacterial Agents. |
AID1286517 | Antibacterial activity against Pseudomonas aeruginosa ATCC 27853 after 20 to 24 hrs in presence of polymyxin B nonapeptide | 2016 | Journal of medicinal chemistry, Mar-10, Volume: 59, Issue:5
| Robenidine Analogues as Gram-Positive Antibacterial Agents. |
AID1286458 | Bactericidal activity against Methicillin-sensitive Staphylococcus aureus ATCC 29213 assessed as log reduction in bacterial cell number at MIC after 24 hrs by time kill curve analysis | 2016 | Journal of medicinal chemistry, Mar-10, Volume: 59, Issue:5
| Robenidine Analogues as Gram-Positive Antibacterial Agents. |
AID1286511 | Antibacterial activity against methicillin-resistant Staphylococcus aureus clinical isolate after 20 to 24 hrs | 2016 | Journal of medicinal chemistry, Mar-10, Volume: 59, Issue:5
| Robenidine Analogues as Gram-Positive Antibacterial Agents. |
AID1286498 | Bactericidal activity against methicillin-sensitive Staphylococcus aureus ATCC 6538 after 24 and 48 hrs | 2016 | Journal of medicinal chemistry, Mar-10, Volume: 59, Issue:5
| Robenidine Analogues as Gram-Positive Antibacterial Agents. |
AID1286518 | Ratio of MIC90 for Escherichia coli ATCC 25922 to MIC90 for Escherichia coli ATCC 25922 in presence of polymyxin B nonapeptide | 2016 | Journal of medicinal chemistry, Mar-10, Volume: 59, Issue:5
| Robenidine Analogues as Gram-Positive Antibacterial Agents. |
AID1286475 | Half life of compound in human liver microsomes | 2016 | Journal of medicinal chemistry, Mar-10, Volume: 59, Issue:5
| Robenidine Analogues as Gram-Positive Antibacterial Agents. |
AID51231 | The compound was tested for anti-coccidial activity in chicken against E. acervulina (DP-761) measured at dose 33(ppm in diet) | 1991 | Journal of medicinal chemistry, Sep, Volume: 34, Issue:9
| Benzylated 1,2,3-triazoles as anticoccidiostats. |
AID51246 | The compound was tested for anti-coccidial activity in chicken against E. hagani(DP-786) measured at dose 33(ppm in diet) | 1991 | Journal of medicinal chemistry, Sep, Volume: 34, Issue:9
| Benzylated 1,2,3-triazoles as anticoccidiostats. |
AID1286489 | Antibacterial activity against methicillin-sensitive Staphylococcus aureus ATCC 25923 after 20 to 24 hrs | 2016 | Journal of medicinal chemistry, Mar-10, Volume: 59, Issue:5
| Robenidine Analogues as Gram-Positive Antibacterial Agents. |
[information is prepared from bioassay data collected from National Library of Medicine (NLM), extracted Dec-2023] |