Page last updated: 2024-08-05 14:59:56

fluorochrome

A fluorescent dye used to stain biological specimens.

ChEBI ID: 51217

Members (120)

MemberDefinitionClass
1,1'-((4,4,7,7-tetramethyl)-4,7-diazaundecamethylene)bis-4-(3-methyl-2,3-dihydro(benzo-1,3-oxazole)-2-methylidine)quinolinium, tetraiodideYoYo-1
1,1'-(4,4,7,7-tetramethyl-4,7-diazaundecamethylene)bis-4-(3-methyl-2,3-dihydro(benzo-1,3-thiazole)-2-methylidene)quinoliniumToTo-1
2-(4-(dimethylamino)styryl)-1-methylpyridinium2-[4-(dimethylamino)styryl]-1-methylpyridinium iodide
2-(5'-chloro-2'-phosphoryloxyphenyl)-6-chloro-4-(3h)-quinazolinone2-(5'-chloro-2'-phosphoryloxyphenyl)-6-chloro-4-(3H)-quinazolinone
2',7'-dichlorofluorescein2',7'-dichlorofluorescein
3-(4-carboxybenzoyl)-2-quinolinecarboxaldehydeCBQCA reagent
3,3'-diethyloxacarbocyanineThe cationic form of a C3 cyanine dye having 3-ethyl-1,3-benzoxazol-2(3H)-yl units at each end.C3-oxacyanine cation
3,3'-diethylthiacarbocyanine iodideC3-thiacarbocyanine
3,3'-diethylthiacarbocyanine iodideC3-thiacarbocyanine
3,3'-dioctadecylindocarbocyanineThe cationic form of a C3 cyanine dye having 3,3-dimethyl-1-octadecylindoleinine units at each end.dilC18(3)(1+)
3,3'-dipentyl-2,2'-oxacarbocyanineThe cationic form of a C3 cyanine dye having 3-pentyl-1,3-benzoxazol-2(3H)-yl units at each end. A fluorescent compound that preferentially stains chronic myelogenic leukemia cells.3,3'-dipentyloxacarbocyanine
4-(4-diethylaminostyryl)-n-methylpyridiniumAn organic iodide salt consisting of pyridinium iodide having a methyl substituent at the 1-position and a 4-diethylaminostyryl substituent at the 4-position.4-(4-diethylaminostyryl)-1-methylpyridinium iodide
4-(4-dihexadecylaminostyryl)-n-methylpyridiumA pyridinium cation with a methyl substituent at the 1-position and a 4-(dihexadecylamino)styryl substituent at the 4-position.4-(4-dihexadecylaminostyryl)-N-methylpyridium
4-carboxyfluorescein5-carboxyfluorescein
4-chloro-7-nitrobenzofurazanA benzoxadiazole that is 2,1,3-benzoxadiazole which is substituted at position 4 by chlorine and at position 7 by a nitro group.4-chloro-7-nitrobenzofurazan
5-carboxytetramethylrhodamineA tetramethylrhodamine compound having a carboxy substituent at the 5-position5-carboxytetramethylrhodamine
5-chloromethylfluorescein diacetate5-chloromethylfluorescein diacetate
5,5',6,6'-tetrachloro-1,1',3,3'-tetraethylbenzimidazolocarbocyanineThe cationic form of a C3 cyanine dye having 1,3-diethyl-5,6-dichloroindoleinine units at each end.1,1',3,3'-tetraethyl-5,5',6,6'-tetrachloroimidacarbocyanine
7-amino-4-methylcoumarincoumarin 120
7-amino-4-trifluoromethylcoumarin7-amino-4-(trifluoromethyl)coumarin
7-methoxycoumarin-4-acetic acid7-methoxycoumarin-4-acetic acid
7-nitrobenzoxadiazole-6-aminohexanoic acidA benzoxadiazole that is 2,1,3-benzoxadiazole which is substituted at positions 4 and 7 by (5-carboxypentyl)amino and nitro groups, respectively.7-nitrobenzoxadiazole-6-aminohexanoic acid
9,10-bis(phenylethynyl)anthracene9,10-bis(phenylethynyl)anthracene
9,10-diphenylanthraceneA member of the class of anthracenes that is anthracene in which both of the hydrogens on the central ring are substituted by phenyl groups.9,10-diphenylanthracene
acridine orangeA member of the class of aminoacridines that is acridine carrying two dimethylamino substituents at positions 3 and 6. The hydrochloride salt is the fluorescent dye 'acridine orange', used for cell cycle determination.acridine orange free base
acridine yellowacridine yellow
alcian yellowAn organic chloride salt composed of {diazenediylbis[(4,1-phenylene)(6-methyl-1,3-benzothiazole-2,5-diyl)methylenesulfanediyl]}bis[(dimethylamino)-N,N-dimethylmethaniminium] and chloride ions in a 1:2 ratio.alcian yellow
alexa fluor 546Alexa Fluor 546
Alexa Fluor 555A fluorescent dye of absorption wavelength 555 nm and emission wavelength 565 nm, derived from a 3,6-diaminoxanthene-4,5-disulfate.Alexa Fluor 555
aurintricarboxylic acidA member of the class of quinomethanes that is 3-methylidene-6-oxocyclohexa-1,4-diene-1-carboxylic acid in which the methylidene hydrogens are replaced by 4-carboxy-3-hydroxyphenyl groups. The trisodium salt is the biological stain 'chrome violet CG' while the triammonium salt is 'aluminon'.aurintricarboxylic acid
basic blue kAn iminium salt composed of 4-{[4-(dimethylamino)phenyl][4-(ethylamino)naphthalen-1-yl]methylidene}-N,N-dimethylcyclohexa-2,5-dien-1-iminium and chloride ions in a 1:1 ratio.victoria blue R
benzophenoneidumA hydrochloride obtained by combining 4,4'-carbonimidoylbis(N,N-dimethylaniline) with one molar equivalent of hydrogen chloride. A fluorescent stain for demonstrating acid fast organisms in a method similar to the Ziehl Neelsen. It also can be used to make a fluorescent Schiff reagent.auramine O
biphenylacetyleneAn arylacetylene that is acetylene in which the hydrogens are replaced by phenyl groups.biphenylacetylene
bisbenzimidazolepibenzimol
bobo 3BoBo-3
brilliant greenAn organic hydrogensulfate salt having 4-{[4-(diethylamino)phenyl](phenyl)methylidene}-N,N-diethylcyclohexa-2,5-dien-1-iminium as the counterion.brilliant green
c.i. direct red 80An organic sodium salt resulting from the formal condensation of Sirius red F3B (acid form) with six equivalents of sodium hydroxide. A polyazo dye used principally in staining methods for collagen and amyloid.Sirius red F3B
