Any compound which can be used to treat or alleviate the symptoms of dyskinesia.
| Protein | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Drugs |
|---|
| 15-hydroxyprostaglandin dehydrogenase [NAD(+)] isoform 1 | Homo sapiens (human) | Potency | 3.9811 | 1 | 1 |
| 15-lipoxygenase, partial | Homo sapiens (human) | Potency | 26.9262 | 1 | 3 |
| 67.9K protein | Vaccinia virus | Potency | 28.1838 | 1 | 1 |
| acetylcholinesterase | Homo sapiens (human) | Potency | 45.6170 | 3 | 5 |
| activating transcription factor 6 | Homo sapiens (human) | Potency | 58.2929 | 2 | 2 |
| aldehyde dehydrogenase 1 family, member A1 | Homo sapiens (human) | Potency | 32.0272 | 1 | 3 |
| apical membrane antigen 1, AMA1 | Plasmodium falciparum 3D7 | Potency | 22.8741 | 1 | 2 |
| AR protein | Homo sapiens (human) | Potency | 20.5956 | 9 | 38 |
| aryl hydrocarbon receptor | Homo sapiens (human) | Potency | 4.3080 | 2 | 2 |
| arylsulfatase A | Homo sapiens (human) | Potency | 15.3451 | 1 | 7 |
| ATAD5 protein, partial | Homo sapiens (human) | Potency | 21.6375 | 3 | 7 |
| Ataxin-2 | Homo sapiens (human) | Potency | 26.5871 | 2 | 10 |
| ATP-dependent phosphofructokinase | Trypanosoma brucei brucei TREU927 | Potency | 16.5281 | 2 | 7 |
| ATPase family AAA domain-containing protein 5 | Homo sapiens (human) | Potency | 21.8730 | 2 | 8 |
| atrial natriuretic peptide receptor 1 precursor | Homo sapiens (human) | Potency | 21.4728 | 1 | 2 |
| Bloom syndrome protein isoform 1 | Homo sapiens (human) | Potency | 12.3079 | 3 | 3 |
| bromodomain adjacent to zinc finger domain 2B | Homo sapiens (human) | Potency | 22.3872 | 1 | 1 |
| caspase 7, apoptosis-related cysteine protease | Homo sapiens (human) | Potency | 49.7016 | 1 | 3 |
| caspase-3 | Cricetulus griseus (Chinese hamster) | Potency | 32.0647 | 1 | 2 |
| caspase-3 | Homo sapiens (human) | Potency | 49.7016 | 1 | 3 |
| Caspase-7 | Cricetulus griseus (Chinese hamster) | Potency | 32.0647 | 1 | 2 |
| Cellular tumor antigen p53 | Homo sapiens (human) | Potency | 39.4887 | 3 | 10 |
| cellular tumor antigen p53 isoform a | Homo sapiens (human) | Potency | 16.9971 | 2 | 5 |
| Chain A, 2-oxoglutarate Oxygenase | Homo sapiens (human) | Potency | 29.8760 | 1 | 4 |
| Chain A, ATP-DEPENDENT DNA HELICASE Q1 | Homo sapiens (human) | Potency | 12.5893 | 1 | 1 |
| Chain A, Beta-lactamase | Escherichia coli K-12 | Potency | 70.7946 | 1 | 1 |
| Chain A, Ferritin light chain | Equus caballus (horse) | Potency | 3.1623 | 1 | 1 |
| Chain A, HADH2 protein | Homo sapiens (human) | Potency | 7.3590 | 2 | 4 |
| Chain A, JmjC domain-containing histone demethylation protein 3A | Homo sapiens (human) | Potency | 39.8107 | 1 | 2 |
| Chain A, MAJOR APURINIC/APYRIMIDINIC ENDONUCLEASE | Homo sapiens (human) | Potency | 8.5072 | 2 | 4 |
| Chain A, Putative fructose-1,6-bisphosphate aldolase | Giardia intestinalis | Potency | 22.3342 | 1 | 1 |
| Chain A, TYROSYL-DNA PHOSPHODIESTERASE | Homo sapiens (human) | Potency | 11.3737 | 1 | 7 |
| Chain B, HADH2 protein | Homo sapiens (human) | Potency | 7.3590 | 2 | 4 |
| chromobox protein homolog 1 | Homo sapiens (human) | Potency | 37.2415 | 2 | 7 |
| cytochrome P450 2C19 precursor | Homo sapiens (human) | Potency | 18.9149 | 1 | 4 |
| cytochrome P450 2C9 precursor | Homo sapiens (human) | Potency | 34.3521 | 1 | 3 |
| cytochrome P450 2C9, partial | Homo sapiens (human) | Potency | 11.4410 | 1 | 3 |
| cytochrome P450 2D6 | Homo sapiens (human) | Potency | 8.9110 | 1 | 6 |
| cytochrome P450 2D6 isoform 1 | Homo sapiens (human) | Potency | 8.0727 | 1 | 9 |
| cytochrome P450 3A4 isoform 1 | Homo sapiens (human) | Potency | 3.6128 | 2 | 12 |
| cytochrome P450 family 3 subfamily A polypeptide 4 | Homo sapiens (human) | Potency | 4.8282 | 2 | 7 |
| cytochrome P450, family 19, subfamily A, polypeptide 1, isoform CRA_a | Homo sapiens (human) | Potency | 31.3262 | 1 | 3 |
| D(1A) dopamine receptor | Homo sapiens (human) | Potency | 6.4288 | 3 | 7 |
| D(1A) dopamine receptor | Sus scrofa (pig) | Potency | 19.8812 | 1 | 2 |
| Disintegrin and metalloproteinase domain-containing protein 17 | Homo sapiens (human) | Potency | 2.5119 | 1 | 1 |
| DNA polymerase eta isoform 1 | Homo sapiens (human) | Potency | 19.5957 | 2 | 2 |
| DNA polymerase III, partial | Bacillus subtilis | Potency | 23.7781 | 1 | 1 |
| DNA polymerase iota isoform a (long) | Homo sapiens (human) | Potency | 16.9549 | 2 | 3 |
| DNA polymerase kappa isoform 1 | Homo sapiens (human) | Potency | 10.1286 | 1 | 7 |
| dopamine D1 receptor | Homo sapiens (human) | Potency | 5.7319 | 1 | 2 |
| endonuclease IV | Escherichia coli | Potency | 10.0000 | 1 | 1 |
| estrogen nuclear receptor alpha | Homo sapiens (human) | Potency | 28.8563 | 10 | 38 |
| estrogen receptor 2 (ER beta) | Homo sapiens (human) | Potency | 18.6330 | 1 | 3 |
| estrogen-related nuclear receptor alpha | Homo sapiens (human) | Potency | 28.2060 | 9 | 28 |
