A substance used as an indicator of a biological state.
| Member | Definition | Class |
|---|
| 1,3,5-trimethoxybenzene | A methoxybenzene carrying methoxy groups at positions 1, 3 and 5. It has been found to be a biomarker of flavonoid consumption in humans. | 1,3,5-trimethoxybenzene |
| 1,6-anhydro-beta-glucopyranose | A anhydrohexose that is the 1,6-anhydro-derivative of beta-D-glucopyranose. | levoglucosan |
| 24-hydroxycholesterol | A 24-hydroxycholesterol that has S configuration at position 24. It is the major metabolic breakdown product of cholesterol in the brain. | (24S)-24-hydroxycholesterol |
| 3-[1-(2,6-dichloro-3-fluorophenyl)ethoxy]-5-[1-(piperidin-4-yl)pyrazol-4-yl]pyridin-2-amine | A racemate comprising equimolar amounts of (R)- and (S)-crizotinib. The active (R)-enantiomer acts as a kinase inhibitor and is used for the treatment of patients with locally advanced or metastatic non-small cell lung cancer. | 3-[1-(2,6-dichloro-3-fluorophenyl)ethoxy]-5-[1-(piperidin-4-yl)pyrazol-4-yl]pyridin-2-amine; rac-crizotinib |
| 3-chloro-L-tyrosine | A chloroamino acid comprising a tyrosine core with a chloro- substituent ortho to the phenolic hydroxy group. | 3-chloro-L-tyrosine zwitterion; 3-chloro-L-tyrosine |
| 3-methoxytyramine | A monomethoxybenzene that is dopamine in which the hydroxy group at position 3 is replaced by a methoxy group. It is a metabolite of the neurotransmitter dopamine and considered a potential biomarker of pheochromocytomas and paragangliomas. | 3-methoxytyramine |
| 3-octanone | A dialkyl ketone that is octane in which the two methylene protons at position 3 have been replaced by an oxo group. | 3-octanone |
| 4-(methylnitrosamino)-1-(3-pyridyl)-1-butan-1-ol | A member of the class of nitrosamines that is butan-1-ol substituted by a pyridin-3-yl group at position 1 and by a methyl(nitroso)amino group at position 4. It is a major metabolite of nitrosamine 4-(methylnitrosamino)-1-(3-pyridyl)-1-butanone (NNK), which is a carcinogen found in tobacco and responsible for inducing lung cancer in smokers. | 4-(methylnitrosamino)-1-(3-pyridyl)-1-butanol |
| 4-heptanone | A dialkyl ketone that is heptane in which the two methylene protons at position 4 have been replaced by an oxo group. | 4-heptanone |
| 5,6-dihydrouridine | The uridine derivative obtained by formal hydrogenation of the endocyclic double bond in the uracil ring. | dihydrouridine |
| 8-epi-prostaglandin f2alpha | An isoprostane that is prostaglandin F2alpha having inverted stereochemistry at the 8-position. | 8-epi-prostaglandin F2alpha |
| 8-hydroxy-2'-deoxyguanosine | Guanosine substituted at the purine 8-position by a hydroxy group. It is used as a biomarker of oxidative DNA damage. | 8-hydroxy-2'-deoxyguanosine |
| 8-nitroguanosine 3',5'-cyclic monophosphate | A 3',5'-cyclic purine nucleotide that is guanosine 3',5'-cyclic monophosphate in which the hydrogen at position 8 on the purine fragment has been replaced by a nitro group. | 8-nitroguanosine 3',5'-cyclic monophosphate |
| apelin-12 peptide | A 12 amino acid oligopeptide fragment of apelin-13 lacking the terminal L-phenylalanine residue. | apelin-12 |
| apelin-13 peptide | A 13 amino acid oligopeptide which is the ligand for the apelin receptor (also known as the APJ receptor). It exhibits hypotensive and neuroprotective effects, and may be a potential prognostic biomarker for acute ischemic stroke and multiple sclerosis. | apelin-13 |
| arginine | An L-alpha-amino acid that is the L-isomer of arginine. | L-arginine |
| brassicasterol | An 3beta-sterol that is (22E)-ergosta-5,22-diene substituted by a hydroxy group at position 3beta. It is a phytosterol found in marine algae, fish, and rapeseed oil. | brassicasterol |
| butyraldehyde | A member of the class of butanals that consists of propane bearing a formyl substituent at the 1-position. The parent of the class of butanals. | butanal |
| carbon monoxide | A one-carbon compound in which the carbon is joined only to a single oxygen. It is a colourless, odourless, tasteless, toxic gas. | carbon monoxide |
| cotinine | An N-alkylpyrrolidine that consists of N-methylpyrrolidinone bearing a pyridin-3-yl substituent at position C-5 (the 5S-enantiomer). It is an alkaloid commonly found in Nicotiana tabacum. | (-)-cotinine |
| crizotinib | A 3-[1-(2,6-dichloro-3-fluorophenyl)ethoxy]-5-[1-(piperidin-4-yl)pyrazol-4-yl]pyridin-2-amine that has R configuration at the chiral centre. The active enantiomer, it acts as a kinase inhibitor and is used for the treatment of patients with locally advanced or metastatic non-small cell lung cancer (NSCLC) | crizotinib |
| cryptoxanthins | A carotenol that exhibits antioxidant activity. It has been isolated from fruits such as papaya and oranges. | beta-cryptoxanthin |
| dehydroergosterol | A phytosterol consiting of ergostane having double bonds at the 5,6-, 7,8- 9,11- and 22,23-positions as well as a 3beta-hydroxy group. | dehydroergosterol |
| delta(9)-tetrahydrocannabinolic acid | A diterpenoid that is 6a,7,8,10a-tetrahydro-6H-benzo[c]chromene substituted at position 1 by a hydroxy group, positions 6, 6 and 9 by methyl groups and at position 3 by a pentyl group. A biosynthetic precursor to Delta(9)-tetrahydrocannabinol, the principal psychoactive constituent of the cannabis plant. | Delta(9)-tetrahydrocannabinolic acid |
| dityrosine | A biphenyl compound comprising two tyrosine residues linked at carbon-3 of their benzene rings. | dityrosine |
| guanosine monophosphate | A purine ribonucleoside 5'-monophosphate having guanine as the nucleobase. | guanosine 5'-monophosphate |
| hawkinsin | A cysteine derivative that is cysteine in which the thiol group is substituted by a [2-(carboxymethyl)-2,5-dihydroxycyclohex-3-en-1-yl]sulfanediyl group. Hawkinsinuria is an inherited disorder which is characterized by the inability to break down the amino acid tyrosine. This results in the finding of certain metabolites in the urine, such as hawkinsin. | hawkinsin |
| heptanal | An n-alkanal resulting from the oxidation of the alcoholic hydroxy group of heptan-1-ol to the corresponding aldehyde. An endogenous aldehyde coming from membrane lipid oxidation, it is found in the blood of lung cancer patients and has been regarded as a potential biomarker of lung cancer. | heptanal |
| homoarginine | An L-lysine derivative that is the L-enantiomer of homoarginine. | L-homoarginine |
| isodesmosine | A pyridinium ion obtained by formal condensation of four molecules of lysine. | isodesmosine |
| isoferulic acid | A ferulic acid consisting of trans-cinnamic acid bearing methoxy and hydroxy substituents at positions 4 and 3 respectively on the phenyl ring. | isoferulic acid |
| malondialdehyde | A dialdehyde that is propane substituted by two oxo groups at the terminal carbon atoms respectively. A biomarker of oxidative damage to lipids caused by smoking, it exists in vivo mainly in the enol form. | malonaldehyde |
| muconic acid | The trans,trans-isomer of muconic acid. It is metabolite of benzene in humans and serves as a biomarker of occupational exposure to benzene. | trans,trans-muconic acid |
| n-acetyltyrosine | An N-acetyltyrosine in which the chiral centre has L configuration. | N-acetyl-L-tyrosine |
| nicotine | A 3-(1-methylpyrrolidin-2-yl)pyridine in which the chiral centre has S-configuration. The naturally occurring and most active enantiomer of nicotine, isolated from Nicotiana tabacum. | (S)-nicotine |
| ophthalmic acid | A L-glutamine derivative that is L-glutamine substituted by a 1-[(carboxymethyl)amino]-1-oxobutan-2-yl at the terminal amino nitrogen atom. | ophthalmic acid |
| pentosidine | An imidazopyridine having norleucine and ornithine residues attached via their side-chains at the 4- and 2-positions respectively. | pentosidine |
| phenylglyoxylic acid | A 2-oxo monocarboxylic acid that is glyoxylic acid in which the aldehyde hydrogen is substituted by a phenyl group. | phenylglyoxylic acid |
| pristane | A norterpene that is an acyclic saturated hydrocarbon derived from phytane by loss of its C-16 terminal methyl group. | pristane |
| rubidium chloride | An inorganic chloride composed of rubidium and chloride ions in a 1:1 ratio. | rubidium chloride |
| s-phenyl-n-acetylcysteine | The S-phenyl derivative of N-acetyl-L-cysteine. It is a urinary metabolite of benzene and used as a biomarker to assess benzene exposure. | N-acetyl-S-phenyl-L-cysteine |
| ubiquinol | A ubiquinol in which the polyprenyl substituent is decaprenyl. | ubiquinol-10 |
| ubiquinone 8 | A ubiquinone whose structure comprises a 2,3-dimethoxy-5-methylbenzoquinone nucleus (common to all ubiquinones) and a side chain of eight isoprenoid units. | ubiquinone-8 |
| Protein | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Drugs |
|---|
| 5-hydroxytryptamine receptor 3A | Homo sapiens (human) | Ki | 71.0000 | 1 | 2 |
| 5-hydroxytryptamine receptor 3B | Homo sapiens (human) | Ki | 71.0000 | 1 | 2 |
| 5-hydroxytryptamine receptor 3C | Homo sapiens (human) | Ki | 71.0000 | 1 | 2 |
| 5-hydroxytryptamine receptor 3D | Homo sapiens (human) | Ki | 71.0000 | 1 | 2 |
| 5-hydroxytryptamine receptor 3E | Homo sapiens (human) | Ki | 71.0000 | 1 | 2 |
| Acetylcholine receptor subunit alpha | Homo sapiens (human) | IC50 | 11.0000 | 2 | 2 |
| Acetylcholine receptor subunit alpha | Tetronarce californica (Pacific electric ray) | IC50 | 0.0025 | 2 | 2 |
| Acetylcholine receptor subunit alpha | Homo sapiens (human) | Ki | 3.3139 | 4 | 4 |
| Acetylcholine receptor subunit alpha | Tetronarce californica (Pacific electric ray) | Ki | 8.1350 | 2 | 2 |
