| Assay ID | Title | Year | Journal | Article |
|---|
| AID365749 | Inhibition of Syk phosphorylation in antigen-stimulated rat RBL-2H3 cells at 50 uM by Western blot analysis in presence of dinitrophenylated bovine serum albumin | 2008 | Bioorganic & medicinal chemistry, Aug-15, Volume: 16, Issue:16
| Inhibitory effects of polymethoxy flavones isolated from Citrus reticulate on degranulation in rat basophilic leukemia RBL-2H3: enhanced inhibition by their combination. |
| AID365748 | Inhibition of Lyn phosphorylation in antigen-stimulated rat RBL-2H3 cells at 50 uM by Western blot analysis in presence of dinitrophenylated bovine serum albumin | 2008 | Bioorganic & medicinal chemistry, Aug-15, Volume: 16, Issue:16
| Inhibitory effects of polymethoxy flavones isolated from Citrus reticulate on degranulation in rat basophilic leukemia RBL-2H3: enhanced inhibition by their combination. |
| AID332775 | Antimicrobial activity against Escherichia coli ATCC 8739 by paper disk method | | | |
| AID1411741 | Inhibition of human recombinant CYP1B1 expressed in HEK293 cells using 7-ethoxyresorufin substrate substrate preincubated for 30 mins followed by substrate addition and measured after 60 mins by fluorescence assay relative to control | 2018 | MedChemComm, Feb-01, Volume: 9, Issue:2
| Identification of karanjin isolated from the Indian beech tree as a potent CYP1 enzyme inhibitor with cellular efficacy |
| AID1230328 | Displacement of [3H]-CP55940 from human CB1 receptor transfected into HEK293 cells at 10 uM by microplate scintillation counting | 2015 | Journal of natural products, Jun-26, Volume: 78, Issue:6
| Flavonoids from Perovskia atriplicifolia and Their in Vitro Displacement of the Respective Radioligands for Human Opioid and Cannabinoid Receptors. |
| AID365751 | Inhibition of ERK1/2 phosphorylation in antigen-stimulated rat RBL-2H3 cells at 50 uM by Western blot analysis in presence of dinitrophenylated bovine serum albumin | 2008 | Bioorganic & medicinal chemistry, Aug-15, Volume: 16, Issue:16
| Inhibitory effects of polymethoxy flavones isolated from Citrus reticulate on degranulation in rat basophilic leukemia RBL-2H3: enhanced inhibition by their combination. |
| AID288087 | Apoptotic activity in HL60 cells after 24 hrs | 2007 | Bioorganic & medicinal chemistry, May-15, Volume: 15, Issue:10
| Isolation and syntheses of polymethoxyflavones and hydroxylated polymethoxyflavones as inhibitors of HL-60 cell lines. |
| AID1546536 | Cytotoxicity against human HeLa cells assessed as reduction in cell viability incubated for 48 hrs by MTT assay | 2020 | Bioorganic & medicinal chemistry, 01-01, Volume: 28, Issue:1
| Artemisia: a promising plant for the treatment of cancer. |
| AID365753 | Inhibition of p38 MAPK phosphorylation in antigen-stimulated rat RBL-2H3 cells at 50 uM by Western blot analysis in presence of dinitrophenylated bovine serum albumin | 2008 | Bioorganic & medicinal chemistry, Aug-15, Volume: 16, Issue:16
| Inhibitory effects of polymethoxy flavones isolated from Citrus reticulate on degranulation in rat basophilic leukemia RBL-2H3: enhanced inhibition by their combination. |
| AID1411736 | Inhibition of recombinant human CYP2C9 expressed in baker's yeast-derived microsomes (Sacchrosomes) at 10 uM using 3-cyano-7-ethoxycoumarin substrate by EROD assay relative to control | 2018 | MedChemComm, Feb-01, Volume: 9, Issue:2
| Identification of karanjin isolated from the Indian beech tree as a potent CYP1 enzyme inhibitor with cellular efficacy |
| AID1411738 | Inhibition of human recombinant CYP1A1 expressed in HEK293 cells at 10 uM using 7-ethoxyresorufin substrate preincubated for 30 mins followed by substrate addition and measured after 60 mins by fluorescence assay relative to control | 2018 | MedChemComm, Feb-01, Volume: 9, Issue:2