| euchromatic histone-lysine N-methyltransferase 2 | Homo sapiens (human) | Potency | 12.0090 | 1 | 13 |
| EWS/FLI fusion protein | Homo sapiens (human) | Potency | 22.5082 | 4 | 8 |
| farnesoid X nuclear receptor | Homo sapiens (human) | Potency | 29.3379 | 3 | 8 |
| flap endonuclease 1 | Homo sapiens (human) | Potency | 20.6366 | 3 | 7 |
| Fumarate hydratase | Homo sapiens (human) | Potency | 32.2233 | 1 | 3 |
| G | Vesicular stomatitis virus | Potency | 11.4410 | 1 | 3 |
| GABA theta subunit | Rattus norvegicus (Norway rat) | Potency | 3.6128 | 1 | 6 |
| GALC protein | Homo sapiens (human) | Potency | 0.7079 | 1 | 1 |
| Gamma-aminobutyric acid receptor subunit alpha-1 | Rattus norvegicus (Norway rat) | Potency | 3.6128 | 1 | 6 |
| Gamma-aminobutyric acid receptor subunit alpha-2 | Rattus norvegicus (Norway rat) | Potency | 3.6128 | 1 | 6 |
| Gamma-aminobutyric acid receptor subunit alpha-3 | Rattus norvegicus (Norway rat) | Potency | 3.6128 | 1 | 6 |
| Gamma-aminobutyric acid receptor subunit alpha-4 | Rattus norvegicus (Norway rat) | Potency | 3.6128 | 1 | 6 |
| Gamma-aminobutyric acid receptor subunit alpha-5 | Rattus norvegicus (Norway rat) | Potency | 3.6128 | 1 | 6 |
| Gamma-aminobutyric acid receptor subunit alpha-6 | Rattus norvegicus (Norway rat) | Potency | 3.6128 | 1 | 6 |
| Gamma-aminobutyric acid receptor subunit beta-1 | Rattus norvegicus (Norway rat) | Potency | 3.6128 | 1 | 6 |
| Gamma-aminobutyric acid receptor subunit beta-2 | Rattus norvegicus (Norway rat) | Potency | 3.6128 | 1 | 6 |
| Gamma-aminobutyric acid receptor subunit beta-3 | Rattus norvegicus (Norway rat) | Potency | 3.6128 | 1 | 6 |
| Gamma-aminobutyric acid receptor subunit delta | Rattus norvegicus (Norway rat) | Potency | 3.6128 | 1 | 6 |
| Gamma-aminobutyric acid receptor subunit epsilon | Rattus norvegicus (Norway rat) | Potency | 3.6128 | 1 | 6 |
| Gamma-aminobutyric acid receptor subunit gamma-1 | Rattus norvegicus (Norway rat) | Potency | 3.6128 | 1 | 6 |
| Gamma-aminobutyric acid receptor subunit gamma-2 | Rattus norvegicus (Norway rat) | Potency | 3.6128 | 1 | 6 |
| Gamma-aminobutyric acid receptor subunit gamma-3 | Rattus norvegicus (Norway rat) | Potency | 3.6128 | 1 | 6 |
| Gamma-aminobutyric acid receptor subunit pi | Rattus norvegicus (Norway rat) | Potency | 3.6128 | 1 | 6 |
| geminin | Homo sapiens (human) | Potency | 12.8341 | 3 | 10 |
| GLI family zinc finger 3 | Homo sapiens (human) | Potency | 16.9144 | 2 | 8 |
| glp-1 receptor, partial | Homo sapiens (human) | Potency | 18.5482 | 1 | 2 |
| GLS protein | Homo sapiens (human) | Potency | 21.2529 | 2 | 10 |
| glucocerebrosidase | Homo sapiens (human) | Potency | 0.7943 | 1 | 1 |
| glucocorticoid receptor [Homo sapiens] | Homo sapiens (human) | Potency | 21.7854 | 3 | 14 |
| glucokinase regulatory protein | Homo sapiens (human) | Potency | 5.0119 | 1 | 1 |
| Glutamate receptor 2 | Rattus norvegicus (Norway rat) | Potency | 37.8552 | 1 | 4 |
| heat shock 70kDa protein 5 (glucose-regulated protein, 78kDa) | Homo sapiens (human) | Potency | 58.4789 | 1 | 1 |
| heat shock protein beta-1 | Homo sapiens (human) | Potency | 34.5200 | 2 | 6 |
| hexokinase-4 isoform 1 | Homo sapiens (human) | Potency | 5.0119 | 1 | 1 |
| Histamine H2 receptor | Cavia porcellus (domestic guinea pig) | Potency | 21.3782 | 2 | 19 |
| histone acetyltransferase KAT2A isoform 1 | Homo sapiens (human) | Potency | 35.4813 | 1 | 1 |
| histone deacetylase 9 isoform 3 | Homo sapiens (human) | Potency | 25.1566 | 2 | 2 |
| Histone H2A.x | Cricetulus griseus (Chinese hamster) | Potency | 44.2604 | 2 | 4 |
| histone-lysine N-methyltransferase 2A isoform 2 precursor | Homo sapiens (human) | Potency | 100.0000 | 1 | 1 |
| HLA class I histocompatibility antigen, B alpha chain | Homo sapiens (human) | Potency | 11.4410 | 1 | 3 |
| huntingtin isoform 2 | Homo sapiens (human) | Potency | 28.9372 | 1 | 3 |
| hypoxia-inducible factor 1 alpha subunit | Homo sapiens (human) | Potency | 21.7615 | 2 | 5 |
| hypoxia-inducible factor 1, alpha subunit (basic helix-loop-helix transcription factor) | Homo sapiens (human) | Potency | 4.6957 | 2 | 8 |
| IDH1 | Homo sapiens (human) | Potency | 16.3601 | 1 | 1 |
| importin subunit beta-1 isoform 1 | Homo sapiens (human) | Potency | 56.2341 | 1 | 1 |
| Inositol hexakisphosphate kinase 1 | Homo sapiens (human) | Potency | 11.4410 | 1 | 6 |
| Inositol monophosphatase 1 | Rattus norvegicus (Norway rat) | Potency | 5.0040 | 2 | 2 |
| Integrin alpha-IIb | Homo sapiens (human) | Potency | 25.1189 | 1 | 2 |
| Integrin beta-3 | Homo sapiens (human) | Potency | 25.1189 | 1 | 2 |
| Interferon beta | Homo sapiens (human) | Potency | 13.6993 | 3 | 7 |
| lamin isoform A-delta10 | Homo sapiens (human) | Potency | 26.2641 | 2 | 9 |
| lethal factor (plasmid) | Bacillus anthracis str. A2012 | Potency | 24.5911 | 1 | 4 |
| Luciferase | Photinus pyralis (common eastern firefly) | Potency | 17.0460 | 1 | 4 |