| Acetylcholine receptor subunit beta | Homo sapiens (human) | IC50 | 1.0000 | 1 | 1 |
| Acetylcholine receptor subunit beta | Tetronarce californica (Pacific electric ray) | IC50 | 0.0025 | 2 | 2 |
| Acetylcholine receptor subunit beta | Homo sapiens (human) | Ki | 3.3139 | 4 | 4 |
| Acetylcholine receptor subunit beta | Tetronarce californica (Pacific electric ray) | Ki | 8.1350 | 2 | 2 |
| Acetylcholine receptor subunit beta-like 2 | Drosophila melanogaster (fruit fly) | IC50 | 4.0000 | 1 | 1 |
| Acetylcholine receptor subunit beta-like 2 | Drosophila melanogaster (fruit fly) | Ki | 2.7000 | 1 | 1 |
| Acetylcholine receptor subunit delta | Homo sapiens (human) | IC50 | 1.0000 | 1 | 1 |
| Acetylcholine receptor subunit delta | Tetronarce californica (Pacific electric ray) | IC50 | 0.0025 | 2 | 2 |
| Acetylcholine receptor subunit delta | Homo sapiens (human) | Ki | 3.3139 | 4 | 4 |
| Acetylcholine receptor subunit delta | Tetronarce californica (Pacific electric ray) | Ki | 8.1350 | 2 | 2 |
| Acetylcholine receptor subunit gamma | Homo sapiens (human) | IC50 | 1.0000 | 1 | 1 |
| Acetylcholine receptor subunit gamma | Tetronarce californica (Pacific electric ray) | IC50 | 0.0025 | 2 | 2 |
| Acetylcholine receptor subunit gamma | Homo sapiens (human) | Ki | 3.3139 | 4 | 4 |
| Acetylcholine receptor subunit gamma | Tetronarce californica (Pacific electric ray) | Ki | 8.1350 | 2 | 2 |
| Acetylcholine-binding protein | Lymnaea stagnalis (great pond snail) | Ki | 0.2236 | 7 | 8 |
| ALK tyrosine kinase receptor | Homo sapiens (human) | GI50 | 0.2130 | 7 | 7 |
| ALK tyrosine kinase receptor | Homo sapiens (human) | IC50 | 13.7068 | 103 | 108 |
| ALK tyrosine kinase receptor | Mus musculus (house mouse) | IC50 | 0.0800 | 1 | 1 |
| ALK tyrosine kinase receptor | Homo sapiens (human) | Ki | 0.0057 | 6 | 6 |
| Alkaline phosphatase, tissue-nonspecific isozyme | Homo sapiens (human) | IC50 | 5.0000 | 1 | 1 |
| Androgen receptor | Homo sapiens (human) | IC50 | 0.0020 | 1 | 1 |
| Angiopoietin-1 receptor | Homo sapiens (human) | IC50 | 0.2265 | 2 | 2 |
| Angiopoietin-1 receptor | Mus musculus (house mouse) | IC50 | 0.4480 | 1 | 1 |
| Apelin receptor | Homo sapiens (human) | Ki | 0.0007 | 1 | 1 |
| ATP-binding cassette sub-family C member 3 | Homo sapiens (human) | IC50 | 133.0000 | 1 | 1 |
| Aurora kinase A-interacting protein | Homo sapiens (human) | IC50 | 10.0000 | 1 | 1 |
| BDNF/NT-3 growth factors receptor | Homo sapiens (human) | IC50 | 0.2005 | 2 | 2 |
| Bile salt export pump | Homo sapiens (human) | IC50 | 422.6667 | 3 | 3 |
| C-terminal-binding protein 2 | Homo sapiens (human) | IC50 | 300.0000 | 1 | 1 |
| Canalicular multispecific organic anion transporter 1 | Homo sapiens (human) | IC50 | 133.0000 | 1 | 1 |
| Cannabinoid receptor 1 | Homo sapiens (human) | Ki | 0.0240 | 1 | 1 |
| Cannabinoid receptor 2 | Homo sapiens (human) | Ki | 0.0560 | 1 | 1 |
| Cationic amino acid transporter 3 | Homo sapiens (human) | IC50 | 283.0000 | 1 | 1 |
| Chain A, HYPOXANTHINE PHOSPHORIBOSYLTRANSFERASE | Escherichia coli | Ki | 526.0000 | 1 | 2 |
| Cyclin-dependent kinase 1 | Homo sapiens (human) | IC50 | 10.0000 | 1 | 1 |
| Cyclin-dependent kinase 7 | Homo sapiens (human) | IC50 | 10.0000 | 1 | 1 |
| Cytidine deaminase | Homo sapiens (human) | Ki | 40.0000 | 1 | 1 |
| Cytochrome P450 1A2 | Homo sapiens (human) | IC50 | 4,750.0000 | 1 | 2 |
| Cytochrome P450 2A13 | Homo sapiens (human) | Ki | 72.0000 | 1 | 1 |
| Cytochrome P450 2A5 | Mus musculus (house mouse) | IC50 | 829.9780 | 2 | 2 |
| Cytochrome P450 2A6 | Homo sapiens (human) | IC50 | 6,072.0048 | 3 | 6 |
| Cytochrome P450 2A6 | Homo sapiens (human) | Ki | 46.2667 | 3 | 3 |
| Cytochrome P450 3A4 | Homo sapiens (human) | IC50 | 146.2667 | 2 | 3 |
| Cytoplasmic tyrosine-protein kinase BMX | Homo sapiens (human) | IC50 | 10.0000 | 1 | 1 |
| Delta-type opioid receptor | Mus musculus (house mouse) | Ki | 0.4400 | 1 | 1 |
| Delta-type opioid receptor | Rattus norvegicus (Norway rat) | Ki | 0.1100 | 1 | 1 |
| Diacylglycerol lipase-alpha | Homo sapiens (human) | IC50 | 27.3000 | 1 | 1 |
| Echinoderm microtubule-associated protein-like 4 | Homo sapiens (human) | IC50 | 0.6542 | 15 | 15 |
| Ephrin type-A receptor 2 | Homo sapiens (human) | IC50 | 1.0000 | 1 | 1 |
| Ephrin type-B receptor 2 | Homo sapiens (human) | IC50 | 10.0000 | 1 | 1 |
| Ephrin type-B receptor 4 | Homo sapiens (human) | IC50 | 10.0000 | 1 | 1 |
| Epidermal growth factor receptor | Homo sapiens (human) | IC50 | 146.9544 | 7 | 7 |
| Fibroblast growth factor receptor 1 | Homo sapiens (human) | IC50 | 1.0000 | 1 | 1 |
| Fibroblast growth factor receptor 3 | Homo sapiens (human) | IC50 | 10.0000 | 1 | 1 |
| G2/mitotic-specific cyclin-B1 | Homo sapiens (human) | IC50 | 10.0000 | 1 | 1 |
| Hepatocyte growth factor receptor | Homo sapiens (human) | IC50 | 0.0063 | 33 | 35 |
| Hepatocyte growth factor receptor | Homo sapiens (human) | Ki | 0.0068 | 3 | 4 |
| High affinity nerve growth factor receptor | Homo sapiens (human) | IC50 | 0.2905 | 2 | 2 |
| HLA class II histocompatibility antigen gamma chain | Homo sapiens (human) | IC50 | 0.0039 | 1 | 1 |
| Hyaluronidase-1 | Homo sapiens (human) | IC50 | 2,000.0000 | 1 | 1 |
| Hypoxanthine-guanine phosphoribosyltransferase | Homo sapiens (human) | Ki | 5.8000 | 2 | 2 |
| Insulin receptor | Homo sapiens (human) | IC50 | 1.0966 | 5 | 5 |
| Insulin-like growth factor 1 receptor | Homo sapiens (human) | IC50 | 3.7143 | 3 | 3 |
| Intestinal-type alkaline phosphatase | Homo sapiens (human) | IC50 | 5.0000 | 1 | 1 |
| L-lactate dehydrogenase A chain | Homo sapiens (human) | Ki | 6.5000 | 1 | 1 |
| Liver carboxylesterase B-1 | Rattus norvegicus (Norway rat) | IC50 | 0.0450 | 1 | 1 |
| Lysine--tRNA ligase | Homo sapiens (human) | IC50 | 10.0000 | 1 | 1 |
| Macrophage colony-stimulating factor 1 receptor | Homo sapiens (human) | IC50 | 10.0000 | 1 | 1 |
| Macrophage-stimulating protein receptor | Homo sapiens (human) | IC50 | 0.2500 | 2 | 2 |
| Macrophage-stimulating protein receptor | Mus musculus (house mouse) | IC50 | 0.0800 | 1 | 1 |
| Mitogen-activated protein kinase 14 | Homo sapiens (human) | IC50 | 10.0000 | 1 | 1 |
| Mitogen-activated protein kinase kinase kinase kinase 3 | Homo sapiens (human) | IC50 | 0.8745 | 2 | 2 |
| Mu-type opioid receptor | Cavia porcellus (domestic guinea pig) | Ki | 0.2260 | 2 | 2 |
| Mu-type opioid receptor | Rattus norvegicus (Norway rat) | Ki | 0.4400 | 1 | 1 |
| Multidrug resistance-associated protein 4 | Homo sapiens (human) | IC50 | 133.0000 | 1 | 1 |
| Muscarinic acetylcholine receptor M1 | Rattus norvegicus (Norway rat) | IC50 | 360.0000 | 1 | 2 |
| Muscarinic acetylcholine receptor M2 | Rattus norvegicus (Norway rat) | IC50 | 360.0000 | 1 | 1 |
| Muscarinic acetylcholine receptor M3 | Rattus norvegicus (Norway rat) | IC50 | 360.0000 | 1 | 1 |
| Muscarinic acetylcholine receptor M4 | Rattus norvegicus (Norway rat) | IC50 | 360.0000 | 1 | 1 |
| Muscarinic acetylcholine receptor M4 | Mus musculus (house mouse) | Ki | 2.1100 | 1 | 1 |
| Muscarinic acetylcholine receptor M4 | Rattus norvegicus (Norway rat) | Ki | 1.0597 | 2 | 2 |
| Muscarinic acetylcholine receptor M5 | Rattus norvegicus (Norway rat) | IC50 | 360.0000 | 1 | 1 |
| N-acylethanolamine-hydrolyzing acid amidase | Homo sapiens (human) | IC50 | 50.0000 | 1 | 1 |
| Neuronal acetylcholine receptor subunit alpha-10 | Rattus norvegicus (Norway rat) | IC50 | 0.0050 | 2 | 2 |
| Neuronal acetylcholine receptor subunit alpha-10 | Rattus norvegicus (Norway rat) | Ki | 0.0070 | 3 | 4 |
| Neuronal acetylcholine receptor subunit alpha-2 | Mus musculus (house mouse) | IC50 | 0.0040 | 1 | 1 |
| Neuronal acetylcholine receptor subunit alpha-2 | Rattus norvegicus (Norway rat) | IC50 | 0.0050 | 2 | 2 |
| Neuronal acetylcholine receptor subunit alpha-2 | Homo sapiens (human) | Ki | 0.0595 | 3 | 3 |
| Neuronal acetylcholine receptor subunit alpha-2 | Mus musculus (house mouse) | Ki | 0.0012 | 1 | 1 |
| Neuronal acetylcholine receptor subunit alpha-2 | Rattus norvegicus (Norway rat) | Ki | 0.0438 | 27 | 28 |
| Neuronal acetylcholine receptor subunit alpha-3 | Homo sapiens (human) | IC50 | 0.3899 | 4 | 4 |
| Neuronal acetylcholine receptor subunit alpha-3 | Mus musculus (house mouse) | IC50 | 0.0040 | 1 | 1 |
| Neuronal acetylcholine receptor subunit alpha-3 | Rattus norvegicus (Norway rat) | IC50 | 5.0025 | 4 | 4 |
| Neuronal acetylcholine receptor subunit alpha-3 | Homo sapiens (human) | Ki | 0.3763 | 20 | 20 |
| Neuronal acetylcholine receptor subunit alpha-3 | Mus musculus (house mouse) | Ki | 0.0841 | 2 | 2 |
| Neuronal acetylcholine receptor subunit alpha-3 | Rattus norvegicus (Norway rat) | Ki | 0.2178 | 37 | 42 |
| Neuronal acetylcholine receptor subunit alpha-4 | Homo sapiens (human) | IC50 | 0.3456 | 10 | 12 |
| Neuronal acetylcholine receptor subunit alpha-4 | Mus musculus (house mouse) | IC50 | 0.0055 | 2 | 2 |
| Neuronal acetylcholine receptor subunit alpha-4 | Rattus norvegicus (Norway rat) | IC50 | 0.0046 | 3 | 3 |
| Neuronal acetylcholine receptor subunit alpha-4 | Gallus gallus (chicken) | Ki | 0.0019 | 1 | 1 |
| Neuronal acetylcholine receptor subunit alpha-4 | Homo sapiens (human) | Ki | 0.3444 | 30 | 30 |
| Neuronal acetylcholine receptor subunit alpha-4 | Mus musculus (house mouse) | Ki | 0.0012 | 1 | 1 |
| Neuronal acetylcholine receptor subunit alpha-4 | Rattus norvegicus (Norway rat) | Ki | 0.0551 | 72 | 86 |
| Neuronal acetylcholine receptor subunit alpha-5 | Mus musculus (house mouse) | IC50 | 0.0040 | 1 | 1 |
