Proteins > XBP1
Page last updated: 2024-08-07 22:51:12

XBP1

[no definition available]

Synonyms

Research

Bioassay Publications (1)

TimeframeStudies on this Protein(%)All Drugs %
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's1 (100.00)24.3611
2020's0 (0.00)2.80

Compounds (73)

Drugs with Inhibition Measurements

DrugTaxonomyMeasurementAverage (mM)Bioassay(s)Publication(s)
fluspirileneHomo sapiens (human)IC5010.000010
terfenadineHomo sapiens (human)IC505.140010
pimozideHomo sapiens (human)IC5010.000010
nsc 3852Homo sapiens (human)IC505.080010
1,6-bismaleimidohexaneHomo sapiens (human)IC505.150010
helenalinHomo sapiens (human)IC502.430010
isovelleralHomo sapiens (human)IC502.350010
9-methoxyellipticineHomo sapiens (human)IC5010.000010
2-phenyl-4,5-dichloro-3-pyridazinoneHomo sapiens (human)IC505.230010
girinimbineHomo sapiens (human)IC5010.000010
3,3-bis(4-hydroxy-3-methylphenyl)-1H-indol-2-oneHomo sapiens (human)IC5010.000010
aromaticinHomo sapiens (human)IC505.710010
angustibalinHomo sapiens (human)IC502.200010
cgp 60474Homo sapiens (human)IC500.160010
2-[(1-cyclohexyl-5-tetrazolyl)thio]-N-(6-ethoxy-1,3-benzothiazol-2-yl)acetamideHomo sapiens (human)IC5010.000010
8-(butan-2-ylthio)-7-[(4-chlorophenyl)methyl]-3-methylpurine-2,6-dioneHomo sapiens (human)IC5010.000010
(1S,2R)-2-(octylamino)-1-[4-(propan-2-ylthio)phenyl]-1-propanolHomo sapiens (human)IC504.760010
1-[5-(trifluoromethyl)-1,3,4-thiadiazol-2-yl]-3-[1,1,1-trifluoro-2-(trifluoromethyl)butan-2-yl]ureaHomo sapiens (human)IC502.000010
4-(cyclohexylamino)-2-(3,5-dimethyl-1-pyrazolyl)-5-pyrimidinecarboxylic acid ethyl esterHomo sapiens (human)IC505.640010
3-(3-benzoyl-6-chloro-4,5-dihydroxy-7-benzofuranyl)pentane-2,4-dioneHomo sapiens (human)IC506.680010
N-[2-[5-[(2,4-dichlorophenyl)methylsulfonyl]-1,3,4-oxadiazol-2-yl]ethyl]carbamic acid tert-butyl esterHomo sapiens (human)IC504.440010
4-chloro-1-methyl-3-nitro-2-quinolinoneHomo sapiens (human)IC505.420010
2-(dichloromethyl)-4-(ethylthio)-6-phenyl-1,3,5-triazineHomo sapiens (human)IC5010.000010
4-chloro-3-ethoxy-N-(4-ethylphenyl)benzenesulfonamideHomo sapiens (human)IC509.300010
LSM-16285Homo sapiens (human)IC507.210010
2-(4-methylsulfonyl-2-nitrophenyl)sulfinylacetic acid (phenylmethyl) esterHomo sapiens (human)IC503.790010
N-(2,5-dimethylphenyl)-2-[[3-(4-ethylphenoxy)-4-oxo-1-benzopyran-7-yl]oxy]acetamideHomo sapiens (human)IC5010.000010
N-[[3-(4-fluorophenyl)-1-phenyl-4-pyrazolyl]methyl]-1-phenylmethanamineHomo sapiens (human)IC5010.000010
5-[(cyclohexylamino)-oxomethyl]-4-methyl-2-[(1-oxo-2-thiophen-2-ylethyl)amino]-3-thiophenecarboxylic acid ethyl esterHomo sapiens (human)IC5010.000010
2-[2-(2,4-dichloro-5-propan-2-yloxyanilino)-2-oxoethyl]sulfinyl-N-[3-(trifluoromethyl)phenyl]acetamideHomo sapiens (human)IC506.300010
(4-chlorophenyl)-[4-[[(2,4-dichlorophenyl)thio]methyl]-4-hydroxy-1-piperidinyl]methanoneHomo sapiens (human)IC5010.000010
3-amino-N-(2-fluorophenyl)-6-(3-pyridinyl)-2-thieno[2,3-b]pyridinecarboxamideHomo sapiens (human)IC5010.000010
2-(3,5-dimethyl-1-pyrazolyl)-4-(4-hydroxyanilino)-5-pyrimidinecarboxylic acid ethyl esterHomo sapiens (human)IC501.260010
4-[bis(2-methylpropyl)sulfamoyl]-N-[5-(3-methoxyphenyl)-1,3,4-oxadiazol-2-yl]benzamideHomo sapiens (human)IC505.000010
6-bromo-2-(3-pyridinyl)-N-[4-(trifluoromethyl)phenyl]-4-quinolinecarboxamideHomo sapiens (human)IC5010.000010
5,6,7,8-tetrafluoro-2-(2,3,4,5,6-pentafluorophenyl)-4h-1-benzopyran-4-oneHomo sapiens (human)IC504.690010
2-(2,6-dichlorophenyl)acetic acid [2-oxo-2-[4-(trifluoromethoxy)anilino]ethyl] esterHomo sapiens (human)IC5010.000010
