Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
fluspirilene | Mus musculus (house mouse) | IC50 | 7.7600 | 1 | 0 |
terfenadine | Mus musculus (house mouse) | IC50 | 4.1200 | 1 | 0 |
pimozide | Mus musculus (house mouse) | IC50 | 6.3400 | 1 | 0 |
nsc 3852 | Mus musculus (house mouse) | IC50 | 8.8300 | 1 | 0 |
1,6-bismaleimidohexane | Mus musculus (house mouse) | IC50 | 4.9400 | 1 | 0 |
helenalin | Mus musculus (house mouse) | IC50 | 2.6100 | 1 | 0 |
isovelleral | Mus musculus (house mouse) | IC50 | 0.8500 | 1 | 0 |
9-methoxyellipticine | Mus musculus (house mouse) | IC50 | 5.2800 | 1 | 0 |
2-phenyl-4,5-dichloro-3-pyridazinone | Mus musculus (house mouse) | IC50 | 9.4500 | 1 | 0 |
girinimbine | Mus musculus (house mouse) | IC50 | 10.0000 | 1 | 0 |
3,3-bis(4-hydroxy-3-methylphenyl)-1H-indol-2-one | Mus musculus (house mouse) | IC50 | 10.0000 | 1 | 0 |
aromaticin | Mus musculus (house mouse) | IC50 | 10.0000 | 1 | 0 |
angustibalin | Mus musculus (house mouse) | IC50 | 2.4800 | 1 | 0 |
cgp 60474 | Mus musculus (house mouse) | IC50 | 0.1600 | 1 | 0 |
2-[(1-cyclohexyl-5-tetrazolyl)thio]-N-(6-ethoxy-1,3-benzothiazol-2-yl)acetamide | Mus musculus (house mouse) | IC50 | 10.0000 | 1 | 0 |
8-(butan-2-ylthio)-7-[(4-chlorophenyl)methyl]-3-methylpurine-2,6-dione | Mus musculus (house mouse) | IC50 | 10.0000 | 1 | 0 |
(1S,2R)-2-(octylamino)-1-[4-(propan-2-ylthio)phenyl]-1-propanol | Mus musculus (house mouse) | IC50 | 2.5300 | 1 | 0 |
1-[5-(trifluoromethyl)-1,3,4-thiadiazol-2-yl]-3-[1,1,1-trifluoro-2-(trifluoromethyl)butan-2-yl]urea | Mus musculus (house mouse) | IC50 | 2.5600 | 1 | 0 |
4-(cyclohexylamino)-2-(3,5-dimethyl-1-pyrazolyl)-5-pyrimidinecarboxylic acid ethyl ester | Mus musculus (house mouse) | IC50 | 10.0000 | 1 | 0 |
3-(3-benzoyl-6-chloro-4,5-dihydroxy-7-benzofuranyl)pentane-2,4-dione | Mus musculus (house mouse) | IC50 | 5.6700 | 1 | 0 |
N-[2-[5-[(2,4-dichlorophenyl)methylsulfonyl]-1,3,4-oxadiazol-2-yl]ethyl]carbamic acid tert-butyl ester | Mus musculus (house mouse) | IC50 | 10.0000 | 1 | 0 |
4-chloro-1-methyl-3-nitro-2-quinolinone | Mus musculus (house mouse) | IC50 | 3.3400 | 1 | 0 |
2-(dichloromethyl)-4-(ethylthio)-6-phenyl-1,3,5-triazine | Mus musculus (house mouse) | IC50 | 6.3200 | 1 | 0 |
4-chloro-3-ethoxy-N-(4-ethylphenyl)benzenesulfonamide | Mus musculus (house mouse) | IC50 | 4.4800 | 1 | 0 |
LSM-16285 | Mus musculus (house mouse) | IC50 | 9.8100 | 1 | 0 |
2-(4-methylsulfonyl-2-nitrophenyl)sulfinylacetic acid (phenylmethyl) ester | Mus musculus (house mouse) | IC50 | 10.0000 | 1 | 0 |
N-(2,5-dimethylphenyl)-2-[[3-(4-ethylphenoxy)-4-oxo-1-benzopyran-7-yl]oxy]acetamide | Mus musculus (house mouse) | IC50 | 5.2300 | 1 | 0 |
N-[[3-(4-fluorophenyl)-1-phenyl-4-pyrazolyl]methyl]-1-phenylmethanamine | Mus musculus (house mouse) | IC50 | 9.6200 | 1 | 0 |