calcein amAn organic heteropentacyclic compound that is calcein in which all four carboxy group hydrogens have been substituted by (acetyloxy)methoxy groups and the hyrodgens of the two hydroxy groups have been substituted by acetyl groups. It is a a non-fluorescent probe cleaved to a fluorescent probe by non-specific intracellular esterases.calcein am
calcium crimsoncalcium crimson
calcium orangeA xanthene dye-based thiourea conjugate.calcium orange
carbocyaninespinacyanol iodide
cascade bluecascade blue
clomipramineA quaternary ammonium salt that is the tetrakis(N,N,N-trimethylmethammonium) salt of 5-({[4-(13-{4-[({3-carboxy-4-[(2,7-dichloro-6-hydroxy-3-oxo-3H-xanthen-9-yl)methyl]phenyl}carbonyl)amino]-2,5-bis(methyloxy)phenyl}-1,4,10-trioxa-7,13-diazacyclopentadecan-7-yl)-2-hydroxy-5-(methyloxy)phenyl]amino}carbonyl)-2-(2,7-dichloro-6-hydroxy-3-oxo-3H-xanthen-9-yl)benzoic acid.sodium green
coumarin 153coumarin 153
coumarin 314coumarin 504
coumarin 343coumarin 343
coumarin 480coumarin 480
coumarin 6coumarin 6
dapiDAPI
dibromobimaneA pyrazolopyrazole that consists of 1H,7H-pyrazolo[1,2-a]pyrazole-1,7-dione bearing two methyl substituents at positions 2 and 6 as well as two bromomethyl substituents at positions 3 and 5.dibromobimane
diphenylhexatriene1,6-diphenylhexatriene
dithiazanineA cationic C3-cyanine dye with 3-ethylbenzothiazol-2-yl groups at both ends.dithiazanine
dithiazanine iodidedithiazanine iodide
DND-167 dyeDND-167 dye
dy-676DY-676
eosine yellowish-(ys)An organic sodium salt that is 2',4',5',7'-tetrabromofluorescein in which the carboxy group and the phenolic hydroxy group have been deprotonated and the resulting charge is neutralised by two sodium ions.eosin YS dye
epicoccononeA natural cell-permeable fluorescent compound isolated from the fungus Epicoccum nigrum.epicocconone
ethidiumThe fluorescent compound widely used in experimental cell biology and biochemistry to reveal double-stranded DNA and RNA.ethidium
ethyl violetAn organic chloride salt that is the monochloride salt of ethyl violet cation. Used for inclusion in mixed dye solutions of the iron resorcin fuchsin type for demonstrating elastic fibres.ethyl violet
evans blueAn organic sodium salt that is the tetrasodium salt of 6,6'-{(3,3'-dimethyl[1,1'-biphenyl]-4,4'-diyl)bis[diazene-2,1-diyl]}bis(4-amino-5-hydroxynaphthalene-1,3-disulfonate). It is sometimes used as a counterstain, especially in fluorescent methods to suppress background autofluorescence.Evans blue
fast green fcfAn organic sodium salt having 2-{(4-{ethyl[(3-sulfonatophenyl)methyl]amino}phenyl)[4-{ethyl[(3-sulfonatophenyl)methyl]iminio}cyclohexa-2,5-dien-1-ylidene]methyl}-5-hydroxybenzene-1-sulfonate as the counterion. Used as a substitute for Light green SF yellowish in Masson's trichrome as it is less likely to fade, and is more brilliant in colour. Also used as a food colouring agent.Fast green FCF
fluo-3Fluo-3
fluorexoncalcein
fm1 43FM 1-43 dye
galleinA xanthene dye that is fluoran carrying four hydroxy substituents at positions 3', 4', 5' and 6'.gallein
herniarinA member of the class of coumarins that is coumarin substituted by a methoxy group at position 7.herniarin
hoe 333422'-(4-ethoxyphenyl)-5-(4-methylpiperazin-1-yl)-2,5'-bibenzimidazole
hydromethylthionineA member of the class of phenothiazines that is 10H-phenothiazine in which the ring hydrogens at positions 3 and 7 have been replaced by dimethylamino groups.leucomethylene blue
indo-1Indo-1 dye
lissamine rhodamine bAn organic sodium salt having 4-[3,6-bis(diethylamino)xanthenium-9-yl]benzene-1,3-disulfonate as the counterion.lissamine rhodamine
lucifer yellowlucifer yellow dye
magnesium greenmagnesium green
malachite greenAn organic chloride salt that is the monochloride salt of malachite green cation. Used as a green-coloured dye, as a counter-stain in histology, and for its anti-fungal properties in aquaculture.malachite green
methylene blueAn organic chloride salt having 3,7-bis(dimethylamino)phenothiazin-5-ium as the counterion. A commonly used dye that also exhibits antioxidant, antimalarial, antidepressant and cardioprotective properties.methylene blue
methylene greenAn organic chloride salt having 3,7-bis(dimethylamino)-4-nitrophenothiazin-5-ium as the counterion. It stains nuclei green and is sometimes used as a counterstain to red or purple primary stains.methylene green
mitotracker orangemitoTracker Orange
monobromobimaneA pyrazolopyrazole that consists of 1H,7H-pyrazolo[1,2-a]pyrazole-1,7-dione bearing three methyl substituents at positions 2, 5 and 6 as well as a bromomethyl substituent at the 3-position.monobromobimane
monochlorobimanemonochlorobimane
monodansylcadaverineA sulfonamide obtained by formal condensation of the sulfo group of 5-(dimethylamino)naphthalene-1-sulfonic acid with one of the amino groups of cadaverine.monodansylcadaverine
new fuchsinA hydrochloride that is the monohydrochloride of 4-[(4-aminophenyl)(4-iminocyclohexa-2,5-dien-1-ylidene)methyl]-2-methylaniline. One of the minor constituents of Basic fuchsin, together with pararosanilin, rosanilin and magenta II.new fuchsin
nile redAn organic heterotetracyclic compound that is 5H-benzo[a]phenoxazin-5-one substituted at position 9 by a diethylamino group.nile red
