Page last updated: 2024-08-05 15:14:08

EC 2.7.11.22 (cyclin-dependent kinase) inhibitor

An EC 2.7.11.* (protein-serine/threonine kinase) inhibitor that interferes with the action of cyclin-dependent kinase (EC 2.7.11.22).

ChEBI ID: 82665

Members (19)

MemberDefinitionClass
((5z)5-(1,3-benzodioxol-5-yl)methylene-2-phenylamino-3,5-dihydro-4h-imidazol-4-one)A member of the class of benzodioxoles that is 1,3-benzodioxole substituted by a (2-anilino-5-oxo-1,5-dihydro-4H-imidazol-4-ylidene)methyl group at position 5. It is an inhibitor of DYRK1A, DYRK2, CLK1, and CLK3 (IC50s = 0.04, 0.035, 0.015, and 4.5 muM, respectively).leucettine L41
(R)-DRF053A member of the class of 2,6-diaminopurines that is 2,6-diamiopurine which is substituted by an isopropyl group at position 9 and in which the amino groups at positions 2 and 6 are substituted by a 1-hydroxybutan-2-yl and 3-(pyridin-2-yl)phenyl groups, respectively (the R enantiomer). A cyclin dependent kinase inhibitor, widely used as its hydrochloride hydrate.(R)-DRF053
5,7-dihydroxy-2-methyl-8-(4-(3-hydroxy-1-methyl)-piperidinyl)-4h-1-benzopyran-4-oneA member of the class of chromones that is 4H-chromen-4-one in which the hydrogens at positions 2,5,7 and 8 are replaced by methyl, hydroxy, hydroxy, and (3S,4R)-3-hydroxy-1-methylpiperidin-4-yl groups, respectively. It is an alkaloid initially isolated from Amoora rohituka and is a precursor of the anti-cancer compound flavopiridol.rohitukine
adapaleneA naphthoic acid that is CD437 in which the phenolic hydroxy group has been converted to its methyl ether.adapalene
alsterpaulloneAn organic heterotetracyclic compound that is 1,3-dihydro-2H-1-benzazepin-2-one which shares its 4-5 bond with the 3-2 bond of 5-nitro-1H-indole.alsterpaullone
alvocidibA synthetic dihydroxyflavone that is 5,7-dihydroxyflavone which is substituted by a 3-hydroxy-1-methylpiperidin-4-yl group at position 8 and by a chlorine at the 2' position (the (-)-3S,4R stereoisomer). A cyclin-dependent kinase 9 (CDK9) inhibitor, it has been studied for the treatment of acute myeloid leukaemia, arthritis and atherosclerotic plaque formation.alvocidib
at 7519A member of the class of pryrazoles that is 4-amino-1H-pyrazole-3-carboxylic acid in which the primary amino group has been acylated by a 2,6-dichlorobenzoyl group and in which the carboxylic acid has been converted into a carboxamide by formal condensation with the primary amino group of 4-aminopiperidine.4-(2,6-dichlorobenzamido)-N-(piperidin-4-yl)-pyrazole-3-carboxamide
bms 387032A secondary carboxamide resulting from the formal condensation of the carboxy group of piperidine-4-carboxylic acid with the amino group of 5-{[(5-tert-butyl-1,3-oxazol-2-yl)methyl]sulfanyl}-1,3-thiazol-2-amine. It is an ATP-competitive inhibitor of CDK2, CDK7 and CDK9 kinases and exhibits anti-cancer properties.N-(5-{[(5-tert-butyl-1,3-oxazol-2-yl)methyl]sulfanyl}-1,3-thiazol-2-yl)piperidine-4-carboxamide
boheminePurine substituted on C-2, C-6 and N-9 with (3-hydroxypropyl)amino, benzylamino and isopropyl groups respectively; a synthetic, cell-permeable, cyclin-dependent kinase (CDK) inhibitor that is structurally similar to olomoucine and roscovitine.bohemine
can 508A member of the class of pyrazoles that is 1H-pyrazole substituted by amino, (4-hydroxyphenyl)diazenyl, and amino groups at positions 3, 4 and 5, respectively. It is a CDK9 inhibitor (IC50 = 0.35 muM) with 38-fold selectivity for CDK9/cyclin T over other CDK/cyclin complexes.CAN-508
CCT251545A chloropyridine that is 3-chloropyridine substituted by a 1-oxo-2,8-diazaspiro[4.5]decan-8-yl group and a 4-(1-methyl-1H-pyrazol-4-yl)phenyl group at positions 4 and 5, respectively. It is an orally bioavailable inhibitor of Wnt signaling (IC50 = 5 nM) and a potent and selective chemical probe for cyclin-dependent kinases CDK8 and CDK19.CCT251545
cyc 2022,6-Diaminopurine carrying benzylamino, (2R)-1-hydroxybutan-2-yl and isopropyl substituents at C-6, C-2-N and N-9 respectively. It is an experimental drug candidate in the family of pharmacological cyclin-dependent kinase (CDK) inhibitors.seliciclib
hmr 1275A hydrochloride salt resulting from the formal reaction of equimolar amounts of alvocidib and hydrogen chloride. A cyclin-dependent kinase 9 (CDK9) inhibitor, it has been studied for the treatment of acute myeloid leukaemia, arthritis and atherosclerotic plaque formation.alvocidib hydrochloride
ldc4297A pyrazolotriazine that is pyrazolo[1,5-a][1,3,5]triazine substituted by a piperidin-3-yloxy group, [2-(1H-pyrazol-1-yl)benzyl]nitrilo group and an isopropyl group at positions 2, 4 and 8 respectively. It is a potent and selective CDK7 inhibitor and exhibits antiviral activity.LDC4297
nsc 664704An indolobenzazepine that is paullone in which the hydrogen at position 9 is replaced by a bromo substituent. It is an ATP-competitive inhibitor of cyclin-dependent kinases (CDKs) and glycogen synthase kinase 3beta (GSK3beta).kenpaullone
olomoucineA 9H-purine that is substituted by a (2-hydroxyethyl)nitrilo, benzylnitrilo and a methyl group at positions 2,6 and 9, respectively. It is a cyclin-dependent kinase inhibitor.olomoucine
palbociclibA member of the class of pyridopyrimidines that is 2-{[5-(piperazin-1-yl)pyridin-2-yl]amino}pyrido[2,3-d]pyrimidin-7-one bearing additional methyl, acetyl and cyclopentyl substituents at positions 5, 6 and 8 respectively. It is used in combination with letrozole for the treatment of metastatic breast cancer.palbociclib
paulloneAn indolobenzazepine that is 5,6,7,12-tetrahydroindolo[3,2-d][1]benzazepine carrying an oxo substituent at position 6.paullone
THZ531A member of the class of indoles that is 5-chloro-4-(1H-indol-3-yl)-N-[(3R)-piperidin-3-yl]pyrimidin-2-amine in which the piperidine NH group is substituted by a 4-{[(2E)-4-(dimethylamino)but-2-enoyl]amino}benzoyl group. It is a first-in-class CDK12 and CDK13 covalent kinase inhibitor with IC50 of 158 nM and 69 nM, respectively.THZ531

Research

Studies (3,131)

TimeframeStudies, Drugs with This Role(%)All Drugs %
pre-19902 (0.06)18.7374
1990's169 (5.40)18.2507
2000's1,030 (32.90)29.6817
2010's1,336 (42.67)24.3611
2020's594 (18.97)2.80

Study Types

Publication TypeStudies, Drugs with this Role (%)All Drugs (%)
Trials352 (9.78%)5.53%
Reviews372 (10.34%)6.00%
Case Studies99 (2.75%)4.05%
Observational17 (0.47%)0.25%
Other2,758 (76.65%)84.16%

Protein Targets (745)