5-[(cyclohexylamino)-oxomethyl]-4-methyl-2-[(1-oxo-2-thiophen-2-ylethyl)amino]-3-thiophenecarboxylic acid ethyl ester | Mus musculus (house mouse) | IC50 | 2.9900 | 1 | 0 |
2-[2-(2,4-dichloro-5-propan-2-yloxyanilino)-2-oxoethyl]sulfinyl-N-[3-(trifluoromethyl)phenyl]acetamide | Mus musculus (house mouse) | IC50 | 7.9900 | 1 | 0 |
(4-chlorophenyl)-[4-[[(2,4-dichlorophenyl)thio]methyl]-4-hydroxy-1-piperidinyl]methanone | Mus musculus (house mouse) | IC50 | 10.0000 | 1 | 0 |
3-amino-N-(2-fluorophenyl)-6-(3-pyridinyl)-2-thieno[2,3-b]pyridinecarboxamide | Mus musculus (house mouse) | IC50 | 10.0000 | 1 | 0 |
2-(3,5-dimethyl-1-pyrazolyl)-4-(4-hydroxyanilino)-5-pyrimidinecarboxylic acid ethyl ester | Mus musculus (house mouse) | IC50 | 1.5100 | 1 | 0 |
4-[bis(2-methylpropyl)sulfamoyl]-N-[5-(3-methoxyphenyl)-1,3,4-oxadiazol-2-yl]benzamide | Mus musculus (house mouse) | IC50 | 4.1300 | 1 | 0 |
6-bromo-2-(3-pyridinyl)-N-[4-(trifluoromethyl)phenyl]-4-quinolinecarboxamide | Mus musculus (house mouse) | IC50 | 3.5900 | 1 | 0 |
5,6,7,8-tetrafluoro-2-(2,3,4,5,6-pentafluorophenyl)-4h-1-benzopyran-4-one | Mus musculus (house mouse) | IC50 | 3.9800 | 1 | 0 |
2-(2,6-dichlorophenyl)acetic acid [2-oxo-2-[4-(trifluoromethoxy)anilino]ethyl] ester | Mus musculus (house mouse) | IC50 | 10.0000 | 1 | 0 |
2-[(3-methoxyphenyl)-oxomethyl]-3,3-bis(methylthio)-2-propenenitrile | Mus musculus (house mouse) | IC50 | 10.0000 | 1 | 0 |
1-hexadecyl-3-methylimidazolium bromide | Mus musculus (house mouse) | IC50 | 0.8600 | 1 | 0 |
N-[1-[[anilino(sulfanylidene)methyl]amino]-2,2,2-trichloroethyl]-2-(4-ethylphenoxy)acetamide | Mus musculus (house mouse) | IC50 | 8.1200 | 1 | 0 |
3-(5-chloro-2-hydroxyphenyl)-3-phenyl-N-[(4-propan-2-yloxyphenyl)methyl]propanamide | Mus musculus (house mouse) | IC50 | 9.5900 | 1 | 0 |
4-oxido-3-(4-phenoxyphenyl)-4a,5,6,7,8,8a-hexahydroquinoxalin-1-ium 1-oxide | Mus musculus (house mouse) | IC50 | 10.0000 | 1 | 0 |
N-cyclohexyl-2-[3-methoxy-N-(1-oxo-2-thiophen-2-ylethyl)-4-(1-tetrazolyl)anilino]-2-(4-methylphenyl)acetamide | Mus musculus (house mouse) | IC50 | 9.9400 | 1 | 0 |
2-[[2-(4-ethoxyphenyl)-5-methyl-4-oxazolyl]methylthio]-N-(2-furanylmethyl)acetamide | Mus musculus (house mouse) | IC50 | 2.2650 | 2 | 1 |
1-(4-methyl-2-prop-2-enylphenoxy)-3-(4-phenyl-1-piperazinyl)-2-propanol | Mus musculus (house mouse) | IC50 | 3.9400 | 1 | 0 |
5-amino-1-(2,3-dihydro-1,4-benzodioxin-6-yl)-N-[2-(3,4-dimethoxyphenyl)ethyl]-4-triazolecarboxamide | Mus musculus (house mouse) | IC50 | 0.6900 | 1 | 0 |
6-[2-butylimino-3-(cyclopentylideneamino)-4-thiazolyl]-4H-1,4-benzoxazin-3-one | Mus musculus (house mouse) | IC50 | 8.0000 | 1 | 0 |
1-(4-butylphenyl)-3-[4-chloro-3-(dimethylsulfamoyl)phenyl]thiourea | Mus musculus (house mouse) | IC50 | 10.0000 | 1 | 0 |
3-[(4-ethylphenoxy)methyl]-4-(6-methylheptan-2-yl)-1H-1,2,4-triazole-5-thione | Mus musculus (house mouse) | IC50 | 2.4400 | 1 | 0 |