| M-phase phosphoprotein 8 | Homo sapiens (human) | Potency | 18.8620 | 1 | 3 |
| Microtubule-associated protein tau | Homo sapiens (human) | Potency | 22.8300 | 2 | 8 |
| mitogen-activated protein kinase 1 | Homo sapiens (human) | Potency | 26.9752 | 2 | 7 |
| muscarinic acetylcholine receptor M1 | Rattus norvegicus (Norway rat) | Potency | 8.8763 | 2 | 9 |
| neuropeptide S receptor isoform A | Homo sapiens (human) | Potency | 9.4494 | 1 | 2 |
| NFKB1 protein, partial | Homo sapiens (human) | Potency | 14.2328 | 2 | 4 |
| nonstructural protein 1 | Influenza A virus (A/WSN/1933(H1N1)) | Potency | 1.7783 | 1 | 1 |
| nuclear factor erythroid 2-related factor 2 isoform 1 | Homo sapiens (human) | Potency | 22.4832 | 4 | 13 |
| nuclear factor erythroid 2-related factor 2 isoform 2 | Homo sapiens (human) | Potency | 18.3564 | 1 | 1 |
| nuclear factor NF-kappa-B p105 subunit isoform 1 | Homo sapiens (human) | Potency | 35.4813 | 1 | 1 |
| nuclear factor of kappa light polypeptide gene enhancer in B-cells 1 (p105), isoform CRA_a | Homo sapiens (human) | Potency | 42.8010 | 2 | 4 |
| nuclear receptor ROR-gamma isoform 1 | Mus musculus (house mouse) | Potency | 30.2649 | 2 | 9 |
| nuclear receptor subfamily 1, group I, member 3 | Homo sapiens (human) | Potency | 33.3149 | 3 | 14 |
| parathyroid hormone/parathyroid hormone-related peptide receptor precursor | Homo sapiens (human) | Potency | 44.6684 | 1 | 1 |
| peptidyl-prolyl cis-trans isomerase NIMA-interacting 1 | Homo sapiens (human) | Potency | 52.3965 | 2 | 3 |
| peripheral myelin protein 22 | Rattus norvegicus (Norway rat) | Potency | 9.7204 | 1 | 5 |
| peripheral myelin protein 22 isoform 1 | Homo sapiens (human) | Potency | 43.4872 | 1 | 2 |
| peroxisome proliferator activated receptor gamma | Homo sapiens (human) | Potency | 20.3369 | 5 | 9 |
| peroxisome proliferator-activated receptor delta | Homo sapiens (human) | Potency | 30.0378 | 5 | 10 |
| phosphoglycerate kinase | Trypanosoma brucei brucei TREU927 | Potency | 12.1739 | 3 | 3 |
| phosphopantetheinyl transferase | Bacillus subtilis | Potency | 64.9975 | 3 | 15 |
| plasminogen precursor | Mus musculus (house mouse) | Potency | 12.5893 | 1 | 1 |
| polyprotein | Zika virus | Potency | 32.2233 | 1 | 3 |
| Polyunsaturated fatty acid lipoxygenase ALOX15B | Homo sapiens (human) | Potency | 9.7017 | 1 | 5 |
| potassium voltage-gated channel subfamily H member 2 isoform d | Homo sapiens (human) | Potency | 12.6561 | 1 | 7 |
| PPM1D protein | Homo sapiens (human) | Potency | 11.7086 | 1 | 2 |
| pregnane X nuclear receptor | Homo sapiens (human) | Potency | 18.5418 | 3 | 6 |
| pregnane X receptor | Rattus norvegicus (Norway rat) | Potency | 50.1187 | 1 | 2 |
| progesterone receptor | Homo sapiens (human) | Potency | 42.9904 | 1 | 4 |
| pyruvate kinase | Leishmania mexicana mexicana | Potency | 25.1189 | 2 | 2 |
| RAR-related orphan receptor gamma | Mus musculus (house mouse) | Potency | 24.4572 | 2 | 9 |
| ras-related protein Rab-9A | Homo sapiens (human) | Potency | 58.0479 | 1 | 1 |
| regulator of G-protein signaling 4 | Homo sapiens (human) | Potency | 5.8241 | 1 | 7 |
| retinoic acid nuclear receptor alpha variant 1 | Homo sapiens (human) | Potency | 40.6884 | 3 | 12 |
| retinoid X nuclear receptor alpha | Homo sapiens (human) | Potency | 11.4215 | 4 | 7 |
| serine/threonine-protein kinase mTOR isoform 1 | Homo sapiens (human) | Potency | 21.0600 | 4 | 7 |
| SMAD family member 2 | Homo sapiens (human) | Potency | 11.1388 | 2 | 5 |
| SMAD family member 3 | Homo sapiens (human) | Potency | 11.1388 | 2 | 5 |
| Smad3 | Homo sapiens (human) | Potency | 0.1122 | 1 | 1 |
| snurportin-1 | Homo sapiens (human) | Potency | 56.2341 | 1 | 1 |
| Spike glycoprotein | Severe acute respiratory syndrome-related coronavirus | Potency | 23.2092 | 1 | 4 |
| survival motor neuron protein isoform d | Homo sapiens (human) | Potency | 19.3810 | 1 | 5 |
| TAR DNA-binding protein 43 | Homo sapiens (human) | Potency | 1.8623 | 1 | 2 |
| TDP1 protein | Homo sapiens (human) | Potency | 16.7942 | 2 | 21 |
| thioredoxin reductase | Rattus norvegicus (Norway rat) | Potency | 18.1988 | 2 | 8 |
| Thrombopoietin | Homo sapiens (human) | Potency | 5.4576 | 2 | 6 |
| thyroid hormone receptor beta isoform 2 | Rattus norvegicus (Norway rat) | Potency | 22.5550 | 3 | 18 |
| thyroid hormone receptor beta isoform a | Homo sapiens (human) | Potency | 70.7946 | 1 | 1 |
| thyroid stimulating hormone receptor | Homo sapiens (human) | Potency | 34.2593 | 4 | 7 |
| transient receptor potential cation channel subfamily V member 1 | Homo sapiens (human) | Potency | 11.2202 | 1 | 1 |
| ubiquitin carboxyl-terminal hydrolase 2 isoform a | Homo sapiens (human) | Potency | 11.6305 | 2 | 2 |
| urokinase plasminogen activator surface receptor precursor | Mus musculus (house mouse) | Potency | 12.5893 | 1 | 1 |
| urokinase-type plasminogen activator precursor | Mus musculus (house mouse) | Potency | 12.5893 | 1 | 1 |
