An EC 3.6.4.10 (non-chaperonin molecular chaperone ATPase) inhibitor that blocks the action of heat shock protein 90.
| Member | Definition | Class |
|---|
| 17-(dimethylaminoethylamino)-17-demethoxygeldanamycin | A 19-membered macrocyle that is geldanamycin in which the methoxy group attached to the benzoquinone moiety has been replaced by a 2-(N,N-dimethylamino)ethylamino group. | alvespimycin |
| 8-(2-chloro-3,4,5-trimethoxybenzyl)-2-fluoro-9-pent-4-yn-1-yl-9H-purin-6-amine | A member of the class of 6-aminopurines that is 2-fluoroadenine carrying additional 2-chloro-3,4,5-trimethoxybenzyl and pent-4-yn-1-yl substituents at positions 8 and 9 respectively. | 8-(2-chloro-3,4,5-trimethoxybenzyl)-2-fluoro-9-pent-4-yn-1-yl-9H-purin-6-amine |
| at 13387 | A member of the class of isoindoles that is isoindole in which the amino group has been acylated by a 2,4-dihydroxy-5-isopropylbenzoyl group and in which position 5 of the isoidole moiety has been substituted by a (4-methylpiperazin-1-yl)methyl group. A second-generation Hsp90 inhibitor. | onalespib |
| cct018159 | A member of the class of pyrazoles that is 1H-pyrazole carrying 1,4-benzodioxane-6-yl and 5-ethyl-2,4-dihydroxyphenyl substituents at positions 4 and 5 respectively. | CCT-018159 |
| celastrol | A pentacyclic triterpenoid that is 24,25,26-trinoroleana-1(10),3,5,7-tetraen-29-oic acid bearing an oxo substituent at position 2, a hydroxy substituent at position 3 and two methyl groups at positions 9 and 13. An antioxidant and anti-inflammatory agent. Potently inhibits lipid peroxidation in mitochondria and inhibits TNF-alpha-induced NFkappaB activation. Also shown to inhibit topoisomerase II activity in vitro (IC50 = 7.41 muM). | celastrol |
| cnf 2024 | A member of the class of 2-aminopurines that is 2-aminopurine which is substituted by a chlorine at position 6 and by a (4-methoxy-3,5-dimethylpyridin-2-yl)methyl group at position 9. | BIIB021 |
| coumermycin | A hydroxycoumarin antibiotic that is obtained from Streptomyces rishiriensis and exhibits potent antibacterial and anticancer activity. | coumermycin A1 |
| dicumarol | A hydroxycoumarin that is methane in which two hydrogens have each been substituted by a 4-hydroxycoumarin-3-yl group. Related to warfarin, it has been used as an anticoagulant. | dicoumarol |
| epigallocatechin gallate | A gallate ester obtained by the formal condensation of gallic acid with the (3R)-hydroxy group of (-)-epigallocatechin. | (-)-epigallocatechin 3-gallate |
| ethoxyquin | A quinoline that is 1,2-dihydroquinoline bearing three methyl substituents at position 2, 2 and 4 as well as an ethoxy substituent at position 6. | ethoxyquin |
| gamendazole | A member of the class of indazoles that is 3-(indazol-3-yl}prop-2-enoic acid carrying additional 2,4-dichlorobenzyl and trifluoromethyl substituents at positions 1 and 6 respectively. An orally active antispermatogenic compound with antifertility effects that is a potential male contraceptive drug. | gamendazole |
| gedunin | A pentacyclic triterpenoid natural product found particularly in Azadirachta indica and Cedrela odorata. | gedunin |
| geldanamycin | An ansamycin consisting of a 19-membered macrocyle incorporating a benzoquinone ring and a lactam functionality. It shows antimicrobial activity against many Gram-positive and some Gram-negative bacteria. | geldanamycin |
| herbimycin | A 19-membered macrocyle incorporating a benzoquinone ring and a lactam functionality. It is an ansamycin antibiotic that induces apoptosis and displays antitumour effects. | herbimycin |
| monascorubrin | | monascorubrin |
| sb 203580 | A member of the class of imidazoles carrying 4-methylsulfinylphenyl, 4-pyridyl and 4-fluorophenyl substituents at positions 2, 4 and 5 respectively. An inhibitor of mitogen-activated protein kinase. | SB 203580 |
| tanespimycin | A 19-membered macrocyle that is geldanamycin in which the methoxy substituent attached to the benzoquinone moiety has been replaced by an allylamino group. It is a potent inhibitor of heat shock protein 90 (Hsp90). A less toxic analogue than geldanamycin, it induces apoptosis and displays antitumour effects. | tanespimycin |
| ver 52296 | A monocarboxylic acid amide obtained by formal condensation of the carboxy group of 5-(2,4-dihydroxy-5-isopropylphenyl)-4-[4-(morpholin-4-ylmethyl)phenyl]-1,2-oxazole-3-carboxylic acid with the amino group of ethylamine. | luminespib |
| ver-49009 | An aromatic amide obtained by formal condensation of the carboxy group of 5-(5-chloro-2,4-dihydroxyphenyl)-4-(4-methoxyphenyl)pyrazole-3-carboxylic acid with the amino group of ethylamine. | 5-(5-chloro-2,4-dihydroxyphenyl)-N-ethyl-4-(4-methoxyphenyl)pyrazole-3-carboxamide |
| Protein | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Drugs |
|---|
| 15-hydroxyprostaglandin dehydrogenase [NAD(+)] isoform 1 | Homo sapiens (human) | Potency | 21.5927 | 1 | 5 |
| 15-lipoxygenase, partial | Homo sapiens (human) | Potency | 19.2203 | 1 | 3 |
| 67.9K protein | Vaccinia virus | Potency | 8.9716 | 2 | 2 |
| acetylcholinesterase | Homo sapiens (human) | Potency | 79.9007 | 1 | 1 |
| acid sphingomyelinase | Homo sapiens (human) | Potency | 25.1189 | 1 | 1 |
| activating transcription factor 6 | Homo sapiens (human) | Potency | 47.8419 | 2 | 5 |
| Adenosine receptor A1 | Rattus norvegicus (Norway rat) | Potency | 10.0000 | 1 | 1 |
| aldehyde dehydrogenase 1 family, member A1 | Homo sapiens (human) | Potency | 25.1647 | 1 | 7 |
| apical membrane antigen 1, AMA1 | Plasmodium falciparum 3D7 | Potency | 22.3872 | 1 | 1 |
| AR protein | Homo sapiens (human) | Potency | 32.2751 | 10 | 26 |
| aryl hydrocarbon receptor | Homo sapiens (human) | Potency | 17.3583 | 2 | 5 |
| ATAD5 protein, partial | Homo sapiens (human) | Potency | 10.1269 | 6 | 6 |
| bromodomain adjacent to zinc finger domain 2B | Homo sapiens (human) | Potency | 29.5156 | 1 | 2 |
| caspase-3 | Cricetulus griseus (Chinese hamster) | Potency | 68.4153 | 1 | 2 |
| Caspase-7 | Cricetulus griseus (Chinese hamster) | Potency | 68.4153 | 1 | 2 |
| Cellular tumor antigen p53 | Homo sapiens (human) | Potency | 26.0844 | 3 | 10 |
| cellular tumor antigen p53 isoform a | Homo sapiens (human) | Potency | 11.2947 | 2 | 2 |
| Chain A, 2-oxoglutarate Oxygenase | Homo sapiens (human) | Potency | 21.4442 | 1 | 5 |
| Chain A, ATP-DEPENDENT DNA HELICASE Q1 | Homo sapiens (human) | Potency | 3.1623 | 1 | 1 |
| Chain A, Beta-lactamase | Escherichia coli K-12 | Potency | 25.1189 | 1 | 1 |
| Chain A, HADH2 protein | Homo sapiens (human) | Potency | 26.4013 | 2 | 8 |
| Chain A, JmjC domain-containing histone demethylation protein 3A | Homo sapiens (human) | Potency | 44.6684 | 1 | 1 |
| Chain A, MAJOR APURINIC/APYRIMIDINIC ENDONUCLEASE | Homo sapiens (human) | Potency | 17.7638 | 1 | 3 |
| Chain A, Putative fructose-1,6-bisphosphate aldolase | Giardia intestinalis | Potency | 11.7908 | 1 | 3 |
| Chain A, TYROSYL-DNA PHOSPHODIESTERASE | Homo sapiens (human) | Potency | 19.9754 | 1 | 4 |
| Chain B, HADH2 protein | Homo sapiens (human) | Potency | 26.4013 | 2 | 8 |
| cytochrome P450 2C19 precursor | Homo sapiens (human) | Potency | 3.3633 | 1 | 3 |
| cytochrome P450 2C9 precursor | Homo sapiens (human) | Potency | 1.3386 | 1 | 3 |
| cytochrome P450 2C9, partial | Homo sapiens (human) | Potency | 7.5515 | 1 | 7 |
| cytochrome P450 2D6 | Homo sapiens (human) | Potency | 7.8024 | 1 | 5 |
| cytochrome P450 2D6 isoform 1 | Homo sapiens (human) | Potency | 21.1613 | 1 | 2 |
| cytochrome P450 3A4 isoform 1 | Homo sapiens (human) | Potency | 7.0420 | 2 | 10 |
| cytochrome P450 family 3 subfamily A polypeptide 4 | Homo sapiens (human) | Potency | 8.7216 | 2 | 8 |
| cytochrome P450, family 19, subfamily A, polypeptide 1, isoform CRA_a | Homo sapiens (human) | Potency | 14.2999 | 1 | 1 |
| DNA polymerase beta | Homo sapiens (human) | Potency | 0.4467 | 1 | 1 |
| DNA polymerase kappa isoform 1 | Homo sapiens (human) | Potency | 23.8770 | 1 | 2 |
| estrogen nuclear receptor alpha | Homo sapiens (human) | Potency | 23.1478 | 10 | 24 |
| estrogen receptor 2 (ER beta) | Homo sapiens (human) | Potency | 11.8832 | 1 | 1 |
| estrogen-related nuclear receptor alpha | Homo sapiens (human) | Potency | 31.7179 | 5 | 11 |
| euchromatic histone-lysine N-methyltransferase 2 | Homo sapiens (human) | Potency | 10.1663 | 1 | 4 |
| EWS/FLI fusion protein | Homo sapiens (human) | Potency | 9.0057 | 4 | 24 |
| farnesoid X nuclear receptor | Homo sapiens (human) | Potency | 24.2130 | 2 | 2 |
| flap endonuclease 1 | Homo sapiens (human) | Potency | 35.4813 | 1 | 1 |
| Fumarate hydratase | Homo sapiens (human) | Potency | 32.8968 | 1 | 4 |
| G | Vesicular stomatitis virus | Potency | 7.5515 | 1 | 7 |
| GABA theta subunit | Rattus norvegicus (Norway rat) | Potency | 7.0420 | 1 | 5 |
| galactokinase | Homo sapiens (human) | Potency | 10.0000 | 1 | 1 |
| Gamma-aminobutyric acid receptor subunit alpha-1 | Rattus norvegicus (Norway rat) | Potency | 7.0420 | 1 | 5 |
| Gamma-aminobutyric acid receptor subunit alpha-2 | Rattus norvegicus (Norway rat) | Potency | 7.0420 | 1 | 5 |
| Gamma-aminobutyric acid receptor subunit alpha-3 | Rattus norvegicus (Norway rat) | Potency | 7.0420 | 1 | 5 |
| Gamma-aminobutyric acid receptor subunit alpha-4 | Rattus norvegicus (Norway rat) | Potency | 7.0420 | 1 | 5 |
| Gamma-aminobutyric acid receptor subunit alpha-5 | Rattus norvegicus (Norway rat) | Potency | 7.0420 | 1 | 5 |
