Page last updated: 2024-08-07 10:20:09

N-acetyltransferase Eis

[no definition available]

Synonyms

EC 2.3.1.-;
Aminoglycoside N-acetyltransferase;
Enhanced intracellular survival protein;
Protein-lysine N-acetyltransferase

Research

Bioassay Publications (1)

TimeframeStudies on this Protein(%)All Drugs %
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's1 (100.00)2.80

Compounds (5)

Drugs with Inhibition Measurements

DrugTaxonomyMeasurementAverage (mM)Bioassay(s)Publication(s)
bromperidolMycobacterium tuberculosis H37RvIC500.520011
bromperidolMycobacterium tuberculosis H37RvKi0.240011
droperidolMycobacterium tuberculosis H37RvIC5012.200011
haloperidolMycobacterium tuberculosis H37RvIC500.390011
haloperidolMycobacterium tuberculosis H37RvKi0.390011
4(4-chlorophenyl)-1-(4-(4-fluorophenyl)-4-oxobutyl)-1,2,3,6-tetrahydropyridineMycobacterium tuberculosis H37RvIC500.560011
1-(3-(4-chlorobenzoyl)propyl)-4-hydroxy-4-(4-chlorophenyl)piperidineMycobacterium tuberculosis H37RvIC505.100011