| USP1 protein, partial | Homo sapiens (human) | Potency | 27.5864 | 3 | 5 |
| v-jun sarcoma virus 17 oncogene homolog (avian) | Homo sapiens (human) | Potency | 23.4472 | 2 | 7 |
| vitamin D (1,25- dihydroxyvitamin D3) receptor | Homo sapiens (human) | Potency | 16.0550 | 4 | 10 |
| vitamin D3 receptor isoform VDRA | Homo sapiens (human) | Potency | 42.6410 | 1 | 6 |
| Voltage-dependent calcium channel gamma-2 subunit | Mus musculus (house mouse) | Potency | 37.8552 | 1 | 4 |
| WRN | Homo sapiens (human) | Potency | 5.4979 | 2 | 2 |
| Protein | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Drugs |
|---|
| 3-beta-hydroxysteroid-Delta(8),Delta(7)-isomerase | Homo sapiens (human) | Ki | 0.1900 | 1 | 1 |
| 5-hydroxytryptamine receptor 1A | Homo sapiens (human) | IC50 | 1.5000 | 1 | 1 |
| 5-hydroxytryptamine receptor 1A | Rattus norvegicus (Norway rat) | IC50 | 3.9224 | 8 | 10 |
| 5-hydroxytryptamine receptor 1A | Homo sapiens (human) | Ki | 1.6119 | 11 | 13 |
| 5-hydroxytryptamine receptor 1A | Rattus norvegicus (Norway rat) | Ki | 1.3808 | 8 | 9 |
| 5-hydroxytryptamine receptor 1B | Rattus norvegicus (Norway rat) | IC50 | 3.5040 | 5 | 6 |
| 5-hydroxytryptamine receptor 1B | Homo sapiens (human) | Ki | 3.5080 | 1 | 1 |
| 5-hydroxytryptamine receptor 1B | Rattus norvegicus (Norway rat) | Ki | 0.0017 | 1 | 2 |
| 5-hydroxytryptamine receptor 1D | Rattus norvegicus (Norway rat) | IC50 | 5.2545 | 4 | 4 |
| 5-hydroxytryptamine receptor 1D | Homo sapiens (human) | Ki | 10.0000 | 1 | 1 |
| 5-hydroxytryptamine receptor 1E | Homo sapiens (human) | Ki | 10.0000 | 1 | 1 |
| 5-hydroxytryptamine receptor 1F | Rattus norvegicus (Norway rat) | IC50 | 5.2545 | 4 | 4 |
| 5-hydroxytryptamine receptor 2A | Homo sapiens (human) | IC50 | 0.3555 | 2 | 6 |
| 5-hydroxytryptamine receptor 2A | Rattus norvegicus (Norway rat) | IC50 | 1.7889 | 12 | 12 |
| 5-hydroxytryptamine receptor 2A | Homo sapiens (human) | Ki | 0.1260 | 17 | 21 |
| 5-hydroxytryptamine receptor 2A | Mus musculus (house mouse) | Ki | 0.0265 | 1 | 1 |
| 5-hydroxytryptamine receptor 2A | Rattus norvegicus (Norway rat) | Ki | 0.0483 | 20 | 21 |
| 5-hydroxytryptamine receptor 2A | Sus scrofa (pig) | Ki | 0.0300 | 1 | 1 |
| 5-hydroxytryptamine receptor 2B | Homo sapiens (human) | IC50 | 1.3145 | 1 | 5 |
| 5-hydroxytryptamine receptor 2B | Rattus norvegicus (Norway rat) | IC50 | 2.3587 | 9 | 9 |
| 5-hydroxytryptamine receptor 2B | Homo sapiens (human) | Ki | 0.7004 | 2 | 6 |
| 5-hydroxytryptamine receptor 2B | Mus musculus (house mouse) | Ki | 0.0265 | 1 | 1 |
| 5-hydroxytryptamine receptor 2B | Rattus norvegicus (Norway rat) | Ki | 0.0261 | 9 | 9 |
| 5-hydroxytryptamine receptor 2C | Homo sapiens (human) | IC50 | 2.5688 | 2 | 6 |
| 5-hydroxytryptamine receptor 2C | Rattus norvegicus (Norway rat) | IC50 | 2.2228 | 10 | 10 |
| 5-hydroxytryptamine receptor 2C | Homo sapiens (human) | Ki | 3.5457 | 11 | 15 |
| 5-hydroxytryptamine receptor 2C | Rattus norvegicus (Norway rat) | Ki | 0.4935 | 10 | 10 |
| 5-hydroxytryptamine receptor 2C | Mus musculus (house mouse) | Ki | 0.0265 | 1 | 1 |
| 5-hydroxytryptamine receptor 3A | Rattus norvegicus (Norway rat) | IC50 | 10.0000 | 2 | 2 |
| 5-hydroxytryptamine receptor 3A | Homo sapiens (human) | Ki | 10.0000 | 1 | 1 |
| 5-hydroxytryptamine receptor 3A | Mus musculus (house mouse) | Ki | 10.0000 | 1 | 1 |
| 5-hydroxytryptamine receptor 3B | Rattus norvegicus (Norway rat) | IC50 | 10.0000 | 2 | 2 |
| 5-hydroxytryptamine receptor 4 | Cavia porcellus (domestic guinea pig) | IC50 | 0.9032 | 2 | 6 |
| 5-hydroxytryptamine receptor 4 | Cavia porcellus (domestic guinea pig) | Ki | 0.8910 | 2 | 6 |
| 5-hydroxytryptamine receptor 4 | Homo sapiens (human) | Ki | 0.0006 | 1 | 1 |
| 5-hydroxytryptamine receptor 4 | Rattus norvegicus (Norway rat) | IC50 | 7.1167 | 3 | 3 |
| 5-hydroxytryptamine receptor 5A | Rattus norvegicus (Norway rat) | IC50 | 10.0000 | 2 | 2 |
| 5-hydroxytryptamine receptor 5A | Homo sapiens (human) | Ki | 10.0000 | 1 | 1 |
| 5-hydroxytryptamine receptor 5B | Rattus norvegicus (Norway rat) | IC50 | 10.0000 | 2 | 2 |
| 5-hydroxytryptamine receptor 6 | Homo sapiens (human) | IC50 | 0.3850 | 1 | 3 |
| 5-hydroxytryptamine receptor 6 | Rattus norvegicus (Norway rat) | IC50 | 10.0000 | 2 | 2 |
| 5-hydroxytryptamine receptor 6 | Homo sapiens (human) | Ki | 2.5267 | 6 | 9 |
| 5-hydroxytryptamine receptor 7 | Cavia porcellus (domestic guinea pig) | IC50 | 58.4333 | 1 | 6 |
| 5-hydroxytryptamine receptor 7 | Homo sapiens (human) | Ki | 0.8268 | 4 | 5 |
| 5-hydroxytryptamine receptor 7 | Rattus norvegicus (Norway rat) | IC50 | 10.0000 | 2 | 2 |
| 5-hydroxytryptamine receptor 7 | Rattus norvegicus (Norway rat) | Ki | 0.1383 | 5 | 6 |
| Acetylcholinesterase | Homo sapiens (human) | IC50 | 0.2700 | 3 | 4 |
| Acetylcholinesterase | Homo sapiens (human) | Ki | 86.6100 | 1 | 2 |
| Acetylcholinesterase | Bos taurus (cattle) | Ki | 173.2000 | 2 | 2 |