1-[(4-chlorophenyl)methyl]-3-(3-fluorophenyl)-1-(3,3,3-trifluoro-2-hydroxypropyl)urea | Mus musculus (house mouse) | IC50 | 3.5800 | 1 | 0 |
2-[[2-(1-adamantyl)-2-oxoethyl]thio]-6-amino-4-(4-chlorophenyl)pyridine-3,5-dicarbonitrile | Mus musculus (house mouse) | IC50 | 10.0000 | 1 | 0 |
[3,5-bis(difluoromethyl)-5-hydroxy-4H-pyrazol-1-yl]-[2-(4-propan-2-ylphenyl)-4-quinolinyl]methanone | Mus musculus (house mouse) | IC50 | 8.3800 | 1 | 0 |
3-[(4-methoxyphenoxy)methyl]-N-(4-nitro-1-pyrazolyl)benzamide | Mus musculus (house mouse) | IC50 | 0.8500 | 1 | 0 |
LSM-24595 | Mus musculus (house mouse) | IC50 | 10.0000 | 1 | 0 |
N,N-dicyclohexyl-5-propyl-3-isoxazolecarboxamide | Mus musculus (house mouse) | IC50 | 10.0000 | 1 | 0 |
bornyl ferulate | Mus musculus (house mouse) | IC50 | 9.5200 | 1 | 0 |
dithiazanine iodide | Mus musculus (house mouse) | IC50 | 0.8700 | 1 | 0 |
kolavenic acid | Mus musculus (house mouse) | IC50 | 9.6800 | 1 | 0 |
cycloheximide | Mus musculus (house mouse) | IC50 | 0.1600 | 1 | 0 |
garcinone e | Mus musculus (house mouse) | IC50 | 9.6700 | 1 | 0 |
protoapigenone | Mus musculus (house mouse) | IC50 | 2.5800 | 1 | 0 |
4-[5-(4-ethoxyphenyl)-3-isoxazolyl]-N-[(4-methylphenyl)methyl]butanamide | Mus musculus (house mouse) | IC50 | 5.9100 | 1 | 0 |
calcimycin | Mus musculus (house mouse) | IC50 | 0.1600 | 1 | 0 |
2-(3-chloro-N-(2-chloro-1-oxoethyl)anilino)-N-cyclohexyl-2-(4-methoxyphenyl)acetamide | Mus musculus (house mouse) | IC50 | 9.5700 | 1 | 0 |
(3E,9E)-5,6-Dihydroxy-9,13,14-trimethyl-16-(2-methylpropyl)-17-azatricyclo[9.7.0.01,15]octadeca-3,9,12-triene-2,18-dione | Mus musculus (house mouse) | IC50 | 9.6900 | 1 | 0 |
(3aS,5S,9aS)-5-[1-(2-methoxyphenyl)-4-pyrazolyl]-2-phenyl-3a,4,5,7,8,9-hexahydro-3H-pyrrolo[3,4-h]pyrrolizin-1-one | Mus musculus (house mouse) | IC50 | 1.8900 | 1 | 0 |
[1-[(7-chloro-3-methyl-1H-indol-2-yl)methyl]-4-(2-phenoxyethyl)-4-piperidinyl]methanol | Mus musculus (house mouse) | IC50 | 9.1300 | 1 | 0 |
4-[3-(4-methoxyphenyl)-1H-pyrazol-5-yl]-1-[[3-(trifluoromethyl)phenyl]methyl]piperidine | Mus musculus (house mouse) | IC50 | 4.1100 | 1 | 0 |
2-[[[4-[(4-chloroanilino)-oxomethyl]-1H-imidazol-5-yl]-oxomethyl]amino]acetic acid tert-butyl ester | Mus musculus (house mouse) | IC50 | 4.6900 | 1 | 0 |
(2S)-2-[[[4-[[4-[[[(2-methylpropan-2-yl)oxy-oxomethyl]amino]methyl]anilino]-oxomethyl]-1H-imidazol-5-yl]-oxomethyl]amino]propanoic acid tert-butyl ester | Mus musculus (house mouse) | IC50 | 10.0000 | 1 | 0 |
N-(1H-benzimidazol-2-yl)-1-ethyl-4-hydroxy-2-oxo-3-quinolinecarboxamide | Mus musculus (house mouse) | IC50 | 5.8400 | 1 | 0 |
2-[(7-methoxy-4-methyl-2-quinazolinyl)amino]-5,6-dimethyl-1H-pyrimidin-4-one | Mus musculus (house mouse) | IC50 | 9.7200 | 1 | 0 |
2-(4-fluoroanilino)-6-methyl-5-(3-methylbutyl)-1H-pyrimidin-4-one | Mus musculus (house mouse) | IC50 | 2.4300 | 1 | 0 |