Potency Measurements

ProteinTaxonomyMeasurementAverage (mM)Bioassay(s)Drugs
15-lipoxygenase, partialHomo sapiens (human)Potency15.848911
67.9K proteinVaccinia virusPotency8.525928
activating transcription factor 6Homo sapiens (human)Potency3.098512
aldehyde dehydrogenase 1 family, member A1Homo sapiens (human)Potency24.350613
AR proteinHomo sapiens (human)Potency6.485479
arylsulfatase AHomo sapiens (human)Potency5.358211
ATAD5 protein, partialHomo sapiens (human)Potency14.745922
Ataxin-2Homo sapiens (human)Potency19.913822
ATP-dependent phosphofructokinaseTrypanosoma brucei brucei TREU927Potency15.848911
ATPase family AAA domain-containing protein 5Homo sapiens (human)Potency0.016811
atrial natriuretic peptide receptor 1 precursorHomo sapiens (human)Potency37.933011
atrial natriuretic peptide receptor 2 precursorHomo sapiens (human)Potency14.689211
Bloom syndrome protein isoform 1Homo sapiens (human)Potency46.884023
BRCA1Homo sapiens (human)Potency18.629812
caspase 7, apoptosis-related cysteine proteaseHomo sapiens (human)Potency0.237111
caspase-3Cricetulus griseus (Chinese hamster)Potency0.266011
caspase-3Homo sapiens (human)Potency0.237111
Caspase-7Cricetulus griseus (Chinese hamster)Potency0.266011
Cellular tumor antigen p53Homo sapiens (human)Potency1.616023
cellular tumor antigen p53 isoform aHomo sapiens (human)Potency19.783022
Chain A, 2-oxoglutarate OxygenaseHomo sapiens (human)Potency25.118912
Chain A, CruzipainTrypanosoma cruziPotency39.810712
Chain A, Ferritin light chainEquus caballus (horse)Potency25.118911
Chain A, HADH2 proteinHomo sapiens (human)Potency39.810711
Chain A, TYROSYL-DNA PHOSPHODIESTERASEHomo sapiens (human)Potency22.395124
Chain B, HADH2 proteinHomo sapiens (human)Potency39.810711
chromobox protein homolog 1Homo sapiens (human)Potency56.234111
cytochrome P450 2C9 precursorHomo sapiens (human)Potency10.000011
cytochrome P450 2C9, partialHomo sapiens (human)Potency9.081012
cytochrome P450 2D6Homo sapiens (human)Potency25.109713
cytochrome P450 2D6 isoform 1Homo sapiens (human)Potency1.606413
cytochrome P450 3A4 isoform 1Homo sapiens (human)Potency13.893125
cytochrome P450 family 3 subfamily A polypeptide 4Homo sapiens (human)Potency11.461213
cytochrome P450, family 19, subfamily A, polypeptide 1, isoform CRA_aHomo sapiens (human)Potency0.112312
D(1A) dopamine receptorHomo sapiens (human)Potency1.633912
DNA dC->dU-editing enzyme APOBEC-3F isoform aHomo sapiens (human)Potency35.481311
DNA dC->dU-editing enzyme APOBEC-3G isoform 1Homo sapiens (human)Potency23.715011
endonuclease IVEscherichia coliPotency6.309611
estrogen nuclear receptor alphaHomo sapiens (human)Potency2.1775814
estrogen receptor 2 (ER beta)Homo sapiens (human)Potency1.678511
estrogen-related nuclear receptor alphaHomo sapiens (human)Potency6.40341017
euchromatic histone-lysine N-methyltransferase 2Homo sapiens (human)Potency23.667713
EWS/FLI fusion proteinHomo sapiens (human)Potency8.3759419
farnesoid X nuclear receptorHomo sapiens (human)Potency13.145023
flap endonuclease 1Homo sapiens (human)Potency4.228411
Fumarate hydrataseHomo sapiens (human)Potency9.950314
GVesicular stomatitis virusPotency9.081012
GABA theta subunitRattus norvegicus (Norway rat)Potency13.675813
Gamma-aminobutyric acid receptor subunit alpha-1Rattus norvegicus (Norway rat)Potency13.675813
Gamma-aminobutyric acid receptor subunit alpha-2Rattus norvegicus (Norway rat)Potency13.675813
Gamma-aminobutyric acid receptor subunit alpha-3Rattus norvegicus (Norway rat)Potency13.675813
Gamma-aminobutyric acid receptor subunit alpha-4Rattus norvegicus (Norway rat)Potency13.675813
Gamma-aminobutyric acid receptor subunit alpha-5Rattus norvegicus (Norway rat)Potency13.675813
Gamma-aminobutyric acid receptor subunit alpha-6Rattus norvegicus (Norway rat)Potency13.675813
Gamma-aminobutyric acid receptor subunit beta-1Rattus norvegicus (Norway rat)Potency13.675813
Gamma-aminobutyric acid receptor subunit beta-2Rattus norvegicus (Norway rat)Potency13.675813
Gamma-aminobutyric acid receptor subunit beta-3Rattus norvegicus (Norway rat)Potency13.675813
Gamma-aminobutyric acid receptor subunit deltaRattus norvegicus (Norway rat)Potency13.675813
Gamma-aminobutyric acid receptor subunit epsilonRattus norvegicus (Norway rat)Potency13.675813
Gamma-aminobutyric acid receptor subunit gamma-1Rattus norvegicus (Norway rat)Potency13.675813
Gamma-aminobutyric acid receptor subunit gamma-2Rattus norvegicus (Norway rat)Potency13.675813
Gamma-aminobutyric acid receptor subunit gamma-3Rattus norvegicus (Norway rat)Potency13.675813
Gamma-aminobutyric acid receptor subunit piRattus norvegicus (Norway rat)Potency13.675813
gemininHomo sapiens (human)Potency9.016648
GLI family zinc finger 3Homo sapiens (human)Potency0.062622
glp-1 receptor, partialHomo sapiens (human)Potency2.578822
GLS proteinHomo sapiens (human)Potency22.387211
glucocorticoid receptor [Homo sapiens]Homo sapiens (human)Potency7.346123
Glutamate receptor 2Rattus norvegicus (Norway rat)Potency0.380812
Glycoprotein hormones alpha chainHomo sapiens (human)Potency0.794311
heat shock 70kDa protein 5 (glucose-regulated protein, 78kDa)Homo sapiens (human)Potency0.052111
heat shock protein beta-1Homo sapiens (human)Potency26.777622
Histamine H2 receptorCavia porcellus (domestic guinea pig)Potency10.000013
histone acetyltransferase KAT2A isoform 1Homo sapiens (human)Potency35.716812
Histone H2A.xCricetulus griseus (Chinese hamster)Potency11.984522
HLA class I histocompatibility antigen, B alpha chain Homo sapiens (human)Potency9.081012
huntingtin isoform 2Homo sapiens (human)Potency1.929323
hypoxia-inducible factor 1 alpha subunitHomo sapiens (human)Potency16.055623
hypoxia-inducible factor 1, alpha subunit (basic helix-loop-helix transcription factor)Homo sapiens (human)Potency3.162322
Inositol hexakisphosphate kinase 1Homo sapiens (human)Potency9.081014
Inositol monophosphatase 1Rattus norvegicus (Norway rat)Potency2.818411
Integrin alpha-IIbHomo sapiens (human)Potency31.622811
Integrin beta-3Homo sapiens (human)Potency31.622811
Interferon betaHomo sapiens (human)Potency7.4729321
lamin isoform A-delta10Homo sapiens (human)Potency12.238924
lethal factor (plasmid)Bacillus anthracis str. A2012Potency12.589311
LuciferasePhotinus pyralis (common eastern firefly)Potency15.848911
lysosomal alpha-glucosidase preproproteinHomo sapiens (human)Potency14.125411
M-phase phosphoprotein 8Homo sapiens (human)Potency25.118911
Microtubule-associated protein tauHomo sapiens (human)Potency44.668411
muscarinic acetylcholine receptor M1Rattus norvegicus (Norway rat)Potency7.079511
NFKB1 protein, partialHomo sapiens (human)Potency4.152424
NPC intracellular cholesterol transporter 1 precursorHomo sapiens (human)Potency0.517411
Nrf2Homo sapiens (human)Potency18.356411
nuclear factor erythroid 2-related factor 2 isoform 1Homo sapiens (human)Potency10.765124
nuclear factor erythroid 2-related factor 2 isoform 2Homo sapiens (human)Potency1.847323
nuclear factor of kappa light polypeptide gene enhancer in B-cells 1 (p105), isoform CRA_aHomo sapiens (human)Potency21.313811
nuclear receptor ROR-gamma isoform 1Mus musculus (house mouse)Potency30.300112
nuclear receptor subfamily 1, group I, member 3Homo sapiens (human)Potency4.281224
Ornithine decarboxylaseRattus norvegicus (Norway rat)Potency3.162311
parathyroid hormone/parathyroid hormone-related peptide receptor precursorHomo sapiens (human)Potency32.749813
ParkinHomo sapiens (human)Potency4.198822
peptidyl-prolyl cis-trans isomerase NIMA-interacting 1Homo sapiens (human)Potency55.008522
peripheral myelin protein 22Rattus norvegicus (Norway rat)Potency7.114422
peripheral myelin protein 22 isoform 1Homo sapiens (human)Potency19.033812
peroxisome proliferator activated receptor gammaHomo sapiens (human)Potency6.854734
peroxisome proliferator-activated receptor deltaHomo sapiens (human)Potency6.898923
polyproteinZika virusPotency9.950314
potassium voltage-gated channel subfamily H member 2 isoform dHomo sapiens (human)Potency35.481311
PPM1D proteinHomo sapiens (human)Potency7.6977112
pregnane X nuclear receptorHomo sapiens (human)Potency0.105911
progesterone receptorHomo sapiens (human)Potency0.084111
pyruvate kinaseLeishmania mexicana mexicanaPotency6.309622
pyruvate kinase PKM isoform bHomo sapiens (human)Potency3.162322
RAR-related orphan receptor gammaMus musculus (house mouse)Potency2.841224
ras-related protein Rab-9AHomo sapiens (human)Potency0.366311
regulator of G-protein signaling 4Homo sapiens (human)Potency31.745012
retinoic acid nuclear receptor alpha variant 1Homo sapiens (human)Potency0.942135
retinoid X nuclear receptor alphaHomo sapiens (human)Potency0.093722
serine/threonine-protein kinase mTOR isoform 1Homo sapiens (human)Potency16.511133
SMAD family member 2Homo sapiens (human)Potency0.674011
SMAD family member 3Homo sapiens (human)Potency0.674011
Smad3Homo sapiens (human)Potency1.435336
Spike glycoproteinSevere acute respiratory syndrome-related coronavirusPotency16.700612
survival motor neuron protein isoform dHomo sapiens (human)Potency15.498318
TDP1 proteinHomo sapiens (human)Potency22.4858216
thioredoxin reductaseRattus norvegicus (Norway rat)Potency22.451035
ThrombopoietinHomo sapiens (human)Potency0.158522
thyroid hormone receptor beta isoform 2Rattus norvegicus (Norway rat)Potency0.664735
thyroid hormone receptor beta isoform aHomo sapiens (human)Potency59.890123
thyroid stimulating hormone receptorHomo sapiens (human)Potency39.810722
tyrosine-protein kinase YesHomo sapiens (human)Potency25.526414
USP1 protein, partialHomo sapiens (human)Potency79.432811
v-jun sarcoma virus 17 oncogene homolog (avian)Homo sapiens (human)Potency0.061722
vitamin D (1,25- dihydroxyvitamin D3) receptorHomo sapiens (human)Potency10.473634
vitamin D3 receptor isoform VDRAHomo sapiens (human)Potency28.183811
Voltage-dependent calcium channel gamma-2 subunitMus musculus (house mouse)Potency0.380812