| Adenosine receptor A1 | Rattus norvegicus (Norway rat) | Ki | 0.3180 | 1 | 1 |
| Adenosine receptor A2a | Homo sapiens (human) | IC50 | 2.3200 | 1 | 1 |
| Adenylate cyclase type 1 | Rattus norvegicus (Norway rat) | IC50 | 2.3000 | 1 | 1 |
| Adenylate cyclase type 2 | Rattus norvegicus (Norway rat) | IC50 | 2.3000 | 1 | 1 |
| Adenylate cyclase type 3 | Rattus norvegicus (Norway rat) | IC50 | 2.3000 | 1 | 1 |
| Adenylate cyclase type 4 | Rattus norvegicus (Norway rat) | IC50 | 2.3000 | 1 | 1 |
| Adenylate cyclase type 5 | Rattus norvegicus (Norway rat) | IC50 | 1.4250 | 2 | 2 |
| Adenylate cyclase type 6 | Rattus norvegicus (Norway rat) | IC50 | 2.3000 | 1 | 1 |
| Adenylate cyclase type 8 | Rattus norvegicus (Norway rat) | IC50 | 2.3000 | 1 | 1 |
| Adenylyl cyclase 7 | Rattus norvegicus (Norway rat) | IC50 | 2.3000 | 1 | 1 |
| Aldo-keto reductase family 1 member B1 | Rattus norvegicus (Norway rat) | IC50 | 2.6813 | 1 | 3 |
| Aldo-keto reductase family 1 member B1 | Rattus norvegicus (Norway rat) | Ki | 2.6587 | 1 | 3 |
| Alpha-1A adrenergic receptor | Rattus norvegicus (Norway rat) | IC50 | 1.3627 | 5 | 6 |
| Alpha-1A adrenergic receptor | Homo sapiens (human) | Ki | 3.3416 | 3 | 3 |
| Alpha-1A adrenergic receptor | Rattus norvegicus (Norway rat) | Ki | 0.0142 | 10 | 12 |
| Alpha-1B adrenergic receptor | Rattus norvegicus (Norway rat) | IC50 | 1.3627 | 5 | 6 |
| Alpha-1B adrenergic receptor | Homo sapiens (human) | Ki | 0.0124 | 2 | 2 |
| Alpha-1B adrenergic receptor | Rattus norvegicus (Norway rat) | Ki | 0.0142 | 10 | 12 |
| Alpha-1D adrenergic receptor | Homo sapiens (human) | IC50 | 0.0517 | 1 | 3 |
| Alpha-1D adrenergic receptor | Rattus norvegicus (Norway rat) | IC50 | 1.3627 | 5 | 6 |
| Alpha-1D adrenergic receptor | Homo sapiens (human) | Ki | 0.0201 | 3 | 5 |
| Alpha-1D adrenergic receptor | Rattus norvegicus (Norway rat) | Ki | 0.0142 | 10 | 12 |
| Alpha-2A adrenergic receptor | Homo sapiens (human) | IC50 | 1.7861 | 1 | 4 |
| Alpha-2A adrenergic receptor | Rattus norvegicus (Norway rat) | IC50 | 0.2885 | 1 | 2 |
| Alpha-2A adrenergic receptor | Homo sapiens (human) | Ki | 1.2926 | 3 | 6 |
| Alpha-2A adrenergic receptor | Rattus norvegicus (Norway rat) | Ki | 9.6000 | 1 | 1 |
| Alpha-2B adrenergic receptor | Homo sapiens (human) | IC50 | 0.8211 | 1 | 4 |
| Alpha-2B adrenergic receptor | Rattus norvegicus (Norway rat) | IC50 | 0.2885 | 1 | 2 |
| Alpha-2B adrenergic receptor | Homo sapiens (human) | Ki | 1.0945 | 3 | 6 |
| Alpha-2B adrenergic receptor | Rattus norvegicus (Norway rat) | Ki | 9.6000 | 1 | 1 |
| Alpha-2C adrenergic receptor | Homo sapiens (human) | IC50 | 0.7898 | 1 | 3 |
| Alpha-2C adrenergic receptor | Rattus norvegicus (Norway rat) | IC50 | 0.2885 | 1 | 2 |
| Alpha-2C adrenergic receptor | Homo sapiens (human) | Ki | 1.0794 | 3 | 5 |
| Alpha-2C adrenergic receptor | Rattus norvegicus (Norway rat) | Ki | 9.6000 | 1 | 1 |
| Alpha-ketoglutarate-dependent dioxygenase FTO | Homo sapiens (human) | IC50 | 3.0000 | 1 | 1 |
| Alpha-synuclein | Homo sapiens (human) | IC50 | 24.7000 | 1 | 1 |
| Androgen receptor | Rattus norvegicus (Norway rat) | IC50 | 2.2810 | 1 | 1 |
| Androgen receptor | Rattus norvegicus (Norway rat) | Ki | 1.5210 | 1 | 1 |
| Angiotensin-converting enzyme | Oryctolagus cuniculus (rabbit) | IC50 | 19.4295 | 2 | 2 |
| Angiotensin-converting enzyme | Oryctolagus cuniculus (rabbit) | Ki | 26.1013 | 1 | 1 |
| AP-2 complex subunit sigma | Rattus norvegicus (Norway rat) | Ki | 0.0242 | 1 | 1 |
| ATP-binding cassette sub-family C member 3 | Homo sapiens (human) | IC50 | 116.6833 | 1 | 6 |
| ATP-dependent translocase ABCB1 | Homo sapiens (human) | IC50 | 2.9750 | 4 | 4 |
| ATP-dependent translocase ABCB1 | Mus musculus (house mouse) | IC50 | 27.4500 | 4 | 4 |
| ATP-dependent translocase ABCB1 | Homo sapiens (human) | Ki | 2.3233 | 3 | 3 |
| ATP-dependent translocase ABCB1 | Mus musculus (house mouse) | Ki | 6.9350 | 2 | 2 |
| Beta-1 adrenergic receptor | Homo sapiens (human) | IC50 | 1.4795 | 1 | 2 |
| Beta-1 adrenergic receptor | Homo sapiens (human) | Ki | 0.8545 | 1 | 2 |
| Beta-1 adrenergic receptor | Rattus norvegicus (Norway rat) | Ki | 10.0000 | 1 | 1 |
| Beta-2 adrenergic receptor | Homo sapiens (human) | IC50 | 0.0410 | 1 | 1 |
| Beta-2 adrenergic receptor | Rattus norvegicus (Norway rat) | IC50 | 2.3000 | 1 | 1 |
| Beta-2 adrenergic receptor | Homo sapiens (human) | Ki | 36.6763 | 3 | 3 |
| Beta-2 adrenergic receptor | Rattus norvegicus (Norway rat) | Ki | 10.0000 | 1 | 1 |
| Beta-3 adrenergic receptor | Homo sapiens (human) | Ki | 10.0000 | 1 | 1 |
| Beta-3 adrenergic receptor | Rattus norvegicus (Norway rat) | Ki | 10.0000 | 1 | 1 |
| Bile salt export pump | Homo sapiens (human) | IC50 | 179.2186 | 3 | 14 |
| C-8 sterol isomerase | Saccharomyces cerevisiae S288C | Ki | 0.0005 | 1 | 1 |
| Calcitonin gene-related peptide type 1 receptor | Homo sapiens (human) | Ki | 0.0004 | 1 | 1 |
