Assay ID | Title | Year | Journal | Article |
AID1105460 | Antifungal activity against Aspergillus fumigatus IPP 210 after 72 hr by broth microdilution method | 2013 | International journal of molecular sciences, Jan-10, Volume: 14, Issue:1
| Synthesis, structure-activity relationships (SAR) and in silico studies of coumarin derivatives with antifungal activity. |
AID1348313 | Inhibition of human carbonic anhydrase 9 incubated for 15 mins prior to testing by stopped-flow CO2 hydration assay | 2018 | European journal of medicinal chemistry, Jan-01, Volume: 143 | Inhibitory effects and structural insights for a novel series of coumarin-based compounds that selectively target human CA IX and CA XII carbonic anhydrases. |
AID1138894 | Antiasthamic activity in Wistar rat tracheal ring assessed as reversal of carbachol-induced contraction | 2014 | European journal of medicinal chemistry, Apr-22, Volume: 77 | Semisynthesis, ex vivo evaluation, and SAR studies of coumarin derivatives as potential antiasthmatic drugs. |
AID1348314 | Inhibition of human carbonic anhydrase 12 incubated for 15 mins prior to testing by stopped-flow CO2 hydration assay | 2018 | European journal of medicinal chemistry, Jan-01, Volume: 143 | Inhibitory effects and structural insights for a novel series of coumarin-based compounds that selectively target human CA IX and CA XII carbonic anhydrases. |
AID1105458 | Antifungal activity against Aspergillus fumigatus ATCC 40640 after 72 hr by broth microdilution method | 2013 | International journal of molecular sciences, Jan-10, Volume: 14, Issue:1
| Synthesis, structure-activity relationships (SAR) and in silico studies of coumarin derivatives with antifungal activity. |
AID1348312 | Inhibition of human carbonic anhydrase 2 incubated for 15 mins prior to testing by stopped-flow CO2 hydration assay | 2018 | European journal of medicinal chemistry, Jan-01, Volume: 143 | Inhibitory effects and structural insights for a novel series of coumarin-based compounds that selectively target human CA IX and CA XII carbonic anhydrases. |
AID1105461 | Antifungal activity against Aspergillus fumigatus ATCC 16913 after 72 hr by broth microdilution method | 2013 | International journal of molecular sciences, Jan-10, Volume: 14, Issue:1
| Synthesis, structure-activity relationships (SAR) and in silico studies of coumarin derivatives with antifungal activity. |
AID1105454 | Antifungal activity against Aspergillus flavus LM 26 after 72 hr by broth microdilution method | 2013 | International journal of molecular sciences, Jan-10, Volume: 14, Issue:1
| Synthesis, structure-activity relationships (SAR) and in silico studies of coumarin derivatives with antifungal activity. |
AID1105459 | Antifungal activity against Aspergillus fumigatus ATCC 46913 after 72 hr by broth microdilution method | 2013 | International journal of molecular sciences, Jan-10, Volume: 14, Issue:1
| Synthesis, structure-activity relationships (SAR) and in silico studies of coumarin derivatives with antifungal activity. |
AID1348311 | Inhibition of human carbonic anhydrase 1 incubated for 15 mins prior to testing by stopped-flow CO2 hydration assay | 2018 | European journal of medicinal chemistry, Jan-01, Volume: 143 | Inhibitory effects and structural insights for a novel series of coumarin-based compounds that selectively target human CA IX and CA XII carbonic anhydrases. |
AID1105456 | Antifungal activity against Aspergillus flavus ATCC 16013 after 72 hr by broth microdilution method | 2013 | International journal of molecular sciences, Jan-10, Volume: 14, Issue:1
| Synthesis, structure-activity relationships (SAR) and in silico studies of coumarin derivatives with antifungal activity. |
AID1105455 | Antifungal activity against Aspergillus flavus LM 210 after 72 hr by broth microdilution method | 2013 | International journal of molecular sciences, Jan-10, Volume: 14, Issue:1
| Synthesis, structure-activity relationships (SAR) and in silico studies of coumarin derivatives with antifungal activity. |
AID1138893 | Antiasthamic activity in Wistar rat tracheal ring assessed as reversal of carbachol-induced contraction at 0.1 to 500 uM relative to control | 2014 | European journal of medicinal chemistry, Apr-22, Volume: 77 | Semisynthesis, ex vivo evaluation, and SAR studies of coumarin derivatives as potential antiasthmatic drugs. |
AID1105457 | Antifungal activity against Aspergillus flavus LM 247 after 72 hr by broth microdilution method | 2013 | International journal of molecular sciences, Jan-10, Volume: 14, Issue:1