nk 5cryptocyanin
nuclear fast redAn organic sodium salt that is the monosodium salt of 4-amino-1,3-dihydroxy-9,10-dioxo-9,10-dihydroanthracene-2-sulfonic acid. It forms bright red lakes with calcium and is a useful red nuclear staining lake with aluminum.nuclear fast red
oregon green 488 carboxylic acidA xanthene dye having two fluoro substituents at the 2- and 7-positions and a 2,4-dicarboxyphenyl group at the 9-position.oregon green 488
oregon green 514OG-514 dye
oxazine 1oxazine-1
pacific blue succinimidyl esterAn N-hydroxysuccinimide ester derived from 6,8-difluoro-7-hydroxycoumarin-3-carboxylic acid (pacific blue). A fluorescent dye of excitation wavelength 403 nm and emission wavelength 455 nm.pacific blue succinimidyl ester
perylenediimideThe 3,4,9,10-tetracarboxylic diimide derivative of perylene.perylenediimide
phenosafranineAn organic chloride salt having 3,7-diamino-5-phenylphenazin-5-ium as the counterion. It is commonly used for staining Gram negative bacteria red in smears to contrast with the blue Gram positive organisms.phenosafranine
ponceau sAn organic sodium salt that is the tetrasodium salt of 3-hydroxy-4-({2-sulfo-4-[(4-sulfophenyl)diazenyl]phenyl}diazenyl)naphthalene-2,7-disulfonic acid.Ponceau S
popopPOPOP
primulineAn organic sodium salt having 2'-(4-aminophenyl)-6-methyl[2,6'-bi-1,3-benzothiazole]-7-sulfonate as the counterion.primuline
propidiumpropidium
pyraninepyranine
quinaldine bluepinacyanol iodide
rhodamine 123rhodamine 123
rhodamine 123A cationic fluorescent dye derived from 9-phenylxanthene.rhodamine 123(1+)
rhodamine 123rhodamine 123
rhodamine bAn organic chloride salt having N-[9-(2-carboxyphenyl)-6-(diethylamino)-3H-xanthen-3-ylidene]-N-ethylethanaminium as the counterion. An amphoteric dye commonly used as a fluorochrome.rhodamine B
rose bengal(2-)The anionic form of a fluorescent dye derived from a polyhalogenated fluorescin.rose bengal(2-)
safranine tAn organic chloride salt having 3,7-diamino-2,8-dimethyl-5-phenylphenazin-5-ium as the counterion. It is commonly used for staining Gram negative bacteria.safranin O
scarlet redA bis(azo) compound that is 2-naphthol substituted at position 1 by a {2-methyl-4-[(2-methylphenyl)diazenyl]phenyl}diazenyl group. A fat-soluble dye predominantly used for demonstrating triglycerides in frozen sections, but which may also stain some protein bound lipids in paraffin sections.Sudan IV
sodium-binding benzofuran isophthalateA crown compound that is 1,4,10-trioxa-7,13-diazacyclopentadecane in which the hydrogens of the amino groups at position 7 and 13 are replaced by 2-(2,4-dicarboxyphenyl)-5-methoxy-1-benzofuran-6-yl groups. It is a cell-impermeant fluorescent sodium indicator.sodium-binding benzofuran isophthalate
stains-allcarbocyanin DBTC
succinyl-leucyl-leucyl-valyl-tyrosyl-methylcoumarinamideA tetrapeptide compound with a succinyl group at the N-terminal and a 7-amino-4-methylcoumarin group at the C-terminal.succinyl-Leu-Leu-Val-Tyr-7-amino-4-methylcoumarin
sudan iiiA bis(azo) compound that is 2-naphthol substituted at position 1 by a 4-{[(2-methylphenyl)diazenyl]phenyl}diazenyl group. A fat-soluble dye predominantly used for demonstrating triglycerides in frozen sections, but which may also stain some protein bound lipids in paraffin sections.Sudan III
sulforhodamine 101sulforhodamine 101
texas redtexas red
thiazole orangeA cyanine dye comprising the thiazole orange cation [1-methyl-4-[(3-methyl-1,3-benzothiazol-2(3H)-ylidene)methyl]quinolinium] with the p-tosylate counterion.thiazole orange
thioflavin tAn organic chloride salt having 2-[4-(dimethylamino)phenyl]-3,6-dimethyl-1,3-benzothiazol-3-ium as the counterion. It is widely used to visualise and quantify the presence of amyloids, both in vitro and in vivo.thioflavine T
to-pro-1A C1 cyanine dye having benzothiazolium-2-yl and quinolinium-4-yl substituents.To-Pro-1
to-pro-3An unsymmetrical C3 cyanine dye having benzothiazolium-2-yl and quinolinium-4-yl substituents.To-Pro-3
tris(2,2'-bipyridine)ruthenium(II)A ruthenium coordination entity consisting of ruthenium(II) bound to three 2,2'-bipyridine units.tris(2,2'-bipyridine)ruthenium(II)
tris(4,7-diphenyl-1,10-phenanthroline)ruthenium (ii)A ruthenium coordination entity consisting of ruthenium(II) bound to three 4,7-diphenyl-1,10-phenanthroline units.tris(4,7-diphenyl-1,10-phenanthroline)ruthenium(II)
uvitex swncoumarin 460
victoria blue 4rAn iminium salt composed of 4-([4-(dimethylamino)phenyl]{4-[methyl(phenyl)amino]naphthalen-1-yl}methylidene)-N,N-dimethylcyclohexa-2,5-dien-1-iminium and chloride ions in a 1:1 ratio. It binds to nucleic acids and can be used in standardised staining techniques suitable for automated cell-pattern recognition.victoria blue 4R
victoria blue bAn iminium salt composed of 4-{(4-anilinonaphthalen-1-yl)[4-(dimethylamino)phenyl]methylidene}-N,N-dimethylcyclohexa-2,5-dien-1-iminium and chloride ions in a 1:1 ratio. It binds to nucleic acids and can be used in standardised staining techniques suitable for automated cell-pattern recognition.victoria blue B
yo-pro 1An unsymmetrical C1 cyanine dye having 1,3-benzoxazol-2-yl and quinolinium-4-yl substituents.Yo-Pro-1
yoyo-3YoYo-3
zn(ii)-phthalocyaninezinc phthalocyanine