| Calcium release-activated calcium channel protein 1 | Homo sapiens (human) | IC50 | 500.0000 | 2 | 2 |
| Canalicular multispecific organic anion transporter 1 | Homo sapiens (human) | IC50 | 133.0000 | 1 | 6 |
| Carboxylic ester hydrolase | Equus caballus (horse) | Ki | 0.0200 | 1 | 1 |
| Catechol O-methyltransferase | Homo sapiens (human) | IC50 | 0.2230 | 2 | 2 |
| Catechol O-methyltransferase | Rattus norvegicus (Norway rat) | IC50 | 1.2750 | 2 | 2 |
| Cholecystokinin receptor type A | Cavia porcellus (domestic guinea pig) | Ki | 0.0500 | 1 | 1 |
| Cholinesterase | Equus caballus (horse) | IC50 | 0.7200 | 1 | 1 |
| Cholinesterase | Homo sapiens (human) | IC50 | 0.2550 | 2 | 2 |
| Cholinesterase | Homo sapiens (human) | Ki | 0.0200 | 2 | 2 |
| Cocaine esterase | Homo sapiens (human) | Ki | 0.0063 | 1 | 1 |
| Cytochrome P450 2C9 | Homo sapiens (human) | IC50 | 27.3450 | 1 | 2 |
| Cytochrome P450 2D6 | Homo sapiens (human) | IC50 | 0.2080 | 1 | 2 |
| Cytochrome P450 2J2 | Homo sapiens (human) | IC50 | 27.3450 | 1 | 2 |
| Cytochrome P450 3A4 | Homo sapiens (human) | IC50 | 3.6885 | 4 | 4 |
| D | Bos taurus (cattle) | IC50 | 0.3268 | 11 | 15 |
| D | Rattus norvegicus (Norway rat) | IC50 | 0.2418 | 21 | 28 |
| D | Bos taurus (cattle) | Ki | 10.0018 | 2 | 2 |
| D | Mus musculus (house mouse) | Ki | 0.1010 | 1 | 1 |
| D | Rattus norvegicus (Norway rat) | Ki | 3.2328 | 26 | 33 |
| D(1A) dopamine receptor | Homo sapiens (human) | IC50 | 0.6404 | 2 | 5 |
| D(1A) dopamine receptor | Homo sapiens (human) | Ki | 0.6878 | 19 | 22 |
| D(1A) dopamine receptor | Sus scrofa (pig) | Ki | 0.0095 | 1 | 1 |
| D(1B) dopamine receptor | Homo sapiens (human) | IC50 | 0.0150 | 1 | 2 |
| D(1B) dopamine receptor | Rattus norvegicus (Norway rat) | IC50 | 0.0590 | 13 | 19 |
| D(1B) dopamine receptor | Homo sapiens (human) | Ki | 1.7365 | 6 | 6 |
| D(1B) dopamine receptor | Rattus norvegicus (Norway rat) | Ki | 0.0017 | 2 | 2 |
| D(2) dopamine receptor | Bos taurus (cattle) | IC50 | 0.9765 | 14 | 19 |
| D(2) dopamine receptor | Homo sapiens (human) | IC50 | 0.6887 | 12 | 16 |
| D(2) dopamine receptor | Rattus norvegicus (Norway rat) | IC50 | 0.0383 | 38 | 51 |
| D(2) dopamine receptor | Bos taurus (cattle) | Ki | 0.0449 | 5 | 5 |
| D(2) dopamine receptor | Chlorocebus aethiops (grivet) | Ki | 0.0049 | 2 | 2 |
| D(2) dopamine receptor | Homo sapiens (human) | Ki | 0.1836 | 133 | 149 |
| D(2) dopamine receptor | Rattus norvegicus (Norway rat) | Ki | 0.0787 | 49 | 74 |
| D(3) dopamine receptor | Homo sapiens (human) | IC50 | 0.0072 | 6 | 9 |
| D(3) dopamine receptor | Rattus norvegicus (Norway rat) | IC50 | 0.0590 | 13 | 19 |
| D(3) dopamine receptor | Chlorocebus aethiops (grivet) | Ki | 0.0030 | 1 | 1 |
| D(3) dopamine receptor | Homo sapiens (human) | Ki | 0.0111 | 70 | 79 |
| D(3) dopamine receptor | Rattus norvegicus (Norway rat) | Ki | 0.0151 | 14 | 14 |
| D(4) dopamine receptor | Homo sapiens (human) | IC50 | 0.0874 | 6 | 7 |
| D(4) dopamine receptor | Rattus norvegicus (Norway rat) | IC50 | 0.0590 | 13 | 19 |
| D(4) dopamine receptor | Homo sapiens (human) | Ki | 0.0195 | 50 | 53 |
| D(4) dopamine receptor | Rattus norvegicus (Norway rat) | Ki | 0.0060 | 2 | 2 |
| Delta-type opioid receptor | Homo sapiens (human) | IC50 | 3.7600 | 1 | 1 |
| Delta-type opioid receptor | Homo sapiens (human) | Ki | 10.0000 | 1 | 1 |
| Delta-type opioid receptor | Rattus norvegicus (Norway rat) | Ki | 7.0700 | 2 | 3 |
| DNA damage-inducible transcript 3 protein | Mus musculus (house mouse) | IC50 | 6.3400 | 1 | 1 |
| E3 ubiquitin-protein ligase Mdm2 | Homo sapiens (human) | IC50 | 10.1367 | 3 | 3 |
| Epidermal growth factor receptor | Homo sapiens (human) | IC50 | 451.4400 | 2 | 2 |
| Gastrin/cholecystokinin type B receptor | Mus musculus (house mouse) | Ki | 0.0234 | 1 | 2 |
| Genome polyprotein | Human rhinovirus sp. | IC50 | 140.0000 | 1 | 1 |
| Genome polyprotein | Zika virus | IC50 | 17.3200 | 2 | 2 |
| Genome polyprotein | Human rhinovirus sp. | Ki | 0.1000 | 1 | 1 |
| Glutamate receptor ionotropic, NMDA 1 | Homo sapiens (human) | Ki | 3.8500 | 1 | 2 |
| Glutamate receptor ionotropic, NMDA 1 | Rattus norvegicus (Norway rat) | Ki | 10.0000 | 1 | 1 |
| Glutamate receptor ionotropic, NMDA 2A | Homo sapiens (human) | Ki | 3.8500 | 1 | 2 |
| Glutamate receptor ionotropic, NMDA 2A | Rattus norvegicus (Norway rat) | Ki | 10.0000 | 1 | 1 |
| Glutamate receptor ionotropic, NMDA 2B | Homo sapiens (human) | Ki | 3.8500 | 1 | 2 |
| Glutamate receptor ionotropic, NMDA 2B | Rattus norvegicus (Norway rat) | Ki | 5.0006 | 2 | 2 |
| Glutamate receptor ionotropic, NMDA 2C | Homo sapiens (human) | Ki | 3.8500 | 1 | 2 |
| Glutamate receptor ionotropic, NMDA 2C | Rattus norvegicus (Norway rat) | Ki | 10.0000 | 1 | 1 |
| Glutamate receptor ionotropic, NMDA 2D | Homo sapiens (human) | Ki | 3.8500 | 1 | 2 |