| Gamma-aminobutyric acid receptor subunit alpha-6 | Rattus norvegicus (Norway rat) | Potency | 7.0420 | 1 | 5 |
| Gamma-aminobutyric acid receptor subunit beta-1 | Rattus norvegicus (Norway rat) | Potency | 7.0420 | 1 | 5 |
| Gamma-aminobutyric acid receptor subunit beta-2 | Rattus norvegicus (Norway rat) | Potency | 7.0420 | 1 | 5 |
| Gamma-aminobutyric acid receptor subunit beta-3 | Rattus norvegicus (Norway rat) | Potency | 7.0420 | 1 | 5 |
| Gamma-aminobutyric acid receptor subunit delta | Rattus norvegicus (Norway rat) | Potency | 7.0420 | 1 | 5 |
| Gamma-aminobutyric acid receptor subunit epsilon | Rattus norvegicus (Norway rat) | Potency | 7.0420 | 1 | 5 |
| Gamma-aminobutyric acid receptor subunit gamma-1 | Rattus norvegicus (Norway rat) | Potency | 7.0420 | 1 | 5 |
| Gamma-aminobutyric acid receptor subunit gamma-2 | Rattus norvegicus (Norway rat) | Potency | 7.0420 | 1 | 5 |
| Gamma-aminobutyric acid receptor subunit gamma-3 | Rattus norvegicus (Norway rat) | Potency | 7.0420 | 1 | 5 |
| Gamma-aminobutyric acid receptor subunit pi | Rattus norvegicus (Norway rat) | Potency | 7.0420 | 1 | 5 |
| geminin | Homo sapiens (human) | Potency | 8.8022 | 2 | 5 |
| GLI family zinc finger 3 | Homo sapiens (human) | Potency | 37.5126 | 2 | 8 |
| glp-1 receptor, partial | Homo sapiens (human) | Potency | 5.6234 | 1 | 1 |
| glucocerebrosidase | Homo sapiens (human) | Potency | 0.7943 | 1 | 1 |
| glucocorticoid receptor [Homo sapiens] | Homo sapiens (human) | Potency | 21.3202 | 2 | 3 |
| Glutamate receptor 2 | Rattus norvegicus (Norway rat) | Potency | 33.4915 | 1 | 1 |
| heat shock 70kDa protein 5 (glucose-regulated protein, 78kDa) | Homo sapiens (human) | Potency | 35.4813 | 1 | 1 |
| heat shock protein beta-1 | Homo sapiens (human) | Potency | 47.5275 | 2 | 5 |
| Histamine H2 receptor | Cavia porcellus (domestic guinea pig) | Potency | 7.1642 | 2 | 15 |
| Histone H2A.x | Cricetulus griseus (Chinese hamster) | Potency | 39.1180 | 2 | 6 |
| HLA class I histocompatibility antigen, B alpha chain | Homo sapiens (human) | Potency | 7.5515 | 1 | 7 |
| hypothetical protein, conserved | Trypanosoma brucei | Potency | 31.6228 | 1 | 1 |
| hypoxia-inducible factor 1 alpha subunit | Homo sapiens (human) | Potency | 37.7491 | 2 | 5 |
| hypoxia-inducible factor 1, alpha subunit (basic helix-loop-helix transcription factor) | Homo sapiens (human) | Potency | 1.2589 | 2 | 2 |
| IDH1 | Homo sapiens (human) | Potency | 10.3225 | 1 | 1 |
| Inositol hexakisphosphate kinase 1 | Homo sapiens (human) | Potency | 7.5515 | 1 | 14 |
| Integrin alpha-IIb | Homo sapiens (human) | Potency | 10.0000 | 1 | 1 |
| Integrin beta-3 | Homo sapiens (human) | Potency | 10.0000 | 1 | 1 |
| Interferon beta | Homo sapiens (human) | Potency | 4.0512 | 3 | 29 |
| lamin isoform A-delta10 | Homo sapiens (human) | Potency | 10.8942 | 1 | 5 |
| lethal factor (plasmid) | Bacillus anthracis str. A2012 | Potency | 22.1060 | 1 | 2 |
| Luciferase | Photinus pyralis (common eastern firefly) | Potency | 39.8537 | 2 | 6 |
| lysosomal alpha-glucosidase preproprotein | Homo sapiens (human) | Potency | 3.9811 | 1 | 1 |
| Microtubule-associated protein tau | Homo sapiens (human) | Potency | 14.8214 | 2 | 5 |
| mitogen-activated protein kinase 1 | Homo sapiens (human) | Potency | 18.8541 | 1 | 2 |
| neuropeptide S receptor isoform A | Homo sapiens (human) | Potency | 12.5893 | 1 | 1 |
| Nrf2 | Homo sapiens (human) | Potency | 19.9526 | 1 | 1 |
| nuclear factor erythroid 2-related factor 2 isoform 1 | Homo sapiens (human) | Potency | 36.2154 | 4 | 13 |
| nuclear factor erythroid 2-related factor 2 isoform 2 | Homo sapiens (human) | Potency | 29.0929 | 1 | 1 |
| nuclear factor NF-kappa-B p105 subunit isoform 1 | Homo sapiens (human) | Potency | 12.5893 | 1 | 1 |
| nuclear factor of kappa light polypeptide gene enhancer in B-cells 1 (p105), isoform CRA_a | Homo sapiens (human) | Potency | 52.9707 | 1 | 1 |
| Nuclear receptor ROR-gamma | Homo sapiens (human) | Potency | 42.1632 | 1 | 1 |
| nuclear receptor ROR-gamma isoform 1 | Mus musculus (house mouse) | Potency | 18.8657 | 2 | 5 |
| nuclear receptor subfamily 1, group I, member 3 | Homo sapiens (human) | Potency | 23.4314 | 3 | 11 |
| parathyroid hormone/parathyroid hormone-related peptide receptor precursor | Homo sapiens (human) | Potency | 44.6684 | 1 | 1 |
| peripheral myelin protein 22 | Rattus norvegicus (Norway rat) | Potency | 0.0721 | 1 | 1 |
| peroxisome proliferator activated receptor gamma | Homo sapiens (human) | Potency | 37.4382 | 5 | 12 |
| peroxisome proliferator-activated receptor delta | Homo sapiens (human) | Potency | 42.0971 | 4 | 6 |
| phosphopantetheinyl transferase | Bacillus subtilis | Potency | 30.6694 | 1 | 2 |
| plasminogen precursor | Mus musculus (house mouse) | Potency | 31.6228 | 1 | 1 |
| polyprotein | Zika virus | Potency | 32.8968 | 1 | 4 |
| polyunsaturated fatty acid lipoxygenase ALOX12 | Homo sapiens (human) | Potency | 12.5893 | 1 | 1 |
| Polyunsaturated fatty acid lipoxygenase ALOX15B | Homo sapiens (human) | Potency | 15.9027 | 1 | 3 |
| potassium voltage-gated channel subfamily H member 2 isoform d | Homo sapiens (human) | Potency | 21.2804 | 1 | 2 |
| PPM1D protein | Homo sapiens (human) | Potency | 1.8181 | 1 | 14 |
| pregnane X nuclear receptor | Homo sapiens (human) | Potency | 38.3088 | 3 | 4 |
| pregnane X receptor | Rattus norvegicus (Norway rat) | Potency | 45.8577 | 1 | 2 |
| progesterone receptor | Homo sapiens (human) | Potency | 30.7538 | 1 | 2 |
| pyruvate kinase PKM isoform a | Homo sapiens (human) | Potency | 3.9811 | 2 | 2 |
| RAR-related orphan receptor gamma | Mus musculus (house mouse) | Potency | 19.6559 | 2 | 3 |
| regulator of G-protein signaling 4 | Homo sapiens (human) | Potency | 1.5912 | 1 | 2 |
| retinoic acid nuclear receptor alpha variant 1 | Homo sapiens (human) | Potency | 54.8276 | 3 | 6 |
| retinoid X nuclear receptor alpha | Homo sapiens (human) | Potency | 26.6729 | 3 | 5 |
| serine/threonine-protein kinase mTOR isoform 1 | Homo sapiens (human) | Potency | 2.4172 | 3 | 3 |
| SMAD family member 2 | Homo sapiens (human) | Potency | 38.7317 | 2 | 4 |
| SMAD family member 3 | Homo sapiens (human) | Potency | 38.7317 | 2 | 4 |
| Smad3 | Homo sapiens (human) | Potency | 1.2450 | 1 | 2 |
| survival motor neuron protein isoform d | Homo sapiens (human) | Potency | 5.3972 | 1 | 2 |
| TDP1 protein | Homo sapiens (human) | Potency | 19.0065 | 2 | 10 |
| thioredoxin glutathione reductase | Schistosoma mansoni | Potency | 50.1727 | 1 | 2 |
| thioredoxin reductase | Rattus norvegicus (Norway rat) | Potency | 89.1251 | 1 | 1 |
| thyroid hormone receptor beta isoform 2 | Rattus norvegicus (Norway rat) | Potency | 30.2658 | 3 | 14 |
| thyroid hormone receptor beta isoform a | Homo sapiens (human) | Potency | 39.1512 | 1 | 2 |
| thyroid stimulating hormone receptor | Homo sapiens (human) | Potency | 33.9558 | 5 | 6 |
| tyrosine-protein kinase Yes | Homo sapiens (human) | Potency | 17.9872 | 1 | 3 |
| urokinase plasminogen activator surface receptor precursor | Mus musculus (house mouse) | Potency | 31.6228 | 1 | 1 |
| urokinase-type plasminogen activator precursor | Mus musculus (house mouse) | Potency | 31.6228 | 1 | 1 |
| USP1 protein, partial | Homo sapiens (human) | Potency | 48.2242 | 2 | 5 |
| v-jun sarcoma virus 17 oncogene homolog (avian) | Homo sapiens (human) | Potency | 29.4962 | 2 | 8 |
| vitamin D (1,25- dihydroxyvitamin D3) receptor | Homo sapiens (human) | Potency | 51.2080 | 4 | 7 |
| vitamin D3 receptor isoform VDRA | Homo sapiens (human) | Potency | 55.3275 | 1 | 5 |
| Voltage-dependent calcium channel gamma-2 subunit | Mus musculus (house mouse) | Potency | 33.4915 | 1 | 1 |
| Vpr | Human immunodeficiency virus 1 | Potency | 0.7943 | 1 | 1 |
| Protein | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Drugs |
|---|
| 10 kDa chaperonin | Escherichia coli | IC50 | 0.4700 | 2 | 2 |
| 10 kDa heat shock protein, mitochondrial | Homo sapiens (human) | IC50 | 2.3000 | 1 | 1 |
| 3-oxoacyl-[acyl-carrier-protein] reductase | Plasmodium falciparum 3D7 | IC50 | 0.3200 | 1 | 1 |
| 3-oxoacyl-acyl-carrier protein reductase | Plasmodium falciparum (malaria parasite P. falciparum) | IC50 | 0.3000 | 1 | 1 |
| 4-galactosyl-N-acetylglucosaminide 3-alpha-L-fucosyltransferase FUT6 | Homo sapiens (human) | IC50 | 7.2833 | 1 | 6 |
| 5-hydroxytryptamine receptor 1A | Rattus norvegicus (Norway rat) | IC50 | 0.0036 | 1 | 1 |
| 6-phosphogluconate dehydrogenase, decarboxylating | Homo sapiens (human) | IC50 | 0.7200 | 1 | 1 |
| 60 kDa chaperonin | Escherichia coli K-12 | IC50 | 250.0000 | 1 | 1 |
| 60 kDa chaperonin | Escherichia coli | IC50 | 0.4700 | 2 | 2 |
| 60 kDa heat shock protein, mitochondrial | Homo sapiens (human) | IC50 | 2.3000 | 1 | 1 |
| 72 kDa type IV collagenase | Homo sapiens (human) | IC50 | 7.6143 | 2 | 7 |
| Adenosine receptor A1 | Homo sapiens (human) | IC50 | 2.9500 | 1 | 1 |
| Adenosine receptor A1 | Homo sapiens (human) | Ki | 1.7210 | 1 | 1 |
| Adenosine receptor A2a | Homo sapiens (human) | IC50 | 6.0680 | 1 | 1 |
| Adenosine receptor A2a | Homo sapiens (human) | Ki | 3.4070 | 1 | 1 |
| Alpha-(1,3)-fucosyltransferase 7 | Homo sapiens (human) | IC50 | 7.2833 | 1 | 6 |
| Alpha-amylase 1A | Homo sapiens (human) | IC50 | 1,400.0000 | 1 | 1 |
| Amine oxidase [flavin-containing] B | Rattus norvegicus (Norway rat) | IC50 | 0.3600 | 1 | 2 |
| Amyloid-beta precursor protein | Homo sapiens (human) | IC50 | 27.0250 | 4 | 4 |