Research

Studies (51,307)

TimeframeStudies, Drugs with This Role(%)All Drugs %
pre-19909,053 (17.64)18.7374
1990's9,927 (19.35)18.2507
2000's13,583 (26.47)29.6817
2010's14,653 (28.56)24.3611
2020's4,091 (7.97)2.80

Study Types

Publication TypeStudies, Drugs with this Role (%)All Drugs (%)
Trials578 (1.00%)5.53%
Reviews945 (1.64%)6.00%
Case Studies1,088 (1.89%)4.05%
Observational25 (0.04%)0.25%
Other54,907 (95.42%)84.16%

Protein Targets (386)

Potency Measurements

ProteinTaxonomyMeasurementAverage (mM)Bioassay(s)Drugs
15-hydroxyprostaglandin dehydrogenase [NAD(+)] isoform 1Homo sapiens (human)Potency18.0454110
15-lipoxygenase, partialHomo sapiens (human)Potency5.928914
2,3-bisphosphoglycerate-independent phosphoglycerate mutaseLeishmania major strain FriedlinPotency30.131311
67.9K proteinVaccinia virusPotency11.781926
acetylcholinesteraseHomo sapiens (human)Potency21.3645424
acid sphingomyelinaseHomo sapiens (human)Potency26.926213
activating transcription factor 6Homo sapiens (human)Potency28.418426
aldehyde dehydrogenase 1 family, member A1Homo sapiens (human)Potency20.2039113
alpha-galactosidaseHomo sapiens (human)Potency35.368827
Alpha-synucleinHomo sapiens (human)Potency8.082715
apical membrane antigen 1, AMA1Plasmodium falciparum 3D7Potency18.230315
AR proteinHomo sapiens (human)Potency18.31671287
aryl hydrocarbon receptorHomo sapiens (human)Potency11.3049219
ATAD5 protein, partialHomo sapiens (human)Potency13.109238
Ataxin-2Homo sapiens (human)Potency9.288816
ATP-dependent phosphofructokinaseTrypanosoma brucei brucei TREU927Potency16.221424
ATPase family AAA domain-containing protein 5Homo sapiens (human)Potency7.064029
Bloom syndrome protein isoform 1Homo sapiens (human)Potency15.4001313
BRCA1Homo sapiens (human)Potency0.891311
bromodomain adjacent to zinc finger domain 2BHomo sapiens (human)Potency17.553017
caspase 7, apoptosis-related cysteine proteaseHomo sapiens (human)Potency11.896015
caspase-1 isoform alpha precursorHomo sapiens (human)Potency10.102215
caspase-3Cricetulus griseus (Chinese hamster)Potency7.616212
caspase-3Homo sapiens (human)Potency11.896015
Caspase-7Cricetulus griseus (Chinese hamster)Potency7.616212
Caspase-7Homo sapiens (human)Potency11.050314
Cellular tumor antigen p53Homo sapiens (human)Potency19.6057319
Chain A, 2-oxoglutarate OxygenaseHomo sapiens (human)Potency24.1773110
Chain A, ATP-DEPENDENT DNA HELICASE Q1Homo sapiens (human)Potency19.3167417
Chain A, Beta-lactamaseEscherichia coli K-12Potency30.305826
Chain A, Breast cancer type 1 susceptibility proteinHomo sapiens (human)Potency14.219112
Chain A, CruzipainTrypanosoma cruziPotency22.912028
Chain A, Ferritin light chainEquus caballus (horse)Potency29.435029
Chain A, HADH2 proteinHomo sapiens (human)Potency16.5439211
Chain A, JmjC domain-containing histone demethylation protein 3AHomo sapiens (human)Potency35.894717
Chain A, MAJOR APURINIC/APYRIMIDINIC ENDONUCLEASEHomo sapiens (human)Potency16.6558316
Chain A, Putative fructose-1,6-bisphosphate aldolaseGiardia intestinalisPotency20.457515
Chain A, TYROSYL-DNA PHOSPHODIESTERASEHomo sapiens (human)Potency13.0874214
Chain B, HADH2 proteinHomo sapiens (human)Potency16.5439211
chaperonin-containing TCP-1 beta subunit homologHomo sapiens (human)Potency51.059414
chromobox protein homolog 1Homo sapiens (human)Potency28.980425
ClpPBacillus subtilisPotency30.741022
core-binding factor subunit beta isoform 2Homo sapiens (human)Potency2.931724
cytochrome P450 2C19 precursorHomo sapiens (human)Potency13.351912
cytochrome P450 2C9 precursorHomo sapiens (human)Potency14.219112
cytochrome P450 2C9, partialHomo sapiens (human)Potency8.675214
cytochrome P450 2D6Homo sapiens (human)Potency9.913215
cytochrome P450 2D6 isoform 1Homo sapiens (human)Potency23.060212
cytochrome P450 3A4 isoform 1Homo sapiens (human)Potency17.216826
cytochrome P450 family 3 subfamily A polypeptide 4Homo sapiens (human)Potency5.094626
cytochrome P450, family 19, subfamily A, polypeptide 1, isoform CRA_aHomo sapiens (human)Potency24.7750114
Disintegrin and metalloproteinase domain-containing protein 17Homo sapiens (human)Potency19.952611
DNA dC->dU-editing enzyme APOBEC-3F isoform aHomo sapiens (human)Potency3.956213
DNA polymerase betaHomo sapiens (human)Potency11.200415
DNA polymerase eta isoform 1Homo sapiens (human)Potency32.056913
DNA polymerase III, partialBacillus subtilisPotency3.358711
DNA polymerase iota isoform a (long)Homo sapiens (human)Potency45.622617
DNA polymerase kappa isoform 1Homo sapiens (human)Potency11.0336112
endonuclease IVEscherichia coliPotency1.473322
Endothelin receptor type BRattus norvegicus (Norway rat)Potency19.118012
Endothelin-1 receptorRattus norvegicus (Norway rat)Potency19.118012
estrogen nuclear receptor alphaHomo sapiens (human)Potency21.30201188
estrogen receptor 2 (ER beta)Homo sapiens (human)Potency32.0712313
estrogen-related nuclear receptor alphaHomo sapiens (human)Potency17.3019770
euchromatic histone-lysine N-methyltransferase 2Homo sapiens (human)Potency18.8114115
EWS/FLI fusion proteinHomo sapiens (human)Potency15.826444
eyes absent homolog 2 isoform aHomo sapiens (human)Potency41.281414
farnesoid X nuclear receptorHomo sapiens (human)Potency24.8871415
flap endonuclease 1Homo sapiens (human)Potency19.842828
