Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
histamine | Homo sapiens (human) | AC50 | 23.0800 | 1 | 0 |
iodoquinol | Homo sapiens (human) | AC50 | 7.4600 | 1 | 0 |
doxorubicin hydrochloride | Homo sapiens (human) | AC50 | 74.4900 | 1 | 0 |
aminoimidazole carboxamide | Homo sapiens (human) | AC50 | 90.4600 | 1 | 0 |
ethyl violet | Homo sapiens (human) | AC50 | 0.7340 | 1 | 0 |
nsc 3852 | Homo sapiens (human) | AC50 | 13.5500 | 1 | 0 |
benserazide hydrochloride | Homo sapiens (human) | AC50 | 13.3100 | 1 | 0 |
Nanaomycin | Homo sapiens (human) | AC50 | 46.9300 | 1 | 0 |
2-(2'-pyridyl)benzimidazole | Homo sapiens (human) | AC50 | 43.9700 | 1 | 0 |
2-(4-hydroxyphenyl)-5,6,7,8-tetrahydroxy-4H-1-benzopyran-4-one | Homo sapiens (human) | AC50 | 63.0200 | 1 | 0 |
8-(methylsulfonylamino)quinoline | Homo sapiens (human) | AC50 | 38.2400 | 1 | 0 |
1-benzylimidazole-4,5-dicarboxylic acid | Homo sapiens (human) | AC50 | 13.7600 | 1 | 0 |
carboline-3-carboxylic acid | Homo sapiens (human) | AC50 | 1.8000 | 1 | 0 |
colchiceine | Homo sapiens (human) | AC50 | 40.7700 | 1 | 0 |
3,6-bis(2-pyridyl)-1,2,4,5-tetrazine | Homo sapiens (human) | AC50 | 28.8400 | 1 | 0 |
dicentrine | Homo sapiens (human) | AC50 | 17.6200 | 1 | 0 |
trimethylcolchicinic acid | Homo sapiens (human) | AC50 | 29.7200 | 1 | 0 |
5-(1,3-benzodioxol-5-yl)-1-methyl-2-imidazolamine | Homo sapiens (human) | AC50 | 38.9900 | 1 | 0 |
L-histidine 2-naphthylamide | Homo sapiens (human) | AC50 | 44.1800 | 1 | 0 |
3-pyridinecarboxylic acid (5-chloro-8-quinolinyl) ester | Homo sapiens (human) | AC50 | 9.5800 | 1 | 0 |
2-(8-quinolinylthio)acetic acid phenacyl ester | Homo sapiens (human) | AC50 | 37.3200 | 1 | 0 |
6-(4-morpholinyl)naphthalene-2,3-dicarbonitrile | Homo sapiens (human) | AC50 | 115.5100 | 1 | 0 |
1,6-dimethyl-3-(2-pyridinyl)pyrimido[5,4-e][1,2,4]triazine-5,7-dione | Homo sapiens (human) | AC50 | 0.5000 | 1 | 0 |
1-(1-pyrrolidinyl)-2-(8-quinolinylthio)ethanone | Homo sapiens (human) | AC50 | 3.2800 | 1 | 0 |
N-[5-(2-chlorophenyl)-1,3,4-oxadiazol-2-yl]-3-pyridinecarboxamide | Homo sapiens (human) | AC50 | 15.7900 | 1 | 0 |
4-(2,6-dimethylphenoxy)-5-methoxy-2-(2-pyridinyl)pyrimidine | Homo sapiens (human) | AC50 | 8.7400 | 1 | 0 |
2-(5-methyl-3-oxo-1H-pyrazol-2-yl)-6-oxo-1H-pyrimidine-5-carboxylic acid ethyl ester | Homo sapiens (human) | AC50 | 0.7540 | 1 | 0 |
N-(5-cyclopropyl-1,3,4-oxadiazol-2-yl)-4-[(4-methyl-1-piperidinyl)sulfonyl]benzamide | Homo sapiens (human) | AC50 | 16.6900 | 1 | 0 |
4-(4-morpholinylsulfonyl)-N-(5-thiophen-2-yl-1,3,4-oxadiazol-2-yl)benzamide | Homo sapiens (human) | AC50 | 17.0900 | 1 | 0 |
6-[[(2-chlorophenyl)methyl-methylamino]methyl]-N2-(2-methylphenyl)-1,3,5-triazine-2,4-diamine | Homo sapiens (human) | AC50 | 53.4600 | 1 | 0 |
N-[4-(2-pyridinyl)-2-thiazolyl]cyclopentanecarboxamide | Homo sapiens (human) | AC50 | 15.5500 | 1 | 0 |