Inhibition Measurements

ProteinTaxonomyMeasurementAverage (mM)Bioassay(s)Drugs
[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1, mitochondrialHomo sapiens (human)IC5010.000011
[Tau protein] kinase Sus scrofa (pig)IC5019.6200910
10 kDa chaperonin Escherichia coliIC503.600022
10 kDa heat shock protein, mitochondrialHomo sapiens (human)IC502.300011
5-hydroxytryptamine receptor 1ARattus norvegicus (Norway rat)IC5040.000011
5-hydroxytryptamine receptor 1BRattus norvegicus (Norway rat)IC5040.000011
5-hydroxytryptamine receptor 1DRattus norvegicus (Norway rat)IC5040.000011
5-hydroxytryptamine receptor 1FRattus norvegicus (Norway rat)IC5040.000011
5-hydroxytryptamine receptor 2ARattus norvegicus (Norway rat)IC50516.500014
60 kDa chaperoninEscherichia coli K-12IC50250.000011
60 kDa chaperonin Escherichia coliIC503.600022
60 kDa heat shock protein, mitochondrialHomo sapiens (human)IC502.300011
AcetylcholinesteraseMus musculus (house mouse)IC500.021011
Alpha-1A adrenergic receptorRattus norvegicus (Norway rat)IC500.437012
Alpha-1B adrenergic receptorRattus norvegicus (Norway rat)IC500.437012
Alpha-1D adrenergic receptorRattus norvegicus (Norway rat)IC500.437012
Aspartate aminotransferase, cytoplasmicHomo sapiens (human)IC5021.790011
ATP-binding cassette sub-family C member 3Homo sapiens (human)IC50133.000011
Aurora kinase AHomo sapiens (human)IC5010.000022
Bile salt export pumpHomo sapiens (human)IC50133.000011
cAMP-dependent protein kinase catalytic subunit alphaBos taurus (cattle)IC50357.935016
cAMP-dependent protein kinase catalytic subunit alphaHomo sapiens (human)IC501,002.000045
cAMP-dependent protein kinase catalytic subunit betaHomo sapiens (human)IC501,002.000045
cAMP-dependent protein kinase catalytic subunit gammaHomo sapiens (human)IC501,002.000045
Canalicular multispecific organic anion transporter 1Homo sapiens (human)IC50133.000011
Cannabinoid receptor 1Homo sapiens (human)IC500.314011
Cannabinoid receptor 2Mus musculus (house mouse)IC500.062011
Casein kinase I isoform alphaHomo sapiens (human)IC5017.503544
Casein kinase I isoform alphaRattus norvegicus (Norway rat)IC50190.1300212
Casein kinase I isoform alphaSus scrofa (pig)IC5010.000012
Casein kinase I isoform deltaHomo sapiens (human)IC5013.500022
Casein kinase I isoform epsilonHomo sapiens (human)IC5017.000011
Casein kinase I isoform gamma-1Homo sapiens (human)IC5017.000011
Casein kinase I isoform gamma-2Homo sapiens (human)IC5017.000011
Casein kinase II subunit alphaHomo sapiens (human)IC506.943333
Casein kinase II subunit alpha 3Homo sapiens (human)IC500.510011
Casein kinase II subunit alpha'Homo sapiens (human)IC500.415022
Casein kinase II subunit betaHomo sapiens (human)IC500.415022
CDK-activating kinase assembly factor MAT1Homo sapiens (human)IC503.2404911
CDK-activating kinase assembly factor MAT1Homo sapiens (human)Ki2.800011
cGMP-dependent protein kinase 1 Bos taurus (cattle)IC50357.935016
Chain A, Cyclin-dependent kinase 9Homo sapiens (human)IC500.740011
Chain A, Extracellular Regulated Kinase 2Rattus norvegicus (Norway rat)IC5027.000012
Chain A, Glycogen Synthase Kinase-3 BetaHomo sapiens (human)IC500.004012
Chain A, Homo sapiens cyclin-dependent kinase 2Homo sapiens (human)IC500.400011
Chain A, MAP KINASE P38Homo sapiens (human)IC5027.000011
Chain A, Protein (glycogen Phosphorylase)Oryctolagus cuniculus (rabbit)IC501.000011
Chain A, PROTEIN (MAP KINASE P38)Homo sapiens (human)IC5027.000013
Chain B, Cell division protein kinase 6Homo sapiens (human)IC500.015012
Chain B, Glycogen Synthase Kinase-3 BetaHomo sapiens (human)IC500.004011
Chain C, Cell division protein kinase 2Homo sapiens (human)IC500.210012
Cyclin homologHerpesvirus saimiri (strain 11)IC500.185014
Cyclin-A1Homo sapiens (human)IC506.65431923
Cyclin-A1Homo sapiens (human)Ki23.146713
Cyclin-A2Homo sapiens (human)IC505.66345576
Cyclin-A2Homo sapiens (human)Ki14.896835
Cyclin-CHomo sapiens (human)IC500.053022
Cyclin-CHomo sapiens (human)Ki0.009011
Cyclin-dependent kinase 1Homo sapiens (human)IC5030.751687154
Cyclin-dependent kinase 1Oryzias latipes (Japanese medaka)IC505.61531035
Cyclin-dependent kinase 1Homo sapiens (human)Ki1.156045
Cyclin-dependent kinase 12Homo sapiens (human)IC502.133755
Cyclin-dependent kinase 13Homo sapiens (human)IC500.265033
Cyclin-dependent kinase 14Homo sapiens (human)IC500.019811
Cyclin-dependent kinase 19Homo sapiens (human)IC500.005522
Cyclin-dependent kinase 2Homo sapiens (human)IC5011.0673133206
Cyclin-dependent kinase 2Homo sapiens (human)Ki8.8562710
Cyclin-dependent kinase 3Homo sapiens (human)IC500.360033
Cyclin-dependent kinase 4Homo sapiens (human)IC5038.020165107
Cyclin-dependent kinase 4Homo sapiens (human)Ki0.258844
Cyclin-dependent kinase 5 activator 1Homo sapiens (human)IC5029.88064481
Cyclin-dependent kinase 5 activator 1Homo sapiens (human)Ki0.018011
Cyclin-dependent kinase 6Homo sapiens (human)IC508.43383138
Cyclin-dependent kinase 6Homo sapiens (human)Ki0.027011
Cyclin-dependent kinase 7Homo sapiens (human)IC506.44754162
Cyclin-dependent kinase 7Homo sapiens (human)Ki3.900022
Cyclin-dependent kinase 8Homo sapiens (human)IC500.037744
Cyclin-dependent kinase 8Homo sapiens (human)Ki0.009011
Cyclin-dependent kinase 9Homo sapiens (human)IC505.09595986
Cyclin-dependent kinase 9Homo sapiens (human)Ki0.230647
Cyclin-dependent-like kinase 5Bos taurus (cattle)IC500.200011
Cyclin-dependent-like kinase 5 Homo sapiens (human)IC5024.013256102
Cyclin-dependent-like kinase 5 Homo sapiens (human)Ki0.018011
Cyclin-HHomo sapiens (human)IC506.56553143
Cyclin-HHomo sapiens (human)Ki3.900022
Cyclin-KHomo sapiens (human)IC500.521388
Cyclin-T1Homo sapiens (human)IC505.35974561
Cyclin-T1Homo sapiens (human)Ki0.321435
Cyclin-YHomo sapiens (human)IC500.019811
Cytochrome P450 1A2Homo sapiens (human)Ki5.000011
Cytochrome P450 2C19Homo sapiens (human)Ki5.000011
Cytochrome P450 2D6Homo sapiens (human)Ki5.000011
Cytochrome P450 3A4Homo sapiens (human)IC500.071011
D(2) dopamine receptorRattus norvegicus (Norway rat)IC5010.000012
Dual specificity mitogen-activated protein kinase kinase 1Homo sapiens (human)IC5010.000011
Dual specificity protein kinase CLK1Homo sapiens (human)IC506.690323
Dual specificity protein kinase CLK1Mus musculus (house mouse)IC500.992077
Dual specificity protein kinase CLK2Mus musculus (house mouse)IC500.470044
Dual specificity protein kinase CLK3Mus musculus (house mouse)IC506.840055
Dual specificity protein kinase CLK4Mus musculus (house mouse)IC500.184544
Dual specificity tyrosine-phosphorylation-regulated kinase 1AHomo sapiens (human)IC509.30961318
Dual specificity tyrosine-phosphorylation-regulated kinase 1AMus musculus (house mouse)IC505.000011
Dual specificity tyrosine-phosphorylation-regulated kinase 1ARattus norvegicus (Norway rat)IC504.484367
Dual specificity tyrosine-phosphorylation-regulated kinase 1BHomo sapiens (human)IC500.284055
Dual specificity tyrosine-phosphorylation-regulated kinase 2Homo sapiens (human)IC500.408455
Dual specificity tyrosine-phosphorylation-regulated kinase 3Homo sapiens (human)IC502.812544
Dual specificity tyrosine-phosphorylation-regulated kinase 4Homo sapiens (human)IC500.520011
Epidermal growth factor receptorHomo sapiens (human)IC50103.120045
Fibroblast growth factor receptor 1Homo sapiens (human)IC5010.000011
Focal adhesion kinase 1Homo sapiens (human)IC5040.000011
G1/S-specific cyclin-D1Homo sapiens (human)IC5047.11425073
G1/S-specific cyclin-D1Homo sapiens (human)Ki0.035022
G1/S-specific cyclin-D2Homo sapiens (human)IC500.168077
G1/S-specific cyclin-D3Homo sapiens (human)IC5014.57151818
G1/S-specific cyclin-D3Homo sapiens (human)Ki0.027011
G1/S-specific cyclin-E1Homo sapiens (human)IC5021.05775588
G1/S-specific cyclin-E1Homo sapiens (human)Ki6.905022
G1/S-specific cyclin-E2Homo sapiens (human)IC5022.24191520
G1/S-specific cyclin-E2Homo sapiens (human)Ki13.300011
G2/mitotic-specific cyclin-BMarthasterias glacialis (spiny starfish)IC505.61531035
G2/mitotic-specific cyclin-B1Homo sapiens (human)IC5034.551566112
G2/mitotic-specific cyclin-B1Homo sapiens (human)Ki2.595022
G2/mitotic-specific cyclin-B2Homo sapiens (human)IC508.54611930
G2/mitotic-specific cyclin-B3Homo sapiens (human)IC508.54611930
Glycogen phosphorylase, muscle formOryctolagus cuniculus (rabbit)IC501.200011
Glycogen synthase kinase 3 Plasmodium falciparum 3D7IC5010.000012
Glycogen synthase kinase-3 alphaHomo sapiens (human)IC5019.1758910
Glycogen synthase kinase-3 alphaHomo sapiens (human)Ki0.231011
Glycogen synthase kinase-3 betaHomo sapiens (human)IC509.03632836
Glycogen synthase kinase-3 betaRattus norvegicus (Norway rat)IC5098.5770422
Glycogen synthase kinase-3 betaHomo sapiens (human)Ki0.345011
Glycogen synthase kinase-3 beta Sus scrofa (pig)IC5019.6200910
Insulin receptorHomo sapiens (human)IC5055.000022
Insulin-like growth factor 1 receptorHomo sapiens (human)IC5025.000011
Kappa-type opioid receptorCavia porcellus (domestic guinea pig)IC505.035522
La-related protein 7Homo sapiens (human)Ki0.003011
Macrophage colony-stimulating factor 1 receptorHomo sapiens (human)IC5010.000011
Mitogen-activated protein kinase 1Homo sapiens (human)IC5023.1625512
Mitogen-activated protein kinase 1Rattus norvegicus (Norway rat)IC5052.333323
Mitogen-activated protein kinase 14Homo sapiens (human)IC5063.500012
Mitogen-activated protein kinase 3 Homo sapiens (human)IC5026.500046
Mitogen-activated protein kinase 8Homo sapiens (human)IC50170.000011
MO15-related protein kinase Pfmrk Plasmodium falciparum (malaria parasite P. falciparum)IC50461.714327
Multidrug resistance-associated protein 4Homo sapiens (human)IC50133.000011
NAD-dependent protein deacetylase sirtuin-1Homo sapiens (human)IC5029.000022
NAD-dependent protein deacetylase sirtuin-2Homo sapiens (human)IC5048.900034
NUAK family SNF1-like kinase 1Homo sapiens (human)IC505.000011
nuclear receptor subfamily 0 group B member 1Homo sapiens (human)IC500.833511
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoformHomo sapiens (human)IC5010.000011
Platelet-derived growth factor receptor betaHomo sapiens (human)IC5010.000011
Poly [ADP-ribose] polymerase tankyrase-1Homo sapiens (human)IC5010.000011
Poly [ADP-ribose] polymerase tankyrase-2Homo sapiens (human)IC5015.000011
Protein kinase C alpha typeHomo sapiens (human)IC5012.466766
Protein kinase C alpha typeRattus norvegicus (Norway rat)IC50507.000012
Protein kinase C beta typeHomo sapiens (human)IC5023.200055
Protein kinase C beta typeRattus norvegicus (Norway rat)IC50507.000012
Protein kinase C delta typeHomo sapiens (human)IC507.972544
Protein kinase C delta typeRattus norvegicus (Norway rat)IC50507.000012
Protein kinase C epsilon typeHomo sapiens (human)IC507.870044
Protein kinase C epsilon typeRattus norvegicus (Norway rat)IC50507.000012
Protein kinase C eta typeHomo sapiens (human)IC5019.000044
Protein kinase C eta typeRattus norvegicus (Norway rat)IC50507.000012
Protein kinase C gamma typeHomo sapiens (human)IC5017.750044
Protein kinase C gamma typeRattus norvegicus (Norway rat)IC50507.000012
Protein kinase C iota typeHomo sapiens (human)IC5010.333333
Protein kinase C theta typeHomo sapiens (human)IC5010.333333
Protein kinase C theta typeRattus norvegicus (Norway rat)IC50507.000012
Protein kinase C theta typeHomo sapiens (human)Ki0.061011
Protein kinase C zeta typeHomo sapiens (human)IC5010.333333
Protein kinase C zeta typeRattus norvegicus (Norway rat)IC50507.000012
Protein Wnt-3aHomo sapiens (human)IC500.007011
Proto-oncogene tyrosine-protein kinase SrcHomo sapiens (human)IC5024.500022
Receptor tyrosine-protein kinase erbB-2Homo sapiens (human)IC5020.400022
Receptor-type tyrosine-protein kinase FLT3Homo sapiens (human)IC505.493333
Replicase polyprotein 1abSevere acute respiratory syndrome coronavirus 2IC501.500012
Retinoic acid receptor alphaHomo sapiens (human)Ki1.100011
Retinoic acid receptor betaHomo sapiens (human)Ki0.034011
Retinoic acid receptor gamma Homo sapiens (human)Ki0.130011
Ribosomal protein S6 kinase beta-1Homo sapiens (human)IC5010.000011
Ribosomal protein S6 kinase beta-2Homo sapiens (human)IC5010.000011
Serine/threonine-protein kinase Chk1Homo sapiens (human)IC5040.000011
Serine/threonine-protein kinase D1Homo sapiens (human)IC5010.333333
Serine/threonine-protein kinase D3Homo sapiens (human)IC5010.333333
Serine/threonine-protein kinase PAK 4Homo sapiens (human)IC506.900011
Serine/threonine-protein kinase pim-1Homo sapiens (human)IC502.060033
Serine/threonine-protein kinase PLK1Homo sapiens (human)IC50100.000011
Squalene synthaseRattus norvegicus (Norway rat)IC500.170011
steroidogenic factor 1Homo sapiens (human)IC5067.518011
Synapsin-1Bos taurus (cattle)IC501.000011
Thiosulfate sulfurtransferaseHomo sapiens (human)IC50100.000011
Tyrosine-protein kinase ABL1Homo sapiens (human)IC5046.000055
Tyrosine-protein kinase FynHomo sapiens (human)IC5010.000011
Tyrosine-protein kinase ITK/TSKHomo sapiens (human)IC5027.425022
Tyrosine-protein kinase JAK3Homo sapiens (human)IC500.063111
Tyrosine-protein kinase LckHomo sapiens (human)IC5011.774045
Tyrosine-protein kinase ZAP-70Homo sapiens (human)IC5045.000022
Vascular endothelial growth factor receptor 2Homo sapiens (human)IC5035.800023
Vitamin K-dependent protein CHomo sapiens (human)IC500.6659432
Voltage-dependent L-type calcium channel subunit alpha-1CHomo sapiens (human)IC5023.400011