| Angiopoietin-1 receptor | Homo sapiens (human) | IC50 | 20.0000 | 1 | 1 |
| Apoptosis regulator Bcl-2 | Homo sapiens (human) | IC50 | 0.4500 | 1 | 1 |
| Apoptosis regulator Bcl-2 | Homo sapiens (human) | Ki | 0.3622 | 2 | 2 |
| ATP phosphoribosyltransferase | Mycobacterium tuberculosis H37Rv | Ki | 60.0000 | 1 | 1 |
| ATP-dependent molecular chaperone HSC82 | Saccharomyces cerevisiae S288C | IC50 | 6.4133 | 1 | 3 |
| ATP-dependent molecular chaperone HSP82 | Saccharomyces cerevisiae S288C | IC50 | 9.1222 | 4 | 9 |
| ATP-dependent translocase ABCB1 | Homo sapiens (human) | IC50 | 0.1234 | 2 | 2 |
| Bcl-2-like protein 1 | Homo sapiens (human) | IC50 | 0.5900 | 1 | 1 |
| Bcl-2-like protein 10 | Homo sapiens (human) | IC50 | 0.3600 | 1 | 1 |
| Bcl-2-like protein 2 | Homo sapiens (human) | IC50 | 2.3300 | 1 | 1 |
| Bcl-2-related protein A1 | Homo sapiens (human) | IC50 | 1.7900 | 1 | 1 |
| Bcl2-associated agonist of cell death | Homo sapiens (human) | Ki | 0.4900 | 1 | 1 |
| Beta-hydroxyacyl-ACP dehydratase precursor (Fatty acid synthesis protein) | Plasmodium falciparum (malaria parasite P. falciparum) | IC50 | 0.2150 | 2 | 2 |
| Beta-secretase 1 | Homo sapiens (human) | IC50 | 1.1785 | 2 | 2 |
| BH3-interacting domain death agonist | Homo sapiens (human) | IC50 | 1.0733 | 6 | 6 |
| Bile salt export pump | Homo sapiens (human) | IC50 | 126.9650 | 2 | 2 |
| Breakpoint cluster region protein | Homo sapiens (human) | IC50 | 3.0000 | 2 | 4 |
| cAMP-dependent protein kinase catalytic subunit alpha | Homo sapiens (human) | IC50 | 50.0000 | 1 | 1 |
| cAMP-dependent protein kinase catalytic subunit beta | Homo sapiens (human) | IC50 | 50.0000 | 1 | 1 |
| cAMP-dependent protein kinase catalytic subunit gamma | Homo sapiens (human) | IC50 | 50.0000 | 1 | 1 |
| Cannabinoid receptor 1 | Homo sapiens (human) | Ki | 33.6000 | 2 | 2 |
| Cannabinoid receptor 2 | Homo sapiens (human) | Ki | 42.8000 | 1 | 1 |
| Casein kinase I isoform delta | Homo sapiens (human) | IC50 | 0.4147 | 3 | 3 |
| Casein kinase I isoform epsilon | Homo sapiens (human) | IC50 | 1.0000 | 1 | 1 |
| cGMP-specific 3',5'-cyclic phosphodiesterase | Homo sapiens (human) | IC50 | 11.4760 | 1 | 1 |
| Chain A, Erk2 | Homo sapiens (human) | Ki | 0.0004 | 1 | 1 |
| Chain A, Heat shock protein HSP 90-alpha | Homo sapiens (human) | IC50 | 0.0190 | 1 | 3 |
| Chain A, Heat shock protein HSP 90-alpha | Homo sapiens (human) | Ki | 0.0017 | 1 | 1 |
| Chain A, POLYMERASE PA | Influenza A virus | IC50 | 1.9000 | 1 | 1 |
| Chain A, Polymerase Pa | Influenza A virus (A/California/04/2009(H1N1)) | IC50 | 1.9000 | 1 | 4 |
| Cholesteryl ester transfer protein | Homo sapiens (human) | IC50 | 0.0400 | 1 | 1 |
| Cholinesterase | Homo sapiens (human) | IC50 | 0.0026 | 1 | 1 |
| Citron Rho-interacting kinase | Homo sapiens (human) | IC50 | 1.0000 | 1 | 1 |
| CMP-N-acetylneuraminate-beta-galactosamide-alpha-2,3-sialyltransferase 1 | Homo sapiens (human) | IC50 | 7.2833 | 1 | 6 |
| Corticotropin releasing hormone receptor 2 | Sus scrofa (pig) | IC50 | 0.0040 | 1 | 1 |
| CPG DNA methylase | Spiroplasma monobiae | Ki | 0.0280 | 1 | 1 |
| CREB-binding protein | Homo sapiens (human) | IC50 | 50.0000 | 2 | 2 |
| Cyclin-G-associated kinase | Homo sapiens (human) | IC50 | 0.4133 | 3 | 3 |
| Cytochrome P450 1A2 | Homo sapiens (human) | IC50 | 1.0070 | 2 | 2 |
| Cytochrome P450 2C19 | Homo sapiens (human) | IC50 | 0.2940 | 2 | 3 |
| Cytochrome P450 2C9 | Homo sapiens (human) | IC50 | 0.3455 | 2 | 4 |
| Cytochrome P450 2C9 | Homo sapiens (human) | Ki | 1.2500 | 2 | 2 |
| Cytochrome P450 2D6 | Homo sapiens (human) | IC50 | 1.0070 | 2 | 2 |
| Cytochrome P450 3A4 | Homo sapiens (human) | IC50 | 0.0380 | 2 | 2 |
| Cytochrome P450 3A43 | Homo sapiens (human) | IC50 | 0.0140 | 1 | 1 |
| Cytochrome P450 3A5 | Homo sapiens (human) | IC50 | 0.0140 | 1 | 1 |
| Cytochrome P450 3A7 | Homo sapiens (human) | IC50 | 0.0140 | 1 | 1 |
| Delta-type opioid receptor | Mus musculus (house mouse) | IC50 | 0.0200 | 1 | 1 |
| Dipeptidyl peptidase 4 | Homo sapiens (human) | IC50 | 10.2100 | 1 | 1 |
| Disintegrin and metalloproteinase domain-containing protein 17 | Homo sapiens (human) | IC50 | 21.0000 | 1 | 1 |
| DNA (cytosine-5)-methyltransferase 1 | Homo sapiens (human) | IC50 | 0.5000 | 1 | 1 |
| DNA repair protein RAD52 homolog | Homo sapiens (human) | IC50 | 2.5108 | 5 | 5 |
| DNA-dependent protein kinase catalytic subunit | Homo sapiens (human) | IC50 | 40.0000 | 1 | 1 |
| Dual specificity mitogen-activated protein kinase kinase 1 | Homo sapiens (human) | IC50 | 61.0000 | 1 | 1 |
| Dual specificity mitogen-activated protein kinase kinase 2 | Homo sapiens (human) | IC50 | 61.0000 | 1 | 1 |
| Dual specificity tyrosine-phosphorylation-regulated kinase 1A | Homo sapiens (human) | IC50 | 2.9324 | 5 | 5 |
| Dual specificity tyrosine-phosphorylation-regulated kinase 1A | Rattus norvegicus (Norway rat) | IC50 | 0.3300 | 1 | 1 |
| Endoplasmin | Canis lupus familiaris (dog) | IC50 | 0.0380 | 2 | 5 |
| Endoplasmin | Homo sapiens (human) | IC50 | 0.0535 | 2 | 2 |
| Endoplasmin | Homo sapiens (human) | Ki | 0.0900 | 1 | 2 |
| Endothelial PAS domain-containing protein 1 | Homo sapiens (human) | IC50 | 7.5252 | 4 | 4 |
| Enoyl-[acyl-carrier-protein] reductase [NADH] | Francisella tularensis subsp. tularensis SCHU S4 | IC50 | 47.0000 | 1 | 1 |
| Enoyl-[acyl-carrier-protein] reductase [NADH] FabI | Escherichia coli K-12 | IC50 | 10.0000 | 2 | 2 |
| Enoyl-acyl-carrier protein reductase | Plasmodium falciparum (malaria parasite P. falciparum) | IC50 | 0.2250 | 2 | 2 |
| Enoyl-acyl-carrier protein reductase | Plasmodium falciparum (malaria parasite P. falciparum) | Ki | 0.0910 | 3 | 3 |
| Ephrin type-B receptor 2 | Homo sapiens (human) | IC50 | 7.8000 | 1 | 1 |
| Epidermal growth factor receptor | Homo sapiens (human) | IC50 | 64.5000 | 2 | 2 |
| Fatty acid synthase | Gallus gallus (chicken) | IC50 | 68.0000 | 3 | 3 |
| Fatty acid synthase | Homo sapiens (human) | IC50 | 51.9700 | 1 | 1 |
| G-protein coupled receptor 35 | Homo sapiens (human) | Ki | 0.0390 | 1 | 1 |
| Genome polyprotein | Zika virus | IC50 | 87.0000 | 1 | 1 |
| Glucose-6-phosphate 1-dehydrogenase | Saccharomyces cerevisiae S288C | IC50 | 0.2500 | 1 | 1 |
| Heat shock protein 75 kDa, mitochondrial | Homo sapiens (human) | IC50 | 0.5507 | 4 | 7 |
| Heat shock protein 75 kDa, mitochondrial | Homo sapiens (human) | Ki | 0.0390 | 1 | 2 |
| Heat shock protein HSP 90 | Oryctolagus cuniculus (rabbit) | IC50 | 1.1410 | 2 | 2 |
| Heat shock protein HSP 90-alpha | Homo sapiens (human) | GI50 | 0.0320 | 1 | 1 |
| Heat shock protein HSP 90-alpha | Homo sapiens (human) | IC50 | 6.5061 | 72 | 100 |
| Heat shock protein HSP 90-alpha | Homo sapiens (human) | Ki | 0.0813 | 7 | 9 |
| Heat shock protein HSP 90-beta | Homo sapiens (human) | IC50 | 7.3081 | 53 | 82 |
| Heat shock protein HSP 90-beta | Homo sapiens (human) | Ki | 0.0542 | 6 | 11 |
| Heat-shock protein | Plasmodium falciparum (malaria parasite P. falciparum) | IC50 | 20.1000 | 1 | 1 |
| Heme oxygenase 1 | Rattus norvegicus (Norway rat) | IC50 | 18.0000 | 1 | 1 |
| Heme oxygenase 2 | Rattus norvegicus (Norway rat) | IC50 | 18.0000 | 1 | 1 |
| Hepatocyte growth factor receptor | Homo sapiens (human) | IC50 | 10.0000 | 1 | 1 |
| Hepatocyte growth factor receptor | Homo sapiens (human) | Ki | 3.3000 | 1 | 1 |
| Histidine kinase | Caulobacter vibrioides | IC50 | 17.6500 | 1 | 2 |
| Histone acetyltransferase KAT2B | Homo sapiens (human) | IC50 | 60.0000 | 2 | 2 |
| Histone acetyltransferase KAT5 | Homo sapiens (human) | IC50 | 70.0000 | 2 | 2 |
| Histone acetyltransferase p300 | Homo sapiens (human) | IC50 | 30.0000 | 2 | 2 |
| Histone deacetylase 1 | Homo sapiens (human) | IC50 | 334.0000 | 3 | 3 |
| Histone deacetylase 11 | Homo sapiens (human) | IC50 | 334.0000 | 3 | 3 |
| Histone deacetylase 2 | Homo sapiens (human) | IC50 | 334.0000 | 3 | 3 |
| Histone deacetylase 3 | Homo sapiens (human) | IC50 | 334.0000 | 3 | 3 |
| Histone deacetylase 4 | Homo sapiens (human) | IC50 | 334.0000 | 3 | 3 |
| Histone deacetylase 5 | Homo sapiens (human) | IC50 | 334.0000 | 3 | 3 |
| Histone deacetylase 6 | Homo sapiens (human) | IC50 | 334.0000 | 3 | 3 |
| Histone deacetylase 7 | Homo sapiens (human) | IC50 | 334.0000 | 3 | 3 |
| Histone deacetylase 8 | Homo sapiens (human) | IC50 | 334.0000 | 3 | 3 |
| Histone deacetylase 9 | Homo sapiens (human) | IC50 | 334.0000 | 3 | 3 |
| Hypoxia-inducible factor 1-alpha | Homo sapiens (human) | IC50 | 4.3521 | 7 | 7 |
| Indoleamine 2,3-dioxygenase 1 | Homo sapiens (human) | IC50 | 8.4100 | 1 | 1 |
| Induced myeloid leukemia cell differentiation protein Mcl-1 | Homo sapiens (human) | IC50 | 0.9200 | 1 | 1 |
| Integrase | Human immunodeficiency virus 1 | IC50 | 166.6667 | 2 | 3 |
| L-ornithine N(5)-monooxygenase | Aspergillus fumigatus Af293 | IC50 | 11.0000 | 2 | 2 |
| Lethal factor | Bacillus anthracis | IC50 | 0.0970 | 1 | 1 |
| Lysine-specific demethylase 4B | Homo sapiens (human) | IC50 | 0.7000 | 1 | 3 |
| Lysine-specific demethylase 4C | Homo sapiens (human) | IC50 | 0.7000 | 1 | 3 |
| Lysine-specific demethylase 5A | Homo sapiens (human) | IC50 | 0.1300 | 1 | 3 |
| Lysine-specific demethylase 6B | Homo sapiens (human) | IC50 | 0.4000 | 1 | 3 |
| MAP kinase-activated protein kinase 5 | Homo sapiens (human) | IC50 | 1.0000 | 1 | 1 |
| Matrilysin | Homo sapiens (human) | IC50 | 9.3143 | 2 | 7 |
| Matrix metalloproteinase-14 | Homo sapiens (human) | IC50 | 6.8000 | 1 | 1 |