| Synthesis, structure-activity relationships (SAR) and in silico studies of coumarin derivatives with antifungal activity. |
AID373105 | Antiamnesic activity against Entamoeba histolytica HM1:IMSS after 72 hrs by microdilution method | 2009 | European journal of medicinal chemistry, May, Volume: 44, Issue:5
| Antiamoebic coumarins from the root bark of Adina cordifolia and their new thiosemicarbazone derivatives. |
AID588501 | High-throughput multiplex microsphere screening for inhibitors of toxin protease, specifically Lethal Factor Protease, MLPCN compound set | 2010 | Current protocols in cytometry, Oct, Volume: Chapter 13 | Microsphere-based flow cytometry protease assays for use in protease activity detection and high-throughput screening. |
AID588501 | High-throughput multiplex microsphere screening for inhibitors of toxin protease, specifically Lethal Factor Protease, MLPCN compound set | 2006 | Cytometry. Part A : the journal of the International Society for Analytical Cytology, May, Volume: 69, Issue:5
| Microsphere-based protease assays and screening application for lethal factor and factor Xa. |
AID588501 | High-throughput multiplex microsphere screening for inhibitors of toxin protease, specifically Lethal Factor Protease, MLPCN compound set | 2010 | Assay and drug development technologies, Feb, Volume: 8, Issue:1
| High-throughput multiplex flow cytometry screening for botulinum neurotoxin type a light chain protease inhibitors. |
AID1745845 | Primary qHTS for Inhibitors of ATXN expression | | | |
AID504810 | Antagonists of the Thyroid Stimulating Hormone Receptor: HTS campaign | 2010 | Endocrinology, Jul, Volume: 151, Issue:7
| A small molecule inverse agonist for the human thyroid-stimulating hormone receptor. |
AID588499 | High-throughput multiplex microsphere screening for inhibitors of toxin protease, specifically Botulinum neurotoxin light chain A protease, MLPCN compound set | 2010 | Current protocols in cytometry, Oct, Volume: Chapter 13 | Microsphere-based flow cytometry protease assays for use in protease activity detection and high-throughput screening. |
AID588499 | High-throughput multiplex microsphere screening for inhibitors of toxin protease, specifically Botulinum neurotoxin light chain A protease, MLPCN compound set | 2006 | Cytometry. Part A : the journal of the International Society for Analytical Cytology, May, Volume: 69, Issue:5
| Microsphere-based protease assays and screening application for lethal factor and factor Xa. |
AID588499 | High-throughput multiplex microsphere screening for inhibitors of toxin protease, specifically Botulinum neurotoxin light chain A protease, MLPCN compound set | 2010 | Assay and drug development technologies, Feb, Volume: 8, Issue:1
| High-throughput multiplex flow cytometry screening for botulinum neurotoxin type a light chain protease inhibitors. |
AID504812 | Inverse Agonists of the Thyroid Stimulating Hormone Receptor: HTS campaign | 2010 | Endocrinology, Jul, Volume: 151, Issue:7
| A small molecule inverse agonist for the human thyroid-stimulating hormone receptor. |
AID588497 | High-throughput multiplex microsphere screening for inhibitors of toxin protease, specifically Botulinum neurotoxin light chain F protease, MLPCN compound set | 2010 | Current protocols in cytometry, Oct, Volume: Chapter 13 | Microsphere-based flow cytometry protease assays for use in protease activity detection and high-throughput screening. |
AID588497 | High-throughput multiplex microsphere screening for inhibitors of toxin protease, specifically Botulinum neurotoxin light chain F protease, MLPCN compound set | 2006 | Cytometry. Part A : the journal of the International Society for Analytical Cytology, May, Volume: 69, Issue:5
| Microsphere-based protease assays and screening application for lethal factor and factor Xa. |
AID588497 | High-throughput multiplex microsphere screening for inhibitors of toxin protease, specifically Botulinum neurotoxin light chain F protease, MLPCN compound set | 2010 | Assay and drug development technologies, Feb, Volume: 8, Issue:1
| High-throughput multiplex flow cytometry screening for botulinum neurotoxin type a light chain protease inhibitors. |
AID651635 | Viability Counterscreen for Primary qHTS for Inhibitors of ATXN expression | | | |
[information is prepared from bioassay data collected from National Library of Medicine (NLM), extracted Dec-2023] |