Activation Measurements

ProteinTaxonomyMeasurementAverage (mM)Bioassay(s)Drugs
26S proteasome regulatory subunit 6BHomo sapiens (human)Kd30.000015
3-phosphoinositide-dependent protein kinase 1Homo sapiens (human)Kd10.000026
5'-AMP-activated protein kinase catalytic subunit alpha-1Homo sapiens (human)Kd17.9000412
5'-AMP-activated protein kinase catalytic subunit alpha-2Homo sapiens (human)Kd10.000026
5'-AMP-activated protein kinase subunit gamma-1Homo sapiens (human)Kd30.000016
5'-AMP-activated protein kinase subunit gamma-2Homo sapiens (human)Kd30.000015
AarF domain-containing protein kinase 1Homo sapiens (human)Kd30.000015
Actin-related protein 2Homo sapiens (human)Kd30.000015
Actin-related protein 3Homo sapiens (human)Kd30.000015
Activated CDC42 kinase 1Homo sapiens (human)Kd20.7692313
Activin receptor type-1Homo sapiens (human)Kd18.6500312
Activin receptor type-1BHomo sapiens (human)Kd20.0000312
Activin receptor type-2AHomo sapiens (human)Kd8.850026
Activin receptor type-2BHomo sapiens (human)Kd17.7091311
Acyl-CoA dehydrogenase family member 10Homo sapiens (human)Kd30.000015
Acyl-CoA dehydrogenase family member 11Homo sapiens (human)Kd30.000015
Adenine phosphoribosyltransferaseHomo sapiens (human)Kd30.000013
Adenosine kinaseHomo sapiens (human)Kd24.488215
Adenylate kinase 2, mitochondrialHomo sapiens (human)Kd30.000015
ADP/ATP translocase 2Homo sapiens (human)Kd30.000015
ADP/ATP translocase 3Homo sapiens (human)Kd30.000015
ALK tyrosine kinase receptorHomo sapiens (human)Kd5.606726
Angiopoietin-1 receptorHomo sapiens (human)Kd10.000026
Ankyrin repeat and protein kinase domain-containing protein 1Homo sapiens (human)Kd10.000026
AP2-associated protein kinase 1Homo sapiens (human)Kd15.8924311
ATP-dependent 6-phosphofructokinase, platelet typeHomo sapiens (human)Kd30.000015
ATP-dependent RNA helicase DDX1Homo sapiens (human)Kd30.000015
ATP-dependent RNA helicase DDX3XHomo sapiens (human)Kd30.000015
ATP-dependent RNA helicase DDX42Homo sapiens (human)Kd30.000013
ATP-dependent RNA helicase DHX30Homo sapiens (human)Kd30.000013
Atypical kinase COQ8A, mitochondrialHomo sapiens (human)Kd19.0909311
Atypical kinase COQ8B, mitochondrialHomo sapiens (human)Kd8.816726
Aurora kinase AHomo sapiens (human)Kd18.6182311
Aurora kinase BHomo sapiens (human)Kd20.0000312
Aurora kinase CHomo sapiens (human)Kd9.166726
BDNF/NT-3 growth factors receptorHomo sapiens (human)Kd10.000026
Beta-adrenergic receptor kinase 1Homo sapiens (human)Kd30.000015
BMP-2-inducible protein kinaseHomo sapiens (human)Kd18.7696311
Bone morphogenetic protein receptor type-1AHomo sapiens (human)Kd19.0909311
Bone morphogenetic protein receptor type-1BHomo sapiens (human)Kd20.064327
Bone morphogenetic protein receptor type-2Homo sapiens (human)Kd19.0909311
Breakpoint cluster region proteinHomo sapiens (human)Kd30.000015
Calcium-dependent protein kinase 1Plasmodium falciparum 3D7Kd10.000013
Calcium/calmodulin-dependent protein kinase kinase 1Homo sapiens (human)Kd5.739637
Calcium/calmodulin-dependent protein kinase kinase 2Homo sapiens (human)Kd12.9132412
Calcium/calmodulin-dependent protein kinase type 1Homo sapiens (human)Kd10.000026
Calcium/calmodulin-dependent protein kinase type 1DHomo sapiens (human)Kd10.000026
Calcium/calmodulin-dependent protein kinase type 1GHomo sapiens (human)Kd10.000026
Calcium/calmodulin-dependent protein kinase type II subunit alphaHomo sapiens (human)Kd6.385737
Calcium/calmodulin-dependent protein kinase type II subunit betaHomo sapiens (human)Kd8.185737
Calcium/calmodulin-dependent protein kinase type II subunit deltaHomo sapiens (human)Kd19.3000312
Calcium/calmodulin-dependent protein kinase type II subunit gammaHomo sapiens (human)Kd18.4182311
Calcium/calmodulin-dependent protein kinase type IVHomo sapiens (human)Kd15.6236311
cAMP-dependent protein kinase catalytic subunit alphaHomo sapiens (human)Kd19.0909311
cAMP-dependent protein kinase catalytic subunit betaHomo sapiens (human)Kd19.0909311
cAMP-dependent protein kinase catalytic subunit gammaHomo sapiens (human)Kd30.000016
cAMP-dependent protein kinase catalytic subunit PRKXHomo sapiens (human)Kd10.000026
cAMP-dependent protein kinase type II-alpha regulatory subunitHomo sapiens (human)Kd30.000015
Casein kinase I isoform alphaHomo sapiens (human)Kd20.512528
Casein kinase I isoform alpha-likeHomo sapiens (human)Kd8.733326
Casein kinase I isoform deltaHomo sapiens (human)Kd14.3345311
Casein kinase I isoform epsilonHomo sapiens (human)Kd13.7324412
Casein kinase I isoform gamma-1Homo sapiens (human)Kd17.0417412
Casein kinase I isoform gamma-2Homo sapiens (human)Kd18.5692413
Casein kinase I isoform gamma-3Homo sapiens (human)Kd19.4083312
Casein kinase II subunit alphaHomo sapiens (human)Kd10.000026
Casein kinase II subunit alpha'Homo sapiens (human)Kd14.2791311
Cell division control protein 2 homologPlasmodium falciparum 3D7Kd7.766713
Cell division cycle 7-related protein kinaseHomo sapiens (human)Kd30.000011
cGMP-dependent protein kinase 1 Homo sapiens (human)Kd19.0909311
cGMP-dependent protein kinase 2Homo sapiens (human)Kd10.000026
Choline-phosphate cytidylyltransferase AHomo sapiens (human)Kd30.000013
Chromodomain-helicase-DNA-binding protein 4Homo sapiens (human)Kd30.000014
Citron Rho-interacting kinaseHomo sapiens (human)Kd14.0780311
Cyclin-A1Homo sapiens (human)EC500.151011
Cyclin-A2Homo sapiens (human)EC500.151011
Cyclin-dependent kinase 1Homo sapiens (human)Kd12.830015
Cyclin-dependent kinase 10Homo sapiens (human)Kd30.000015
Cyclin-dependent kinase 11AHomo sapiens (human)Kd5.016926
Cyclin-dependent kinase 11BHomo sapiens (human)Kd5.034126
Cyclin-dependent kinase 12Homo sapiens (human)Kd12.114815
Cyclin-dependent kinase 13Homo sapiens (human)Kd7.853728
Cyclin-dependent kinase 14Homo sapiens (human)Kd1.936026
Cyclin-dependent kinase 15Homo sapiens (human)Kd0.377313
Cyclin-dependent kinase 16Homo sapiens (human)Kd3.5428413
Cyclin-dependent kinase 17Homo sapiens (human)Kd3.8431311
Cyclin-dependent kinase 18Homo sapiens (human)Kd6.043137
Cyclin-dependent kinase 19Mus musculus (house mouse)EC500.020011
Cyclin-dependent kinase 19Homo sapiens (human)Kd2.552326
Cyclin-dependent kinase 2Homo sapiens (human)EC500.151011
Cyclin-dependent kinase 2Homo sapiens (human)Kd5.3445413
Cyclin-dependent kinase 3Homo sapiens (human)Kd14.6356311
Cyclin-dependent kinase 4Homo sapiens (human)Kd5.8951311
Cyclin-dependent kinase 6Homo sapiens (human)Kd6.956415
Cyclin-dependent kinase 7Homo sapiens (human)Kd3.7594311
Cyclin-dependent kinase 8Mus musculus (house mouse)EC500.020011
Cyclin-dependent kinase 8Homo sapiens (human)Kd3.773326
Cyclin-dependent kinase 9Homo sapiens (human)Kd2.2337311
Cyclin-dependent kinase-like 1Homo sapiens (human)Kd10.000013
Cyclin-dependent kinase-like 2Homo sapiens (human)Kd3.680313
Cyclin-dependent kinase-like 3Homo sapiens (human)Kd7.133313
Cyclin-dependent kinase-like 5Homo sapiens (human)Kd15.001926
Cyclin-dependent-like kinase 5 Homo sapiens (human)Kd5.5304413
Cyclin-G-associated kinaseHomo sapiens (human)Kd14.6200412
Cysteine--tRNA ligase, cytoplasmicHomo sapiens (human)Kd30.000012
Cytochrome c1, heme protein, mitochondrialHomo sapiens (human)Kd30.000014
Cytoplasmic tyrosine-protein kinase BMXHomo sapiens (human)Kd10.000026
dCTP pyrophosphatase 1Homo sapiens (human)Kd30.000017
Death-associated protein kinase 1Homo sapiens (human)Kd10.000026
Death-associated protein kinase 2Homo sapiens (human)Kd10.000026
Death-associated protein kinase 3Homo sapiens (human)Kd10.000039
Delta(24)-sterol reductaseHomo sapiens (human)Kd30.000015
Deoxycytidine kinaseHomo sapiens (human)Kd30.000016
Discoidin domain-containing receptor 2Homo sapiens (human)Kd19.0909311
DNA replication licensing factor MCM4Homo sapiens (human)Kd30.000015
DNA topoisomerase 2-alphaHomo sapiens (human)Kd30.000015
DNA topoisomerase 2-betaHomo sapiens (human)Kd30.000015
DnaJ homolog subfamily A member 1Homo sapiens (human)Kd30.000015
Dual serine/threonine and tyrosine protein kinaseHomo sapiens (human)Kd8.066713
Dual specificity mitogen-activated protein kinase kinase 1Homo sapiens (human)Kd20.0000312
Dual specificity mitogen-activated protein kinase kinase 2Homo sapiens (human)Kd19.0909311
Dual specificity mitogen-activated protein kinase kinase 3Homo sapiens (human)Kd18.2909311
Dual specificity mitogen-activated protein kinase kinase 4Homo sapiens (human)Kd12.616839
Dual specificity mitogen-activated protein kinase kinase 5Homo sapiens (human)Kd21.272528
Dual specificity mitogen-activated protein kinase kinase 6Homo sapiens (human)Kd19.0909311
Dual specificity mitogen-activated protein kinase kinase 7Homo sapiens (human)Kd10.000013
Dual specificity protein kinase CLK1Homo sapiens (human)Kd5.5263514