2-[3-(4-pyridyl)-1H-1,2,4-triazol-5-yl]pyridine | Homo sapiens (human) | AC50 | 1.1160 | 2 | 0 |
N-[2-furanyl-(8-hydroxy-7-quinolinyl)methyl]-2-methylpropanamide | Homo sapiens (human) | AC50 | 0.7045 | 2 | 0 |
5-chloro-7-[3-pyridinyl-(2-pyridinylamino)methyl]-8-quinolinol | Homo sapiens (human) | AC50 | 5.6700 | 1 | 0 |
N-[1-oxo-1-[[4-(2-pyridinyl)-2-thiazolyl]amino]propan-2-yl]-2-furancarboxamide | Homo sapiens (human) | AC50 | 4.5200 | 1 | 0 |
3-[5-[bis(3-methyl-5-oxo-1,2-dihydropyrazol-4-yl)methyl]-2-furanyl]benzoic acid methyl ester | Homo sapiens (human) | AC50 | 87.9100 | 1 | 0 |
N-cycloheptyl-3-(5,7-dioxo-6-pyrrolo[3,4-b]pyridinyl)propanamide | Homo sapiens (human) | AC50 | 76.8900 | 1 | 0 |
2-pyridinecarboxylic acid [2-(5-chloro-2-thiophenyl)-2-oxoethyl] ester | Homo sapiens (human) | AC50 | 18.8300 | 1 | 0 |
5-chloro-7-[1-piperidinyl(2-pyridinyl)methyl]-8-quinolinol | Homo sapiens (human) | AC50 | 1.3300 | 1 | 0 |
5-chloro-7-[(4-ethyl-1-piperazinyl)-(3-pyridinyl)methyl]-8-quinolinol | Homo sapiens (human) | AC50 | 4.0300 | 1 | 0 |
4-chloro-N-[5-(2,3-dihydro-1,4-dioxin-5-yl)-1,3,4-oxadiazol-2-yl]benzamide | Homo sapiens (human) | AC50 | 17.6700 | 1 | 0 |
5-methyl-4-[(3-methyl-5-oxo-1,2-dihydropyrazol-4-yl)-[1-(1-naphthalenylmethyl)-3-indolyl]methyl]-1,2-dihydropyrazol-3-one | Homo sapiens (human) | AC50 | 19.8600 | 1 | 0 |
N-(5-cyclopropyl-1,3,4-oxadiazol-2-yl)-4-[(3-methyl-1-piperidinyl)sulfonyl]benzamide | Homo sapiens (human) | AC50 | 31.9500 | 1 | 0 |
5-nitro-2-thiophenecarboxylic acid [2-oxo-2-[(phenylmethyl)amino]ethyl] ester | Homo sapiens (human) | AC50 | 37.0400 | 1 | 0 |
N-(5-cyclopropyl-1,3,4-thiadiazol-2-yl)-2-(2-fluorophenyl)sulfonyl-3,4-dihydro-1H-isoquinoline-3-carboxamide | Homo sapiens (human) | AC50 | 30.9800 | 1 | 0 |
1-(4-morpholinyl)-2-[[3-(2-pyridinyl)-[1,2,4]triazolo[4,3-b]pyridazin-6-yl]thio]ethanone | Homo sapiens (human) | AC50 | 21.2600 | 1 | 0 |
centaureidin | Homo sapiens (human) | AC50 | 101.2800 | 1 | 0 |
N-methyl-6-phenyl-3-(2-pyridinyl)-1,2,4-triazin-5-amine | Homo sapiens (human) | AC50 | 0.5000 | 1 | 0 |
3-(2-pyridinyl)-6-(2-pyridinylmethylthio)pyridazine | Homo sapiens (human) | AC50 | 0.8950 | 1 | 0 |
N-(4-acetylphenyl)-2-[[3-(2-pyridinyl)-[1,2,4]triazolo[4,3-b]pyridazin-6-yl]thio]acetamide | Homo sapiens (human) | AC50 | 18.1900 | 1 | 0 |
N-cyclohexyl-2-[[6-(2-pyridinyl)-3-pyridazinyl]thio]acetamide | Homo sapiens (human) | AC50 | 2.0950 | 2 | 0 |
N-cyclopentyl-2-[[6-(2-pyridinyl)-3-pyridazinyl]thio]acetamide | Homo sapiens (human) | AC50 | 2.6400 | 1 | 0 |
R-(-)-actinodaphnine | Homo sapiens (human) | AC50 | 27.6600 | 1 | 0 |
8-{1-[4-(dimethylamino)phenyl]-3-(pyrrolidin-1-yl)propyl}-5,7-dimethoxy-4-pentyl-2H-chromen-2-one | Homo sapiens (human) | AC50 | 6.8600 | 1 | 0 |
5-[[4-(4-methyl-1-piperazinyl)-1-piperidinyl]methyl]-8-quinolinol | Homo sapiens (human) | AC50 | 2.3000 | 1 | 0 |
ml228 probe | Homo sapiens (human) | AC50 | 1.6000 | 1 | 0 |