| Microtubule-associated protein tau | Homo sapiens (human) | IC50 | 1.8000 | 1 | 1 |
| Mitogen-activated protein kinase 1 | Homo sapiens (human) | IC50 | 4.4260 | 1 | 1 |
| Mitogen-activated protein kinase 1 | Rattus norvegicus (Norway rat) | IC50 | 500.0240 | 1 | 2 |
| Mitogen-activated protein kinase 10 | Homo sapiens (human) | IC50 | 0.6933 | 3 | 3 |
| Mitogen-activated protein kinase 10 | Homo sapiens (human) | Ki | 0.0900 | 1 | 1 |
| Mitogen-activated protein kinase 11 | Homo sapiens (human) | IC50 | 0.2646 | 26 | 27 |
| Mitogen-activated protein kinase 12 | Homo sapiens (human) | IC50 | 0.2329 | 21 | 22 |
| Mitogen-activated protein kinase 13 | Homo sapiens (human) | IC50 | 0.2329 | 21 | 22 |
| Mitogen-activated protein kinase 14 | Homo sapiens (human) | IC50 | 15.1567 | 74 | 77 |
| Mitogen-activated protein kinase 14 | Homo sapiens (human) | Ki | 0.0375 | 2 | 2 |
| Mitogen-activated protein kinase 14 | Mus musculus (house mouse) | IC50 | 0.0560 | 1 | 3 |
| Mitogen-activated protein kinase 2 | Pneumocystis carinii | IC50 | 0.1050 | 1 | 1 |
| Mitogen-activated protein kinase 9 | Homo sapiens (human) | IC50 | 2.3871 | 7 | 7 |
| Muscarinic acetylcholine receptor M1 | Homo sapiens (human) | IC50 | 10.6660 | 1 | 1 |
| Muscarinic acetylcholine receptor M1 | Homo sapiens (human) | Ki | 2.5690 | 1 | 1 |
| Myeloperoxidase | Homo sapiens (human) | Ki | 0.0900 | 1 | 1 |
| Myotonin-protein kinase | Homo sapiens (human) | IC50 | 1.0000 | 1 | 1 |
| NAD | Homo sapiens (human) | IC50 | 0.2585 | 7 | 8 |
| NAD | Rattus norvegicus (Norway rat) | Ki | 0.0010 | 1 | 1 |
| NAD kinase | Homo sapiens (human) | IC50 | 0.9600 | 1 | 1 |
| NAD kinase | Homo sapiens (human) | Ki | 3.2800 | 1 | 1 |
| Neuronal acetylcholine receptor subunit alpha-4 | Rattus norvegicus (Norway rat) | Ki | 0.0900 | 1 | 1 |
| Neuronal acetylcholine receptor subunit beta-2 | Rattus norvegicus (Norway rat) | Ki | 0.0900 | 1 | 1 |
| Neutrophil elastase | Homo sapiens (human) | IC50 | 6.4125 | 2 | 2 |
| P2X purinoceptor 7 | Homo sapiens (human) | IC50 | 5.0000 | 1 | 1 |
| P2X purinoceptor 7 | Rattus norvegicus (Norway rat) | IC50 | 30.0000 | 1 | 1 |
| Peptidyl-prolyl cis-trans isomerase NIMA-interacting 1 | Homo sapiens (human) | IC50 | 20.0000 | 1 | 1 |
| Phosphatidylinositol 3,4,5-trisphosphate 3-phosphatase and dual-specificity protein phosphatase PTEN | Homo sapiens (human) | IC50 | 13.3000 | 1 | 1 |
| Phosphoglycerate mutase 1 | Homo sapiens (human) | IC50 | 0.4900 | 2 | 2 |
| Plasminogen activator inhibitor 1 | Homo sapiens (human) | IC50 | 0.0910 | 1 | 1 |
| Polyamine deacetylase HDAC10 | Homo sapiens (human) | IC50 | 334.0000 | 3 | 3 |
| Polymerase acidic protein | Influenza A virus (A/Puerto Rico/8/1934(H1N1)) | IC50 | 5.8600 | 1 | 1 |
| Proprotein convertase subtilisin/kexin type 7 | Homo sapiens (human) | IC50 | 1.3000 | 1 | 1 |
| Prostaglandin E synthase | Homo sapiens (human) | IC50 | 1.8000 | 1 | 1 |
| Prostaglandin G/H synthase 1 | Homo sapiens (human) | IC50 | 3.5000 | 2 | 2 |
| Proteasome subunit beta type-5 | Homo sapiens (human) | IC50 | 6.3620 | 3 | 3 |
| Protein kinase C alpha type | Homo sapiens (human) | IC50 | 75.0000 | 1 | 1 |
| Protein kinase C beta type | Homo sapiens (human) | IC50 | 75.0000 | 1 | 1 |
| Protein kinase C delta type | Homo sapiens (human) | IC50 | 75.0000 | 1 | 1 |
| Protein kinase C epsilon type | Homo sapiens (human) | IC50 | 75.0000 | 1 | 1 |
| Protein kinase C eta type | Homo sapiens (human) | IC50 | 75.0000 | 1 | 1 |
| Protein kinase C gamma type | Homo sapiens (human) | IC50 | 75.0000 | 1 | 1 |
| Protein kinase C iota type | Homo sapiens (human) | IC50 | 75.0000 | 1 | 1 |
| Protein kinase C theta type | Homo sapiens (human) | IC50 | 75.0000 | 1 | 1 |
| Protein kinase C zeta type | Homo sapiens (human) | IC50 | 75.0000 | 1 | 1 |
| Proto-oncogene tyrosine-protein kinase Src | Homo sapiens (human) | IC50 | 5.0000 | 1 | 1 |
| Putative heat shock protein HSP 90-alpha A4 | Homo sapiens (human) | IC50 | 0.4600 | 1 | 2 |
| RAF proto-oncogene serine/threonine-protein kinase | Homo sapiens (human) | IC50 | 0.7575 | 4 | 4 |
| Receptor tyrosine-protein kinase erbB-2 | Homo sapiens (human) | IC50 | 9.4635 | 2 | 2 |
| Receptor-interacting serine/threonine-protein kinase 2 | Homo sapiens (human) | IC50 | 1.0359 | 7 | 8 |
| Receptor-type tyrosine-protein phosphatase epsilon | Homo sapiens (human) | IC50 | 500.0000 | 1 | 1 |
| Receptor-type tyrosine-protein phosphatase eta | Homo sapiens (human) | IC50 | 111.5000 | 1 | 1 |
| Regulator of G-protein signaling 17 | Homo sapiens (human) | IC50 | 27.9338 | 5 | 5 |
| Replicase polyprotein 1ab | Betacoronavirus England 1 | IC50 | 10.0000 | 1 | 2 |
| Replicase polyprotein 1ab | Severe acute respiratory syndrome coronavirus 2 | IC50 | 4.2000 | 2 | 3 |
| Replicase polyprotein 1ab | Severe acute respiratory syndrome-related coronavirus | IC50 | 10.3000 | 2 | 2 |
| Replicase polyprotein 1ab | Severe acute respiratory syndrome coronavirus 2 | Ki | 4.2000 | 1 | 1 |
| Replicase polyprotein 1ab | Severe acute respiratory syndrome-related coronavirus | Ki | 4.2000 | 2 | 2 |
| Reverse transcriptase/RNaseH | Human immunodeficiency virus 1 | IC50 | 0.7300 | 1 | 1 |
| Sarcoplasmic/endoplasmic reticulum calcium ATPase 1 | Oryctolagus cuniculus (rabbit) | IC50 | 12.0000 | 1 | 1 |
| Serine/threonine-protein kinase 36 | Homo sapiens (human) | IC50 | 1.0000 | 1 | 1 |
| Serine/threonine-protein kinase B-raf | Homo sapiens (human) | IC50 | 1.0000 | 1 | 1 |
| Serine/threonine-protein kinase D1 | Homo sapiens (human) | IC50 | 75.0000 | 1 | 1 |
| Serine/threonine-protein kinase D3 | Homo sapiens (human) | IC50 | 75.0000 | 1 | 1 |
| Serine/threonine-protein kinase NLK | Homo sapiens (human) | IC50 | 1.0000 | 1 | 1 |
| Sigma non-opioid intracellular receptor 1 | Cavia porcellus (domestic guinea pig) | IC50 | 10.0000 | 1 | 1 |
| Sodium-dependent serotonin transporter | Rattus norvegicus (Norway rat) | IC50 | 0.0100 | 1 | 1 |
| Squalene monooxygenase | Rattus norvegicus (Norway rat) | IC50 | 0.6900 | 2 | 2 |
| Telomerase reverse transcriptase | Homo sapiens (human) | IC50 | 1.0100 | 4 | 4 |
| TGF-beta receptor type-1 | Homo sapiens (human) | IC50 | 18.0000 | 2 | 2 |
| Thiosulfate sulfurtransferase | Homo sapiens (human) | IC50 | 7.3000 | 1 | 1 |
| Thromboxane-A synthase | Homo sapiens (human) | IC50 | 0.4940 | 1 | 1 |
| Tissue-type plasminogen activator | Homo sapiens (human) | IC50 | 0.0910 | 1 | 1 |
| TRAF2 and NCK-interacting protein kinase | Homo sapiens (human) | IC50 | 1.0000 | 1 | 1 |
| Tryptophan 2,3-dioxygenase | Homo sapiens (human) | IC50 | 100.0000 | 1 | 1 |
| Tyrosinase | Mus musculus (house mouse) | IC50 | 0.0340 | 1 | 1 |
| Tyrosine-protein kinase ABL1 | Homo sapiens (human) | IC50 | 3.0000 | 2 | 4 |
| Tyrosine-protein kinase Lck | Homo sapiens (human) | IC50 | 3.4500 | 1 | 1 |
| Tyrosine-protein phosphatase non-receptor type 1 | Homo sapiens (human) | IC50 | 6.7000 | 3 | 3 |
| Tyrosine-protein phosphatase non-receptor type 11 | Homo sapiens (human) | IC50 | 3.5667 | 3 | 3 |
| Tyrosine-protein phosphatase non-receptor type 2 | Homo sapiens (human) | IC50 | 20.9000 | 2 | 2 |
| Tyrosine-protein phosphatase non-receptor type 6 | Homo sapiens (human) | IC50 | 15.4500 | 2 | 2 |
| Tyrosine-protein phosphatase non-receptor type 7 | Homo sapiens (human) | IC50 | 75.7000 | 1 | 1 |
| Ubiquitin carboxyl-terminal hydrolase 15 | Homo sapiens (human) | IC50 | 31.4000 | 1 | 5 |
| Ubiquitin carboxyl-terminal hydrolase 2 | Homo sapiens (human) | IC50 | 31.4000 | 1 | 5 |
| Ubiquitin carboxyl-terminal hydrolase isozyme L1 | Homo sapiens (human) | IC50 | 31.4000 | 1 | 5 |
| Ubiquitin carboxyl-terminal hydrolase isozyme L3 | Homo sapiens (human) | IC50 | 31.4000 | 1 | 5 |
| Ubiquitin carboxyl-terminal hydrolase isozyme L5 | Homo sapiens (human) | IC50 | 31.4000 | 1 | 5 |
| Urease | Canavalia ensiformis (jack bean) | IC50 | 15.0728 | 2 | 2 |
| Urokinase-type plasminogen activator | Homo sapiens (human) | IC50 | 0.0910 | 1 | 1 |
| Urokinase-type plasminogen activator | Mus musculus (house mouse) | IC50 | 0.0910 | 1 | 1 |
| Virulence sensor histidine kinase PhoQ | Salmonella enterica subsp. enterica serovar Typhimurium str. LT2 | IC50 | 261.0000 | 1 | 1 |
| Protein | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Drugs |
|---|
| 3-phosphoinositide-dependent protein kinase 1 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| 5'-AMP-activated protein kinase catalytic subunit alpha-1 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| 5'-AMP-activated protein kinase catalytic subunit alpha-2 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Activated CDC42 kinase 1 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Activin receptor type-1 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Activin receptor type-1B | Homo sapiens (human) | Kd | 3.0000 | 2 | 2 |
| Activin receptor type-2A | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Activin receptor type-2B | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| ALK tyrosine kinase receptor | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Angiopoietin-1 receptor | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Ankyrin repeat and protein kinase domain-containing protein 1 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| AP2-associated protein kinase 1 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| ATP-dependent molecular chaperone HSP82 | Saccharomyces cerevisiae S288C | Kd | 1.2000 | 1 | 1 |