| Neuronal acetylcholine receptor subunit alpha-5 | Rattus norvegicus (Norway rat) | IC50 | 0.0050 | 2 | 2 |
| Neuronal acetylcholine receptor subunit alpha-5 | Mus musculus (house mouse) | Ki | 0.0012 | 1 | 1 |
| Neuronal acetylcholine receptor subunit alpha-5 | Rattus norvegicus (Norway rat) | Ki | 0.0070 | 3 | 4 |
| Neuronal acetylcholine receptor subunit alpha-6 | Homo sapiens (human) | IC50 | 0.0848 | 1 | 1 |
| Neuronal acetylcholine receptor subunit alpha-6 | Mus musculus (house mouse) | IC50 | 0.0040 | 1 | 1 |
| Neuronal acetylcholine receptor subunit alpha-6 | Rattus norvegicus (Norway rat) | IC50 | 0.0050 | 2 | 2 |
| Neuronal acetylcholine receptor subunit alpha-6 | Mus musculus (house mouse) | Ki | 0.0012 | 1 | 1 |
| Neuronal acetylcholine receptor subunit alpha-6 | Rattus norvegicus (Norway rat) | Ki | 0.0070 | 3 | 4 |
| Neuronal acetylcholine receptor subunit alpha-7 | Homo sapiens (human) | IC50 | 14.3000 | 2 | 2 |
| Neuronal acetylcholine receptor subunit alpha-7 | Mus musculus (house mouse) | IC50 | 0.0040 | 1 | 1 |
| Neuronal acetylcholine receptor subunit alpha-7 | Rattus norvegicus (Norway rat) | IC50 | 0.0087 | 3 | 3 |
| Neuronal acetylcholine receptor subunit alpha-7 | Homo sapiens (human) | Ki | 5.9317 | 17 | 19 |
| Neuronal acetylcholine receptor subunit alpha-7 | Mus musculus (house mouse) | Ki | 0.2406 | 2 | 2 |
| Neuronal acetylcholine receptor subunit alpha-7 | Rattus norvegicus (Norway rat) | Ki | 3.1729 | 16 | 20 |
| Neuronal acetylcholine receptor subunit alpha-9 | Rattus norvegicus (Norway rat) | IC50 | 0.0041 | 3 | 3 |
| Neuronal acetylcholine receptor subunit alpha-9 | Rattus norvegicus (Norway rat) | Ki | 0.0070 | 3 | 4 |
| Neuronal acetylcholine receptor subunit beta-2 | Homo sapiens (human) | IC50 | 0.3256 | 11 | 13 |
| Neuronal acetylcholine receptor subunit beta-2 | Mus musculus (house mouse) | IC50 | 0.0040 | 1 | 1 |
| Neuronal acetylcholine receptor subunit beta-2 | Rattus norvegicus (Norway rat) | IC50 | 0.0046 | 3 | 3 |
| Neuronal acetylcholine receptor subunit beta-2 | Homo sapiens (human) | Ki | 0.3399 | 30 | 30 |
| Neuronal acetylcholine receptor subunit beta-2 | Mus musculus (house mouse) | Ki | 0.0024 | 2 | 2 |
| Neuronal acetylcholine receptor subunit beta-2 | Rattus norvegicus (Norway rat) | Ki | 0.0471 | 76 | 86 |
| Neuronal acetylcholine receptor subunit beta-3 | Homo sapiens (human) | IC50 | 0.0848 | 1 | 1 |
| Neuronal acetylcholine receptor subunit beta-3 | Mus musculus (house mouse) | IC50 | 0.0040 | 1 | 1 |
| Neuronal acetylcholine receptor subunit beta-3 | Rattus norvegicus (Norway rat) | IC50 | 0.0050 | 2 | 2 |
| Neuronal acetylcholine receptor subunit beta-3 | Mus musculus (house mouse) | Ki | 0.0012 | 1 | 1 |
| Neuronal acetylcholine receptor subunit beta-3 | Rattus norvegicus (Norway rat) | Ki | 0.0070 | 3 | 4 |
| Neuronal acetylcholine receptor subunit beta-4 | Homo sapiens (human) | IC50 | 0.7150 | 2 | 2 |
| Neuronal acetylcholine receptor subunit beta-4 | Mus musculus (house mouse) | IC50 | 0.0040 | 1 | 1 |
| Neuronal acetylcholine receptor subunit beta-4 | Rattus norvegicus (Norway rat) | IC50 | 5.0025 | 4 | 4 |
| Neuronal acetylcholine receptor subunit beta-4 | Homo sapiens (human) | Ki | 0.3463 | 22 | 22 |
| Neuronal acetylcholine receptor subunit beta-4 | Mus musculus (house mouse) | Ki | 0.0572 | 3 | 3 |
| Neuronal acetylcholine receptor subunit beta-4 | Rattus norvegicus (Norway rat) | Ki | 0.1748 | 54 | 63 |
| Non-receptor tyrosine-protein kinase TYK2 | Homo sapiens (human) | IC50 | 1.2690 | 1 | 1 |
| Nucleophosmin | Homo sapiens (human) | IC50 | 0.0510 | 1 | 1 |
| Phenylethanolamine N-methyltransferase | Bos taurus (cattle) | IC50 | 109.0000 | 1 | 1 |
| Phosphatidylinositol 3,4,5-trisphosphate 5-phosphatase 2 | Homo sapiens (human) | IC50 | 5.5000 | 2 | 2 |
| Phospholipase A-2-activating protein | Homo sapiens (human) | IC50 | 5.0000 | 1 | 1 |
| Platelet-derived growth factor receptor alpha | Homo sapiens (human) | IC50 | 1.0000 | 1 | 1 |
| Platelet-derived growth factor receptor beta | Homo sapiens (human) | IC50 | 7.0000 | 3 | 3 |
| Polyphenol oxidase 2 | Agaricus bisporus | IC50 | 115.2000 | 1 | 1 |
| Potassium voltage-gated channel subfamily H member 2 | Homo sapiens (human) | IC50 | 245.0807 | 5 | 6 |
| Proto-oncogene tyrosine-protein kinase receptor Ret | Homo sapiens (human) | IC50 | 10.0000 | 1 | 1 |
| Proto-oncogene tyrosine-protein kinase ROS | Homo sapiens (human) | IC50 | 0.5458 | 13 | 13 |
| Proto-oncogene tyrosine-protein kinase ROS | Homo sapiens (human) | Ki | 0.0842 | 4 | 4 |
| Proto-oncogene tyrosine-protein kinase Src | Homo sapiens (human) | IC50 | 5.5000 | 2 | 2 |
| Purine nucleoside phosphorylase | Homo sapiens (human) | Ki | 1,500.0000 | 1 | 1 |
| RAC-beta serine/threonine-protein kinase | Homo sapiens (human) | IC50 | 10.0000 | 1 | 1 |
| Receptor tyrosine-protein kinase erbB-2 | Homo sapiens (human) | IC50 | 1.0000 | 1 | 1 |
| Receptor-type tyrosine-protein kinase FLT3 | Homo sapiens (human) | IC50 | 1.0000 | 1 | 1 |
| Ribosomal protein S6 kinase beta-1 | Homo sapiens (human) | IC50 | 10.0000 | 1 | 1 |
| Serine/threonine-protein kinase D1 | Homo sapiens (human) | IC50 | 10.0000 | 1 | 1 |
| Serine/threonine-protein kinase N2 | Homo sapiens (human) | IC50 | 10.0000 | 1 | 1 |
| Sigma intracellular receptor 2 | Rattus norvegicus (Norway rat) | IC50 | 1,000.0000 | 1 | 1 |
| Sodium-dependent phosphate transport protein 2B | Homo sapiens (human) | IC50 | 0.0510 | 1 | 1 |
| Soluble acetylcholine receptor | Aplysia californica (California sea hare) | Ki | 1.0466 | 3 | 3 |
| Solute carrier family 22 member 1 | Rattus norvegicus (Norway rat) | Ki | 64.3000 | 1 | 1 |
| Solute carrier family 22 member 2 | Rattus norvegicus (Norway rat) | Ki | 50.5000 | 1 | 1 |
| Stromelysin-1 | Homo sapiens (human) | IC50 | 500.0000 | 1 | 1 |
| Substance-P receptor | Cavia porcellus (domestic guinea pig) | IC50 | 500.0000 | 1 | 3 |
| Translocator protein | Rattus norvegicus (Norway rat) | Ki | 0.5063 | 2 | 4 |
| Transporter | Rattus norvegicus (Norway rat) | Ki | 5.5000 | 1 | 1 |
| Tyrosine-protein kinase ABL1 | Homo sapiens (human) | IC50 | 0.7277 | 3 | 3 |
| Tyrosine-protein kinase ABL1 | Mus musculus (house mouse) | IC50 | 1.1590 | 1 | 1 |
| Tyrosine-protein kinase BTK | Homo sapiens (human) | IC50 | 10.0000 | 1 | 1 |
| Tyrosine-protein kinase Fgr | Homo sapiens (human) | IC50 | 10.0000 | 1 | 1 |
| Tyrosine-protein kinase Fyn | Homo sapiens (human) | IC50 | 10.0000 | 1 | 1 |
| Tyrosine-protein kinase JAK1 | Homo sapiens (human) | IC50 | 0.5630 | 1 | 1 |
| Tyrosine-protein kinase JAK2 | Homo sapiens (human) | IC50 | 0.0595 | 1 | 2 |
| Tyrosine-protein kinase JAK3 | Homo sapiens (human) | IC50 | 1.3600 | 1 | 1 |
| Tyrosine-protein kinase Lck | Homo sapiens (human) | IC50 | 1.8277 | 3 | 3 |
| Tyrosine-protein kinase Mer | Homo sapiens (human) | IC50 | 0.1000 | 1 | 1 |
| Tyrosine-protein kinase receptor TYRO3 | Homo sapiens (human) | IC50 | 5.0500 | 2 | 2 |
| Tyrosine-protein kinase receptor UFO | Homo sapiens (human) | IC50 | 0.1978 | 5 | 5 |
| Tyrosine-protein phosphatase non-receptor type 1 | Homo sapiens (human) | IC50 | 2,700.0000 | 1 | 1 |
| Vascular endothelial growth factor receptor 1 | Homo sapiens (human) | IC50 | 1.0000 | 1 | 1 |
| Vascular endothelial growth factor receptor 2 | Homo sapiens (human) | IC50 | 7.7500 | 4 | 4 |
| Protein | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Drugs |
|---|
| 26S proteasome regulatory subunit 6B | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| 3-phosphoinositide-dependent protein kinase 1 | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| 5'-AMP-activated protein kinase catalytic subunit alpha-1 | Homo sapiens (human) | Kd | 16.2000 | 2 | 2 |
| 5'-AMP-activated protein kinase catalytic subunit alpha-2 | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| 5'-AMP-activated protein kinase subunit gamma-1 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| 5'-AMP-activated protein kinase subunit gamma-2 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| AarF domain-containing protein kinase 1 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Acetylcholine receptor subunit alpha | Homo sapiens (human) | EC50 | 25.3333 | 3 | 3 |
| Acetylcholine receptor subunit alpha | Tetronarce californica (Pacific electric ray) | EC50 | 60.0000 | 1 | 1 |
| Acetylcholine receptor subunit beta | Homo sapiens (human) | EC50 | 29.0000 | 3 | 3 |
| Acetylcholine receptor subunit beta | Tetronarce californica (Pacific electric ray) | EC50 | 60.0000 | 1 | 1 |
| Acetylcholine receptor subunit delta | Homo sapiens (human) | EC50 | 33.0000 | 2 | 2 |
| Acetylcholine receptor subunit delta | Tetronarce californica (Pacific electric ray) | EC50 | 110.0000 | 2 | 2 |
| Acetylcholine receptor subunit epsilon | Homo sapiens (human) | EC50 | 65.0000 | 1 | 1 |
| Acetylcholine receptor subunit gamma | Homo sapiens (human) | EC50 | 33.0000 | 2 | 2 |
| Acetylcholine receptor subunit gamma | Tetronarce californica (Pacific electric ray) | EC50 | 60.0000 | 1 | 1 |
| Acetylcholine-binding protein | Lymnaea stagnalis (great pond snail) | Kd | 0.2931 | 3 | 5 |
| Actin-related protein 2 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Actin-related protein 3 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Activated CDC42 kinase 1 | Homo sapiens (human) | Kd | 15.3800 | 2 | 2 |
| Activin receptor type-1 | Homo sapiens (human) | Kd | 15.2200 | 2 | 2 |
| Activin receptor type-1B | Homo sapiens (human) | Kd | 15.4300 | 2 | 2 |