Fumarate hydrataseHomo sapiens (human)Potency10.665412
GVesicular stomatitis virusPotency8.675214
GABA theta subunitRattus norvegicus (Norway rat)Potency17.216813
galactokinaseHomo sapiens (human)Potency14.125411
Gamma-aminobutyric acid receptor subunit alpha-1Rattus norvegicus (Norway rat)Potency17.216813
Gamma-aminobutyric acid receptor subunit alpha-2Rattus norvegicus (Norway rat)Potency17.216813
Gamma-aminobutyric acid receptor subunit alpha-3Rattus norvegicus (Norway rat)Potency17.216813
Gamma-aminobutyric acid receptor subunit alpha-4Rattus norvegicus (Norway rat)Potency17.216813
Gamma-aminobutyric acid receptor subunit alpha-5Rattus norvegicus (Norway rat)Potency17.216813
Gamma-aminobutyric acid receptor subunit alpha-6Rattus norvegicus (Norway rat)Potency17.216813
Gamma-aminobutyric acid receptor subunit beta-1Rattus norvegicus (Norway rat)Potency17.216813
Gamma-aminobutyric acid receptor subunit beta-2Rattus norvegicus (Norway rat)Potency17.216813
Gamma-aminobutyric acid receptor subunit beta-3Rattus norvegicus (Norway rat)Potency17.216813
Gamma-aminobutyric acid receptor subunit deltaRattus norvegicus (Norway rat)Potency17.216813
Gamma-aminobutyric acid receptor subunit epsilonRattus norvegicus (Norway rat)Potency17.216813
Gamma-aminobutyric acid receptor subunit gamma-1Rattus norvegicus (Norway rat)Potency17.216813
Gamma-aminobutyric acid receptor subunit gamma-2Rattus norvegicus (Norway rat)Potency17.216813
Gamma-aminobutyric acid receptor subunit gamma-3Rattus norvegicus (Norway rat)Potency17.216813
Gamma-aminobutyric acid receptor subunit piRattus norvegicus (Norway rat)Potency17.216813
gemininHomo sapiens (human)Potency17.4545310
GLI family zinc finger 3Homo sapiens (human)Potency12.1759221
glp-1 receptor, partialHomo sapiens (human)Potency12.427714
GLS proteinHomo sapiens (human)Potency6.878824
glucocerebrosidaseHomo sapiens (human)Potency35.716812
glucocorticoid receptor [Homo sapiens]Homo sapiens (human)Potency27.5010518
glucokinase regulatory proteinHomo sapiens (human)Potency10.699233
Glutamate receptor 1Rattus norvegicus (Norway rat)Potency0.056211
Glutamate receptor 2Rattus norvegicus (Norway rat)Potency16.6913211
Glutamate receptor 3Rattus norvegicus (Norway rat)Potency0.056211
Glutamate receptor 4Rattus norvegicus (Norway rat)Potency0.056211
Glycoprotein hormones alpha chainHomo sapiens (human)Potency22.982614
GTP-binding nuclear protein Ran isoform 1Homo sapiens (human)Potency29.216815
Guanine nucleotide-binding protein GHomo sapiens (human)Potency17.633528
guanine nucleotide-binding protein G(i) subunit alpha-1 isoform 1Homo sapiens (human)Potency15.848911
heat shock protein beta-1Homo sapiens (human)Potency34.606128
hemoglobin subunit betaHomo sapiens (human)Potency31.622811
hexokinase-4 isoform 1Homo sapiens (human)Potency10.699233
Histamine H2 receptorCavia porcellus (domestic guinea pig)Potency11.7825214
histone acetyltransferase KAT2A isoform 1Homo sapiens (human)Potency14.9171112
histone deacetylase 9 isoform 3Homo sapiens (human)Potency15.8871211
Histone H2A.xCricetulus griseus (Chinese hamster)Potency30.7562218
histone-lysine N-methyltransferase 2A isoform 2 precursorHomo sapiens (human)Potency17.176716
HLA class I histocompatibility antigen, B alpha chain Homo sapiens (human)Potency8.675214
huntingtin isoform 2Homo sapiens (human)Potency9.575613
hypothetical protein, conservedTrypanosoma bruceiPotency28.443324
hypoxia-inducible factor 1 alpha subunitHomo sapiens (human)Potency33.3931211
hypoxia-inducible factor 1, alpha subunit (basic helix-loop-helix transcription factor)Homo sapiens (human)Potency23.282333
IDH1Homo sapiens (human)Potency7.708214
importin subunit beta-1 isoform 1Homo sapiens (human)Potency43.188327
Inositol hexakisphosphate kinase 1Homo sapiens (human)Potency8.675218
inositol monophosphatase 1Rattus norvegicus (Norway rat)Potency15.640539
Interferon betaHomo sapiens (human)Potency13.5030311
interleukin 8Homo sapiens (human)Potency66.824212
isocitrate dehydrogenase 1, partialHomo sapiens (human)Potency33.008813
lamin isoform A-delta10Homo sapiens (human)Potency9.084013
lethal factor (plasmid)Bacillus anthracis str. A2012Potency14.219114
lethal(3)malignant brain tumor-like protein 1 isoform IHomo sapiens (human)Potency18.801013
LuciferasePhotinus pyralis (common eastern firefly)Potency21.4016421
luciferasePhoturis pensylvanica (Pennsylania firefly)Potency10.863113
luteinizing hormone receptorHomo sapiens (human)Potency84.921411
lysosomal alpha-glucosidase preproproteinHomo sapiens (human)Potency27.720946
M-phase phosphoprotein 8Homo sapiens (human)Potency0.207812
Microtubule-associated protein tauHomo sapiens (human)Potency13.8921214
mitogen-activated protein kinase 1Homo sapiens (human)Potency16.015823
muscleblind-like protein 1 isoform 1Homo sapiens (human)Potency6.902016
Neuronal acetylcholine receptor subunit alpha-4Rattus norvegicus (Norway rat)Potency25.665112
Neuronal acetylcholine receptor subunit beta-2Rattus norvegicus (Norway rat)Potency25.665112
neuropeptide S receptor isoform AHomo sapiens (human)Potency6.015935
nonstructural protein 1Influenza A virus (A/WSN/1933(H1N1))Potency2.794412
NPC intracellular cholesterol transporter 1 precursorHomo sapiens (human)Potency1.608413
nuclear factor erythroid 2-related factor 2 isoform 1Homo sapiens (human)Potency20.0136420
