Page last updated: 2024-08-07 18:38:48
Acetylcholine-binding protein
[no definition available]
Synonyms
ACh-binding protein;
AchBP
Research
Bioassay Publications (13)
Timeframe | Studies on this Protein(%) | All Drugs % |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 0 (0.00) | 18.2507 |
2000's | 1 (7.69) | 29.6817 |
2010's | 11 (84.62) | 24.3611 |
2020's | 1 (7.69) | 2.80 |
Compounds (22)
Drugs with Inhibition Measurements
Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
---|---|---|---|---|---|
3-(1-methylpyrrolidin-2-yl)pyridine | Lymnaea stagnalis (great pond snail) | Ki | 0.0863 | 1 | 3 |
epibatidine | Lymnaea stagnalis (great pond snail) | Ki | 0.0003 | 1 | 1 |
LSM-22634 | Lymnaea stagnalis (great pond snail) | Ki | 0.1014 | 1 | 3 |
nicotine | Lymnaea stagnalis (great pond snail) | Ki | 0.2236 | 7 | 8 |
lobeline | Lymnaea stagnalis (great pond snail) | Ki | 0.6310 | 1 | 1 |
thiacloprid | Lymnaea stagnalis (great pond snail) | Ki | 0.2200 | 1 | 1 |
aaptamine | Lymnaea stagnalis (great pond snail) | Ki | 3.0000 | 1 | 1 |
dibenzheptropine | Lymnaea stagnalis (great pond snail) | Ki | 1.1967 | 2 | 2 |
prizes | Lymnaea stagnalis (great pond snail) | Ki | 1.2000 | 1 | 1 |
harmicine | Lymnaea stagnalis (great pond snail) | Ki | 1.2589 | 1 | 1 |
tropacocaine | Lymnaea stagnalis (great pond snail) | Ki | 4.1524 | 1 | 2 |
epibatidine | Lymnaea stagnalis (great pond snail) | Ki | 0.0061 | 1 | 3 |
pnu-282987 | Lymnaea stagnalis (great pond snail) | Ki | 2.0893 | 1 | 1 |
desnitroimidacloprid | Lymnaea stagnalis (great pond snail) | Ki | 0.0180 | 1 | 1 |
rhizochaline | Lymnaea stagnalis (great pond snail) | Ki | 28.0000 | 1 | 1 |
monanchocidin | Lymnaea stagnalis (great pond snail) | Ki | 2.5000 | 1 | 1 |
alpha-conotoxin pnia | Lymnaea stagnalis (great pond snail) | Ki | 9.1201 | 1 | 1 |
imidacloprid | Lymnaea stagnalis (great pond snail) | Ki | 0.9700 | 1 | 1 |
debromohymenialdisine | Lymnaea stagnalis (great pond snail) | Ki | 1,000.0000 | 1 | 2 |
Drugs with Activation Measurements
Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
---|---|---|---|---|---|
nicotine | Lymnaea stagnalis (great pond snail) | Kd | 0.2931 | 3 | 5 |
lobeline | Lymnaea stagnalis (great pond snail) | Kd | 0.6305 | 1 | 2 |
epibatidine | Lymnaea stagnalis (great pond snail) | Kd | 0.0014 | 1 | 2 |
3-(2,4-dimethoxybenzylidene)anabaseine | Lymnaea stagnalis (great pond snail) | Kd | 0.0190 | 1 | 1 |
pnu-282987 | Lymnaea stagnalis (great pond snail) | Kd | 3.6308 | 1 | 1 |
3-(4-hydroxy-2-methoxybenzylidene)anabaseine | Lymnaea stagnalis (great pond snail) | Kd | 0.0004 | 1 | 1 |