| Activin receptor type-2A | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Activin receptor type-2B | Homo sapiens (human) | Kd | 20.0000 | 2 | 2 |
| Acyl-CoA dehydrogenase family member 10 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Acyl-CoA dehydrogenase family member 11 | Homo sapiens (human) | Kd | 1.9160 | 1 | 1 |
| Adenine phosphoribosyltransferase | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Adenosine kinase | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Adenylate kinase 2, mitochondrial | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| ADP/ATP translocase 2 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| ADP/ATP translocase 3 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| ALK tyrosine kinase receptor | Homo sapiens (human) | EC50 | 6.3644 | 4 | 4 |
| ALK tyrosine kinase receptor | Homo sapiens (human) | Kd | 0.0036 | 3 | 3 |
| Angiopoietin-1 receptor | Homo sapiens (human) | Kd | 0.2700 | 1 | 1 |
| Ankyrin repeat and protein kinase domain-containing protein 1 | Homo sapiens (human) | Kd | 0.7800 | 1 | 1 |
| AP2-associated protein kinase 1 | Homo sapiens (human) | Kd | 16.1500 | 2 | 2 |
| Apelin receptor | Homo sapiens (human) | EC50 | 0.0170 | 5 | 5 |
| ATP-dependent 6-phosphofructokinase, platelet type | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| ATP-dependent RNA helicase DDX1 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| ATP-dependent RNA helicase DDX3X | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| ATP-dependent RNA helicase DDX42 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| ATP-dependent RNA helicase DHX30 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Atypical kinase COQ8A, mitochondrial | Homo sapiens (human) | Kd | 23.3333 | 2 | 3 |
| Atypical kinase COQ8B, mitochondrial | Homo sapiens (human) | Kd | 1.1000 | 1 | 1 |
| Aurora kinase A | Homo sapiens (human) | Kd | 0.2877 | 3 | 3 |
| Aurora kinase B | Homo sapiens (human) | Kd | 0.6580 | 2 | 2 |
| Aurora kinase C | Homo sapiens (human) | Kd | 4.3000 | 1 | 1 |
| BDNF/NT-3 growth factors receptor | Homo sapiens (human) | Kd | 0.0370 | 1 | 1 |
| Beta-adrenergic receptor kinase 1 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| BMP-2-inducible protein kinase | Homo sapiens (human) | Kd | 15.3700 | 2 | 2 |
| Bone morphogenetic protein receptor type-1A | Homo sapiens (human) | Kd | 20.0000 | 2 | 2 |
| Bone morphogenetic protein receptor type-1B | Homo sapiens (human) | Kd | 15.1150 | 2 | 2 |
| Bone morphogenetic protein receptor type-2 | Homo sapiens (human) | Kd | 20.0000 | 2 | 2 |
| Breakpoint cluster region protein | Homo sapiens (human) | Kd | 2.4850 | 1 | 1 |
| Calcium-dependent protein kinase 1 | Plasmodium falciparum 3D7 | Kd | 10.0000 | 1 | 1 |
| Calcium/calmodulin-dependent protein kinase kinase 1 | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Calcium/calmodulin-dependent protein kinase kinase 2 | Homo sapiens (human) | Kd | 15.7500 | 2 | 2 |
| Calcium/calmodulin-dependent protein kinase type 1 | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Calcium/calmodulin-dependent protein kinase type 1D | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Calcium/calmodulin-dependent protein kinase type 1G | Homo sapiens (human) | Kd | 20.0000 | 2 | 2 |
| Calcium/calmodulin-dependent protein kinase type II subunit alpha | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Calcium/calmodulin-dependent protein kinase type II subunit beta | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Calcium/calmodulin-dependent protein kinase type II subunit delta | Homo sapiens (human) | Kd | 20.0000 | 2 | 2 |
| Calcium/calmodulin-dependent protein kinase type II subunit gamma | Homo sapiens (human) | Kd | 20.0000 | 2 | 2 |
| Calcium/calmodulin-dependent protein kinase type IV | Homo sapiens (human) | Kd | 20.0000 | 2 | 2 |
| cAMP-dependent protein kinase catalytic subunit alpha | Homo sapiens (human) | Kd | 20.0000 | 2 | 2 |
| cAMP-dependent protein kinase catalytic subunit beta | Homo sapiens (human) | Kd | 20.0000 | 2 | 2 |
| cAMP-dependent protein kinase catalytic subunit gamma | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| cAMP-dependent protein kinase catalytic subunit PRKX | Homo sapiens (human) | Kd | 20.0000 | 2 | 2 |
| cAMP-dependent protein kinase type II-alpha regulatory subunit | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Casein kinase I isoform alpha | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Casein kinase I isoform alpha-like | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Casein kinase I isoform delta | Homo sapiens (human) | Kd | 20.0000 | 2 | 2 |
| Casein kinase I isoform epsilon | Homo sapiens (human) | Kd | 20.0000 | 2 | 2 |
| Casein kinase I isoform gamma-1 | Homo sapiens (human) | Kd | 20.0000 | 2 | 2 |
| Casein kinase I isoform gamma-2 | Homo sapiens (human) | Kd | 20.0000 | 2 | 2 |
| Casein kinase I isoform gamma-3 | Homo sapiens (human) | Kd | 20.0000 | 2 | 2 |
| Casein kinase II subunit alpha | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Casein kinase II subunit alpha' | Homo sapiens (human) | Kd | 20.0000 | 2 | 2 |
| Cell division control protein 2 homolog | Plasmodium falciparum 3D7 | Kd | 10.0000 | 1 | 1 |
| Cell division cycle 7-related protein kinase | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| cGMP-dependent protein kinase 1 | Homo sapiens (human) | Kd | 20.0000 | 2 | 2 |
| cGMP-dependent protein kinase 2 | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Chain A, Avidin | Gallus gallus (chicken) | Kd | 117.0000 | 1 | 2 |
| Chain A, HYPOXANTHINE-GUANINE PHOSPHORIBOSYLTRANSFERASE | Toxoplasma gondii RH | Kd | 7.1000 | 1 | 2 |
| Chain A, Xanthine phosphoribosyltransferase | Bacillus subtilis | Kd | 4.5000 | 1 | 1 |
| Chain B, Avidin | Gallus gallus (chicken) | Kd | 117.0000 | 1 | 1 |
| Chain B, HYPOXANTHINE-GUANINE PHOSPHORIBOSYLTRANSFERASE | Toxoplasma gondii RH | Kd | 7.1000 | 1 | 1 |
| Chain E, LYSINE, ARGININE, ORNITHINE-BINDING PROTEIN | Salmonella enterica subsp. enterica serovar Typhimurium | Kd | 0.0140 | 1 | 3 |
| Choline-phosphate cytidylyltransferase A | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Chromodomain-helicase-DNA-binding protein 4 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Citron Rho-interacting kinase | Homo sapiens (human) | Kd | 20.0000 | 2 | 2 |
| Cyclin-dependent kinase 1 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Cyclin-dependent kinase 10 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Cyclin-dependent kinase 11A | Homo sapiens (human) | Kd | 0.4200 | 1 | 1 |
| Cyclin-dependent kinase 11B | Homo sapiens (human) | Kd | 0.7600 | 1 | 1 |
| Cyclin-dependent kinase 12 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Cyclin-dependent kinase 13 | Homo sapiens (human) | Kd | 20.0000 | 2 | 2 |
| Cyclin-dependent kinase 14 | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Cyclin-dependent kinase 15 | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Cyclin-dependent kinase 16 | Homo sapiens (human) | Kd | 20.0000 | 2 | 2 |
| Cyclin-dependent kinase 17 | Homo sapiens (human) | Kd | 20.0000 | 2 | 2 |
| Cyclin-dependent kinase 18 | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Cyclin-dependent kinase 19 | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Cyclin-dependent kinase 2 | Homo sapiens (human) | Kd | 20.0000 | 2 | 2 |
| Cyclin-dependent kinase 3 | Homo sapiens (human) | Kd | 20.0000 | 2 | 2 |
| Cyclin-dependent kinase 4 | Homo sapiens (human) | Kd | 16.6667 | 3 | 3 |
| Cyclin-dependent kinase 6 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Cyclin-dependent kinase 7 | Homo sapiens (human) | Kd | 15.1650 | 2 | 2 |
| Cyclin-dependent kinase 8 | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Cyclin-dependent kinase 9 | Homo sapiens (human) | Kd | 20.0000 | 2 | 2 |
| Cyclin-dependent kinase-like 1 | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Cyclin-dependent kinase-like 2 | Homo sapiens (human) | Kd | 2.1000 | 1 | 1 |
| Cyclin-dependent kinase-like 3 | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Cyclin-dependent kinase-like 5 | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Cyclin-dependent-like kinase 5 | Homo sapiens (human) | Kd | 20.0000 | 2 | 2 |
| Cyclin-G-associated kinase | Homo sapiens (human) | Kd | 20.0000 | 2 | 2 |
| Cysteine--tRNA ligase, cytoplasmic | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Cytochrome c1, heme protein, mitochondrial | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Cytochrome P450 2A13 | Homo sapiens (human) | Kd | 54.0000 | 1 | 1 |
| Cytochrome P450 2A6 | Homo sapiens (human) | Kd | 470.0000 | 1 | 1 |
| Cytoplasmic tyrosine-protein kinase BMX | Homo sapiens (human) | Kd | 3.6000 | 1 | 1 |
| D(2) dopamine receptor | Rattus norvegicus (Norway rat) | Kd | 150.4000 | 4 | 5 |
| dCTP pyrophosphatase 1 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Death-associated protein kinase 1 | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Death-associated protein kinase 2 | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Death-associated protein kinase 3 | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Delta(24)-sterol reductase | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Deoxycytidine kinase | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Discoidin domain-containing receptor 2 | Homo sapiens (human) | Kd | 20.0000 | 2 | 2 |
| DNA replication licensing factor MCM4 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| DNA topoisomerase 2-alpha | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| DNA topoisomerase 2-beta | Homo sapiens (human) | Kd | 30.0000 | 1 | 2 |