nuclear factor erythroid 2-related factor 2 isoform 2Homo sapiens (human)Potency6.082027
nuclear factor NF-kappa-B p105 subunit isoform 1Homo sapiens (human)Potency39.810711
nuclear factor of kappa light polypeptide gene enhancer in B-cells 1 (p105), isoform CRA_aHomo sapiens (human)Potency34.959828
Nuclear receptor ROR-gammaHomo sapiens (human)Potency11.046812
nuclear receptor ROR-gamma isoform 1Mus musculus (house mouse)Potency11.4807212
nuclear receptor subfamily 1, group I, member 2Rattus norvegicus (Norway rat)Potency8.318612
nuclear receptor subfamily 1, group I, member 3Homo sapiens (human)Potency24.0535336
Ornithine decarboxylaseRattus norvegicus (Norway rat)Potency0.158511
parathyroid hormone/parathyroid hormone-related peptide receptor precursorHomo sapiens (human)Potency11.095712
ParkinHomo sapiens (human)Potency1.584911
peptidyl-prolyl cis-trans isomerase NIMA-interacting 1Homo sapiens (human)Potency40.888726
peripheral myelin protein 22Rattus norvegicus (Norway rat)Potency28.695411
peripheral myelin protein 22 isoform 1Homo sapiens (human)Potency67.455511
peroxisome proliferator activated receptor gammaHomo sapiens (human)Potency31.5857515
peroxisome proliferator-activated receptor deltaHomo sapiens (human)Potency30.8128516
phosphoglycerate kinaseTrypanosoma brucei brucei TREU927Potency13.859636
phosphopantetheinyl transferaseBacillus subtilisPotency46.0230310
Photinus pyralis luciferaseShuttle vector pANFlucPotency16.944111
PINK1Homo sapiens (human)Potency1.584911
plasminogen precursorMus musculus (house mouse)Potency1.748812
polyproteinZika virusPotency10.665412
polyunsaturated fatty acid lipoxygenase ALOX12Homo sapiens (human)Potency18.989513
Polyunsaturated fatty acid lipoxygenase ALOX15BHomo sapiens (human)Potency9.955114
potassium voltage-gated channel subfamily H member 2 isoform dHomo sapiens (human)Potency9.493913
PPM1D proteinHomo sapiens (human)Potency13.423014
pregnane X nuclear receptorHomo sapiens (human)Potency15.6340311
pregnane X receptorRattus norvegicus (Norway rat)Potency29.396912
progesterone receptorHomo sapiens (human)Potency31.7533314
pyruvate kinaseLeishmania mexicana mexicanaPotency19.118024
pyruvate kinase PKM isoform aHomo sapiens (human)Potency32.464824
pyruvate kinase PKM isoform bHomo sapiens (human)Potency0.158522
Rap guanine nucleotide exchange factor 3Homo sapiens (human)Potency59.583324
Rap guanine nucleotide exchange factor 4Homo sapiens (human)Potency81.998523
RAR-related orphan receptor gammaMus musculus (house mouse)Potency18.1632223
ras-related protein Rab-9AHomo sapiens (human)Potency1.316713
regulator of G-protein signaling 4Homo sapiens (human)Potency40.559013
relaxin receptor 1 isoform 1Homo sapiens (human)Potency28.183811
retinoic acid nuclear receptor alpha variant 1Homo sapiens (human)Potency14.5383329
retinoid X nuclear receptor alphaHomo sapiens (human)Potency19.3760319
RGS12Homo sapiens (human)Potency15.848911
runt-related transcription factor 1 isoform AML1bHomo sapiens (human)Potency2.931724
serine-protein kinase ATM isoform aHomo sapiens (human)Potency19.018847
serine/threonine-protein kinase PLK1Homo sapiens (human)Potency12.609413
Single-stranded DNA cytosine deaminaseHomo sapiens (human)Potency79.373524
SMAD family member 2Homo sapiens (human)Potency25.8436315
SMAD family member 3Homo sapiens (human)Potency25.8436315
Smad3Homo sapiens (human)Potency11.713816
snurportin-1Homo sapiens (human)Potency43.188327
Spike glycoproteinSevere acute respiratory syndrome-related coronavirusPotency39.810712
survival motor neuron protein isoform dHomo sapiens (human)Potency5.889615
T cell receptor, partialHomo sapiens (human)Potency4.027612
TAR DNA-binding protein 43Homo sapiens (human)Potency10.619214
TDP1 proteinHomo sapiens (human)Potency7.1767228
thioredoxin glutathione reductaseSchistosoma mansoniPotency45.991913
thioredoxin reductaseRattus norvegicus (Norway rat)Potency45.7179212
ThrombopoietinHomo sapiens (human)Potency3.162322
thyroid hormone receptor beta isoform 2Rattus norvegicus (Norway rat)Potency17.4691328
thyroid hormone receptor beta isoform aHomo sapiens (human)Potency24.7864417
thyroid stimulating hormone receptorHomo sapiens (human)Potency17.2215738
thyrotropin-releasing hormone receptorHomo sapiens (human)Potency21.789324
transcriptional regulator ERG isoform 3Homo sapiens (human)Potency4.928812
TSHR proteinHomo sapiens (human)Potency15.503522
tumor susceptibility gene 101 proteinHomo sapiens (human)Potency14.276335
ubiquitin carboxyl-terminal hydrolase 2 isoform aHomo sapiens (human)Potency9.950536
urokinase plasminogen activator surface receptor precursorMus musculus (house mouse)Potency1.748812
urokinase-type plasminogen activator precursorMus musculus (house mouse)Potency1.748812
USP1 protein, partialHomo sapiens (human)Potency26.219127
v-jun sarcoma virus 17 oncogene homolog (avian)Homo sapiens (human)Potency21.0396217
vitamin D (1,25- dihydroxyvitamin D3) receptorHomo sapiens (human)Potency24.4790517
vitamin D3 receptor isoform VDRAHomo sapiens (human)Potency21.4924110
Voltage-dependent calcium channel gamma-2 subunitMus musculus (house mouse)Potency18.3549110
VprHuman immunodeficiency virus 1Potency16.792114
WRNHomo sapiens (human)Potency52.796814

