Page last updated: 2024-08-07 16:18:45
Beta-3 adrenergic receptor
A beta-3 adrenergic receptor that is encoded in the genome of rat. [OMA:P26255, PRO:DNx]
Synonyms
Beta-3 adrenoreceptor;
Beta-3 adrenoceptor
Research
Bioassay Publications (19)
| Timeframe | Studies on this Protein(%) | All Drugs % |
|---|
| pre-1990 | 8 (42.11) | 18.7374 |
| 1990's | 7 (36.84) | 18.2507 |
| 2000's | 3 (15.79) | 29.6817 |
| 2010's | 1 (5.26) | 24.3611 |
| 2020's | 0 (0.00) | 2.80 |
Compounds (26)
Drugs with Inhibition Measurements
Drugs with Activation Measurements
Syntheses of 2,5- and 2,6-difluoronorepinephrine, 2,5-difluoroepinephrine, and 2,6-difluorophenylephrine: effect of disubstitution with fluorine on adrenergic activity.Journal of medicinal chemistry, , Nov-26, Volume: 36, Issue:24, 1993
Discovery of novel N-phenylglycine derivatives as potent and selective beta(3)-adrenoceptor agonists for the treatment of frequent urination and urinary incontinence.Journal of medicinal chemistry, , Apr-26, Volume: 44, Issue:9, 2001
Effect of fluorine substitution on the adrenergic properties of 3-(tert-butylamino)-1-(3,4-dihydroxyphenoxy)-2-propanol.Journal of medicinal chemistry, , Volume: 34, Issue:3, 1991
Carbostyril derivatives having potent beta-adrenergic agonist properties.Journal of medicinal chemistry, , Volume: 30, Issue:9, 1987
Syntheses and adrenergic agonist properties of ring-fluorinated isoproterenols.Journal of medicinal chemistry, , Volume: 25, Issue:6, 1982
Synthesis and adrenergic activity of a new series of N-aryl dicyclopropyl ketone oxime ethers: SAR and stereochemical aspects.Journal of medicinal chemistry, , May-07, Volume: 41, Issue:10, 1998
Flavones. 2. Synthesis and structure-activity relationship of flavodilol and its analogues, a novel class of antihypertensive agents with catecholamine depleting properties.Journal of medicinal chemistry, , Volume: 32, Issue:1, 1989
Syntheses and adrenergic agonist properties of ring-fluorinated isoproterenols.Journal of medicinal chemistry, , Volume: 25, Issue:6, 1982
Syntheses of 2,5- and 2,6-difluoronorepinephrine, 2,5-difluoroepinephrine, and 2,6-difluorophenylephrine: effect of disubstitution with fluorine on adrenergic activity.Journal of medicinal chemistry, , Nov-26, Volume: 36, Issue:24, 1993
Novel and potent human and rat beta3-adrenergic receptor agonists containing substituted 3-indolylalkylamines.Bioorganic & medicinal chemistry letters, , Apr-07, Volume: 13, Issue:7, 2003
Discovery of novel N-phenylglycine derivatives as potent and selective beta(3)-adrenoceptor agonists for the treatment of frequent urination and urinary incontinence.Journal of medicinal chemistry, , Apr-26, Volume: 44, Issue:9, 2001