| Atypical kinase COQ8A, mitochondrial | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Atypical kinase COQ8B, mitochondrial | Homo sapiens (human) | Kd | 3.1000 | 2 | 2 |
| Aurora kinase A | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Aurora kinase B | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Aurora kinase C | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| BDNF/NT-3 growth factors receptor | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| BMP-2-inducible protein kinase | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Bone morphogenetic protein receptor type-1A | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Bone morphogenetic protein receptor type-1B | Homo sapiens (human) | Kd | 3.3000 | 1 | 1 |
| Bone morphogenetic protein receptor type-2 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Calcium-dependent protein kinase 1 | Plasmodium falciparum 3D7 | Kd | 0.8500 | 1 | 1 |
| Calcium/calmodulin-dependent protein kinase kinase 1 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Calcium/calmodulin-dependent protein kinase kinase 2 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Calcium/calmodulin-dependent protein kinase type 1 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Calcium/calmodulin-dependent protein kinase type 1D | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Calcium/calmodulin-dependent protein kinase type 1G | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Calcium/calmodulin-dependent protein kinase type II subunit alpha | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Calcium/calmodulin-dependent protein kinase type II subunit beta | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Calcium/calmodulin-dependent protein kinase type II subunit delta | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Calcium/calmodulin-dependent protein kinase type II subunit gamma | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Calcium/calmodulin-dependent protein kinase type IV | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| cAMP-dependent protein kinase catalytic subunit alpha | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| cAMP-dependent protein kinase catalytic subunit beta | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| cAMP-dependent protein kinase catalytic subunit PRKX | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Casein kinase I isoform alpha | Homo sapiens (human) | Kd | 0.0750 | 1 | 1 |
| Casein kinase I isoform alpha-like | Homo sapiens (human) | Kd | 1.7000 | 2 | 2 |
| Casein kinase I isoform delta | Homo sapiens (human) | Kd | 0.0370 | 2 | 2 |
| Casein kinase I isoform epsilon | Homo sapiens (human) | Kd | 0.1400 | 3 | 3 |
| Casein kinase I isoform gamma-1 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Casein kinase I isoform gamma-2 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Casein kinase I isoform gamma-3 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Casein kinase II subunit alpha | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Casein kinase II subunit alpha' | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Cell division control protein 2 homolog | Plasmodium falciparum 3D7 | Kd | 10.0000 | 1 | 1 |
| cGMP-dependent protein kinase 1 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| cGMP-dependent protein kinase 2 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Chain A, Peptidyl-prolyl cis-trans isomerase NIMA-interacting 1 | Homo sapiens (human) | Kd | 21.6000 | 1 | 1 |
| Chain A, Troponin C, slow skeletal and cardiac muscles | Homo sapiens (human) | Kd | 1,100.0000 | 1 | 1 |
| Cholesteryl ester transfer protein | Homo sapiens (human) | Kd | 0.1235 | 1 | 4 |
| Citron Rho-interacting kinase | Homo sapiens (human) | Kd | 0.4200 | 2 | 2 |
| Cyclin-dependent kinase 11A | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Cyclin-dependent kinase 11B | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Cyclin-dependent kinase 13 | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Cyclin-dependent kinase 14 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Cyclin-dependent kinase 15 | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Cyclin-dependent kinase 16 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Cyclin-dependent kinase 17 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Cyclin-dependent kinase 18 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Cyclin-dependent kinase 19 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Cyclin-dependent kinase 2 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Cyclin-dependent kinase 3 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Cyclin-dependent kinase 4 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Cyclin-dependent kinase 7 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Cyclin-dependent kinase 8 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Cyclin-dependent kinase 9 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Cyclin-dependent kinase-like 1 | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Cyclin-dependent kinase-like 2 | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Cyclin-dependent kinase-like 3 | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Cyclin-dependent kinase-like 5 | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Cyclin-dependent-like kinase 5 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Cyclin-G-associated kinase | Homo sapiens (human) | Kd | 0.0257 | 3 | 3 |
| Cytoplasmic tyrosine-protein kinase BMX | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Death-associated protein kinase 1 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Death-associated protein kinase 2 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Death-associated protein kinase 3 | Homo sapiens (human) | Kd | 10.0000 | 3 | 3 |
| Discoidin domain-containing receptor 2 | Homo sapiens (human) | Kd | 5.0000 | 2 | 2 |
| Dual serine/threonine and tyrosine protein kinase | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Dual specificity mitogen-activated protein kinase kinase 1 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Dual specificity mitogen-activated protein kinase kinase 2 | Homo sapiens (human) | Kd | 9.6000 | 2 | 2 |
| Dual specificity mitogen-activated protein kinase kinase 3 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Dual specificity mitogen-activated protein kinase kinase 4 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Dual specificity mitogen-activated protein kinase kinase 5 | Homo sapiens (human) | Kd | 1.4000 | 1 | 1 |
| Dual specificity mitogen-activated protein kinase kinase 6 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Dual specificity mitogen-activated protein kinase kinase 7 | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Dual specificity protein kinase CLK1 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Dual specificity protein kinase CLK2 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Dual specificity protein kinase CLK3 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Dual specificity protein kinase CLK4 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Dual specificity protein kinase TTK | Homo sapiens (human) | Kd | 2.5000 | 2 | 2 |
| Dual specificity testis-specific protein kinase 1 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Dual specificity tyrosine-phosphorylation-regulated kinase 1A | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Dual specificity tyrosine-phosphorylation-regulated kinase 1B | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Dual specificity tyrosine-phosphorylation-regulated kinase 2 | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| eIF-2-alpha kinase GCN2 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Endoplasmin | Canis lupus familiaris (dog) | EC50 | 0.0945 | 1 | 2 |
| Ephrin type-A receptor 1 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Ephrin type-A receptor 2 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Ephrin type-A receptor 3 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Ephrin type-A receptor 4 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Ephrin type-A receptor 5 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Ephrin type-A receptor 6 | Homo sapiens (human) | Kd | 1.2000 | 2 | 2 |
| Ephrin type-A receptor 7 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Ephrin type-A receptor 8 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Ephrin type-B receptor 1 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Ephrin type-B receptor 2 | Homo sapiens (human) | Kd | 8.9333 | 3 | 3 |
| Ephrin type-B receptor 3 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Ephrin type-B receptor 4 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Ephrin type-B receptor 6 | Homo sapiens (human) | Kd | 3.1000 | 1 | 1 |
| Epidermal growth factor receptor | Homo sapiens (human) | Kd | 1.6783 | 23 | 23 |
| Epithelial discoidin domain-containing receptor 1 | Homo sapiens (human) | Kd | 1.0000 | 2 | 2 |
| Eukaryotic translation initiation factor 2-alpha kinase 1 | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Fibroblast growth factor receptor 1 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Fibroblast growth factor receptor 2 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Fibroblast growth factor receptor 3 | Homo sapiens (human) | Kd | 10.0000 | 4 | 4 |
