Proteins > Muscarinic acetylcholine receptor M4
Page last updated: 2024-08-07 16:29:44
Muscarinic acetylcholine receptor M4
A muscarinic acetylcholine receptor M4 that is encoded in the genome of mouse. [OMA:P32211, PRO:DNx]
Synonyms
Mm4 mAChR
Research
Bioassay Publications (5)
| Timeframe | Studies on this Protein(%) | All Drugs % |
|---|
| pre-1990 | 3 (60.00) | 18.7374 |
| 1990's | 0 (0.00) | 18.2507 |
| 2000's | 1 (20.00) | 29.6817 |
| 2010's | 1 (20.00) | 24.3611 |
| 2020's | 0 (0.00) | 2.80 |
Compounds (10)
Drugs with Inhibition Measurements
| Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
|---|
| pirenzepine | Mus musculus (house mouse) | IC50 | 0.7500 | 1 | 3 |
| pinacidil | Mus musculus (house mouse) | IC50 | 8.9000 | 1 | 3 |
| dexetimide | Mus musculus (house mouse) | IC50 | 0.0033 | 1 | 3 |
| nicotine | Mus musculus (house mouse) | Ki | 2.1100 | 1 | 1 |
| varenicline | Mus musculus (house mouse) | Ki | 0.1250 | 1 | 1 |
| atropine | Mus musculus (house mouse) | Ki | 0.0005 | 1 | 1 |
Drugs with Activation Measurements
| Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
|---|
| phencyclidine | Mus musculus (house mouse) | Kd | 9.1000 | 1 | 1 |
Drugs with Other Measurements