| Glutamate receptor ionotropic, NMDA 2D | Rattus norvegicus (Norway rat) | Ki | 10.0000 | 1 | 1 |
| Glutamate receptor ionotropic, NMDA 3A | Homo sapiens (human) | Ki | 3.8500 | 1 | 2 |
| Glutamate receptor ionotropic, NMDA 3A | Rattus norvegicus (Norway rat) | Ki | 10.0000 | 1 | 1 |
| Glutamate receptor ionotropic, NMDA 3B | Homo sapiens (human) | Ki | 3.8500 | 1 | 2 |
| Glutamate receptor ionotropic, NMDA 3B | Rattus norvegicus (Norway rat) | Ki | 10.0000 | 1 | 1 |
| Histamine H1 receptor | Homo sapiens (human) | IC50 | 19.9766 | 2 | 6 |
| Histamine H1 receptor | Rattus norvegicus (Norway rat) | IC50 | 1.0000 | 1 | 2 |
| Histamine H1 receptor | Homo sapiens (human) | Ki | 0.2856 | 6 | 9 |
| Histamine H1 receptor | Rattus norvegicus (Norway rat) | Ki | 2.1000 | 1 | 1 |
| Histamine H2 receptor | Homo sapiens (human) | IC50 | 3.0557 | 1 | 3 |
| Histamine H2 receptor | Homo sapiens (human) | Ki | 5.1002 | 3 | 5 |
| Histamine H4 receptor | Homo sapiens (human) | Ki | 18.2193 | 3 | 3 |
| integrase, partial | Human immunodeficiency virus 1 | IC50 | 0.5939 | 2 | 2 |
| Integrin alpha-4 | Homo sapiens (human) | Ki | 0.0039 | 1 | 1 |
| Integrin beta-1 | Homo sapiens (human) | Ki | 0.0039 | 1 | 1 |
| Kappa-type opioid receptor | Homo sapiens (human) | IC50 | 0.9900 | 1 | 1 |
| Kappa-type opioid receptor | Cavia porcellus (domestic guinea pig) | Ki | 0.0026 | 1 | 1 |
| Kappa-type opioid receptor | Rattus norvegicus (Norway rat) | Ki | 7.0700 | 2 | 3 |
| Large neutral amino acids transporter small subunit 1 | Homo sapiens (human) | IC50 | 100.0000 | 1 | 1 |
| lens epithelium-derived growth factor p75 | Homo sapiens (human) | IC50 | 0.5939 | 2 | 2 |
| Lysine-specific demethylase 4E | Homo sapiens (human) | Ki | 1.9800 | 1 | 1 |
| Mu-type opioid receptor | Homo sapiens (human) | IC50 | 1.4075 | 2 | 2 |
| Mu-type opioid receptor | Homo sapiens (human) | Ki | 4.4873 | 3 | 3 |
| Mu-type opioid receptor | Rattus norvegicus (Norway rat) | Ki | 7.0700 | 2 | 3 |
| Multidrug and toxin extrusion protein 1 | Homo sapiens (human) | IC50 | 282.5000 | 2 | 2 |
| Multidrug and toxin extrusion protein 2 | Homo sapiens (human) | IC50 | 300.0000 | 2 | 2 |
| Multidrug resistance-associated protein 4 | Homo sapiens (human) | IC50 | 111.9667 | 1 | 6 |
| Muscarinic acetylcholine receptor M1 | Homo sapiens (human) | IC50 | 2.8735 | 3 | 4 |
| Muscarinic acetylcholine receptor M1 | Rattus norvegicus (Norway rat) | IC50 | 0.2205 | 2 | 4 |
| Muscarinic acetylcholine receptor M1 | Homo sapiens (human) | Ki | 2.5702 | 6 | 7 |
| Muscarinic acetylcholine receptor M1 | Rattus norvegicus (Norway rat) | Ki | 4.6306 | 4 | 5 |
| Muscarinic acetylcholine receptor M2 | Homo sapiens (human) | IC50 | 0.7130 | 1 | 2 |
| Muscarinic acetylcholine receptor M2 | Rattus norvegicus (Norway rat) | IC50 | 0.3870 | 2 | 2 |
| Muscarinic acetylcholine receptor M2 | Homo sapiens (human) | Ki | 3.0381 | 4 | 5 |
| Muscarinic acetylcholine receptor M2 | Rattus norvegicus (Norway rat) | Ki | 5.2542 | 5 | 5 |
| Muscarinic acetylcholine receptor M3 | Homo sapiens (human) | IC50 | 0.4110 | 1 | 2 |
| Muscarinic acetylcholine receptor M3 | Rattus norvegicus (Norway rat) | IC50 | 0.3870 | 2 | 2 |
| Muscarinic acetylcholine receptor M3 | Homo sapiens (human) | Ki | 2.9700 | 4 | 5 |
| Muscarinic acetylcholine receptor M3 | Rattus norvegicus (Norway rat) | Ki | 8.7066 | 2 | 2 |
| Muscarinic acetylcholine receptor M4 | Homo sapiens (human) | IC50 | 0.2485 | 1 | 2 |
| Muscarinic acetylcholine receptor M4 | Rattus norvegicus (Norway rat) | IC50 | 0.3870 | 2 | 2 |
| Muscarinic acetylcholine receptor M4 | Homo sapiens (human) | Ki | 1.1928 | 3 | 4 |
| Muscarinic acetylcholine receptor M4 | Rattus norvegicus (Norway rat) | Ki | 8.7066 | 2 | 2 |
| Muscarinic acetylcholine receptor M5 | Homo sapiens (human) | IC50 | 1.3600 | 1 | 3 |
| Muscarinic acetylcholine receptor M5 | Rattus norvegicus (Norway rat) | IC50 | 0.3870 | 2 | 2 |
| Muscarinic acetylcholine receptor M5 | Homo sapiens (human) | Ki | 1.9002 | 2 | 4 |
| Muscarinic acetylcholine receptor M5 | Rattus norvegicus (Norway rat) | Ki | 8.7066 | 2 | 2 |
| N-acetyltransferase Eis | Mycobacterium tuberculosis H37Rv | IC50 | 0.3900 | 1 | 1 |
| N-acetyltransferase Eis | Mycobacterium tuberculosis H37Rv | Ki | 0.3900 | 1 | 1 |
| Nuclear receptor subfamily 3 group C member 3 | Bos taurus (cattle) | IC50 | 31.8590 | 1 | 1 |
| Nuclear receptor subfamily 3 group C member 3 | Bos taurus (cattle) | Ki | 26.1013 | 1 | 1 |
| Polyunsaturated fatty acid lipoxygenase ALOX15 | Oryctolagus cuniculus (rabbit) | IC50 | 2.2580 | 1 | 1 |
| Potassium channel subfamily K member 2 | Homo sapiens (human) | IC50 | 3.6500 | 1 | 2 |
| Potassium voltage-gated channel subfamily H member 2 | Homo sapiens (human) | IC50 | 3.4478 | 20 | 37 |
| Potassium voltage-gated channel subfamily H member 2 | Homo sapiens (human) | Ki | 6.6938 | 3 | 4 |
| Protease | Human immunodeficiency virus 1 | IC50 | 125.0000 | 1 | 1 |