Inhibition Measurements

ProteinTaxonomyMeasurementAverage (mM)Bioassay(s)Drugs
10 kDa chaperonin Escherichia coliIC500.399024
10 kDa heat shock protein, mitochondrialHomo sapiens (human)IC501.685012
60 kDa chaperoninEscherichia coli K-12IC50205.500012
60 kDa chaperonin Escherichia coliIC500.399024
60 kDa heat shock protein, mitochondrialHomo sapiens (human)IC501.685012
AcetylcholinesteraseHomo sapiens (human)IC5017.263013
AcetylcholinesteraseHomo sapiens (human)Ki4.140023
AcetylcholinesteraseMus musculus (house mouse)Ki0.660011
Acetylcholinesterase Bos taurus (cattle)IC5017.263013
Aldo-keto reductase family 1 member B1Homo sapiens (human)IC5099.250022
Aldo-keto reductase family 1 member B1Rattus norvegicus (Norway rat)IC500.370011
alkaline phosphatase, germ cell type preproproteinHomo sapiens (human)IC50100.000011
alkaline phosphatase, intestinalHomo sapiens (human)IC50100.000011
alkaline phosphatase, tissue-nonspecific isozyme isoform 1 preproproteinHomo sapiens (human)IC5074.800011
Alpha-1A adrenergic receptorRattus norvegicus (Norway rat)IC500.500011
Alpha-1B adrenergic receptorRattus norvegicus (Norway rat)IC500.500011
Alpha-1D adrenergic receptorRattus norvegicus (Norway rat)IC500.500011
Amine oxidase [flavin-containing] AHomo sapiens (human)IC500.070011
Amyloid-beta precursor proteinHomo sapiens (human)IC500.550022
Amyloid-beta precursor proteinHomo sapiens (human)Ki0.963366
Apoptotic peptidase activating factor 1Homo sapiens (human)IC5059.075024
AromataseHomo sapiens (human)IC5010.000011
B1 bradykinin receptorHomo sapiens (human)IC5068.925512
Bcl-2-like protein 1Homo sapiens (human)Ki0.000911
bcrHomo sapiens (human)IC5035.070011
Beta lactamase (plasmid)Pseudomonas aeruginosaIC5020.196234
Beta-secretase 1Homo sapiens (human)IC50500.000011
BZLF2Human herpesvirus 4 type 2 (Epstein-Barr virus type 2)IC500.420011
Carbonic anhydrase 1Homo sapiens (human)Ki5.730022
Carbonic anhydrase 12Homo sapiens (human)Ki9.415022
Carbonic anhydrase 13Mus musculus (house mouse)Ki8.900011
Carbonic anhydrase 14Homo sapiens (human)Ki9.000011
Carbonic anhydrase 15Mus musculus (house mouse)Ki8.400011
Carbonic anhydrase 2Homo sapiens (human)Ki350.000022
Carbonic anhydrase 3Homo sapiens (human)Ki96.000011
Carbonic anhydrase 4Homo sapiens (human)Ki8.300011
Carbonic anhydrase 5A, mitochondrialHomo sapiens (human)Ki5.100011
Carbonic anhydrase 5B, mitochondrialHomo sapiens (human)Ki500.000011
Carbonic anhydrase 6Homo sapiens (human)Ki5.500011
Carbonic anhydrase 7Homo sapiens (human)Ki2.400011
Carbonic anhydrase 9Homo sapiens (human)Ki8.720022
caspase recruitment domain family, member 15Homo sapiens (human)IC5010.895011
caspase-1 isoform alpha precursorHomo sapiens (human)IC50100.000011
caspase-3 isoform a preproproteinHomo sapiens (human)IC5034.900012
caspase-9 isoform alpha precursorHomo sapiens (human)IC5034.900012
catenin beta-1 isoform 1Homo sapiens (human)IC503.730011
Chain A, AcetylcholinesteraseTetronarce californica (Pacific electric ray)Ki0.033111
Chain E, Fibrin beta chainHomo sapiens (human)IC5046.265522
CholinesteraseHomo sapiens (human)IC5017.263013
CholinesteraseHomo sapiens (human)Ki3.247524
Complement component C9Homo sapiens (human)IC500.500011
core protein, partialIC5049.751011
CruzipainTrypanosoma cruziIC5055.250044
Cystathionine beta-synthaseHomo sapiens (human)IC50181.800044
Cystathionine gamma-lyaseHomo sapiens (human)IC5094.50001010
Cystathionine gamma-lyaseMus musculus (house mouse)IC5043.200011
Cystathionine gamma-lyaseHomo sapiens (human)Ki0.600011
Cysteine protease ATG4BHomo sapiens (human)IC5010.475044
Delta-type opioid receptorRattus norvegicus (Norway rat)IC501.800011
Dihydrolipoyl dehydrogenase Plasmodium falciparum (malaria parasite P. falciparum)IC501,000.000011
Dihydrolipoyl dehydrogenase, mitochondrialSus scrofa (pig)IC501,000.000011
DNA damage-inducible transcript 3 proteinMus musculus (house mouse)IC500.870011
DNA polymerase etaHomo sapiens (human)IC500.075011
DNA polymerase iotaHomo sapiens (human)IC500.075011
DNA repair protein RAD52 homologHomo sapiens (human)IC505.000011
DNA topoisomerase 1Homo sapiens (human)IC5036.430012
DNA topoisomerase 2-alphaHomo sapiens (human)IC5028.920011
DNA-(apurinic or apyrimidinic site) endonucleaseHomo sapiens (human)IC503.370033
DNA-3-methyladenine glycosylaseHomo sapiens (human)IC500.200011
Dual specificity mitogen-activated protein kinase kinase 3Homo sapiens (human)IC5014.060011
Ectonucleotide pyrophosphatase/phosphodiesterase family member 2Homo sapiens (human)IC500.922011
Ectonucleotide pyrophosphatase/phosphodiesterase family member 2Homo sapiens (human)Ki0.824011
exodeoxyribonuclease V subunit RecBEscherichia coli str. K-12 substr. MG1655IC5080.908011
exodeoxyribonuclease V subunit RecCEscherichia coli str. K-12 substr. MG1655IC5080.908011
exodeoxyribonuclease V subunit RecDEscherichia coli str. K-12 substr. MG1655IC5080.908011
Exportin-1Homo sapiens (human)IC5025.000011
G-protein coupled receptor 35 isoform aHomo sapiens (human)IC501.370711
Glandular kallikreinSus scrofa (pig)Ki2.700011
glucose-6-phosphate 1-dehydrogenase isoform bHomo sapiens (human)IC5044.700011
glucose-6-phosphate dehydrogenase-6-phosphogluconolactonasePlasmodium bergheiIC5022.000033
Glutathione reductasePlasmodium falciparum 3D7IC506.400011
Glutathione reductase, mitochondrialHomo sapiens (human)IC5016.200022
Glutathione S-transferase PHomo sapiens (human)IC500.051211
Guanine nucleotide-binding protein G(I)/G(S)/G(O) subunit gamma-2Homo sapiens (human)IC500.200011
Guanine nucleotide-binding protein G(I)/G(S)/G(T) subunit beta-1Homo sapiens (human)IC500.200011
Inhibitor of nuclear factor kappa-B kinase subunit betaHomo sapiens (human)IC505.400011
integrase, partialHuman immunodeficiency virus 1IC5019.240522
intestinal alkaline phosphatase precursorMus musculus (house mouse)IC501.550011
Kappa-type opioid receptorCavia porcellus (domestic guinea pig)IC50282.900011
large T antigenBetapolyomavirus macacaeIC501.930011
lens epithelium-derived growth factor p75Homo sapiens (human)IC5019.240522
Luciferin 4-monooxygenasePhotinus pyralis (common eastern firefly)IC5011.040055
matrix metalloproteinase-14 preproproteinHomo sapiens (human)IC5080.000011
metallo beta-lactamasePseudomonas aeruginosaIC5040.852512
metallo-beta-lactamase IMP-1Pseudomonas aeruginosaIC5068.925512
Microtubule-associated protein tauHomo sapiens (human)IC509.425044
Monocarboxylate transporter 4Homo sapiens (human)IC500.730011
Mu-type opioid receptorRattus norvegicus (Norway rat)IC503.300011
Muscarinic acetylcholine receptor M1Homo sapiens (human)Ki500.022022
Muscarinic acetylcholine receptor M2Homo sapiens (human)Ki0.055011
Muscarinic acetylcholine receptor M3Homo sapiens (human)Ki0.030011
Muscarinic acetylcholine receptor M4Homo sapiens (human)Ki0.103011
Muscarinic acetylcholine receptor M5Homo sapiens (human)Ki0.083011
Myc proto-oncogene proteinHomo sapiens (human)IC5014.060011
NACHT, LRR and PYD domains-containing protein 1 isoform 1Homo sapiens (human)IC5019.500011
neutrophil cytosol factor 1Homo sapiens (human)IC500.390011
nonstructural protein 1Influenza A virus (A/California/07/2009(H1N1))IC505.253012
nuclear receptor corepressor 2 isoform 2Homo sapiens (human)IC501.025011
peroxisome proliferator-activated receptor gamma isoform 2Homo sapiens (human)IC501.025011
phospholipase A2, group IIIHomo sapiens (human)IC5040.587011
photoreceptor-specific nuclear receptorHomo sapiens (human)IC5039.841012
Prothrombin Bos taurus (cattle)Ki8.370011
Proto-oncogene tyrosine-protein kinase SrcHomo sapiens (human)IC5030.900011
rac GTPase-activating protein 1 isoform aHomo sapiens (human)IC5015.575022
receptor-interacting serine/threonine-protein kinase 2 isoform 1Homo sapiens (human)IC5010.895011
Replicase polyprotein 1abBetacoronavirus England 1IC50141.000011
Retinal dehydrogenase 1Homo sapiens (human)IC500.760022
Retinal dehydrogenase 1Homo sapiens (human)Ki1.035022
Retinal dehydrogenase 2Homo sapiens (human)IC5010.000011
Reverse transcriptase/RNaseH Human immunodeficiency virus 1IC5051.525044
rho GTPase-activating protein 1Homo sapiens (human)IC5022.080011
Solute carrier organic anion transporter family member 1B1Homo sapiens (human)IC5019.000011
Solute carrier organic anion transporter family member 1B1Homo sapiens (human)Ki18.000011
Solute carrier organic anion transporter family member 1B3Homo sapiens (human)IC5018.000011
Solute carrier organic anion transporter family member 1B3Homo sapiens (human)Ki16.000011
Solute carrier organic anion transporter family member 2B1 Homo sapiens (human)IC5051.000011
Solute carrier organic anion transporter family member 2B1 Homo sapiens (human)Ki20.000011
Sorbitol dehydrogenaseHomo sapiens (human)IC50124.000011
Telomerase reverse transcriptaseHomo sapiens (human)IC5012.200033
Thioredoxin reductase 1, cytoplasmicHomo sapiens (human)IC5030.000011
Thiosulfate sulfurtransferaseHomo sapiens (human)IC5054.350012
toll-like receptor 9Homo sapiens (human)IC508.421011
TransthyretinHomo sapiens (human)IC5011.000011
Tyrosine-protein phosphatase 1Saccharomyces cerevisiae S288CIC501.200011
Tyrosine-protein phosphatase non-receptor type 1Homo sapiens (human)IC501.300011
Tyrosyl-DNA phosphodiesterase 1Homo sapiens (human)IC500.017022
Vesicular glutamate transporter 3Rattus norvegicus (Norway rat)Ki0.040011
XBP1Homo sapiens (human)IC502.400011