| DnaJ homolog subfamily A member 1 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Dual serine/threonine and tyrosine protein kinase | Homo sapiens (human) | Kd | 0.4500 | 1 | 1 |
| Dual specificity mitogen-activated protein kinase kinase 1 | Homo sapiens (human) | Kd | 20.0000 | 2 | 2 |
| Dual specificity mitogen-activated protein kinase kinase 2 | Homo sapiens (human) | Kd | 20.0000 | 2 | 2 |
| Dual specificity mitogen-activated protein kinase kinase 3 | Homo sapiens (human) | Kd | 16.6500 | 2 | 2 |
| Dual specificity mitogen-activated protein kinase kinase 4 | Homo sapiens (human) | Kd | 23.3333 | 2 | 3 |
| Dual specificity mitogen-activated protein kinase kinase 5 | Homo sapiens (human) | Kd | 20.0000 | 2 | 2 |
| Dual specificity mitogen-activated protein kinase kinase 6 | Homo sapiens (human) | Kd | 23.3333 | 2 | 3 |
| Dual specificity mitogen-activated protein kinase kinase 7 | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Dual specificity protein kinase CLK1 | Homo sapiens (human) | Kd | 20.0000 | 2 | 2 |
| Dual specificity protein kinase CLK2 | Homo sapiens (human) | Kd | 20.0000 | 2 | 2 |
| Dual specificity protein kinase CLK3 | Homo sapiens (human) | Kd | 20.0000 | 2 | 2 |
| Dual specificity protein kinase CLK4 | Homo sapiens (human) | Kd | 23.3333 | 2 | 3 |
| Dual specificity protein kinase TTK | Homo sapiens (human) | Kd | 20.0000 | 2 | 2 |
| Dual specificity testis-specific protein kinase 1 | Homo sapiens (human) | Kd | 15.1900 | 2 | 2 |
| Dual specificity testis-specific protein kinase 2 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Dual specificity tyrosine-phosphorylation-regulated kinase 1A | Homo sapiens (human) | Kd | 20.0000 | 2 | 2 |
| Dual specificity tyrosine-phosphorylation-regulated kinase 1B | Homo sapiens (human) | Kd | 20.0000 | 2 | 2 |
| Dual specificity tyrosine-phosphorylation-regulated kinase 2 | Homo sapiens (human) | Kd | 4.0000 | 1 | 1 |
| Dynamin-like 120 kDa protein, mitochondrial | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| eIF-2-alpha kinase GCN2 | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| EKC/KEOPS complex subunit TP53RK | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Electron transfer flavoprotein subunit beta | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Elongation factor Tu, mitochondrial | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Ephrin type-A receptor 1 | Homo sapiens (human) | Kd | 15.0700 | 2 | 2 |
| Ephrin type-A receptor 2 | Homo sapiens (human) | Kd | 0.7127 | 3 | 3 |
| Ephrin type-A receptor 3 | Homo sapiens (human) | Kd | 0.7000 | 1 | 1 |
| Ephrin type-A receptor 4 | Homo sapiens (human) | Kd | 15.1800 | 2 | 2 |
| Ephrin type-A receptor 5 | Homo sapiens (human) | Kd | 15.5000 | 2 | 2 |
| Ephrin type-A receptor 6 | Homo sapiens (human) | Kd | 0.0650 | 1 | 1 |
| Ephrin type-A receptor 7 | Homo sapiens (human) | Kd | 0.4700 | 1 | 1 |
| Ephrin type-A receptor 8 | Homo sapiens (human) | Kd | 0.2800 | 1 | 1 |
| Ephrin type-B receptor 1 | Homo sapiens (human) | Kd | 0.1200 | 1 | 1 |
| Ephrin type-B receptor 2 | Homo sapiens (human) | Kd | 20.0000 | 2 | 2 |
| Ephrin type-B receptor 3 | Homo sapiens (human) | Kd | 20.0000 | 2 | 2 |
| Ephrin type-B receptor 4 | Homo sapiens (human) | Kd | 15.2850 | 2 | 2 |
| Ephrin type-B receptor 6 | Homo sapiens (human) | Kd | 0.2755 | 2 | 2 |
| Epidermal growth factor receptor | Homo sapiens (human) | Kd | 10.4154 | 13 | 13 |
| Epithelial discoidin domain-containing receptor 1 | Homo sapiens (human) | Kd | 15.2550 | 2 | 2 |
| Eukaryotic translation initiation factor 2-alpha kinase 1 | Homo sapiens (human) | Kd | 20.0000 | 2 | 2 |
| Eukaryotic translation initiation factor 5B | Homo sapiens (human) | Kd | 30.0000 | 1 | 2 |
| Exosome RNA helicase MTR4 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Ferrochelatase, mitochondrial | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Fibroblast growth factor receptor 1 | Homo sapiens (human) | Kd | 20.0000 | 2 | 2 |
| Fibroblast growth factor receptor 2 | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Fibroblast growth factor receptor 3 | Homo sapiens (human) | Kd | 3.1000 | 2 | 2 |
| Fibroblast growth factor receptor 4 | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Focal adhesion kinase 1 | Homo sapiens (human) | Kd | 0.4525 | 2 | 2 |
| G protein-coupled receptor kinase 4 | Homo sapiens (human) | Kd | 4.2000 | 1 | 1 |
| G protein-coupled receptor kinase 6 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| General transcription and DNA repair factor IIH helicase subunit XPD | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Glutamate receptor ionotropic, NMDA 1 | Homo sapiens (human) | EC50 | 0.2825 | 4 | 4 |
| Glutamate receptor ionotropic, NMDA 1 | Rattus norvegicus (Norway rat) | EC50 | 0.6500 | 1 | 1 |
| Glutamate receptor ionotropic, NMDA 2A | Homo sapiens (human) | EC50 | 0.2000 | 3 | 3 |
| Glutamate receptor ionotropic, NMDA 2A | Rattus norvegicus (Norway rat) | EC50 | 0.6500 | 1 | 1 |
| Glutamate receptor ionotropic, NMDA 2B | Homo sapiens (human) | EC50 | 0.5300 | 1 | 1 |
| Glycine--tRNA ligase | Homo sapiens (human) | Kd | 30.0000 | 1 | 2 |
| Glycogen phosphorylase, brain form | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Glycogen phosphorylase, liver form | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Glycogen synthase kinase-3 alpha | Homo sapiens (human) | Kd | 20.0000 | 2 | 2 |
| Glycogen synthase kinase-3 beta | Homo sapiens (human) | Kd | 20.0000 | 2 | 2 |
| Glycoprotein IIb | Oryctolagus cuniculus (rabbit) | EC50 | 1.5068 | 1 | 4 |
| GTP-binding nuclear protein Ran | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Guanine nucleotide-binding protein G(i) subunit alpha-2 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Heme oxygenase 2 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Hepatocyte growth factor receptor | Homo sapiens (human) | Kd | 0.0024 | 6 | 6 |
| High affinity nerve growth factor receptor | Homo sapiens (human) | Kd | 15.0475 | 2 | 2 |
| Histidine triad nucleotide-binding protein 1 | Homo sapiens (human) | Kd | 67.0000 | 1 | 1 |
| Homeodomain-interacting protein kinase 1 | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Homeodomain-interacting protein kinase 2 | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Homeodomain-interacting protein kinase 3 | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Homeodomain-interacting protein kinase 4 | Homo sapiens (human) | Kd | 3.6000 | 1 | 1 |
| Hormonally up-regulated neu tumor-associated kinase | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Inhibitor of nuclear factor kappa-B kinase subunit alpha | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Inhibitor of nuclear factor kappa-B kinase subunit beta | Homo sapiens (human) | Kd | 5.5000 | 1 | 1 |
| Inhibitor of nuclear factor kappa-B kinase subunit epsilon | Homo sapiens (human) | Kd | 1.7190 | 2 | 2 |
| Inosine-5'-monophosphate dehydrogenase 2 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Insulin receptor | Homo sapiens (human) | Kd | 15.1700 | 2 | 2 |
| Insulin receptor-related protein | Homo sapiens (human) | Kd | 0.6000 | 1 | 1 |
| Insulin-like growth factor 1 receptor | Homo sapiens (human) | Kd | 15.3900 | 2 | 2 |
| Integrin beta | Oryctolagus cuniculus (rabbit) | EC50 | 1.5068 | 1 | 4 |
| Integrin-linked protein kinase | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Interferon-induced, double-stranded RNA-activated protein kinase | Homo sapiens (human) | Kd | 1.1000 | 1 | 1 |
| Interleukin-1 receptor-associated kinase 1 | Homo sapiens (human) | Kd | 1.9955 | 2 | 2 |
| Interleukin-1 receptor-associated kinase 3 | Homo sapiens (human) | Kd | 0.3270 | 2 | 2 |
| Interleukin-1 receptor-associated kinase 4 | Homo sapiens (human) | Kd | 16.8000 | 2 | 2 |
| Isoleucine--tRNA ligase, mitochondrial | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Leucine-rich repeat serine/threonine-protein kinase 2 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Leukocyte tyrosine kinase receptor | Homo sapiens (human) | Kd | 0.0120 | 1 | 1 |
| Leukotriene C4 synthase | Cavia porcellus (domestic guinea pig) | Kd | 10.0000 | 1 | 1 |
| LIM domain kinase 1 | Homo sapiens (human) | Kd | 1.3600 | 2 | 2 |
| LIM domain kinase 2 | Homo sapiens (human) | Kd | 2.5150 | 2 | 2 |
| Long-chain-fatty-acid--CoA ligase 5 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Macrophage colony-stimulating factor 1 receptor | Homo sapiens (human) | Kd | 0.2100 | 1 | 1 |
| Macrophage-stimulating protein receptor | Homo sapiens (human) | Kd | 0.0505 | 2 | 2 |
| MAP kinase-activated protein kinase 2 | Homo sapiens (human) | Kd | 20.0000 | 2 | 2 |
| MAP kinase-activated protein kinase 5 | Homo sapiens (human) | Kd | 20.0000 | 2 | 2 |
| MAP kinase-interacting serine/threonine-protein kinase 1 | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| MAP kinase-interacting serine/threonine-protein kinase 2 | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| MAP/microtubule affinity-regulating kinase 3 | Homo sapiens (human) | Kd | 20.0000 | 2 | 2 |
| MAP/microtubule affinity-regulating kinase 4 | Homo sapiens (human) | Kd | 20.0000 | 2 | 2 |
| Mast/stem cell growth factor receptor Kit | Homo sapiens (human) | Kd | 10.5000 | 9 | 9 |
| Maternal embryonic leucine zipper kinase | Homo sapiens (human) | Kd | 20.0000 | 2 | 2 |