| Identification of karanjin isolated from the Indian beech tree as a potent CYP1 enzyme inhibitor with cellular efficacy |
| AID332774 | Antimicrobial activity against Pseudomonas aeruginosa ATCC 1539 by paper disk method | | | |
| AID365747 | Antioxidant activity assessed as DPPH radical scavenging activity | 2008 | Bioorganic & medicinal chemistry, Aug-15, Volume: 16, Issue:16
| Inhibitory effects of polymethoxy flavones isolated from Citrus reticulate on degranulation in rat basophilic leukemia RBL-2H3: enhanced inhibition by their combination. |
| AID361717 | Suppression of degranulation in IgE-sensitized rat RBL-2H3 cells assessed as inhibition of antigen-stimulated histamine release after 30 mins in presence of dinitrophenylated bovine serum albumin | 2008 | Bioorganic & medicinal chemistry, Aug-15, Volume: 16, Issue:16
| Inhibitory effects of polymethoxy flavones isolated from Citrus reticulate on degranulation in rat basophilic leukemia RBL-2H3: enhanced inhibition by their combination. |
| AID1546537 | Cytotoxicity against human MCF7 cells assessed as reduction in cell viability incubated for 48 hrs by MTT assay | 2020 | Bioorganic & medicinal chemistry, 01-01, Volume: 28, Issue:1
| Artemisia: a promising plant for the treatment of cancer. |
| AID1411739 | Inhibition of human recombinant CYP1A1 expressed in HEK293 cells using 7-ethoxyresorufin substrate preincubated for 30 mins followed by substrate addition and measured after 60 mins by fluorescence assay relative to control | 2018 | MedChemComm, Feb-01, Volume: 9, Issue:2
| Identification of karanjin isolated from the Indian beech tree as a potent CYP1 enzyme inhibitor with cellular efficacy |
| AID1230329 | Displacement of [3H]-CP55940 from human CB2 receptor transfected into HEK293 cells at 10 uM by microplate scintillation counting | 2015 | Journal of natural products, Jun-26, Volume: 78, Issue:6
| Flavonoids from Perovskia atriplicifolia and Their in Vitro Displacement of the Respective Radioligands for Human Opioid and Cannabinoid Receptors. |
| AID365750 | Inhibition of PLC-gamma-1/gamma-2 phosphorylation in antigen-stimulated rat RBL-2H3 cells at 50 uM by Western blot analysis in presence of dinitrophenylated bovine serum albumin | 2008 | Bioorganic & medicinal chemistry, Aug-15, Volume: 16, Issue:16
| Inhibitory effects of polymethoxy flavones isolated from Citrus reticulate on degranulation in rat basophilic leukemia RBL-2H3: enhanced inhibition by their combination. |
| AID381260 | Cytotoxicity against human KB cells | | | |
| AID1411744 | Inhibition of human recombinant CYP2C19 expressed in HEK293 cells using 3-cyano-7-ethoxycoumarin substrate substrate preincubated for 30 mins followed by substrate addition and measured after 60 mins by fluorescence assay relative to control | 2018 | MedChemComm, Feb-01, Volume: 9, Issue:2
| Identification of karanjin isolated from the Indian beech tree as a potent CYP1 enzyme inhibitor with cellular efficacy |
| AID1411743 | Inhibition of human recombinant CYP2C9 expressed in HEK293 cells using 3-cyano-7-ethoxycoumarin substrate substrate preincubated for 30 mins followed by substrate addition and measured after 60 mins by fluorescence assay relative to control | 2018 | MedChemComm, Feb-01, Volume: 9, Issue:2
| Identification of karanjin isolated from the Indian beech tree as a potent CYP1 enzyme inhibitor with cellular efficacy |
| AID1411740 | Inhibition of human recombinant CYP1A2 expressed in HEK293 cells using 3-cyano-7-ethoxycoumarin substrate preincubated for 30 mins followed by substrate addition and measured after 60 mins by fluorescence assay relative to control | 2018 | MedChemComm, Feb-01, Volume: 9, Issue:2