| Fibroblast growth factor receptor 4 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Focal adhesion kinase 1 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| G protein-coupled receptor kinase 4 | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| G-protein coupled receptor 35 | Homo sapiens (human) | EC50 | 4.1267 | 3 | 3 |
| GABA theta subunit | Rattus norvegicus (Norway rat) | EC50 | 0.0325 | 1 | 2 |
| Gamma-aminobutyric acid receptor subunit alpha-1 | Rattus norvegicus (Norway rat) | EC50 | 0.0325 | 1 | 2 |
| Gamma-aminobutyric acid receptor subunit alpha-2 | Rattus norvegicus (Norway rat) | EC50 | 0.0325 | 1 | 2 |
| Gamma-aminobutyric acid receptor subunit alpha-3 | Rattus norvegicus (Norway rat) | EC50 | 0.0325 | 1 | 2 |
| Gamma-aminobutyric acid receptor subunit alpha-4 | Rattus norvegicus (Norway rat) | EC50 | 0.0325 | 1 | 2 |
| Gamma-aminobutyric acid receptor subunit alpha-5 | Rattus norvegicus (Norway rat) | EC50 | 0.0325 | 1 | 2 |
| Gamma-aminobutyric acid receptor subunit alpha-6 | Rattus norvegicus (Norway rat) | EC50 | 0.0325 | 1 | 2 |
| Gamma-aminobutyric acid receptor subunit beta-1 | Rattus norvegicus (Norway rat) | EC50 | 0.0325 | 1 | 2 |
| Gamma-aminobutyric acid receptor subunit beta-2 | Rattus norvegicus (Norway rat) | EC50 | 0.0325 | 1 | 2 |
| Gamma-aminobutyric acid receptor subunit beta-3 | Rattus norvegicus (Norway rat) | EC50 | 0.0325 | 1 | 2 |
| Gamma-aminobutyric acid receptor subunit delta | Rattus norvegicus (Norway rat) | EC50 | 0.0325 | 1 | 2 |
| Gamma-aminobutyric acid receptor subunit epsilon | Rattus norvegicus (Norway rat) | EC50 | 0.0325 | 1 | 2 |
| Gamma-aminobutyric acid receptor subunit gamma-1 | Rattus norvegicus (Norway rat) | EC50 | 0.0325 | 1 | 2 |
| Gamma-aminobutyric acid receptor subunit gamma-2 | Rattus norvegicus (Norway rat) | EC50 | 0.0325 | 1 | 2 |
| Gamma-aminobutyric acid receptor subunit gamma-3 | Rattus norvegicus (Norway rat) | EC50 | 0.0325 | 1 | 2 |
| Gamma-aminobutyric acid receptor subunit pi | Rattus norvegicus (Norway rat) | EC50 | 0.0325 | 1 | 2 |
| Glycogen synthase kinase-3 alpha | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Glycogen synthase kinase-3 beta | Homo sapiens (human) | Kd | 1.7000 | 2 | 2 |
| Heat shock factor protein 1 | Homo sapiens (human) | EC50 | 1.8500 | 2 | 2 |
| Heat shock protein 90, putative | Plasmodium falciparum 3D7 | Kd | 0.2435 | 2 | 2 |
| Heat shock protein HSP 90-alpha | Homo sapiens (human) | EC50 | 0.1674 | 17 | 28 |
| Heat shock protein HSP 90-alpha | Homo sapiens (human) | Kd | 0.4963 | 17 | 20 |
| Heat shock protein HSP 90-beta | Homo sapiens (human) | EC50 | 0.2809 | 12 | 18 |
| Heat shock protein HSP 90-beta | Homo sapiens (human) | Kd | 0.5639 | 10 | 13 |
| Hepatocyte growth factor receptor | Homo sapiens (human) | Kd | 9.4750 | 4 | 4 |
| High affinity nerve growth factor receptor | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Homeodomain-interacting protein kinase 1 | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Homeodomain-interacting protein kinase 2 | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Homeodomain-interacting protein kinase 3 | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Homeodomain-interacting protein kinase 4 | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Hormonally up-regulated neu tumor-associated kinase | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Inhibitor of nuclear factor kappa-B kinase subunit alpha | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Inhibitor of nuclear factor kappa-B kinase subunit beta | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Inhibitor of nuclear factor kappa-B kinase subunit epsilon | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Insulin receptor | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Insulin receptor-related protein | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Insulin-like growth factor 1 receptor | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Interferon-induced, double-stranded RNA-activated protein kinase | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Interleukin-1 receptor-associated kinase 1 | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Interleukin-1 receptor-associated kinase 3 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Interleukin-1 receptor-associated kinase 4 | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| L-ornithine N(5)-monooxygenase | Aspergillus fumigatus Af293 | Kd | 1.4000 | 2 | 2 |
| Leucine-rich repeat serine/threonine-protein kinase 2 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Leukocyte tyrosine kinase receptor | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Leukotriene C4 synthase | Cavia porcellus (domestic guinea pig) | Kd | 10.0000 | 1 | 1 |
| LIM domain kinase 1 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| LIM domain kinase 2 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Macrophage colony-stimulating factor 1 receptor | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Macrophage-stimulating protein receptor | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| MAP kinase-activated protein kinase 2 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| MAP kinase-activated protein kinase 5 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| MAP kinase-interacting serine/threonine-protein kinase 1 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| MAP kinase-interacting serine/threonine-protein kinase 2 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| MAP/microtubule affinity-regulating kinase 3 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| MAP/microtubule affinity-regulating kinase 4 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Mast/stem cell growth factor receptor Kit | Homo sapiens (human) | Kd | 10.0000 | 15 | 15 |
| Maternal embryonic leucine zipper kinase | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Megakaryocyte-associated tyrosine-protein kinase | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Membrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinase | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Microtubule-associated serine/threonine-protein kinase 1 | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Misshapen-like kinase 1 | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Mitogen-activated protein kinase 1 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Mitogen-activated protein kinase 10 | Homo sapiens (human) | Kd | 0.0383 | 3 | 3 |
| Mitogen-activated protein kinase 11 | Homo sapiens (human) | EC50 | 0.0600 | 1 | 1 |
| Mitogen-activated protein kinase 11 | Homo sapiens (human) | Kd | 0.1000 | 4 | 4 |
| Mitogen-activated protein kinase 12 | Homo sapiens (human) | EC50 | 0.0600 | 1 | 1 |
| Mitogen-activated protein kinase 12 | Homo sapiens (human) | Kd | 1.1775 | 4 | 4 |
| Mitogen-activated protein kinase 13 | Homo sapiens (human) | EC50 | 0.0600 | 1 | 1 |
| Mitogen-activated protein kinase 13 | Homo sapiens (human) | Kd | 5.0050 | 2 | 2 |
| Mitogen-activated protein kinase 14 | Homo sapiens (human) | EC50 | 0.0600 | 2 | 2 |
| Mitogen-activated protein kinase 14 | Homo sapiens (human) | Kd | 0.0128 | 6 | 6 |
| Mitogen-activated protein kinase 14 | Mus musculus (house mouse) | Kd | 0.0200 | 2 | 2 |
| Mitogen-activated protein kinase 15 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Mitogen-activated protein kinase 3 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Mitogen-activated protein kinase 4 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Mitogen-activated protein kinase 6 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Mitogen-activated protein kinase 7 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Mitogen-activated protein kinase 8 | Homo sapiens (human) | Kd | 1.1333 | 3 | 3 |
| Mitogen-activated protein kinase 9 | Homo sapiens (human) | Kd | 0.1183 | 3 | 3 |
| Mitogen-activated protein kinase kinase kinase 1 | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Mitogen-activated protein kinase kinase kinase 10 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Mitogen-activated protein kinase kinase kinase 11 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Mitogen-activated protein kinase kinase kinase 12 | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Mitogen-activated protein kinase kinase kinase 13 | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Mitogen-activated protein kinase kinase kinase 15 | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Mitogen-activated protein kinase kinase kinase 19 | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Mitogen-activated protein kinase kinase kinase 2 | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Mitogen-activated protein kinase kinase kinase 20 | Homo sapiens (human) | Kd | 4.4000 | 2 | 2 |
| Mitogen-activated protein kinase kinase kinase 3 | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Mitogen-activated protein kinase kinase kinase 4 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Mitogen-activated protein kinase kinase kinase 5 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Mitogen-activated protein kinase kinase kinase 6 | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Mitogen-activated protein kinase kinase kinase 7 | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Mitogen-activated protein kinase kinase kinase 9 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Mitogen-activated protein kinase kinase kinase kinase 1 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Mitogen-activated protein kinase kinase kinase kinase 2 | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Mitogen-activated protein kinase kinase kinase kinase 3 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Mitogen-activated protein kinase kinase kinase kinase 4 | Homo sapiens (human) | Kd | 3.7000 | 2 | 2 |