| Protease | Human immunodeficiency virus 1 | Ki | 50.0500 | 2 | 2 |
| Protein orai-2 | Homo sapiens (human) | IC50 | 500.0000 | 2 | 2 |
| Protein orai-3 | Homo sapiens (human) | IC50 | 500.0000 | 2 | 2 |
| Sigma intracellular receptor 2 | Homo sapiens (human) | Ki | 0.0616 | 6 | 6 |
| Sigma intracellular receptor 2 | Rattus norvegicus (Norway rat) | Ki | 0.0721 | 11 | 11 |
| Sigma non-opioid intracellular receptor 1 | Homo sapiens (human) | IC50 | 1.3112 | 7 | 8 |
| Sigma non-opioid intracellular receptor 1 | Rattus norvegicus (Norway rat) | IC50 | 0.0013 | 4 | 5 |
| Sigma non-opioid intracellular receptor 1 | Cavia porcellus (domestic guinea pig) | Ki | 0.0048 | 36 | 36 |
| Sigma non-opioid intracellular receptor 1 | Homo sapiens (human) | Ki | 0.1114 | 38 | 42 |
| Sigma non-opioid intracellular receptor 1 | Rattus norvegicus (Norway rat) | Ki | 0.0148 | 7 | 7 |
| Sodium channel protein type 1 subunit alpha | Homo sapiens (human) | IC50 | 3.5270 | 2 | 2 |
| Sodium channel protein type 10 subunit alpha | Homo sapiens (human) | IC50 | 3.5270 | 2 | 2 |
| Sodium channel protein type 11 subunit alpha | Homo sapiens (human) | IC50 | 3.5270 | 2 | 2 |
| Sodium channel protein type 2 subunit alpha | Homo sapiens (human) | IC50 | 3.5270 | 2 | 2 |
| Sodium channel protein type 2 subunit alpha | Rattus norvegicus (Norway rat) | IC50 | 0.3400 | 1 | 1 |
| Sodium channel protein type 3 subunit alpha | Homo sapiens (human) | IC50 | 3.5270 | 2 | 2 |
| Sodium channel protein type 4 subunit alpha | Homo sapiens (human) | IC50 | 3.5270 | 2 | 2 |
| Sodium channel protein type 5 subunit alpha | Homo sapiens (human) | IC50 | 16.0180 | 3 | 3 |
| Sodium channel protein type 7 subunit alpha | Homo sapiens (human) | IC50 | 3.5270 | 2 | 2 |
| Sodium channel protein type 8 subunit alpha | Homo sapiens (human) | IC50 | 3.5270 | 2 | 2 |
| Sodium channel protein type 9 subunit alpha | Homo sapiens (human) | IC50 | 3.5270 | 2 | 2 |
| Sodium-dependent dopamine transporter | Rattus norvegicus (Norway rat) | Ki | 2.0237 | 2 | 3 |
| Sodium-dependent noradrenaline transporter | Homo sapiens (human) | IC50 | 2.6813 | 1 | 3 |
| Sodium-dependent noradrenaline transporter | Homo sapiens (human) | Ki | 3.3690 | 2 | 4 |
| Sodium-dependent serotonin transporter | Homo sapiens (human) | IC50 | 1.9220 | 1 | 2 |
| Sodium-dependent serotonin transporter | Homo sapiens (human) | Ki | 1.4105 | 3 | 4 |
| Sodium-dependent serotonin transporter | Rattus norvegicus (Norway rat) | Ki | 0.0342 | 1 | 1 |
| Solute carrier family 15 member 1 | Homo sapiens (human) | IC50 | 141,200.0000 | 1 | 1 |
| Solute carrier family 22 member 1 | Rattus norvegicus (Norway rat) | IC50 | 24.0000 | 1 | 1 |
| Solute carrier family 22 member 1 | Homo sapiens (human) | IC50 | 59.1520 | 3 | 5 |
| Solute carrier family 22 member 2 | Homo sapiens (human) | IC50 | 18.3500 | 2 | 2 |
| Solute carrier family 22 member 2 | Rattus norvegicus (Norway rat) | IC50 | 32.0000 | 1 | 1 |
| Transient receptor potential cation channel subfamily V member 1 | Rattus norvegicus (Norway rat) | Ki | 0.0050 | 1 | 1 |
| Transient receptor potential cation channel subfamily V member 2 | Rattus norvegicus (Norway rat) | Ki | 0.0050 | 1 | 1 |
| Transient receptor potential cation channel subfamily V member 4 | Rattus norvegicus (Norway rat) | Ki | 0.0050 | 1 | 1 |
| Transporter | Rattus norvegicus (Norway rat) | Ki | 5.5000 | 1 | 1 |
| Tryptophan 5-hydroxylase 1 | Rattus norvegicus (Norway rat) | IC50 | 0.2200 | 1 | 1 |
| Tyrosinase | Homo sapiens (human) | IC50 | 8,400.0000 | 1 | 1 |
| Tyrosine-protein kinase Fyn | Homo sapiens (human) | IC50 | 2.9385 | 1 | 2 |
| Tyrosine-protein kinase Lck | Homo sapiens (human) | IC50 | 5.2620 | 1 | 2 |
| Ubiquitin carboxyl-terminal hydrolase 1 | Homo sapiens (human) | IC50 | 2.0000 | 2 | 2 |
| UDP-glucuronosyltransferase 1A9 | Homo sapiens (human) | Ki | 344.0000 | 1 | 1 |
| UDP-glucuronosyltransferase 2B7 | Homo sapiens (human) | Ki | 590.0000 | 1 | 1 |
| Vesicular acetylcholine transporter | Rattus norvegicus (Norway rat) | Ki | 0.3910 | 1 | 1 |
| Vitamin D-binding protein | Rattus norvegicus (Norway rat) | Ki | 0.0037 | 1 | 1 |
| Voltage-dependent L-type calcium channel subunit alpha-1C | Cavia porcellus (domestic guinea pig) | IC50 | 1.7000 | 1 | 1 |
| Voltage-dependent L-type calcium channel subunit alpha-1C | Homo sapiens (human) | IC50 | 0.8505 | 4 | 4 |
| Voltage-dependent L-type calcium channel subunit alpha-1D | Homo sapiens (human) | IC50 | 0.8505 | 4 | 4 |
| Voltage-dependent L-type calcium channel subunit alpha-1F | Homo sapiens (human) | IC50 | 0.8505 | 4 | 4 |
| Voltage-dependent L-type calcium channel subunit alpha-1S | Homo sapiens (human) | IC50 | 0.8505 | 4 | 4 |
| WD repeat-containing protein 48 | Homo sapiens (human) | IC50 | 2.0000 | 1 | 1 |
| XBP1 | Homo sapiens (human) | IC50 | 10.0000 | 1 | 1 |
| Zinc finger protein 664 | Cavia porcellus (domestic guinea pig) | Ki | 0.0066 | 1 | 1 |