| Identification of karanjin isolated from the Indian beech tree as a potent CYP1 enzyme inhibitor with cellular efficacy |
| AID365746 | Effect on antigen-stimulated intracellular ROS production in IgE-sensitized CM-H2DCF-DA-treated rat RBL-2H3 cells assessed as increase in 2',7'-dichlorofluorescein oxidation at 50 uM after 30 mins in presence of dinitrophenylated bovine serum albumin | 2008 | Bioorganic & medicinal chemistry, Aug-15, Volume: 16, Issue:16
| Inhibitory effects of polymethoxy flavones isolated from Citrus reticulate on degranulation in rat basophilic leukemia RBL-2H3: enhanced inhibition by their combination. |
| AID365752 | Inhibition of JNK1/2 phosphorylation in antigen-stimulated rat RBL-2H3 cells at 50 uM by Western blot analysis in presence of dinitrophenylated bovine serum albumin | 2008 | Bioorganic & medicinal chemistry, Aug-15, Volume: 16, Issue:16
| Inhibitory effects of polymethoxy flavones isolated from Citrus reticulate on degranulation in rat basophilic leukemia RBL-2H3: enhanced inhibition by their combination. |
| AID1230324 | Displacement of [3H]DPDPE from delta opioid receptor (unknown origin) transfected into HEK293 cells at 10 uM by microplate scintillation counting | 2015 | Journal of natural products, Jun-26, Volume: 78, Issue:6
| Flavonoids from Perovskia atriplicifolia and Their in Vitro Displacement of the Respective Radioligands for Human Opioid and Cannabinoid Receptors. |
| AID1411732 | Inhibition of recombinant human CYP1A2 expressed in baker's yeast-derived microsomes (Sacchrosomes) at 10 uM using 3-cyano-7-ethoxycoumarin substrate by EROD assay relative to control | 2018 | MedChemComm, Feb-01, Volume: 9, Issue:2
| Identification of karanjin isolated from the Indian beech tree as a potent CYP1 enzyme inhibitor with cellular efficacy |
| AID1230327 | Displacement of [3H]DPDPE from delta opioid receptor (unknown origin) transfected into HEK293 cells by microplate scintillation counting | 2015 | Journal of natural products, Jun-26, Volume: 78, Issue:6
| Flavonoids from Perovskia atriplicifolia and Their in Vitro Displacement of the Respective Radioligands for Human Opioid and Cannabinoid Receptors. |
| AID1411737 | Inhibition of recombinant human CYP2C19 expressed in baker's yeast-derived microsomes (Sacchrosomes) at 10 uM using 3-cyano-7-ethoxycoumarin substrate by EROD assay relative to control | 2018 | MedChemComm, Feb-01, Volume: 9, Issue:2
| Identification of karanjin isolated from the Indian beech tree as a potent CYP1 enzyme inhibitor with cellular efficacy |
| AID1230326 | Displacement of [3H]DAMGO from mu opioid receptor (unknown origin) transfected into HEK293 cells at 10 uM by microplate scintillation counting | 2015 | Journal of natural products, Jun-26, Volume: 78, Issue:6
| Flavonoids from Perovskia atriplicifolia and Their in Vitro Displacement of the Respective Radioligands for Human Opioid and Cannabinoid Receptors. |
| AID1411745 | Inhibition of human recombinant CYP3A4 expressed in HEK293 cells using dibenzylfluorescein substrate substrate preincubated for 30 mins followed by substrate addition and measured after 60 mins by fluorescence assay relative to control | 2018 | MedChemComm, Feb-01, Volume: 9, Issue:2
| Identification of karanjin isolated from the Indian beech tree as a potent CYP1 enzyme inhibitor with cellular efficacy |
| AID1230330 | Agonist activity at human delta opioid receptor transfected into HEK293 cells assessed as effect on [35S]-GTPgammaS binding at 300 uM | 2015 | Journal of natural products, Jun-26, Volume: 78, Issue:6
| Flavonoids from Perovskia atriplicifolia and Their in Vitro Displacement of the Respective Radioligands for Human Opioid and Cannabinoid Receptors. |
