Proteins > Soluble acetylcholine receptor
Page last updated: 2024-08-08 00:06:22
Soluble acetylcholine receptor
[no definition available]
Synonyms
Research
Bioassay Publications (3)
| Timeframe | Studies on this Protein(%) | All Drugs % |
|---|
| pre-1990 | 0 (0.00) | 18.7374 |
| 1990's | 0 (0.00) | 18.2507 |
| 2000's | 0 (0.00) | 29.6817 |
| 2010's | 3 (100.00) | 24.3611 |
| 2020's | 0 (0.00) | 2.80 |
Compounds (9)
Drugs with Inhibition Measurements
| Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
|---|
| epibatidine | Aplysia californica (California sea hare) | Ki | 0.0010 | 1 | 1 |
| nicotine | Aplysia californica (California sea hare) | Ki | 1.0466 | 3 | 3 |
| lobeline | Aplysia californica (California sea hare) | Ki | 0.0025 | 1 | 1 |
| thiacloprid | Aplysia californica (California sea hare) | Ki | 0.0039 | 1 | 1 |
| dibenzheptropine | Aplysia californica (California sea hare) | Ki | 6.3096 | 1 | 1 |
| prizes | Aplysia californica (California sea hare) | Ki | 0.0320 | 1 | 1 |
| tropacocaine | Aplysia californica (California sea hare) | Ki | 9.9150 | 1 | 2 |
| desnitroimidacloprid | Aplysia californica (California sea hare) | Ki | 0.0150 | 1 | 1 |
| imidacloprid | Aplysia californica (California sea hare) | Ki | 0.0190 | 1 | 1 |
Structure-based design, synthesis and structure-activity relationships of dibenzosuberyl- and benzoate-substituted tropines as ligands for acetylcholine-binding protein.Bioorganic & medicinal chemistry letters, , Feb-01, Volume: 22, Issue:3, 2012
Insights into the structural determinants required for high-affinity binding of chiral cyclopropane-containing ligands to α4β2-nicotinic acetylcholine receptors: an integrated approach to behaviorally active nicotinic ligands.Journal of medicinal chemistry, , Sep-27, Volume: 55, Issue:18, 2012
Unique neonicotinoid binding conformations conferring selective receptor interactions.Journal of agricultural and food chemistry, , Apr-13, Volume: 59, Issue:7, 2011