| Megakaryocyte-associated tyrosine-protein kinase | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Membrane-associated progesterone receptor component 1 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Membrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinase | Homo sapiens (human) | Kd | 20.0000 | 2 | 2 |
| Microtubule-associated serine/threonine-protein kinase 1 | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Midasin | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Misshapen-like kinase 1 | Homo sapiens (human) | Kd | 17.2000 | 2 | 2 |
| Mitogen-activated protein kinase 1 | Homo sapiens (human) | Kd | 20.0000 | 2 | 2 |
| Mitogen-activated protein kinase 10 | Homo sapiens (human) | Kd | 23.3333 | 2 | 3 |
| Mitogen-activated protein kinase 11 | Homo sapiens (human) | Kd | 20.0000 | 2 | 2 |
| Mitogen-activated protein kinase 12 | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Mitogen-activated protein kinase 13 | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Mitogen-activated protein kinase 14 | Homo sapiens (human) | Kd | 20.0000 | 2 | 2 |
| Mitogen-activated protein kinase 15 | Homo sapiens (human) | Kd | 20.0000 | 2 | 2 |
| Mitogen-activated protein kinase 3 | Homo sapiens (human) | Kd | 20.0000 | 2 | 2 |
| Mitogen-activated protein kinase 4 | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Mitogen-activated protein kinase 6 | Homo sapiens (human) | Kd | 6.7000 | 2 | 2 |
| Mitogen-activated protein kinase 7 | Homo sapiens (human) | Kd | 15.2550 | 2 | 2 |
| Mitogen-activated protein kinase 8 | Homo sapiens (human) | Kd | 20.0000 | 2 | 2 |
| Mitogen-activated protein kinase 9 | Homo sapiens (human) | Kd | 20.0000 | 2 | 2 |
| Mitogen-activated protein kinase kinase kinase 1 | Homo sapiens (human) | Kd | 1.4835 | 2 | 2 |
| Mitogen-activated protein kinase kinase kinase 10 | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Mitogen-activated protein kinase kinase kinase 11 | Homo sapiens (human) | Kd | 20.0000 | 2 | 2 |
| Mitogen-activated protein kinase kinase kinase 12 | Homo sapiens (human) | Kd | 0.1700 | 1 | 1 |
| Mitogen-activated protein kinase kinase kinase 13 | Homo sapiens (human) | Kd | 0.2300 | 1 | 1 |
| Mitogen-activated protein kinase kinase kinase 15 | Homo sapiens (human) | Kd | 2.8000 | 1 | 1 |
| Mitogen-activated protein kinase kinase kinase 19 | Homo sapiens (human) | Kd | 0.9800 | 1 | 1 |
| Mitogen-activated protein kinase kinase kinase 2 | Homo sapiens (human) | Kd | 15.0360 | 2 | 2 |
| Mitogen-activated protein kinase kinase kinase 20 | Homo sapiens (human) | Kd | 20.0000 | 2 | 2 |
| Mitogen-activated protein kinase kinase kinase 3 | Homo sapiens (human) | Kd | 15.0550 | 2 | 2 |
| Mitogen-activated protein kinase kinase kinase 4 | Homo sapiens (human) | Kd | 20.0000 | 2 | 2 |
| Mitogen-activated protein kinase kinase kinase 5 | Homo sapiens (human) | Kd | 20.0000 | 2 | 2 |
| Mitogen-activated protein kinase kinase kinase 6 | Homo sapiens (human) | Kd | 20.0000 | 2 | 2 |
| Mitogen-activated protein kinase kinase kinase 7 | Homo sapiens (human) | Kd | 1.8000 | 1 | 1 |
| Mitogen-activated protein kinase kinase kinase 9 | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Mitogen-activated protein kinase kinase kinase kinase 1 | Homo sapiens (human) | Kd | 1.0035 | 2 | 2 |
| Mitogen-activated protein kinase kinase kinase kinase 2 | Homo sapiens (human) | Kd | 0.1310 | 2 | 2 |
| Mitogen-activated protein kinase kinase kinase kinase 3 | Homo sapiens (human) | Kd | 0.9123 | 3 | 3 |
| Mitogen-activated protein kinase kinase kinase kinase 4 | Homo sapiens (human) | Kd | 20.0000 | 2 | 2 |
| Mitogen-activated protein kinase kinase kinase kinase 5 | Homo sapiens (human) | Kd | 0.6050 | 2 | 2 |
| Mitotic checkpoint serine/threonine-protein kinase BUB1 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Mixed lineage kinase domain-like protein | Homo sapiens (human) | Kd | 0.2170 | 1 | 1 |
| Multifunctional protein ADE2 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Muscle, skeletal receptor tyrosine-protein kinase | Homo sapiens (human) | Kd | 0.2300 | 1 | 1 |
| Myosin light chain kinase 2, skeletal/cardiac muscle | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Myosin light chain kinase 3 | Homo sapiens (human) | Kd | 20.0000 | 2 | 2 |
| Myosin light chain kinase family member 4 | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Myosin light chain kinase, smooth muscle | Homo sapiens (human) | Kd | 20.0000 | 2 | 2 |
| Myosin-10 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Myosin-14 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Myosin-IIIa | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Myosin-IIIb | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Myotonin-protein kinase | Homo sapiens (human) | Kd | 1.4000 | 1 | 1 |
| NADH dehydrogenase [ubiquinone] 1 alpha subcomplex subunit 13 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Neuronal acetylcholine receptor subunit alpha-10 | Rattus norvegicus (Norway rat) | EC50 | 40.6667 | 2 | 3 |
| Neuronal acetylcholine receptor subunit alpha-10 | Rattus norvegicus (Norway rat) | Kd | 14,352.0000 | 3 | 3 |
| Neuronal acetylcholine receptor subunit alpha-2 | Rattus norvegicus (Norway rat) | EC50 | 35.5000 | 2 | 2 |
| Neuronal acetylcholine receptor subunit alpha-2 | Rattus norvegicus (Norway rat) | Kd | 14,352.0000 | 3 | 3 |
| Neuronal acetylcholine receptor subunit alpha-3 | Homo sapiens (human) | EC50 | 21.3260 | 14 | 15 |
| Neuronal acetylcholine receptor subunit alpha-3 | Rattus norvegicus (Norway rat) | EC50 | 30.2517 | 7 | 8 |
| Neuronal acetylcholine receptor subunit alpha-3 | Rattus norvegicus (Norway rat) | Kd | 14,352.0000 | 3 | 3 |
| Neuronal acetylcholine receptor subunit alpha-4 | Homo sapiens (human) | EC50 | 3.1424 | 20 | 24 |
| Neuronal acetylcholine receptor subunit alpha-4 | Mus musculus (house mouse) | EC50 | 0.7222 | 1 | 2 |
| Neuronal acetylcholine receptor subunit alpha-4 | Rattus norvegicus (Norway rat) | EC50 | 11.5290 | 12 | 13 |
| Neuronal acetylcholine receptor subunit alpha-4 | Rattus norvegicus (Norway rat) | Kd | 14,352.0000 | 3 | 3 |
| Neuronal acetylcholine receptor subunit alpha-5 | Homo sapiens (human) | EC50 | 30.0000 | 1 | 1 |
| Neuronal acetylcholine receptor subunit alpha-5 | Rattus norvegicus (Norway rat) | EC50 | 35.5000 | 2 | 2 |
| Neuronal acetylcholine receptor subunit alpha-5 | Rattus norvegicus (Norway rat) | Kd | 14,352.0000 | 3 | 3 |
| Neuronal acetylcholine receptor subunit alpha-6 | Homo sapiens (human) | EC50 | 0.1270 | 1 | 1 |
| Neuronal acetylcholine receptor subunit alpha-6 | Rattus norvegicus (Norway rat) | EC50 | 35.5000 | 2 | 2 |
| Neuronal acetylcholine receptor subunit alpha-6 | Rattus norvegicus (Norway rat) | Kd | 14,352.0000 | 3 | 3 |
| Neuronal acetylcholine receptor subunit alpha-7 | Homo sapiens (human) | EC50 | 55.2158 | 6 | 6 |
| Neuronal acetylcholine receptor subunit alpha-7 | Rattus norvegicus (Norway rat) | EC50 | 3,948.0836 | 10 | 11 |
| Neuronal acetylcholine receptor subunit alpha-7 | Homo sapiens (human) | Kd | 0.0011 | 1 | 1 |
| Neuronal acetylcholine receptor subunit alpha-7 | Rattus norvegicus (Norway rat) | Kd | 14,352.0000 | 3 | 3 |
| Neuronal acetylcholine receptor subunit alpha-9 | Rattus norvegicus (Norway rat) | EC50 | 35.5000 | 2 | 2 |
| Neuronal acetylcholine receptor subunit alpha-9 | Rattus norvegicus (Norway rat) | Kd | 14,352.0000 | 3 | 3 |
| Neuronal acetylcholine receptor subunit beta-2 | Homo sapiens (human) | EC50 | 9.3127 | 23 | 27 |
| Neuronal acetylcholine receptor subunit beta-2 | Mus musculus (house mouse) | EC50 | 0.7222 | 1 | 2 |
| Neuronal acetylcholine receptor subunit beta-2 | Rattus norvegicus (Norway rat) | EC50 | 11.5290 | 12 | 13 |
| Neuronal acetylcholine receptor subunit beta-2 | Rattus norvegicus (Norway rat) | Kd | 14,352.0000 | 3 | 3 |
| Neuronal acetylcholine receptor subunit beta-3 | Homo sapiens (human) | EC50 | 10.5635 | 2 | 2 |
| Neuronal acetylcholine receptor subunit beta-3 | Rattus norvegicus (Norway rat) | EC50 | 35.5000 | 2 | 2 |
| Neuronal acetylcholine receptor subunit beta-3 | Rattus norvegicus (Norway rat) | Kd | 14,352.0000 | 3 | 3 |
| Neuronal acetylcholine receptor subunit beta-4 | Homo sapiens (human) | EC50 | 13.6576 | 14 | 15 |
| Neuronal acetylcholine receptor subunit beta-4 | Rattus norvegicus (Norway rat) | EC50 | 30.2517 | 7 | 8 |
| Neuronal acetylcholine receptor subunit beta-4 | Rattus norvegicus (Norway rat) | Kd | 14,352.0000 | 3 | 3 |
| Nitric oxide synthase, inducible | Homo sapiens (human) | Kd | 7.0000 | 2 | 2 |
| Non-receptor tyrosine-protein kinase TNK1 | Homo sapiens (human) | Kd | 15.1600 | 2 | 2 |
| Non-receptor tyrosine-protein kinase TYK2 | Homo sapiens (human) | Kd | 10.7367 | 3 | 3 |
| NT-3 growth factor receptor | Homo sapiens (human) | Kd | 0.0820 | 1 | 1 |
| NUAK family SNF1-like kinase 1 | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| NUAK family SNF1-like kinase 2 | Homo sapiens (human) | Kd | 20.0400 | 2 | 3 |
| Nucleolar GTP-binding protein 1 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Obg-like ATPase 1 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Oxysterols receptor LXR-alpha | Homo sapiens (human) | EC50 | 0.1300 | 2 | 2 |
| PAS domain-containing serine/threonine-protein kinase | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Peripheral plasma membrane protein CASK | Homo sapiens (human) | Kd | 0.1400 | 1 | 1 |