| AID1230325 | Displacement of [3H]U69593 from kappa opioid receptor (unknown origin) transfected into HEK293 cells at 10 uM by microplate scintillation counting | 2015 | Journal of natural products, Jun-26, Volume: 78, Issue:6
| Flavonoids from Perovskia atriplicifolia and Their in Vitro Displacement of the Respective Radioligands for Human Opioid and Cannabinoid Receptors. |
| AID361718 | Suppression of degranulation in IgE-sensitized rat RBL-2H3 cells assessed as inhibition of A-23187-stimulated histamine release after 30 mins | 2008 | Bioorganic & medicinal chemistry, Aug-15, Volume: 16, Issue:16
| Inhibitory effects of polymethoxy flavones isolated from Citrus reticulate on degranulation in rat basophilic leukemia RBL-2H3: enhanced inhibition by their combination. |
| AID288086 | Antiproliferative activity against HL60 after 24 hrs | 2007 | Bioorganic & medicinal chemistry, May-15, Volume: 15, Issue:10
| Isolation and syntheses of polymethoxyflavones and hydroxylated polymethoxyflavones as inhibitors of HL-60 cell lines. |
| AID288088 | Cytotoxicity against human PMN cells at 100 uM | 2007 | Bioorganic & medicinal chemistry, May-15, Volume: 15, Issue:10
| Isolation and syntheses of polymethoxyflavones and hydroxylated polymethoxyflavones as inhibitors of HL-60 cell lines. |
| AID1411734 | Inhibition of recombinant human CYP2D6 expressed in baker's yeast-derived microsomes (Sacchrosomes) at 10 uM using 7-ethoxy-methyloxy-3-cyanocoumarin substrate by EROD assay relative to control | 2018 | MedChemComm, Feb-01, Volume: 9, Issue:2
| Identification of karanjin isolated from the Indian beech tree as a potent CYP1 enzyme inhibitor with cellular efficacy |
| AID361966 | Inhibition of degranulation in IgE-sensitized rat RBL-2H3 cells assessed as inhibition of antigen-stimulated intracellular calcium elevation after 30 mins in presence of dinitrophenylated bovine serum albumin | 2008 | Bioorganic & medicinal chemistry, Aug-15, Volume: 16, Issue:16
| Inhibitory effects of polymethoxy flavones isolated from Citrus reticulate on degranulation in rat basophilic leukemia RBL-2H3: enhanced inhibition by their combination. |
| AID1411735 | Inhibition of recombinant human CYP3A4 expressed in baker's yeast-derived microsomes (Sacchrosomes) at 10 uM using dibenzylfluorescein substrate by EROD assay relative to control | 2018 | MedChemComm, Feb-01, Volume: 9, Issue:2
| Identification of karanjin isolated from the Indian beech tree as a potent CYP1 enzyme inhibitor with cellular efficacy |
| AID1411730 | Inhibition of recombinant human CYP1A1 expressed in baker's yeast-derived microsomes (Sacchrosomes) at 10 uM using 7-ethoxyresorufin substrate by EROD assay relative to control | 2018 | MedChemComm, Feb-01, Volume: 9, Issue:2
| Identification of karanjin isolated from the Indian beech tree as a potent CYP1 enzyme inhibitor with cellular efficacy |
| AID1411742 | Inhibition of human recombinant CYP2D6 expressed in HEK293 cells using 7-ethoxy-methyloxy-3-cyanocoumarin substrate substrate preincubated for 30 mins followed by substrate addition and measured after 60 mins by fluorescence assay relative to control | 2018 | MedChemComm, Feb-01, Volume: 9, Issue:2
| Identification of karanjin isolated from the Indian beech tree as a potent CYP1 enzyme inhibitor with cellular efficacy |
| AID1411733 | Inhibition of recombinant human CYP1B1 expressed in baker's yeast-derived microsomes (Sacchrosomes) at 10 uM using 7-ethoxyresorufin substrate by EROD assay relative to control | 2018 | MedChemComm, Feb-01, Volume: 9, Issue:2
| Identification of karanjin isolated from the Indian beech tree as a potent CYP1 enzyme inhibitor with cellular efficacy |
| [information is prepared from bioassay data collected from National Library of Medicine (NLM), extracted Dec-2023] |