| Mitogen-activated protein kinase kinase kinase kinase 5 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Muscle, skeletal receptor tyrosine-protein kinase | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Myosin light chain kinase 2, skeletal/cardiac muscle | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Myosin light chain kinase 3 | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Myosin light chain kinase family member 4 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Myosin light chain kinase, smooth muscle | Gallus gallus (chicken) | Kd | 10.0000 | 1 | 1 |
| Myosin light chain kinase, smooth muscle | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Myosin-IIIa | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Myosin-IIIb | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Myotonin-protein kinase | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| NAD kinase | Homo sapiens (human) | Kd | 1.7800 | 1 | 1 |
| Non-receptor tyrosine-protein kinase TNK1 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Non-receptor tyrosine-protein kinase TYK2 | Homo sapiens (human) | Kd | 7.3333 | 3 | 3 |
| NT-3 growth factor receptor | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| NUAK family SNF1-like kinase 1 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| NUAK family SNF1-like kinase 2 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Nuclear receptor subfamily 4 group A member 1 | Homo sapiens (human) | Kd | 0.3000 | 3 | 3 |
| Peripheral plasma membrane protein CASK | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Phosphatidylinositol 4-kinase beta | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Phosphatidylinositol 4-phosphate 3-kinase C2 domain-containing subunit beta | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Phosphatidylinositol 4-phosphate 3-kinase C2 domain-containing subunit gamma | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Phosphatidylinositol 4-phosphate 5-kinase type-1 alpha | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Phosphatidylinositol 4-phosphate 5-kinase type-1 gamma | Homo sapiens (human) | Kd | 2.6000 | 1 | 1 |
| Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform | Homo sapiens (human) | Kd | 10.0000 | 12 | 12 |
| Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Phosphatidylinositol 5-phosphate 4-kinase type-2 beta | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Phosphatidylinositol 5-phosphate 4-kinase type-2 gamma | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Phosphorylase b kinase gamma catalytic chain, liver/testis isoform | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Phosphorylase b kinase gamma catalytic chain, skeletal muscle/heart isoform | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Platelet-derived growth factor receptor alpha | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Platelet-derived growth factor receptor beta | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Polycomb protein EED | Homo sapiens (human) | Kd | 15.1000 | 1 | 1 |
| POsterior Segregation | Caenorhabditis elegans | EC50 | 5.8920 | 1 | 1 |
| Prostaglandin G/H synthase 2 | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Protein kinase C delta type | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Protein kinase C epsilon type | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Protein kinase C eta type | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Protein kinase C iota type | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Protein kinase C theta type | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Protein-tyrosine kinase 2-beta | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Protein-tyrosine kinase 6 | Homo sapiens (human) | Kd | 5.6000 | 3 | 3 |
| Proto-oncogene tyrosine-protein kinase receptor Ret | Homo sapiens (human) | Kd | 10.0000 | 6 | 6 |
| Proto-oncogene tyrosine-protein kinase ROS | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Proto-oncogene tyrosine-protein kinase Src | Homo sapiens (human) | Kd | 5.3000 | 2 | 2 |
| RAC-alpha serine/threonine-protein kinase | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| RAC-beta serine/threonine-protein kinase | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| RAC-gamma serine/threonine-protein kinase | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| RAF proto-oncogene serine/threonine-protein kinase | Homo sapiens (human) | Kd | 0.9800 | 2 | 2 |
| Receptor tyrosine-protein kinase erbB-2 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Receptor tyrosine-protein kinase erbB-3 | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Receptor tyrosine-protein kinase erbB-4 | Homo sapiens (human) | Kd | 4.8000 | 1 | 1 |
| Receptor-interacting serine/threonine-protein kinase 1 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Receptor-interacting serine/threonine-protein kinase 2 | Homo sapiens (human) | Kd | 0.7160 | 3 | 3 |
| Receptor-interacting serine/threonine-protein kinase 4 | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Receptor-type tyrosine-protein kinase FLT3 | Homo sapiens (human) | Kd | 10.0000 | 12 | 12 |
| recombinase A | Mycobacterium tuberculosis H37Rv | EC50 | 87.1000 | 2 | 2 |
| Rho-associated protein kinase 1 | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Rho-associated protein kinase 2 | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Rhodopsin kinase GRK1 | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Rhodopsin kinase GRK7 | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Ribosomal protein S6 kinase alpha-1 | Homo sapiens (human) | Kd | 5.1600 | 4 | 4 |
| Ribosomal protein S6 kinase alpha-2 | Homo sapiens (human) | Kd | 10.0000 | 4 | 4 |
| Ribosomal protein S6 kinase alpha-3 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Ribosomal protein S6 kinase alpha-4 | Homo sapiens (human) | Kd | 10.0000 | 4 | 4 |
| Ribosomal protein S6 kinase alpha-5 | Homo sapiens (human) | Kd | 10.0000 | 4 | 4 |
| Ribosomal protein S6 kinase alpha-6 | Homo sapiens (human) | Kd | 5.1250 | 4 | 4 |
| Ribosomal protein S6 kinase beta-1 | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Serine/threonine-protein kinase 10 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Serine/threonine-protein kinase 16 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Serine/threonine-protein kinase 17A | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Serine/threonine-protein kinase 17B | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Serine/threonine-protein kinase 24 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Serine/threonine-protein kinase 25 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Serine/threonine-protein kinase 26 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Serine/threonine-protein kinase 3 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Serine/threonine-protein kinase 32A | Homo sapiens (human) | Kd | 1.3000 | 1 | 1 |
| Serine/threonine-protein kinase 32B | Homo sapiens (human) | Kd | 2.1000 | 2 | 2 |
| Serine/threonine-protein kinase 32C | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Serine/threonine-protein kinase 33 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Serine/threonine-protein kinase 35 | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Serine/threonine-protein kinase 36 | Homo sapiens (human) | Kd | 1.1533 | 3 | 3 |
| Serine/threonine-protein kinase 38 | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Serine/threonine-protein kinase 38-like | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Serine/threonine-protein kinase 4 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Serine/threonine-protein kinase B-raf | Homo sapiens (human) | Kd | 0.6200 | 4 | 4 |
| Serine/threonine-protein kinase BRSK1 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Serine/threonine-protein kinase BRSK2 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Serine/threonine-protein kinase Chk1 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Serine/threonine-protein kinase Chk2 | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Serine/threonine-protein kinase D1 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Serine/threonine-protein kinase D2 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Serine/threonine-protein kinase D3 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Serine/threonine-protein kinase DCLK1 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Serine/threonine-protein kinase DCLK2 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Serine/threonine-protein kinase DCLK3 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Serine/threonine-protein kinase ICK | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Serine/threonine-protein kinase LATS1 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Serine/threonine-protein kinase LATS2 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Serine/threonine-protein kinase MAK | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Serine/threonine-protein kinase MARK1 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Serine/threonine-protein kinase MARK2 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Serine/threonine-protein kinase MRCK alpha | Homo sapiens (human) | Kd | 6.2000 | 2 | 2 |