Dual specificity protein kinase CLK2Homo sapiens (human)Kd11.5164514
Dual specificity protein kinase CLK3Homo sapiens (human)Kd8.6984511
Dual specificity protein kinase CLK4Homo sapiens (human)Kd13.5975512
Dual specificity protein kinase TTKHomo sapiens (human)Kd15.7909411
Dual specificity testis-specific protein kinase 1Homo sapiens (human)Kd19.0909311
Dual specificity testis-specific protein kinase 2Homo sapiens (human)Kd30.000013
Dual specificity tyrosine-phosphorylation-regulated kinase 1AHomo sapiens (human)Kd8.476339
Dual specificity tyrosine-phosphorylation-regulated kinase 1BHomo sapiens (human)Kd4.012248
Dual specificity tyrosine-phosphorylation-regulated kinase 2Homo sapiens (human)Kd4.387524
Dynamin-like 120 kDa protein, mitochondrialHomo sapiens (human)Kd30.000015
eIF-2-alpha kinase GCN2Homo sapiens (human)Kd10.000026
EKC/KEOPS complex subunit TP53RKHomo sapiens (human)Kd30.000015
Electron transfer flavoprotein subunit betaHomo sapiens (human)Kd30.000015
Elongation factor Tu, mitochondrialHomo sapiens (human)Kd30.000015
Ephrin type-A receptor 1Homo sapiens (human)Kd14.037538
Ephrin type-A receptor 2Homo sapiens (human)Kd17.7273311
Ephrin type-A receptor 3Homo sapiens (human)Kd7.766726
Ephrin type-A receptor 4Homo sapiens (human)Kd19.0909311
Ephrin type-A receptor 5Homo sapiens (human)Kd17.2917412
Ephrin type-A receptor 6Homo sapiens (human)Kd10.000026
Ephrin type-A receptor 7Homo sapiens (human)Kd19.0909311
Ephrin type-A receptor 8Homo sapiens (human)Kd10.000026
Ephrin type-B receptor 1Homo sapiens (human)Kd7.671437
Ephrin type-B receptor 2Homo sapiens (human)Kd19.0909311
Ephrin type-B receptor 3Homo sapiens (human)Kd20.0000312
Ephrin type-B receptor 4Homo sapiens (human)Kd19.0909311
Ephrin type-B receptor 6Homo sapiens (human)Kd21.428627
Epidermal growth factor receptorHomo sapiens (human)Kd9.82072371
Epithelial discoidin domain-containing receptor 1Homo sapiens (human)Kd19.0909311
Eukaryotic translation initiation factor 2-alpha kinase 1Homo sapiens (human)Kd17.616028
Eukaryotic translation initiation factor 5BHomo sapiens (human)Kd30.000011
Exosome RNA helicase MTR4Homo sapiens (human)Kd30.000015
Ferrochelatase, mitochondrialHomo sapiens (human)Kd30.000015
Fibroblast growth factor receptor 1Homo sapiens (human)Kd19.0909311
Fibroblast growth factor receptor 2Homo sapiens (human)Kd10.000026
Fibroblast growth factor receptor 3Homo sapiens (human)Kd10.0000412
Fibroblast growth factor receptor 4Homo sapiens (human)Kd10.000026
Focal adhesion kinase 1Homo sapiens (human)Kd19.0909311
G protein-coupled receptor kinase 4Homo sapiens (human)Kd10.000013
G protein-coupled receptor kinase 6Homo sapiens (human)Kd30.000012
General transcription and DNA repair factor IIH helicase subunit XPDHomo sapiens (human)Kd14.810215
Glycine receptor subunit alpha-1Homo sapiens (human)EC501.300011
Glycine--tRNA ligaseHomo sapiens (human)Kd30.000016
Glycogen phosphorylase, brain formHomo sapiens (human)Kd24.713815
Glycogen phosphorylase, liver formHomo sapiens (human)Kd25.353516
Glycogen synthase kinase-3 alphaHomo sapiens (human)Kd6.2022412
Glycogen synthase kinase-3 betaHomo sapiens (human)Kd6.6038311
GTP-binding nuclear protein RanHomo sapiens (human)Kd30.000015
Guanine nucleotide-binding protein G(i) subunit alpha-2Homo sapiens (human)Kd30.000014
Heme oxygenase 2Homo sapiens (human)Kd30.000015
Hepatocyte growth factor receptorHomo sapiens (human)Kd14.2155517
High affinity nerve growth factor receptorHomo sapiens (human)Kd16.666739
Homeodomain-interacting protein kinase 1Homo sapiens (human)Kd4.705024
Homeodomain-interacting protein kinase 2Homo sapiens (human)Kd5.233313
Homeodomain-interacting protein kinase 3Homo sapiens (human)Kd4.132524
Homeodomain-interacting protein kinase 4Homo sapiens (human)Kd7.333313
Hormonally up-regulated neu tumor-associated kinaseHomo sapiens (human)Kd10.000013
Inhibitor of nuclear factor kappa-B kinase subunit alphaHomo sapiens (human)Kd10.000013
Inhibitor of nuclear factor kappa-B kinase subunit betaHomo sapiens (human)Kd10.000013
Inhibitor of nuclear factor kappa-B kinase subunit epsilonHomo sapiens (human)Kd17.8364311
Inosine-5'-monophosphate dehydrogenase 2Homo sapiens (human)Kd30.000014
Insulin receptorHomo sapiens (human)Kd19.0909311
Insulin receptor-related proteinHomo sapiens (human)Kd10.000026
Insulin-like growth factor 1 receptorHomo sapiens (human)Kd19.0909311
Integrin-linked protein kinaseHomo sapiens (human)Kd30.000014
Interferon-induced, double-stranded RNA-activated protein kinaseHomo sapiens (human)Kd8.400026
Interleukin-1 receptor-associated kinase 1Homo sapiens (human)Kd19.052239
Interleukin-1 receptor-associated kinase 3Homo sapiens (human)Kd17.8000311
Interleukin-1 receptor-associated kinase 4Homo sapiens (human)Kd21.437528
Isoleucine--tRNA ligase, mitochondrialHomo sapiens (human)Kd30.000013
Leucine-rich repeat serine/threonine-protein kinase 2Homo sapiens (human)Kd7.166726
Leukocyte tyrosine kinase receptorHomo sapiens (human)Kd7.400026
Leukotriene C4 synthaseCavia porcellus (domestic guinea pig)Kd7.066713
LIM domain kinase 1Homo sapiens (human)Kd19.0909311
LIM domain kinase 2Homo sapiens (human)Kd20.0000312
Long-chain-fatty-acid--CoA ligase 5Homo sapiens (human)Kd30.000013
Macrophage colony-stimulating factor 1 receptorHomo sapiens (human)Kd7.600026
Macrophage-stimulating protein receptorHomo sapiens (human)Kd22.500028
MAP kinase-activated protein kinase 2Homo sapiens (human)Kd19.0909311
MAP kinase-activated protein kinase 5Homo sapiens (human)Kd19.0909311
MAP kinase-interacting serine/threonine-protein kinase 1Homo sapiens (human)Kd7.933326
MAP kinase-interacting serine/threonine-protein kinase 2Homo sapiens (human)Kd6.085737
MAP/microtubule affinity-regulating kinase 3Homo sapiens (human)Kd19.0909311
MAP/microtubule affinity-regulating kinase 4Homo sapiens (human)Kd19.0909311
Mast/stem cell growth factor receptor KitHomo sapiens (human)Kd9.59111545
Maternal embryonic leucine zipper kinaseHomo sapiens (human)Kd18.2909311
Megakaryocyte-associated tyrosine-protein kinaseHomo sapiens (human)Kd10.000013
Membrane-associated progesterone receptor component 1Homo sapiens (human)Kd30.000013
Membrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinaseHomo sapiens (human)Kd20.0000312
Microtubule-associated serine/threonine-protein kinase 1Homo sapiens (human)Kd8.733313
MidasinHomo sapiens (human)Kd30.000015
Misshapen-like kinase 1Homo sapiens (human)Kd12.825024
Mitogen-activated protein kinase 1Homo sapiens (human)Kd19.0909311
Mitogen-activated protein kinase 10Homo sapiens (human)Kd17.9000311
Mitogen-activated protein kinase 11Homo sapiens (human)Kd19.0909311
Mitogen-activated protein kinase 12Homo sapiens (human)Kd10.000026
Mitogen-activated protein kinase 13Homo sapiens (human)Kd10.000013
Mitogen-activated protein kinase 14Homo sapiens (human)Kd19.0909311
Mitogen-activated protein kinase 15Homo sapiens (human)Kd14.6382311
Mitogen-activated protein kinase 3 Homo sapiens (human)Kd19.0909311
Mitogen-activated protein kinase 4Homo sapiens (human)Kd8.033326
Mitogen-activated protein kinase 6Homo sapiens (human)Kd6.833326
Mitogen-activated protein kinase 7Homo sapiens (human)Kd9.7498311
Mitogen-activated protein kinase 8Homo sapiens (human)Kd18.3273311
Mitogen-activated protein kinase 9Homo sapiens (human)Kd16.6233311
Mitogen-activated protein kinase kinase kinase 1Homo sapiens (human)Kd22.500028
Mitogen-activated protein kinase kinase kinase 10Homo sapiens (human)Kd8.400026
Mitogen-activated protein kinase kinase kinase 11Homo sapiens (human)Kd19.0909311
Mitogen-activated protein kinase kinase kinase 12Homo sapiens (human)Kd10.000013
Mitogen-activated protein kinase kinase kinase 13Homo sapiens (human)Kd10.000013
Mitogen-activated protein kinase kinase kinase 15Homo sapiens (human)Kd10.000013
Mitogen-activated protein kinase kinase kinase 19Homo sapiens (human)Kd10.000013
Mitogen-activated protein kinase kinase kinase 2Homo sapiens (human)Kd22.012528
Mitogen-activated protein kinase kinase kinase 20Homo sapiens (human)Kd19.0909311
Mitogen-activated protein kinase kinase kinase 3Homo sapiens (human)Kd22.487528
Mitogen-activated protein kinase kinase kinase 4Homo sapiens (human)Kd20.0000312
Mitogen-activated protein kinase kinase kinase 5Homo sapiens (human)Kd19.0909311
Mitogen-activated protein kinase kinase kinase 6Homo sapiens (human)Kd22.500028
Mitogen-activated protein kinase kinase kinase 7Homo sapiens (human)Kd4.766713
Mitogen-activated protein kinase kinase kinase 9Homo sapiens (human)Kd8.566726
Mitogen-activated protein kinase kinase kinase kinase 1Homo sapiens (human)Kd17.8727311
Mitogen-activated protein kinase kinase kinase kinase 2Homo sapiens (human)Kd21.261128