| Peroxisomal acyl-coenzyme A oxidase 1 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Peroxisomal acyl-coenzyme A oxidase 3 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Phenylalanine--tRNA ligase beta subunit | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Phosphatidylethanolamine-binding protein 1 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Phosphatidylinositol 4-kinase beta | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Phosphatidylinositol 4-phosphate 3-kinase C2 domain-containing subunit beta | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Phosphatidylinositol 4-phosphate 3-kinase C2 domain-containing subunit gamma | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Phosphatidylinositol 4-phosphate 5-kinase type-1 alpha | Homo sapiens (human) | Kd | 3.2000 | 1 | 1 |
| Phosphatidylinositol 4-phosphate 5-kinase type-1 gamma | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform | Homo sapiens (human) | Kd | 10.0000 | 10 | 10 |
| Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Phosphatidylinositol 5-phosphate 4-kinase type-2 alpha | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Phosphatidylinositol 5-phosphate 4-kinase type-2 beta | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Phosphatidylinositol 5-phosphate 4-kinase type-2 gamma | Homo sapiens (human) | Kd | 20.0000 | 2 | 2 |
| Phosphorylase b kinase gamma catalytic chain, liver/testis isoform | Homo sapiens (human) | Kd | 20.0000 | 2 | 2 |
| Phosphorylase b kinase gamma catalytic chain, skeletal muscle/heart isoform | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Platelet-derived growth factor receptor alpha | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Platelet-derived growth factor receptor beta | Homo sapiens (human) | Kd | 20.0000 | 2 | 2 |
| Probable ATP-dependent RNA helicase DDX6 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Prostaglandin G/H synthase 2 | Homo sapiens (human) | Kd | 6.1000 | 1 | 1 |
| Protein kinase C alpha type | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Protein kinase C beta type | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Protein kinase C delta type | Homo sapiens (human) | Kd | 20.0000 | 2 | 2 |
| Protein kinase C epsilon type | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Protein kinase C eta type | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Protein kinase C iota type | Homo sapiens (human) | Kd | 20.0000 | 2 | 2 |
| Protein kinase C theta type | Homo sapiens (human) | Kd | 20.0000 | 2 | 2 |
| Protein-tyrosine kinase 2-beta | Homo sapiens (human) | Kd | 15.0950 | 2 | 2 |
| Protein-tyrosine kinase 6 | Homo sapiens (human) | Kd | 20.0000 | 2 | 2 |
| Proto-oncogene tyrosine-protein kinase receptor Ret | Homo sapiens (human) | Kd | 10.6800 | 5 | 5 |
| Proto-oncogene tyrosine-protein kinase ROS | Homo sapiens (human) | Kd | 0.0041 | 1 | 1 |
| Proto-oncogene tyrosine-protein kinase Src | Homo sapiens (human) | Kd | 15.2800 | 2 | 2 |
| Putative heat shock protein HSP 90-beta 2 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Pyridoxal kinase | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Rab-like protein 3 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| RAC-alpha serine/threonine-protein kinase | Homo sapiens (human) | Kd | 20.0000 | 2 | 2 |
| RAC-beta serine/threonine-protein kinase | Homo sapiens (human) | Kd | 20.0000 | 2 | 2 |
| RAC-gamma serine/threonine-protein kinase | Homo sapiens (human) | Kd | 20.0000 | 2 | 2 |
| RAF proto-oncogene serine/threonine-protein kinase | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Ras-related protein Rab-10 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Ras-related protein Rab-27A | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Ras-related protein Rab-6A | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Receptor tyrosine-protein kinase erbB-2 | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Receptor tyrosine-protein kinase erbB-3 | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Receptor tyrosine-protein kinase erbB-4 | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Receptor-interacting serine/threonine-protein kinase 1 | Homo sapiens (human) | Kd | 1.4500 | 2 | 2 |
| Receptor-interacting serine/threonine-protein kinase 2 | Homo sapiens (human) | Kd | 15.4500 | 2 | 2 |
| Receptor-interacting serine/threonine-protein kinase 3 | Homo sapiens (human) | Kd | 18.3500 | 2 | 2 |
| Receptor-interacting serine/threonine-protein kinase 4 | Homo sapiens (human) | Kd | 2.1000 | 1 | 1 |
| Receptor-type tyrosine-protein kinase FLT3 | Homo sapiens (human) | Kd | 4.6312 | 8 | 8 |
| Rho-associated protein kinase 1 | Homo sapiens (human) | Kd | 16.8500 | 2 | 2 |
| Rho-associated protein kinase 2 | Homo sapiens (human) | Kd | 16.6500 | 2 | 2 |
| Rhodopsin kinase GRK1 | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Rhodopsin kinase GRK7 | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Ribosomal protein S6 kinase alpha-1 | Homo sapiens (human) | Kd | 16.6667 | 3 | 3 |
| Ribosomal protein S6 kinase alpha-2 | Homo sapiens (human) | Kd | 10.0000 | 2 | 2 |
| Ribosomal protein S6 kinase alpha-3 | Homo sapiens (human) | Kd | 20.0000 | 2 | 2 |
| Ribosomal protein S6 kinase alpha-4 | Homo sapiens (human) | Kd | 16.6667 | 3 | 3 |
| Ribosomal protein S6 kinase alpha-5 | Homo sapiens (human) | Kd | 20.0000 | 3 | 4 |
| Ribosomal protein S6 kinase alpha-6 | Homo sapiens (human) | Kd | 16.6667 | 3 | 3 |
| Ribosomal protein S6 kinase beta-1 | Homo sapiens (human) | Kd | 15.3200 | 2 | 2 |
| Ribosyldihydronicotinamide dehydrogenase [quinone] | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| RNA cytidine acetyltransferase | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| S-adenosylmethionine synthase isoform type-2 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Septin-9 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Serine/threonine-protein kinase 10 | Homo sapiens (human) | Kd | 1.4335 | 2 | 2 |
| Serine/threonine-protein kinase 16 | Homo sapiens (human) | Kd | 20.0000 | 2 | 2 |
| Serine/threonine-protein kinase 17A | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Serine/threonine-protein kinase 17B | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Serine/threonine-protein kinase 24 | Homo sapiens (human) | Kd | 20.0000 | 2 | 2 |
| Serine/threonine-protein kinase 25 | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Serine/threonine-protein kinase 26 | Homo sapiens (human) | Kd | 16.4000 | 2 | 2 |
| Serine/threonine-protein kinase 3 | Homo sapiens (human) | Kd | 15.4950 | 2 | 2 |
| Serine/threonine-protein kinase 32A | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Serine/threonine-protein kinase 32B | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Serine/threonine-protein kinase 32C | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Serine/threonine-protein kinase 33 | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Serine/threonine-protein kinase 35 | Homo sapiens (human) | Kd | 0.6100 | 1 | 1 |
| Serine/threonine-protein kinase 36 | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Serine/threonine-protein kinase 38 | Homo sapiens (human) | Kd | 20.0000 | 2 | 2 |
| Serine/threonine-protein kinase 38-like | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Serine/threonine-protein kinase 4 | Homo sapiens (human) | Kd | 15.2900 | 2 | 2 |
| Serine/threonine-protein kinase A-Raf | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Serine/threonine-protein kinase B-raf | Homo sapiens (human) | Kd | 16.6667 | 3 | 3 |
| Serine/threonine-protein kinase BRSK1 | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Serine/threonine-protein kinase BRSK2 | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Serine/threonine-protein kinase Chk1 | Homo sapiens (human) | Kd | 20.0000 | 2 | 2 |
| Serine/threonine-protein kinase Chk2 | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Serine/threonine-protein kinase D1 | Homo sapiens (human) | Kd | 0.9900 | 1 | 1 |
| Serine/threonine-protein kinase D2 | Homo sapiens (human) | Kd | 8.2440 | 2 | 2 |
| Serine/threonine-protein kinase D3 | Homo sapiens (human) | Kd | 0.6885 | 2 | 2 |
| Serine/threonine-protein kinase DCLK1 | Homo sapiens (human) | Kd | 0.3300 | 1 | 1 |
| Serine/threonine-protein kinase DCLK2 | Homo sapiens (human) | Kd | 0.3700 | 1 | 1 |
| Serine/threonine-protein kinase DCLK3 | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Serine/threonine-protein kinase ICK | Homo sapiens (human) | Kd | 20.0000 | 2 | 2 |
| Serine/threonine-protein kinase LATS1 | Homo sapiens (human) | Kd | 20.0000 | 2 | 2 |
| Serine/threonine-protein kinase LATS2 | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Serine/threonine-protein kinase MAK | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Serine/threonine-protein kinase MARK1 | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Serine/threonine-protein kinase MARK2 | Homo sapiens (human) | Kd | 20.0000 | 2 | 2 |
| Serine/threonine-protein kinase MRCK alpha | Homo sapiens (human) | Kd | 20.0000 | 2 | 2 |
| Serine/threonine-protein kinase MRCK beta | Homo sapiens (human) | Kd | 20.0000 | 2 | 2 |
| Serine/threonine-protein kinase MRCK gamma | Homo sapiens (human) | Kd | 23.3333 | 2 | 3 |
| Serine/threonine-protein kinase mTOR | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Serine/threonine-protein kinase N1 | Homo sapiens (human) | Kd | 20.0000 | 2 | 2 |
| Serine/threonine-protein kinase N2 | Homo sapiens (human) | Kd | 20.0000 | 2 | 2 |
| Serine/threonine-protein kinase N3 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Serine/threonine-protein kinase Nek1 | Homo sapiens (human) | Kd | 20.0000 | 2 | 2 |
| Serine/threonine-protein kinase Nek11 | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Serine/threonine-protein kinase Nek2 | Homo sapiens (human) | Kd | 20.0000 | 2 | 2 |
