Page last updated: 2024-08-07 22:59:07

kelch-like ECH-associated protein 1

[no definition available]

Synonyms

Research

Bioassay Publications (0)

TimeframeStudies on this Protein(%)All Drugs %
pre-19900 (0)18.7374
1990's0 (0)18.2507
2000's0 (0)29.6817
2010's0 (0)24.3611
2020's0 (0)2.80

Compounds (26)

Drugs with Other Measurements

DrugTaxonomyMeasurementAverage (mM)Bioassay(s)Publication(s)
dipyridamoleHomo sapiens (human)AC504.030010
dipyridamoleHomo sapiens (human)Max_Activity_Concentration_uM 50.000010
fusaric acidHomo sapiens (human)Max_Activity_Concentration_uM 0.380010
ns 1619Homo sapiens (human)Max_Activity_Concentration_uM 26.000010
alizarinHomo sapiens (human)AC5052.000010
alizarinHomo sapiens (human)Max_Activity_Concentration_uM 26.000010
5-amino-2-naphthalenesulfonateHomo sapiens (human)Max_Activity_Concentration_uM 12.000010
2,4-dihydroxybenzophenoneHomo sapiens (human)AC5011.130010
2,4-dihydroxybenzophenoneHomo sapiens (human)Max_Activity_Concentration_uM 6.000010
3-aminofluorantheneHomo sapiens (human)AC502.010010
3-aminofluorantheneHomo sapiens (human)Max_Activity_Concentration_uM 50.000010
3-aminofluorantheneHomo sapiens (human)Max_Concentration(uM) 6.000010
s-2678Homo sapiens (human)AC5052.000010
s-2678Homo sapiens (human)Max_Activity_Concentration_uM 50.000010
s-2678Homo sapiens (human)Max_Concentration(uM) 50.000010
topotecan hydrochlorideHomo sapiens (human)AC503.700010
topotecan hydrochlorideHomo sapiens (human)Max_Activity_Concentration_uM 0.380010
coumarin 153Homo sapiens (human)AC502.800010
coumarin 153Homo sapiens (human)Max_Activity_Concentration_uM 1.600010
agroclavineHomo sapiens (human)AC5038.410010
agroclavineHomo sapiens (human)Max_Activity_Concentration_uM 50.000010
brazilinHomo sapiens (human)Max_Activity_Concentration_uM 0.380010
raubasineHomo sapiens (human)AC5052.000010
raubasineHomo sapiens (human)Max_Activity_Concentration_uM 26.000010
n,n-dimethyldaunorubicinHomo sapiens (human)AC5052.000010
n,n-dimethyldaunorubicinHomo sapiens (human)Max_Activity_Concentration_uM 50.000010
doxorubicin hydrochlorideHomo sapiens (human)AC5043.410010
doxorubicin hydrochlorideHomo sapiens (human)Max_Activity_Concentration_uM 50.000010
3-[3,4-dihydro-1H-isoquinolin-2-yl-[1-(2-methylbutan-2-yl)-5-tetrazolyl]methyl]-7-methoxy-1H-quinolin-2-oneHomo sapiens (human)Max_Activity_Concentration_uM 6.000010
3-[3,4-dihydro-1H-isoquinolin-2-yl-[1-(2-methylbutan-2-yl)-5-tetrazolyl]methyl]-7-methoxy-1H-quinolin-2-oneHomo sapiens (human)Max_Concentration(uM) 26.000010
N-(2-oxolanylmethyl)-1-phenyl-4-pyrazolo[3,4-d]pyrimidinamineHomo sapiens (human)Max_Activity_Concentration_uM 0.800010
2-cyano-2-[3-(4-morpholinyl)-2-quinoxalinyl]acetic acid hexyl esterHomo sapiens (human)Max_Activity_Concentration_uM 0.800010
N-(4-amino-2-oxo-1-benzopyran-3-yl)acetamideHomo sapiens (human)Max_Activity_Concentration_uM 0.800010
N-(4-amino-2-oxo-1-benzopyran-3-yl)acetamideHomo sapiens (human)Max_Concentration(uM) 50.000010
3-amino-N-(2-fluorophenyl)-6-(phenylmethyl)-4-(trifluoromethyl)-2-thieno[2,3-b]pyridinecarboxamideHomo sapiens (human)Max_Activity_Concentration_uM 12.000010
2-[[2-[(3,7-dimethyl-2-quinolinyl)thio]-1-oxoethyl]amino]-4,5-dimethoxybenzoic acidHomo sapiens (human)Max_Activity_Concentration_uM 3.000010
2-[[2-[(3,7-dimethyl-2-quinolinyl)thio]-1-oxoethyl]amino]-4,5-dimethoxybenzoic acidHomo sapiens (human)Max_Concentration(uM) 50.000010
N-(3-chlorophenyl)-2-[[2-(2-pyridinyl)-2,3-dihydro-1,3,4-thiadiazol-5-yl]thio]acetamideHomo sapiens (human)Max_Activity_Concentration_uM 3.000010
2-(3-hydroxyphenyl)-6-(1-piperidinyl)benzo[de]isoquinoline-1,3-dioneHomo sapiens (human)Max_Activity_Concentration_uM 0.800010
2-(3-hydroxyphenyl)-6-(1-piperidinyl)benzo[de]isoquinoline-1,3-dioneHomo sapiens (human)Max_Concentration(uM) 50.000010
6-amino-3-methyl-4-(2-methylpropyl)-2,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrileHomo sapiens (human)Max_Activity_Concentration_uM 0.380010
6-amino-3-methyl-4-(2-methylpropyl)-2,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrileHomo sapiens (human)Max_Concentration(uM) 50.000010
LSM-24581Homo sapiens (human)Max_Activity_Concentration_uM 0.380010
LSM-24581Homo sapiens (human)Max_Concentration(uM) 50.000010
(1S,2R)-2-[[(1S)-1-[(1,3-dioxo-2-isoindolyl)methyl]-3,4-dihydro-1H-isoquinolin-2-yl]-oxomethyl]-1-cyclohexanecarboxylic acidHomo sapiens (human)AbsAC40_uM13.185010
(1S,2R)-2-[[(1S)-1-[(1,3-dioxo-2-isoindolyl)methyl]-3,4-dihydro-1H-isoquinolin-2-yl]-oxomethyl]-1-cyclohexanecarboxylic acidHomo sapiens (human)AC502.496730
(1S,2R)-2-[[(1S)-1-[(1,3-dioxo-2-isoindolyl)methyl]-3,4-dihydro-1H-isoquinolin-2-yl]-oxomethyl]-1-cyclohexanecarboxylic acidHomo sapiens (human)Max_Delta_Tm_Conc_uM19.500010