Mitogen-activated protein kinase kinase kinase kinase 3Homo sapiens (human)Kd18.0909311
Mitogen-activated protein kinase kinase kinase kinase 4Homo sapiens (human)Kd19.0909311
Mitogen-activated protein kinase kinase kinase kinase 5Homo sapiens (human)Kd19.0909311
Mitotic checkpoint serine/threonine-protein kinase BUB1Homo sapiens (human)Kd30.000013
Multifunctional protein ADE2Homo sapiens (human)Kd30.000015
Muscle, skeletal receptor tyrosine-protein kinaseHomo sapiens (human)Kd10.000026
Myosin light chain kinase 2, skeletal/cardiac muscleHomo sapiens (human)Kd6.993326
Myosin light chain kinase 3Homo sapiens (human)Kd20.242927
Myosin light chain kinase family member 4Homo sapiens (human)Kd8.733326
Myosin light chain kinase, smooth muscleGallus gallus (chicken)Kd7.233313
Myosin light chain kinase, smooth muscleHomo sapiens (human)Kd20.0000312
Myosin-10Homo sapiens (human)Kd30.000015
Myosin-14Homo sapiens (human)Kd30.000015
Myosin-IIIaHomo sapiens (human)Kd10.000026
Myosin-IIIbHomo sapiens (human)Kd10.000026
Myotonin-protein kinaseHomo sapiens (human)Kd5.400026
NADH dehydrogenase [ubiquinone] 1 alpha subcomplex subunit 13Homo sapiens (human)Kd30.000015
Non-receptor tyrosine-protein kinase TNK1Homo sapiens (human)Kd19.0909311
Non-receptor tyrosine-protein kinase TYK2Homo sapiens (human)Kd13.8345414
NPYLR7BAedes aegypti (yellow fever mosquito)EC5020.000011
NT-3 growth factor receptorHomo sapiens (human)Kd10.000026
NUAK family SNF1-like kinase 1Homo sapiens (human)Kd10.000026
NUAK family SNF1-like kinase 2Homo sapiens (human)Kd14.6200310
Nucleolar GTP-binding protein 1Homo sapiens (human)Kd30.000015
Nucleoside diphosphate kinase BHomo sapiens (human)Kd30.000011
Obg-like ATPase 1Homo sapiens (human)Kd30.000014
PAS domain-containing serine/threonine-protein kinaseHomo sapiens (human)Kd30.000015
Peripheral plasma membrane protein CASKHomo sapiens (human)Kd3.474713
Peroxisomal acyl-coenzyme A oxidase 1Homo sapiens (human)Kd30.000015
Peroxisomal acyl-coenzyme A oxidase 3Homo sapiens (human)Kd30.000016
Phenylalanine--tRNA ligase beta subunitHomo sapiens (human)Kd30.000015
Phosphatidylethanolamine-binding protein 1Homo sapiens (human)Kd30.000014
Phosphatidylinositol 4-kinase betaHomo sapiens (human)Kd10.000013
Phosphatidylinositol 4-phosphate 3-kinase C2 domain-containing subunit betaHomo sapiens (human)Kd10.000013
Phosphatidylinositol 4-phosphate 3-kinase C2 domain-containing subunit gammaHomo sapiens (human)Kd10.000013
Phosphatidylinositol 4-phosphate 5-kinase type-1 alphaHomo sapiens (human)Kd10.000026
Phosphatidylinositol 4-phosphate 5-kinase type-1 gammaHomo sapiens (human)Kd7.533313
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoformHomo sapiens (human)Kd10.00001236
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoformHomo sapiens (human)Kd10.000013
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoformHomo sapiens (human)Kd10.000013
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform Homo sapiens (human)Kd10.000013
Phosphatidylinositol 5-phosphate 4-kinase type-2 alphaHomo sapiens (human)Kd24.041615
Phosphatidylinositol 5-phosphate 4-kinase type-2 betaHomo sapiens (human)Kd10.000026
Phosphatidylinositol 5-phosphate 4-kinase type-2 gammaHomo sapiens (human)Kd14.429528
Phosphorylase b kinase gamma catalytic chain, liver/testis isoformHomo sapiens (human)Kd15.6883412
Phosphorylase b kinase gamma catalytic chain, skeletal muscle/heart isoformHomo sapiens (human)Kd5.333326
Platelet-derived growth factor receptor alphaHomo sapiens (human)Kd9.316726
Platelet-derived growth factor receptor betaHomo sapiens (human)Kd19.0909311
Probable ATP-dependent RNA helicase DDX6Homo sapiens (human)Kd30.000016
Prostaglandin G/H synthase 2Homo sapiens (human)Kd10.000013
Protein kinase C alpha typeHomo sapiens (human)Kd30.000015
Protein kinase C beta typeHomo sapiens (human)Kd30.000015
Protein kinase C delta typeHomo sapiens (human)Kd14.7975311
Protein kinase C epsilon typeHomo sapiens (human)Kd6.793326
Protein kinase C eta typeHomo sapiens (human)Kd6.783326
Protein kinase C iota typeHomo sapiens (human)Kd22.500028
Protein kinase C theta typeHomo sapiens (human)Kd17.3364311
Protein kinase C zeta typeHomo sapiens (human)Kd30.000013
Protein-tyrosine kinase 2-betaHomo sapiens (human)Kd18.4636311
Protein-tyrosine kinase 6Homo sapiens (human)Kd19.0909311
Proto-oncogene tyrosine-protein kinase receptor RetHomo sapiens (human)Kd14.3478723
Proto-oncogene tyrosine-protein kinase ROSHomo sapiens (human)Kd10.000026
Proto-oncogene tyrosine-protein kinase SrcHomo sapiens (human)Kd19.0909311
Putative heat shock protein HSP 90-beta 2Homo sapiens (human)Kd30.000015
Pyridoxal kinaseHomo sapiens (human)Kd30.000016
Rab-like protein 3Homo sapiens (human)Kd30.000015
RAC-alpha serine/threonine-protein kinaseHomo sapiens (human)Kd19.0909311
RAC-beta serine/threonine-protein kinaseHomo sapiens (human)Kd19.0909311
RAC-gamma serine/threonine-protein kinaseHomo sapiens (human)Kd19.0909311
RAF proto-oncogene serine/threonine-protein kinaseHomo sapiens (human)Kd10.000026
Ras-related protein Rab-10Homo sapiens (human)Kd30.000015
Ras-related protein Rab-27AHomo sapiens (human)Kd30.000015
Ras-related protein Rab-6AHomo sapiens (human)Kd30.000014
Receptor tyrosine-protein kinase erbB-2Homo sapiens (human)Kd10.000026
Receptor tyrosine-protein kinase erbB-3Homo sapiens (human)Kd9.733313
Receptor tyrosine-protein kinase erbB-4Homo sapiens (human)Kd8.333313
Receptor-interacting serine/threonine-protein kinase 1Homo sapiens (human)Kd10.000026
Receptor-interacting serine/threonine-protein kinase 2Homo sapiens (human)Kd19.0909311
Receptor-interacting serine/threonine-protein kinase 3Homo sapiens (human)Kd30.000015
Receptor-interacting serine/threonine-protein kinase 4Homo sapiens (human)Kd10.000013
Receptor-type tyrosine-protein kinase FLT3Homo sapiens (human)Kd10.94391341
Retinoic acid receptor alphaHomo sapiens (human)EC500.022011
Retinoic acid receptor betaHomo sapiens (human)EC500.002011
Retinoic acid receptor gamma Homo sapiens (human)EC500.003111
Rho-associated protein kinase 1Homo sapiens (human)Kd21.400028
Rho-associated protein kinase 2Homo sapiens (human)Kd21.437528
Rhodopsin kinase GRK1Homo sapiens (human)Kd6.883313
Rhodopsin kinase GRK7Homo sapiens (human)Kd6.993313
Ribosomal protein S6 kinase alpha-1Homo sapiens (human)Kd12.2576517
Ribosomal protein S6 kinase alpha-2Homo sapiens (human)Kd7.2929514
Ribosomal protein S6 kinase alpha-3Homo sapiens (human)Kd18.2727311
Ribosomal protein S6 kinase alpha-4Homo sapiens (human)Kd14.8588517
Ribosomal protein S6 kinase alpha-5Homo sapiens (human)Kd15.0556618
Ribosomal protein S6 kinase alpha-6Homo sapiens (human)Kd14.3353517
Ribosomal protein S6 kinase beta-1Homo sapiens (human)Kd21.712528
Ribosyldihydronicotinamide dehydrogenase [quinone]Homo sapiens (human)Kd30.000015
RNA cytidine acetyltransferaseHomo sapiens (human)Kd30.000016
S-adenosylmethionine synthase isoform type-2Homo sapiens (human)Kd30.000015
Septin-9Homo sapiens (human)Kd30.000015
Serine/threonine-protein kinase 10Homo sapiens (human)Kd19.0909311
Serine/threonine-protein kinase 16Homo sapiens (human)Kd17.2699311
Serine/threonine-protein kinase 17AHomo sapiens (human)Kd5.830026
Serine/threonine-protein kinase 17BHomo sapiens (human)Kd6.985737
Serine/threonine-protein kinase 24Homo sapiens (human)Kd16.666739
Serine/threonine-protein kinase 25Homo sapiens (human)Kd10.000026
Serine/threonine-protein kinase 26Homo sapiens (human)Kd19.0909311
Serine/threonine-protein kinase 3Homo sapiens (human)Kd18.9818311
Serine/threonine-protein kinase 32AHomo sapiens (human)Kd8.500013
Serine/threonine-protein kinase 32BHomo sapiens (human)Kd10.000026
Serine/threonine-protein kinase 32CHomo sapiens (human)Kd10.000026
Serine/threonine-protein kinase 33Homo sapiens (human)Kd7.233326
Serine/threonine-protein kinase 35Homo sapiens (human)Kd6.816713
Serine/threonine-protein kinase 36Homo sapiens (human)Kd6.753326
Serine/threonine-protein kinase 38Homo sapiens (human)Kd15.000024
Serine/threonine-protein kinase 38-likeHomo sapiens (human)Kd12.857137
Serine/threonine-protein kinase 4Homo sapiens (human)Kd20.0000312
Serine/threonine-protein kinase A-RafHomo sapiens (human)Kd30.000015
Serine/threonine-protein kinase ATRHomo sapiens (human)Kd30.000011
Serine/threonine-protein kinase B-rafHomo sapiens (human)Kd14.8765517
Serine/threonine-protein kinase BRSK1Homo sapiens (human)Kd10.000026
Serine/threonine-protein kinase BRSK2Homo sapiens (human)Kd9.266726
Serine/threonine-protein kinase Chk1Homo sapiens (human)Kd19.0909311
Serine/threonine-protein kinase Chk2Homo sapiens (human)Kd10.000013
Serine/threonine-protein kinase D1Homo sapiens (human)Kd3.906726