| Serine/threonine-protein kinase MRCK beta | Homo sapiens (human) | Kd | 2.7000 | 2 | 2 |
| Serine/threonine-protein kinase MRCK gamma | Homo sapiens (human) | Kd | 0.4000 | 2 | 2 |
| Serine/threonine-protein kinase mTOR | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Serine/threonine-protein kinase N1 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Serine/threonine-protein kinase N2 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Serine/threonine-protein kinase Nek1 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Serine/threonine-protein kinase Nek11 | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Serine/threonine-protein kinase Nek2 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Serine/threonine-protein kinase Nek3 | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Serine/threonine-protein kinase Nek4 | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Serine/threonine-protein kinase Nek5 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Serine/threonine-protein kinase Nek6 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Serine/threonine-protein kinase Nek7 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Serine/threonine-protein kinase Nek9 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Serine/threonine-protein kinase NIM1 | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Serine/threonine-protein kinase NLK | Homo sapiens (human) | Kd | 0.0250 | 2 | 2 |
| Serine/threonine-protein kinase OSR1 | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Serine/threonine-protein kinase PAK 1 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Serine/threonine-protein kinase PAK 2 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Serine/threonine-protein kinase PAK 3 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Serine/threonine-protein kinase PAK 4 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Serine/threonine-protein kinase PAK 5 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Serine/threonine-protein kinase PAK 6 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Serine/threonine-protein kinase pim-1 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Serine/threonine-protein kinase pim-2 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Serine/threonine-protein kinase pim-3 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Serine/threonine-protein kinase PknB | Mycobacterium tuberculosis H37Rv | Kd | 10.0000 | 1 | 1 |
| Serine/threonine-protein kinase PLK1 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Serine/threonine-protein kinase PLK2 | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Serine/threonine-protein kinase PLK3 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Serine/threonine-protein kinase PLK4 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Serine/threonine-protein kinase PRP4 homolog | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Serine/threonine-protein kinase receptor R3 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Serine/threonine-protein kinase RIO1 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Serine/threonine-protein kinase RIO2 | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Serine/threonine-protein kinase RIO3 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Serine/threonine-protein kinase SBK1 | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Serine/threonine-protein kinase Sgk3 | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Serine/threonine-protein kinase SIK1 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Serine/threonine-protein kinase SIK2 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Serine/threonine-protein kinase SIK3 | Homo sapiens (human) | Kd | 3.9000 | 1 | 1 |
| Serine/threonine-protein kinase STK11 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Serine/threonine-protein kinase TAO1 | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Serine/threonine-protein kinase TAO2 | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Serine/threonine-protein kinase TAO3 | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Serine/threonine-protein kinase TBK1 | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Serine/threonine-protein kinase TNNI3K | Homo sapiens (human) | Kd | 3.5000 | 2 | 2 |
| Serine/threonine-protein kinase tousled-like 1 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Serine/threonine-protein kinase tousled-like 2 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Serine/threonine-protein kinase ULK1 | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Serine/threonine-protein kinase ULK2 | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Serine/threonine-protein kinase ULK3 | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Serine/threonine-protein kinase VRK2 | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Serine/threonine-protein kinase/endoribonuclease IRE1 | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Signal transducer and activator of transcription 1-alpha/beta | Homo sapiens (human) | Kd | 0.7000 | 1 | 1 |
| SNF-related serine/threonine-protein kinase | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Sodium-dependent noradrenaline transporter | Homo sapiens (human) | EC50 | 0.7270 | 1 | 1 |
| SRSF protein kinase 1 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| SRSF protein kinase 2 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| SRSF protein kinase 3 | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| STE20-like serine/threonine-protein kinase | Homo sapiens (human) | Kd | 4.0000 | 3 | 3 |
| STE20/SPS1-related proline-alanine-rich protein kinase | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Testis-specific serine/threonine-protein kinase 1 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| TGF-beta receptor type-1 | Homo sapiens (human) | Kd | 7.1000 | 2 | 2 |
| TGF-beta receptor type-2 | Homo sapiens (human) | Kd | 1.8000 | 2 | 2 |
| TRAF2 and NCK-interacting protein kinase | Homo sapiens (human) | Kd | 1.0467 | 3 | 3 |
| Transient receptor potential cation channel subfamily M member 6 | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Transthyretin | Homo sapiens (human) | Kd | 0.4000 | 2 | 2 |
| Tubulin alpha-1A chain | Rattus norvegicus (Norway rat) | Kd | 10.0000 | 1 | 1 |
| Tyrosine-protein kinase ABL1 | Homo sapiens (human) | Kd | 9.3864 | 22 | 22 |
| Tyrosine-protein kinase ABL2 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Tyrosine-protein kinase Blk | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Tyrosine-protein kinase BTK | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Tyrosine-protein kinase CSK | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Tyrosine-protein kinase Fer | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Tyrosine-protein kinase Fes/Fps | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Tyrosine-protein kinase Fgr | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Tyrosine-protein kinase FRK | Homo sapiens (human) | Kd | 2.6667 | 3 | 3 |
| Tyrosine-protein kinase Fyn | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Tyrosine-protein kinase HCK | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Tyrosine-protein kinase ITK/TSK | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Tyrosine-protein kinase JAK1 | Homo sapiens (human) | Kd | 10.0000 | 3 | 3 |
| Tyrosine-protein kinase JAK2 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Tyrosine-protein kinase JAK3 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Tyrosine-protein kinase Lck | Homo sapiens (human) | Kd | 2.8000 | 2 | 2 |
| Tyrosine-protein kinase Lyn | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Tyrosine-protein kinase Mer | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Tyrosine-protein kinase receptor Tie-1 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Tyrosine-protein kinase receptor TYRO3 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Tyrosine-protein kinase receptor UFO | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Tyrosine-protein kinase Srms | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Tyrosine-protein kinase SYK | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Tyrosine-protein kinase Tec | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Tyrosine-protein kinase TXK | Homo sapiens (human) | Kd | 4.5000 | 2 | 2 |
| Tyrosine-protein kinase Yes | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Tyrosine-protein kinase ZAP-70 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Tyrosine-protein phosphatase non-receptor type 1 | Homo sapiens (human) | Kd | 6.0800 | 1 | 1 |
| Uncharacterized serine/threonine-protein kinase SBK3 | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Vascular endothelial growth factor receptor 1 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Vascular endothelial growth factor receptor 2 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Vascular endothelial growth factor receptor 3 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Wee1-like protein kinase | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Wee1-like protein kinase 2 | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Zinc finger protein mex-5 | Caenorhabditis elegans | EC50 | 0.7270 | 1 | 1 |