Proteins > TSHR protein
Page last updated: 2024-08-07 20:58:48

TSHR protein

[no definition available]

Synonyms

Research

Bioassay Publications (0)

TimeframeStudies on this Protein(%)All Drugs %
pre-19900 (0)18.7374
1990's0 (0)18.2507
2000's0 (0)29.6817
2010's0 (0)24.3611
2020's0 (0)2.80

Compounds (59)

Drugs with Potency Measurements

DrugTaxonomyMeasurementAverage (mM)Bioassay(s)Publication(s)
dichlorophenHomo sapiens (human)Potency30.131310
hexachloropheneHomo sapiens (human)Potency2.133110
niclosamideHomo sapiens (human)Potency92.537420
methylene blueHomo sapiens (human)Potency15.503520
strophanthidinHomo sapiens (human)Potency0.849210
bisphenol a-glycidyl methacrylateHomo sapiens (human)Potency21.331310
2,4-diacetylphloroglucinolHomo sapiens (human)Potency30.131310
1,6-bismaleimidohexaneHomo sapiens (human)Potency37.933020
clioxanideHomo sapiens (human)Potency1.901210
rafoxanideHomo sapiens (human)Potency1.510110
closantelHomo sapiens (human)Potency2.133110
lobaric acidHomo sapiens (human)Potency25.376020
4-(2-thiazolylazo)resorcinolHomo sapiens (human)Potency75.686310
nsc 95397Homo sapiens (human)Potency96.747920
nsc228155Homo sapiens (human)Potency304.845020
2,3-dichloro-5,8-dimethoxy-1,4-naphthoquinoneHomo sapiens (human)Potency33.807810
N-[1-[(2-bromophenyl)methyl]-2-oxo-3-pyridinyl]butanamideHomo sapiens (human)Potency75.686310
3-chloro-4-[4-(4-fluorophenyl)sulfonyl-1-piperazinyl]-N,N-dimethylbenzenesulfonamideHomo sapiens (human)Potency47.754810
1-[(3,4-dimethoxyphenyl)-[1-(thiophen-2-ylmethyl)-5-tetrazolyl]methyl]-4-phenylpiperazineHomo sapiens (human)Potency16.944110
2',2'-dimethyl-3-spiro[5,6,7,8a-tetrahydrothiazolo[3,2-a]pyridine-8,4'-thiane]oneHomo sapiens (human)Potency16.944110
4-chloro-1-methyl-3-nitro-2-quinolinoneHomo sapiens (human)Potency30.131310
4-chloro-1-ethyl-3-nitro-2-quinolinoneHomo sapiens (human)Potency75.686310
1-(1-naphthalenylmethoxy)benzotriazoleHomo sapiens (human)Potency151.014010
N-[[3-chloro-4-(4-morpholinyl)anilino]-sulfanylidenemethyl]-2-(4-methoxyphenoxy)acetamideHomo sapiens (human)Potency19.011510
3-chloro-4-[2-(3,4-dimethoxyphenyl)ethylamino]-1-(2-phenylethyl)pyrrole-2,5-dioneHomo sapiens (human)Potency26.854510
2-amino-4-[(4-bromophenyl)methylthio]-3-azaspiro[5.5]undeca-1,4-diene-1,5-dicarbonitrileHomo sapiens (human)Potency23.934110
4-(dimethylsulfamoyl)-N-(4-thiophen-2-yl-2-thiazolyl)benzamideHomo sapiens (human)Potency10.456420
6-fluoro-2-(2-methylphenyl)-1,2-benzothiazol-3-oneHomo sapiens (human)Potency19.011510
SMER 28Homo sapiens (human)Potency42.561510
2-[(6-amino-3,5-dicyano-4-thiophen-2-yl-2-pyridinyl)thio]-N-[(2-methoxyphenyl)methyl]acetamideHomo sapiens (human)Potency37.933010
3-[2-oxo-2-[4-(phenylmethyl)-1-piperidinyl]ethyl]-1,3-diazaspiro[4.6]undecane-2,4-dioneHomo sapiens (human)Potency21.331310
1-[(2-chlorophenyl)methyl]-3-methyl-N-(4-methyl-2-thiazolyl)-5-thieno[2,3-c]pyrazolecarboxamideHomo sapiens (human)Potency75.686310