Serine/threonine-protein kinase D2Homo sapiens (human)Kd11.5399311
Serine/threonine-protein kinase D3Homo sapiens (human)Kd9.2847311
Serine/threonine-protein kinase DCLK1Homo sapiens (human)Kd4.566726
Serine/threonine-protein kinase DCLK2Homo sapiens (human)Kd5.766726
Serine/threonine-protein kinase DCLK3Homo sapiens (human)Kd2.750026
Serine/threonine-protein kinase ICKHomo sapiens (human)Kd18.769928
Serine/threonine-protein kinase LATS1Homo sapiens (human)Kd19.0909311
Serine/threonine-protein kinase LATS2Homo sapiens (human)Kd10.000026
Serine/threonine-protein kinase MAKHomo sapiens (human)Kd0.808313
Serine/threonine-protein kinase MARK1Homo sapiens (human)Kd10.000026
Serine/threonine-protein kinase MARK2Homo sapiens (human)Kd19.0909311
Serine/threonine-protein kinase MRCK alphaHomo sapiens (human)Kd17.5473311
Serine/threonine-protein kinase MRCK betaHomo sapiens (human)Kd20.5504312
Serine/threonine-protein kinase MRCK gammaHomo sapiens (human)Kd19.0909311
Serine/threonine-protein kinase mTORHomo sapiens (human)Kd10.000013
Serine/threonine-protein kinase N1Homo sapiens (human)Kd17.2165312
Serine/threonine-protein kinase N2Homo sapiens (human)Kd20.0000312
Serine/threonine-protein kinase N3Homo sapiens (human)Kd30.000013
Serine/threonine-protein kinase Nek1Homo sapiens (human)Kd19.0909311
Serine/threonine-protein kinase Nek11Homo sapiens (human)Kd10.000013
Serine/threonine-protein kinase Nek2Homo sapiens (human)Kd19.0909311
Serine/threonine-protein kinase Nek3Homo sapiens (human)Kd22.500028
Serine/threonine-protein kinase Nek4Homo sapiens (human)Kd10.000013
Serine/threonine-protein kinase Nek5Homo sapiens (human)Kd10.000026
Serine/threonine-protein kinase Nek6Homo sapiens (human)Kd10.000026
Serine/threonine-protein kinase Nek7Homo sapiens (human)Kd18.0000310
Serine/threonine-protein kinase Nek9Homo sapiens (human)Kd19.0909311
Serine/threonine-protein kinase NIM1Homo sapiens (human)Kd10.000013
Serine/threonine-protein kinase NLKHomo sapiens (human)Kd19.0909311
Serine/threonine-protein kinase OSR1Homo sapiens (human)Kd10.000013
Serine/threonine-protein kinase PAK 1Homo sapiens (human)Kd10.000026
Serine/threonine-protein kinase PAK 2Homo sapiens (human)Kd15.000038
Serine/threonine-protein kinase PAK 3Homo sapiens (human)Kd7.833326
Serine/threonine-protein kinase PAK 4Homo sapiens (human)Kd16.8204311
Serine/threonine-protein kinase PAK 5Homo sapiens (human)Kd10.000026
Serine/threonine-protein kinase PAK 6Homo sapiens (human)Kd15.000038
Serine/threonine-protein kinase pim-1Homo sapiens (human)Kd15.9700412
Serine/threonine-protein kinase pim-2Homo sapiens (human)Kd16.0158412
Serine/threonine-protein kinase pim-3Homo sapiens (human)Kd6.866726
Serine/threonine-protein kinase PknBMycobacterium tuberculosis H37RvKd10.000013
Serine/threonine-protein kinase PLK1Homo sapiens (human)Kd16.666739
Serine/threonine-protein kinase PLK2Homo sapiens (human)Kd10.000013
Serine/threonine-protein kinase PLK3Homo sapiens (human)Kd10.000026
Serine/threonine-protein kinase PLK4Homo sapiens (human)Kd18.5769413
Serine/threonine-protein kinase PRP4 homologHomo sapiens (human)Kd10.000013
Serine/threonine-protein kinase receptor R3Homo sapiens (human)Kd12.071437
Serine/threonine-protein kinase RIO1Homo sapiens (human)Kd10.000026
Serine/threonine-protein kinase RIO2Homo sapiens (human)Kd7.166713
Serine/threonine-protein kinase RIO3Homo sapiens (human)Kd10.000026
Serine/threonine-protein kinase SBK1Homo sapiens (human)Kd10.000013
Serine/threonine-protein kinase Sgk3Homo sapiens (human)Kd10.000013
Serine/threonine-protein kinase SIK1Homo sapiens (human)Kd10.000026
Serine/threonine-protein kinase SIK2Homo sapiens (human)Kd19.0909311
Serine/threonine-protein kinase SIK3Homo sapiens (human)Kd23.333329
Serine/threonine-protein kinase STK11Homo sapiens (human)Kd19.0909311
Serine/threonine-protein kinase TAO1Homo sapiens (human)Kd10.828739
Serine/threonine-protein kinase TAO2Homo sapiens (human)Kd15.101228
Serine/threonine-protein kinase TAO3Homo sapiens (human)Kd10.916828
Serine/threonine-protein kinase TBK1Homo sapiens (human)Kd19.157729
Serine/threonine-protein kinase TNNI3KHomo sapiens (human)Kd6.685026
Serine/threonine-protein kinase tousled-like 1Homo sapiens (human)Kd8.733326
Serine/threonine-protein kinase tousled-like 2Homo sapiens (human)Kd10.000026
Serine/threonine-protein kinase ULK1Homo sapiens (human)Kd22.533329
Serine/threonine-protein kinase ULK2Homo sapiens (human)Kd6.823313
Serine/threonine-protein kinase ULK3Homo sapiens (human)Kd23.333329
Serine/threonine-protein kinase VRK2Homo sapiens (human)Kd6.687713
Serine/threonine-protein kinase/endoribonuclease IRE1Homo sapiens (human)Kd23.333329
Serine/threonine-protein kinase/endoribonuclease IRE2Homo sapiens (human)Kd30.000016
Signal recognition particle receptor subunit alphaHomo sapiens (human)Kd30.000016
SNF-related serine/threonine-protein kinaseHomo sapiens (human)Kd10.000013
SRSF protein kinase 1Homo sapiens (human)Kd10.000026
SRSF protein kinase 2Homo sapiens (human)Kd10.000026
SRSF protein kinase 3Homo sapiens (human)Kd10.000013
STE20-like serine/threonine-protein kinase Homo sapiens (human)Kd18.7182311
STE20-related kinase adapter protein alphaHomo sapiens (human)Kd25.467816
STE20/SPS1-related proline-alanine-rich protein kinaseHomo sapiens (human)Kd10.000013
Structural maintenance of chromosomes protein 1AHomo sapiens (human)Kd30.000013
Structural maintenance of chromosomes protein 2Homo sapiens (human)Kd30.000015
Succinate--CoA ligase [ADP-forming] subunit beta, mitochondrialHomo sapiens (human)Kd30.000012
Testis-specific serine/threonine-protein kinase 1Homo sapiens (human)Kd10.000026
TGF-beta receptor type-1Homo sapiens (human)Kd20.0000312
TGF-beta receptor type-2Homo sapiens (human)Kd16.9091311
Thyroid hormone receptor-associated protein 3Homo sapiens (human)Kd30.000014
TRAF2 and NCK-interacting protein kinaseHomo sapiens (human)Kd20.0000312
Transient receptor potential cation channel subfamily M member 6Homo sapiens (human)Kd10.000013
Tubulin alpha-1A chainRattus norvegicus (Norway rat)Kd10.000013
Tyrosine--tRNA ligase, cytoplasmicHomo sapiens (human)Kd30.000015
Tyrosine-protein kinase ABL1Homo sapiens (human)Kd10.09142371
Tyrosine-protein kinase ABL2Homo sapiens (human)Kd19.0909311
Tyrosine-protein kinase BlkHomo sapiens (human)Kd10.000026
Tyrosine-protein kinase BTKHomo sapiens (human)Kd19.0909311
Tyrosine-protein kinase CSKHomo sapiens (human)Kd19.0909311
Tyrosine-protein kinase FerHomo sapiens (human)Kd19.0909311
Tyrosine-protein kinase Fes/FpsHomo sapiens (human)Kd19.0909311
Tyrosine-protein kinase FgrHomo sapiens (human)Kd15.000038
Tyrosine-protein kinase FRKHomo sapiens (human)Kd18.2909311
Tyrosine-protein kinase FynHomo sapiens (human)Kd19.0909311
Tyrosine-protein kinase HCKHomo sapiens (human)Kd19.0909311
Tyrosine-protein kinase ITK/TSKHomo sapiens (human)Kd10.000026
Tyrosine-protein kinase JAK1Homo sapiens (human)Kd17.1429414
Tyrosine-protein kinase JAK2Homo sapiens (human)Kd18.6818311
Tyrosine-protein kinase JAK3Homo sapiens (human)Kd8.600026
Tyrosine-protein kinase LckHomo sapiens (human)Kd20.0000312
Tyrosine-protein kinase LynHomo sapiens (human)Kd19.0909311
Tyrosine-protein kinase MerHomo sapiens (human)Kd11.942937
Tyrosine-protein kinase receptor Tie-1Homo sapiens (human)Kd10.000026
Tyrosine-protein kinase receptor TYRO3Homo sapiens (human)Kd10.000026
Tyrosine-protein kinase receptor UFOHomo sapiens (human)Kd7.833326
Tyrosine-protein kinase SrmsHomo sapiens (human)Kd7.133326
Tyrosine-protein kinase SYKHomo sapiens (human)Kd19.0909311
Tyrosine-protein kinase TecHomo sapiens (human)Kd19.0909311
Tyrosine-protein kinase TXKHomo sapiens (human)Kd10.000026
Tyrosine-protein kinase YesHomo sapiens (human)Kd19.0909311
Tyrosine-protein kinase ZAP-70Homo sapiens (human)Kd10.000026
U5 small nuclear ribonucleoprotein 200 kDa helicaseHomo sapiens (human)Kd30.000015
UMP-CMP kinase Homo sapiens (human)Kd30.000014
Uncharacterized aarF domain-containing protein kinase 5Homo sapiens (human)Kd30.000012
Uncharacterized protein FLJ45252Homo sapiens (human)Kd29.555716
Uncharacterized serine/threonine-protein kinase SBK3Homo sapiens (human)Kd10.000013
Vascular endothelial growth factor receptor 1 Homo sapiens (human)Kd9.983326
Vascular endothelial growth factor receptor 2Homo sapiens (human)Kd10.000026
Vascular endothelial growth factor receptor 3Homo sapiens (human)Kd10.000026
Very long-chain specific acyl-CoA dehydrogenase, mitochondrialHomo sapiens (human)Kd30.000016
Voltage-dependent N-type calcium channel subunit alpha-1BHomo sapiens (human)EC50675.860013
Wee1-like protein kinaseHomo sapiens (human)Kd19.0909311
Wee1-like protein kinase 2Homo sapiens (human)Kd10.000013