Activation Measurements

ProteinTaxonomyMeasurementAverage (mM)Bioassay(s)Drugs
AlbuminHomo sapiens (human)Kd2.500011
Cell division protein FtsZEscherichia coli K-12Kd16.600011
Cystathionine gamma-lyaseHomo sapiens (human)Kd3.400011
G-protein coupled receptor 55Homo sapiens (human)EC500.500011
Hsf1 proteinMus musculus (house mouse)EC50260.000011
Immunoglobulin lambda variable 6-57Homo sapiens (human)EC505.666723
karyopherin alpha 2 (RAG cohort 1, importin alpha 1), isoform CRA_bHomo sapiens (human)EC50119.500011
Microtubule-associated protein tauHomo sapiens (human)EC500.360022
NPYLR7BAedes aegypti (yellow fever mosquito)EC504.830011
POsterior SegregationCaenorhabditis elegansEC50186.681011
recombinase AMycobacterium tuberculosis H37RvEC5078.650022
regulator of G-protein signaling 16Homo sapiens (human)EC506.670011
regulator of G-protein signaling 19Homo sapiens (human)EC5030.000011
regulator of G-protein signaling 4Homo sapiens (human)EC503.410011
RGS7, partialHomo sapiens (human)EC5030.000011
Serine/threonine-protein kinase mTORHomo sapiens (human)Kd130.000011
Sodium-dependent noradrenaline transporter Homo sapiens (human)EC50113.886011
streptokinase A precursorStreptococcus pyogenes M1 GASEC502.154011
Tyrosine-protein kinase LckHomo sapiens (human)Kd2.500011
Zinc finger protein mex-5Caenorhabditis elegansEC50113.886011

Other Measurements

ProteinTaxonomyMeasurementAverage (mM)Bioassay(s)Drugs
AlbuminBos taurus (cattle)Kdiss2.900011
aryl hydrocarbon receptor nuclear translocatorHomo sapiens (human)AC500.734011
ATP-dependent translocase ABCB1Homo sapiens (human)Ki10.110011
ATP-dependent translocase ABCB1Homo sapiens (human)Ki23.400011
Broad substrate specificity ATP-binding cassette transporter ABCG2Homo sapiens (human)Kact4.500011
Canalicular multispecific organic anion transporter 1Rattus norvegicus (Norway rat)Km3.700011
Caspase 6, apoptosis-related cysteine peptidaseHomo sapiens (human)AC501.600011
CDK5Homo sapiens (human)AC5012.323011
Cell death-related nuclease 4Caenorhabditis elegansINH100.000011
Cell division protein FtsZEscherichia coli K-12Km29.400011
Cyclin-dependent kinase 5, regulatory subunit 1 (p35)Homo sapiens (human)AC5012.323011
Cystathionine gamma-lyaseHomo sapiens (human)alphaKi4.200011
Dihydrolipoyl dehydrogenase Plasmodium falciparum (malaria parasite P. falciparum)Km49.000011
Dihydrolipoyl dehydrogenase, mitochondrialSus scrofa (pig)Km28.000011
DNA repair protein RAD52 homolog isoform aHomo sapiens (human)AC500.936011
DNA topoisomerase 2-betaHomo sapiens (human)Ka0.274012
FAD-linked sulfhydryl oxidase ALRHomo sapiens (human)AC500.522011
Glucocorticoid receptorHomo sapiens (human)Kis453.000011
Glutathione reductase, mitochondrialHomo sapiens (human)Km6.300011
glycogen synthase kinase-3 alphaHomo sapiens (human)AC5024.610011
heat shock protein 90, putativePlasmodium falciparum 3D7AC500.735011
heat shock protein HSP 90-alpha isoform 2Homo sapiens (human)AC500.570011
histone-lysine N-methyltransferase NSD2 isoform 1Homo sapiens (human)AC5010.505012
Hsf1 proteinMus musculus (house mouse)AbsAC40_uM26.000011
kelch-like ECH-associated protein 1Homo sapiens (human)AC502.800011
kelch-like ECH-associated protein 1Homo sapiens (human)Max_Activity_Concentration_uM 1.600011
Multidrug resistance-associated protein 1 Homo sapiens (human)Km97.333333
nuclear factor erythroid 2-related factor 2 isoform 2Homo sapiens (human)AC502.800011
Nuclear factor NF-kappa-B p105 subunitHomo sapiens (human)Concentration100.000011
protein AF-9 isoform aHomo sapiens (human)AC502.116512
replicative DNA helicaseMycobacterium tuberculosis H37RvAC5058.180022
Ribonuclease TEscherichia coli K-12INH10.000011
Thioredoxin reductase 1, cytoplasmicHomo sapiens (human)Km95.000011
transforming acidic coiled-coil-containing protein 3Homo sapiens (human)AC500.734011