1-(4-bromo-2-fluorophenyl)-3-(3-chlorophenyl)ureaHomo sapiens (human)Potency16.011220
3-[[[4-(phenylmethyl)-5-thiophen-2-yl-1,2,4-triazol-3-yl]thio]methyl]-1,2,3-benzotriazin-4-oneHomo sapiens (human)Potency47.754810
12-oxo-N-(4-phenyl-2-thiazolyl)-7,8,9,10-tetrahydro-6H-azepino[2,1-b]quinazoline-3-carboxamideHomo sapiens (human)Potency8.857620
2-[4-[benzenesulfonyl(methyl)amino]phenoxy]-N-(1,3-benzothiazol-2-yl)acetamideHomo sapiens (human)Potency379.330010
LSM-28486Homo sapiens (human)Potency37.933010
6-(2,3-dihydro-1,4-benzodioxin-3-ylmethylamino)-N-ethyl-N-phenyl-3-pyridinesulfonamideHomo sapiens (human)Potency37.933010
2-[[2,2,2-trichloro-1-[(2-methyl-1-oxopropyl)amino]ethyl]amino]-5,6-dihydro-4H-cyclopenta[b]thiophene-3-carboxylic acid ethyl esterHomo sapiens (human)Potency47.754810
2-(4-chlorophenoxy)-N-(5-nitro-2-thiazolyl)acetamideHomo sapiens (human)Potency9.528310
N-[[3-[(3-chlorophenyl)sulfamoyl]-4-methylanilino]-sulfanylidenemethyl]-4-fluorobenzamideHomo sapiens (human)Potency30.131310
2-[2-[5-amino-4-(3-thiophenyl)-1-pyrazolyl]-4-phenyl-5-thiazolyl]acetic acidHomo sapiens (human)Potency37.933010
3,3-bis(4-hydroxyphenyl)-7-methyl-1,3-dihydro-2h-indol-2-oneHomo sapiens (human)Potency75.686310
2-(1H-benzimidazol-2-ylthio)-1-[2,5-dimethyl-1-(2-oxolanylmethyl)-3-pyrrolyl]ethanoneHomo sapiens (human)Potency21.331310
N-[3-[(2-methoxyphenyl)sulfamoyl]phenyl]-2-quinolinecarboxamideHomo sapiens (human)Potency239.341010
2-[[3-(3-oxo-1,2-benzothiazol-2-yl)phenyl]sulfonylamino]benzoic acidHomo sapiens (human)Potency23.934110
digitoxigeninHomo sapiens (human)Potency0.477510
3-[2,2-dichloro-1-(3-fluoro-4-methylphenyl)ethyl]-1,1-bis(phenylmethyl)ureaHomo sapiens (human)Potency75.686310
N-[4-chloro-3-[(4-chlorophenyl)sulfamoyl]phenyl]-4-propan-2-yloxybenzamideHomo sapiens (human)Potency21.331310
4-cyano-N-[4-thiophen-2-yl-5-(2,2,2-trifluoro-1-oxoethyl)-2-thiazolyl]benzamideHomo sapiens (human)Potency6.012010
N-[4-chloro-3-(4-morpholinylsulfonyl)phenyl]-4-(2-oxolanylmethoxy)benzamideHomo sapiens (human)Potency14.280220
[(10R,13S,17R)-17-Ethynyl-13-methyl-3-oxo-1,2,6,7,8,9,10,11,12,14,15,16-dodecahydrocyclopenta[a]phenanthren-17-yl] acetateHomo sapiens (human)Potency13.459110
quinaldine redHomo sapiens (human)Potency314.026220
lasalocid sodiumHomo sapiens (human)Potency4.775510
calcimycinHomo sapiens (human)Potency11.505320
4-(5-methyl-3-nitro-1-pyrazolyl)-N-[3-(4-methylphenoxy)-5-nitrophenyl]butanamideHomo sapiens (human)Potency75.686310
5-chloro-2-[(4-methylphenyl)methylsulfonyl]-N-(5-propan-2-yl-1,3,4-thiadiazol-2-yl)-4-pyrimidinecarboxamideHomo sapiens (human)Potency20.439120
2-[(6-chloro-3-pyridinyl)sulfonylamino]-N-[(4-methylphenyl)methyl]benzamideHomo sapiens (human)Potency119.955010
5-[(2-bromophenyl)methyl]-1-tert-butyl-4-pyrazolo[3,4-d]pyrimidinoneHomo sapiens (human)Potency47.754810