2-[(3-methoxyphenyl)-oxomethyl]-3,3-bis(methylthio)-2-propenenitrileHomo sapiens (human)IC5010.000010
1-hexadecyl-3-methylimidazolium bromideHomo sapiens (human)IC502.210010
N-[1-[[anilino(sulfanylidene)methyl]amino]-2,2,2-trichloroethyl]-2-(4-ethylphenoxy)acetamideHomo sapiens (human)IC5010.000010
3-(5-chloro-2-hydroxyphenyl)-3-phenyl-N-[(4-propan-2-yloxyphenyl)methyl]propanamideHomo sapiens (human)IC5010.000010
4-oxido-3-(4-phenoxyphenyl)-4a,5,6,7,8,8a-hexahydroquinoxalin-1-ium 1-oxideHomo sapiens (human)IC5010.000010
N-cyclohexyl-2-[3-methoxy-N-(1-oxo-2-thiophen-2-ylethyl)-4-(1-tetrazolyl)anilino]-2-(4-methylphenyl)acetamideHomo sapiens (human)IC5010.000010
2-[[2-(4-ethoxyphenyl)-5-methyl-4-oxazolyl]methylthio]-N-(2-furanylmethyl)acetamideHomo sapiens (human)IC503.805021
1-(4-methyl-2-prop-2-enylphenoxy)-3-(4-phenyl-1-piperazinyl)-2-propanolHomo sapiens (human)IC509.690010
5-amino-1-(2,3-dihydro-1,4-benzodioxin-6-yl)-N-[2-(3,4-dimethoxyphenyl)ethyl]-4-triazolecarboxamideHomo sapiens (human)IC5010.000010
6-[2-butylimino-3-(cyclopentylideneamino)-4-thiazolyl]-4H-1,4-benzoxazin-3-oneHomo sapiens (human)IC508.070010
1-(4-butylphenyl)-3-[4-chloro-3-(dimethylsulfamoyl)phenyl]thioureaHomo sapiens (human)IC5010.000010
3-[(4-ethylphenoxy)methyl]-4-(6-methylheptan-2-yl)-1H-1,2,4-triazole-5-thioneHomo sapiens (human)IC505.530010
1-[(4-chlorophenyl)methyl]-3-(3-fluorophenyl)-1-(3,3,3-trifluoro-2-hydroxypropyl)ureaHomo sapiens (human)IC506.090010
2-[[2-(1-adamantyl)-2-oxoethyl]thio]-6-amino-4-(4-chlorophenyl)pyridine-3,5-dicarbonitrileHomo sapiens (human)IC5010.000010
[3,5-bis(difluoromethyl)-5-hydroxy-4H-pyrazol-1-yl]-[2-(4-propan-2-ylphenyl)-4-quinolinyl]methanoneHomo sapiens (human)IC505.020010
3-[(4-methoxyphenoxy)methyl]-N-(4-nitro-1-pyrazolyl)benzamideHomo sapiens (human)IC500.330010
LSM-24595Homo sapiens (human)IC5010.000010
N,N-dicyclohexyl-5-propyl-3-isoxazolecarboxamideHomo sapiens (human)IC5010.000010
bornyl ferulateHomo sapiens (human)IC5010.000010
dithiazanine iodideHomo sapiens (human)IC502.400010
kolavenic acidHomo sapiens (human)IC5010.000010
cycloheximideHomo sapiens (human)IC500.210010
garcinone eHomo sapiens (human)IC505.240010
protoapigenoneHomo sapiens (human)IC503.840010
4-[5-(4-ethoxyphenyl)-3-isoxazolyl]-N-[(4-methylphenyl)methyl]butanamideHomo sapiens (human)IC500.290010
calcimycinHomo sapiens (human)IC501.410010
2-(3-chloro-N-(2-chloro-1-oxoethyl)anilino)-N-cyclohexyl-2-(4-methoxyphenyl)acetamideHomo sapiens (human)IC509.490010
(3E,9E)-5,6-Dihydroxy-9,13,14-trimethyl-16-(2-methylpropyl)-17-azatricyclo[9.7.0.01,15]octadeca-3,9,12-triene-2,18-dioneHomo sapiens (human)IC506.340010
(3aS,5S,9aS)-5-[1-(2-methoxyphenyl)-4-pyrazolyl]-2-phenyl-3a,4,5,7,8,9-hexahydro-3H-pyrrolo[3,4-h]pyrrolizin-1-oneHomo sapiens (human)IC500.740010
[1-[(7-chloro-3-methyl-1H-indol-2-yl)methyl]-4-(2-phenoxyethyl)-4-piperidinyl]methanolHomo sapiens (human)IC5010.000010
4-[3-(4-methoxyphenyl)-1H-pyrazol-5-yl]-1-[[3-(trifluoromethyl)phenyl]methyl]piperidineHomo sapiens (human)IC507.130010
2-[[[4-[(4-chloroanilino)-oxomethyl]-1H-imidazol-5-yl]-oxomethyl]amino]acetic acid tert-butyl esterHomo sapiens (human)IC509.830010
(2S)-2-[[[4-[[4-[[[(2-methylpropan-2-yl)oxy-oxomethyl]amino]methyl]anilino]-oxomethyl]-1H-imidazol-5-yl]-oxomethyl]amino]propanoic acid tert-butyl esterHomo sapiens (human)IC506.190010
N-(1H-benzimidazol-2-yl)-1-ethyl-4-hydroxy-2-oxo-3-quinolinecarboxamideHomo sapiens (human)IC507.940010
2-[(7-methoxy-4-methyl-2-quinazolinyl)amino]-5,6-dimethyl-1H-pyrimidin-4-oneHomo sapiens (human)IC500.160010
2-(4-fluoroanilino)-6-methyl-5-(3-methylbutyl)-1H-pyrimidin-4-oneHomo sapiens (human)IC506.000010