Other Measurements

ProteinTaxonomyMeasurementAverage (mM)Bioassay(s)Drugs
Cannabinoid receptor 1Homo sapiens (human)Kb2.200011
Casein kinase I isoform alphaHomo sapiens (human)EC4.980022
Casein kinase I isoform deltaHomo sapiens (human)EC4.980022
Cyclin-A1Homo sapiens (human)ID500.100011
Cyclin-A2Homo sapiens (human)ID500.100011
Cyclin-dependent kinase 1Homo sapiens (human)ID502.217127
Cyclin-dependent kinase 1Homo sapiens (human)INH24.500011
Cyclin-dependent kinase 10Homo sapiens (human)INH24.500011
Cyclin-dependent kinase 11BHomo sapiens (human)INH24.500011
Cyclin-dependent kinase 12Homo sapiens (human)INH24.500011
Cyclin-dependent kinase 13Homo sapiens (human)INH24.500011
Cyclin-dependent kinase 14Homo sapiens (human)INH24.500011
Cyclin-dependent kinase 15Homo sapiens (human)INH24.500011
Cyclin-dependent kinase 16Homo sapiens (human)INH24.500011
Cyclin-dependent kinase 17Homo sapiens (human)INH24.500011
Cyclin-dependent kinase 18Homo sapiens (human)INH24.500011
Cyclin-dependent kinase 19Homo sapiens (human)INH24.500011
Cyclin-dependent kinase 2Homo sapiens (human)Cell cycle0.02101010
Cyclin-dependent kinase 2Homo sapiens (human)ID503.550022
Cyclin-dependent kinase 2Homo sapiens (human)INH24.500011
Cyclin-dependent kinase 20Homo sapiens (human)INH24.500011
Cyclin-dependent kinase 3Homo sapiens (human)INH24.500011
Cyclin-dependent kinase 4Homo sapiens (human)ID500.400011
Cyclin-dependent kinase 4Homo sapiens (human)INH24.500011
Cyclin-dependent kinase 6Homo sapiens (human)INH24.500011
Cyclin-dependent kinase 7Homo sapiens (human)INH24.500011
Cyclin-dependent kinase 8Homo sapiens (human)INH24.500011
Cyclin-dependent kinase 9Homo sapiens (human)INH24.500011
Cyclin-dependent-like kinase 5 Homo sapiens (human)INH24.500011
G1/S-specific cyclin-D1Homo sapiens (human)ID500.400011
G1/S-specific cyclin-D2Homo sapiens (human)ID500.400011
G1/S-specific cyclin-D3Homo sapiens (human)ID500.400011
G1/S-specific cyclin-E1Homo sapiens (human)ID507.000011
G1/S-specific cyclin-E2Homo sapiens (human)ID507.000011
G2/mitotic-specific cyclin-B1Homo sapiens (human)ID502.217127
G2/mitotic-specific cyclin-B2Homo sapiens (human)ID502.217127
G2/mitotic-specific cyclin-B3Homo sapiens (human)ID502.217127
UDP-glucuronosyltransferase 1A9Homo sapiens (human)Km37.000011