Proteins > Acetylcholine receptor subunit delta
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Acetylcholine receptor subunit delta
[no definition available]
Synonyms
Research
Bioassay Publications (7)
| Timeframe | Studies on this Protein(%) | All Drugs % |
|---|
| pre-1990 | 1 (14.29) | 18.7374 |
| 1990's | 3 (42.86) | 18.2507 |
| 2000's | 2 (28.57) | 29.6817 |
| 2010's | 1 (14.29) | 24.3611 |
| 2020's | 0 (0.00) | 2.80 |
Compounds (16)
Drugs with Inhibition Measurements
| Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
|---|
| nornicotine | Tetronarce californica (Pacific electric ray) | IC50 | 0.2000 | 2 | 2 |
| epibatidine | Tetronarce californica (Pacific electric ray) | Ki | 0.0014 | 2 | 2 |
| cytisine | Tetronarce californica (Pacific electric ray) | Ki | 0.2500 | 1 | 1 |
| nicotine | Tetronarce californica (Pacific electric ray) | IC50 | 0.0025 | 2 | 2 |
| nicotine | Tetronarce californica (Pacific electric ray) | Ki | 8.1350 | 2 | 2 |
| 3-methyl-5-(1-methyl-2-pyrrolidinyl)isoxazole | Tetronarce californica (Pacific electric ray) | Ki | 10.0000 | 1 | 1 |
| aaptamine | Tetronarce californica (Pacific electric ray) | Ki | 34.0000 | 1 | 1 |
| anatoxin a | Tetronarce californica (Pacific electric ray) | IC50 | 0.0006 | 2 | 2 |
| etomidate | Tetronarce californica (Pacific electric ray) | IC50 | 41.0000 | 1 | 1 |
| rhizochaline | Tetronarce californica (Pacific electric ray) | Ki | 22.0000 | 1 | 1 |
| monanchocidin | Tetronarce californica (Pacific electric ray) | Ki | 8.0000 | 1 | 1 |
| debromohymenialdisine | Tetronarce californica (Pacific electric ray) | Ki | 1,000.0000 | 1 | 1 |
Drugs with Activation Measurements
Emerging molecular approaches to pain therapy.Journal of medicinal chemistry, , May-06, Volume: 42, Issue:9, 1999
Neuronal nicotinic acetylcholine receptors as targets for drug discovery.Journal of medicinal chemistry, , Dec-19, Volume: 40, Issue:26, 1997
Varenicline: an alpha4beta2 nicotinic receptor partial agonist for smoking cessation.Journal of medicinal chemistry, , May-19, Volume: 48, Issue:10, 2005
Neuronal nicotinic acetylcholine receptors as targets for drug discovery.Journal of medicinal chemistry, , Dec-19, Volume: 40, Issue:26, 1997
Varenicline: an alpha4beta2 nicotinic receptor partial agonist for smoking cessation.Journal of medicinal chemistry, , May-19, Volume: 48, Issue:10, 2005
Neuronal nicotinic acetylcholine receptors as targets for drug discovery.Journal of medicinal chemistry, , Dec-19, Volume: 40, Issue:26, 1997
Synthesis and biological characterization of pyridohomotropanes. Structure-activity relationships of conformationally restricted nicotinoids.Journal of medicinal chemistry, , Volume: 31, Issue:3, 1988