| Serine/threonine-protein kinase Nek3 | Homo sapiens (human) | Kd | 20.0000 | 2 | 2 |
| Serine/threonine-protein kinase Nek4 | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Serine/threonine-protein kinase Nek5 | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Serine/threonine-protein kinase Nek6 | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Serine/threonine-protein kinase Nek7 | Homo sapiens (human) | Kd | 5.7000 | 1 | 1 |
| Serine/threonine-protein kinase Nek9 | Homo sapiens (human) | Kd | 15.3950 | 2 | 2 |
| Serine/threonine-protein kinase NIM1 | Homo sapiens (human) | Kd | 4.6000 | 1 | 1 |
| Serine/threonine-protein kinase NLK | Homo sapiens (human) | Kd | 20.0000 | 2 | 2 |
| Serine/threonine-protein kinase OSR1 | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Serine/threonine-protein kinase PAK 1 | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Serine/threonine-protein kinase PAK 2 | Homo sapiens (human) | Kd | 20.0000 | 2 | 2 |
| Serine/threonine-protein kinase PAK 3 | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Serine/threonine-protein kinase PAK 4 | Homo sapiens (human) | Kd | 20.0000 | 2 | 2 |
| Serine/threonine-protein kinase PAK 5 | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Serine/threonine-protein kinase PAK 6 | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Serine/threonine-protein kinase pim-1 | Homo sapiens (human) | Kd | 20.0000 | 2 | 2 |
| Serine/threonine-protein kinase pim-2 | Homo sapiens (human) | Kd | 20.0000 | 2 | 2 |
| Serine/threonine-protein kinase pim-3 | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Serine/threonine-protein kinase PknB | Mycobacterium tuberculosis H37Rv | Kd | 10.0000 | 1 | 1 |
| Serine/threonine-protein kinase PLK1 | Homo sapiens (human) | Kd | 20.0000 | 2 | 2 |
| Serine/threonine-protein kinase PLK2 | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Serine/threonine-protein kinase PLK3 | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Serine/threonine-protein kinase PLK4 | Homo sapiens (human) | Kd | 15.0300 | 2 | 2 |
| Serine/threonine-protein kinase PRP4 homolog | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Serine/threonine-protein kinase receptor R3 | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Serine/threonine-protein kinase RIO1 | Homo sapiens (human) | Kd | 6.1000 | 1 | 1 |
| Serine/threonine-protein kinase RIO2 | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Serine/threonine-protein kinase RIO3 | Homo sapiens (human) | Kd | 4.0000 | 1 | 1 |
| Serine/threonine-protein kinase SBK1 | Homo sapiens (human) | Kd | 1.3000 | 1 | 1 |
| Serine/threonine-protein kinase Sgk3 | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Serine/threonine-protein kinase SIK1 | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Serine/threonine-protein kinase SIK2 | Homo sapiens (human) | Kd | 15.1000 | 2 | 2 |
| Serine/threonine-protein kinase SIK3 | Homo sapiens (human) | Kd | 20.0000 | 2 | 2 |
| Serine/threonine-protein kinase STK11 | Homo sapiens (human) | Kd | 20.0000 | 2 | 2 |
| Serine/threonine-protein kinase TAO1 | Homo sapiens (human) | Kd | 15.6000 | 2 | 2 |
| Serine/threonine-protein kinase TAO2 | Homo sapiens (human) | Kd | 15.4500 | 2 | 2 |
| Serine/threonine-protein kinase TAO3 | Homo sapiens (human) | Kd | 15.2450 | 2 | 2 |
| Serine/threonine-protein kinase TBK1 | Homo sapiens (human) | Kd | 20.2300 | 2 | 3 |
| Serine/threonine-protein kinase TNNI3K | Homo sapiens (human) | Kd | 0.1100 | 1 | 1 |
| Serine/threonine-protein kinase tousled-like 1 | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Serine/threonine-protein kinase tousled-like 2 | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Serine/threonine-protein kinase ULK1 | Homo sapiens (human) | Kd | 15.5000 | 2 | 2 |
| Serine/threonine-protein kinase ULK2 | Homo sapiens (human) | Kd | 1.6000 | 1 | 1 |
| Serine/threonine-protein kinase ULK3 | Homo sapiens (human) | Kd | 18.3500 | 2 | 2 |
| Serine/threonine-protein kinase VRK2 | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Serine/threonine-protein kinase/endoribonuclease IRE1 | Homo sapiens (human) | Kd | 20.0000 | 2 | 2 |
| Serine/threonine-protein kinase/endoribonuclease IRE2 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Signal recognition particle receptor subunit alpha | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| SNF-related serine/threonine-protein kinase | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| SRSF protein kinase 1 | Homo sapiens (human) | Kd | 1.8000 | 1 | 1 |
| SRSF protein kinase 2 | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| SRSF protein kinase 3 | Homo sapiens (human) | Kd | 8.2000 | 1 | 1 |
| STE20-like serine/threonine-protein kinase | Homo sapiens (human) | Kd | 0.5985 | 2 | 2 |
| STE20-related kinase adapter protein alpha | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| STE20/SPS1-related proline-alanine-rich protein kinase | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Structural maintenance of chromosomes protein 1A | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Structural maintenance of chromosomes protein 2 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Succinate--CoA ligase [ADP-forming] subunit beta, mitochondrial | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Testis-specific serine/threonine-protein kinase 1 | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| TGF-beta receptor type-1 | Homo sapiens (human) | Kd | 2.2460 | 2 | 2 |
| TGF-beta receptor type-2 | Homo sapiens (human) | Kd | 20.0000 | 2 | 2 |
| Thyroid hormone receptor-associated protein 3 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Trace amine-associated receptor 1 | Homo sapiens (human) | EC50 | 0.3080 | 1 | 1 |
| TRAF2 and NCK-interacting protein kinase | Homo sapiens (human) | Kd | 20.0000 | 2 | 2 |
| Transient receptor potential cation channel subfamily A member 1 | Homo sapiens (human) | EC50 | 152,369.0000 | 2 | 3 |
| Transient receptor potential cation channel subfamily A member 1 | Mus musculus (house mouse) | EC50 | 10.0000 | 1 | 1 |
| Transient receptor potential cation channel subfamily M member 6 | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Transporter | Rattus norvegicus (Norway rat) | EC50 | 51.0000 | 1 | 1 |
| Tyrosine--tRNA ligase, cytoplasmic | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Tyrosine-protein kinase ABL1 | Homo sapiens (human) | Kd | 0.5482 | 16 | 16 |
| Tyrosine-protein kinase ABL2 | Homo sapiens (human) | Kd | 0.4435 | 2 | 2 |
| Tyrosine-protein kinase Blk | Homo sapiens (human) | Kd | 0.1100 | 1 | 1 |
| Tyrosine-protein kinase BTK | Homo sapiens (human) | Kd | 18.9000 | 2 | 2 |
| Tyrosine-protein kinase CSK | Homo sapiens (human) | Kd | 20.0000 | 2 | 2 |
| Tyrosine-protein kinase Fer | Homo sapiens (human) | Kd | 15.1350 | 2 | 2 |
| Tyrosine-protein kinase Fes/Fps | Homo sapiens (human) | Kd | 20.1500 | 2 | 3 |
| Tyrosine-protein kinase Fgr | Homo sapiens (human) | Kd | 15.3350 | 2 | 2 |
| Tyrosine-protein kinase FRK | Homo sapiens (human) | Kd | 16.4500 | 2 | 2 |
| Tyrosine-protein kinase Fyn | Homo sapiens (human) | Kd | 15.6500 | 2 | 2 |
| Tyrosine-protein kinase HCK | Homo sapiens (human) | Kd | 20.0000 | 2 | 2 |
| Tyrosine-protein kinase ITK/TSK | Homo sapiens (human) | Kd | 2.0000 | 1 | 1 |
| Tyrosine-protein kinase JAK1 | Homo sapiens (human) | Kd | 13.4433 | 3 | 3 |
| Tyrosine-protein kinase JAK2 | Homo sapiens (human) | Kd | 10.1003 | 3 | 3 |
| Tyrosine-protein kinase JAK3 | Homo sapiens (human) | Kd | 0.2000 | 1 | 1 |
| Tyrosine-protein kinase Lck | Homo sapiens (human) | Kd | 0.7220 | 2 | 2 |
| Tyrosine-protein kinase Lyn | Homo sapiens (human) | Kd | 15.4700 | 2 | 2 |
| Tyrosine-protein kinase Mer | Homo sapiens (human) | Kd | 0.0036 | 1 | 1 |
| Tyrosine-protein kinase receptor Tie-1 | Homo sapiens (human) | Kd | 0.1100 | 1 | 1 |
| Tyrosine-protein kinase receptor TYRO3 | Homo sapiens (human) | Kd | 0.8000 | 1 | 1 |
| Tyrosine-protein kinase receptor UFO | Homo sapiens (human) | Kd | 0.0078 | 1 | 1 |
| Tyrosine-protein kinase Srms | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Tyrosine-protein kinase SYK | Homo sapiens (human) | Kd | 16.2500 | 2 | 2 |
| Tyrosine-protein kinase Tec | Homo sapiens (human) | Kd | 20.0000 | 2 | 2 |
| Tyrosine-protein kinase TXK | Homo sapiens (human) | Kd | 0.8500 | 1 | 1 |
| Tyrosine-protein kinase Yes | Homo sapiens (human) | Kd | 15.3850 | 2 | 2 |
| Tyrosine-protein kinase ZAP-70 | Homo sapiens (human) | Kd | 4.2000 | 1 | 1 |
| U5 small nuclear ribonucleoprotein 200 kDa helicase | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| UMP-CMP kinase | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Uncharacterized aarF domain-containing protein kinase 5 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Uncharacterized protein FLJ45252 | Homo sapiens (human) | Kd | 30.0000 | 1 | 1 |
| Uncharacterized serine/threonine-protein kinase SBK3 | Homo sapiens (human) | Kd | 0.2400 | 1 | 1 |
| Vascular endothelial growth factor receptor 1 | Homo sapiens (human) | Kd | 2.3000 | 1 | 1 |
| Vascular endothelial growth factor receptor 2 | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Vascular endothelial growth factor receptor 3 | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |
| Very long-chain specific acyl-CoA dehydrogenase, mitochondrial | Homo sapiens (human) | Kd | 30.0000 | 1 | 2 |
| Wee1-like protein kinase | Homo sapiens (human) | Kd | 20.0000 | 2 | 2 |
| Wee1-like protein kinase 2 | Homo sapiens (human) | Kd | 10.0000 | 1 | 1 |