A protein that is a translation product of the CCKAR gene in guinea pig. [PRO:DNx, UniProtKB:Q63931]
CCK-A receptor;
CCK-AR;
Cholecystokinin-1 receptor;
CCK1-R
| Timeframe | Studies on this Protein(%) | All Drugs % |
|---|---|---|
| pre-1990 | 4 (20.00) | 18.7374 |
| 1990's | 12 (60.00) | 18.2507 |
| 2000's | 3 (15.00) | 29.6817 |
| 2010's | 0 (0.00) | 24.3611 |
| 2020's | 1 (5.00) | 2.80 |
| Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
|---|---|---|---|---|---|
| alprazolam | Cavia porcellus (domestic guinea pig) | IC50 | 64.0000 | 1 | 1 |
| haloperidol | Cavia porcellus (domestic guinea pig) | Ki | 0.0500 | 1 | 1 |
| lorglumide | Cavia porcellus (domestic guinea pig) | IC50 | 2.2000 | 1 | 1 |
| proglumide | Cavia porcellus (domestic guinea pig) | IC50 | 800.0000 | 1 | 1 |
| triazolam | Cavia porcellus (domestic guinea pig) | IC50 | 39.0000 | 1 | 1 |
| ci 988 | Cavia porcellus (domestic guinea pig) | Ki | 0.6310 | 1 | 1 |
| a 71623 | Cavia porcellus (domestic guinea pig) | IC50 | 1.9000 | 1 | 2 |
| devazepide | Cavia porcellus (domestic guinea pig) | IC50 | 0.2700 | 1 | 1 |
| tetragastrin | Cavia porcellus (domestic guinea pig) | Ki | 36.1330 | 2 | 2 |
| benzotript | Cavia porcellus (domestic guinea pig) | IC50 | 100.0000 | 1 | 1 |
| a 65186 | Cavia porcellus (domestic guinea pig) | IC50 | 1.1701 | 3 | 3 |
| cholecystokinin (27-33), tert-butyloxycarbonyl-nle(28,31)- | Cavia porcellus (domestic guinea pig) | IC50 | 0.0009 | 1 | 1 |
| cholecystokinin (27-33), tert-butyloxycarbonyl-nle(28,31)- | Cavia porcellus (domestic guinea pig) | Ki | 0.0009 | 1 | 1 |
| l 365260 | Cavia porcellus (domestic guinea pig) | IC50 | 0.0440 | 2 | 2 |
| l 365260 | Cavia porcellus (domestic guinea pig) | Ki | 0.3920 | 2 | 2 |
| sincalide | Cavia porcellus (domestic guinea pig) | IC50 | 0.0004 | 1 | 1 |
| sincalide | Cavia porcellus (domestic guinea pig) | Ki | 0.0005 | 7 | 7 |
| yf 476 | Cavia porcellus (domestic guinea pig) | Ki | 0.3981 | 1 | 1 |
| butyloxycarbonyl-tryptophyl-methionyl-aspartyl-phenylalaninamide | Cavia porcellus (domestic guinea pig) | IC50 | 1.8000 | 4 | 4 |
| butyloxycarbonyl-tryptophyl-methionyl-aspartyl-phenylalaninamide | Cavia porcellus (domestic guinea pig) | Ki | 11.9000 | 1 | 1 |
| clozapine | Cavia porcellus (domestic guinea pig) | Ki | 0.0600 | 1 | 1 |