Assay ID | Title | Year | Journal | Article |
AID540299 | A screen for compounds that inhibit the MenB enzyme of Mycobacterium tuberculosis | 2010 | Bioorganic & medicinal chemistry letters, Nov-01, Volume: 20, Issue:21
| Synthesis and SAR studies of 1,4-benzoxazine MenB inhibitors: novel antibacterial agents against Mycobacterium tuberculosis. |
AID588519 | A screen for compounds that inhibit viral RNA polymerase binding and polymerization activities | 2011 | Antiviral research, Sep, Volume: 91, Issue:3
| High-throughput screening identification of poliovirus RNA-dependent RNA polymerase inhibitors. |
AID288086 | Antiproliferative activity against HL60 after 24 hrs | 2007 | Bioorganic & medicinal chemistry, May-15, Volume: 15, Issue:10
| Isolation and syntheses of polymethoxyflavones and hydroxylated polymethoxyflavones as inhibitors of HL-60 cell lines. |
AID1190339 | Displacement of [3H]DPDPE from delta opioid receptor in CD1 mouse whole brain minus cerebellum membranes by liquid scintillation counting | 2015 | Journal of natural products, Jan-23, Volume: 78, Issue:1
| Methoxyflavones from Stachys glutinosa with binding affinity to opioid receptors: in silico, in vitro, and in vivo studies. |
AID381260 | Cytotoxicity against human KB cells | | | |
AID761700 | Antiproliferative activity against human WI38 cells after 48 hrs by MTT assay | 2013 | European journal of medicinal chemistry, Aug, Volume: 66 | Selective cytotoxic effects on human breast carcinoma of new methoxylated flavonoids from Euryops arabicus grown in Saudi Arabia. |
AID288088 | Cytotoxicity against human PMN cells at 100 uM | 2007 | Bioorganic & medicinal chemistry, May-15, Volume: 15, Issue:10
| Isolation and syntheses of polymethoxyflavones and hydroxylated polymethoxyflavones as inhibitors of HL-60 cell lines. |
AID761702 | Antiproliferative activity against human MCF7 cells after 48 hrs by MTT assay | 2013 | European journal of medicinal chemistry, Aug, Volume: 66 | Selective cytotoxic effects on human breast carcinoma of new methoxylated flavonoids from Euryops arabicus grown in Saudi Arabia. |
AID288087 | Apoptotic activity in HL60 cells after 24 hrs | 2007 | Bioorganic & medicinal chemistry, May-15, Volume: 15, Issue:10
| Isolation and syntheses of polymethoxyflavones and hydroxylated polymethoxyflavones as inhibitors of HL-60 cell lines. |
AID761701 | Antiproliferative activity against african green monkey Vero cells after 48 hrs by MTT assay | 2013 | European journal of medicinal chemistry, Aug, Volume: 66 | Selective cytotoxic effects on human breast carcinoma of new methoxylated flavonoids from Euryops arabicus grown in Saudi Arabia. |
AID371774 | Induction of apoptosis in human HL60 cells assessed as caspase 3/7 activation at 100 uM relative to control | 2009 | Bioorganic & medicinal chemistry letters, Jul-01, Volume: 19, Issue:13
| Semisynthesis and antiproliferative evaluation of a series of 3'-aminoflavones. |
AID761704 | Antioxidant activity assessed as ABTS free radical scavenging activity by spectrophotometry | 2013 | European journal of medicinal chemistry, Aug, Volume: 66 | Selective cytotoxic effects on human breast carcinoma of new methoxylated flavonoids from Euryops arabicus grown in Saudi Arabia. |
AID1766165 | Antagonist activity at PPARgamma (unknown origin) expressed in human LNCaP cells assessed as suppression of pioglitazone-induced PPAR response element driven firefly luciferase activity measured after 24 hrs by dual luciferase reporter assay | 2021 | Bioorganic & medicinal chemistry, 09-15, Volume: 46 | Virtual screening and biological evaluation of PPARĪ³ antagonists as potential anti-prostate cancer agents. |
AID1100871 | Antifeedant activity against Spodoptera litura in compound treated cork borer from fresh sweet potato leaves by Choice Leaf-Disk Bioassay | 2000 | Journal of agricultural and food chemistry, May, Volume: 48, Issue:5
| Insect antifeedant flavonoids from Gnaphalium affine D. Don. |
AID371771 | Cytotoxicity against human KB cells at 1 uM after 72 hrs by MTS assay | 2009 | Bioorganic & medicinal chemistry letters, Jul-01, Volume: 19, Issue:13
| Semisynthesis and antiproliferative evaluation of a series of 3'-aminoflavones. |
AID761699 | Antiproliferative activity against human HepG2 cells after 48 hrs by MTT assay | 2013 | European journal of medicinal chemistry, Aug, Volume: 66 | Selective cytotoxic effects on human breast carcinoma of new methoxylated flavonoids from Euryops arabicus grown in Saudi Arabia. |
AID403015 | Induction of quinone reductase | 2005 | Journal of natural products, Jul, Volume: 68, Issue:7
| Limnophilaspiroketone, a highly oxygenated phenolic derivative from Limnophila geoffrayi. |
AID761703 | Immunostimulant activity in PHA-stimulated human PBL assessed as lymphocyte transformation at 2 mM after 72 hrs by Giemsa staining method | 2013 | European journal of medicinal chemistry, Aug, Volume: 66 | Selective cytotoxic effects on human breast carcinoma of new methoxylated flavonoids from Euryops arabicus grown in Saudi Arabia. |
AID1190338 | Displacement of [3H]DAMGO from mu opioid receptor in CD1 mouse whole brain minus cerebellum membranes by liquid scintillation counting | 2015 | Journal of natural products, Jan-23, Volume: 78, Issue:1
| Methoxyflavones from Stachys glutinosa with binding affinity to opioid receptors: in silico, in vitro, and in vivo studies. |
AID651635 | Viability Counterscreen for Primary qHTS for Inhibitors of ATXN expression | | | |
AID588497 | High-throughput multiplex microsphere screening for inhibitors of toxin protease, specifically Botulinum neurotoxin light chain F protease, MLPCN compound set | 2010 | Current protocols in cytometry, Oct, Volume: Chapter 13 | Microsphere-based flow cytometry protease assays for use in protease activity detection and high-throughput screening. |
AID588497 | High-throughput multiplex microsphere screening for inhibitors of toxin protease, specifically Botulinum neurotoxin light chain F protease, MLPCN compound set | 2006 | Cytometry. Part A : the journal of the International Society for Analytical Cytology, May, Volume: 69, Issue:5
| Microsphere-based protease assays and screening application for lethal factor and factor Xa. |
AID588497 | High-throughput multiplex microsphere screening for inhibitors of toxin protease, specifically Botulinum neurotoxin light chain F protease, MLPCN compound set | 2010 | Assay and drug development technologies, Feb, Volume: 8, Issue:1
| High-throughput multiplex flow cytometry screening for botulinum neurotoxin type a light chain protease inhibitors. |
AID1745845 | Primary qHTS for Inhibitors of ATXN expression | | | |
AID588499 | High-throughput multiplex microsphere screening for inhibitors of toxin protease, specifically Botulinum neurotoxin light chain A protease, MLPCN compound set | 2010 | Current protocols in cytometry, Oct, Volume: Chapter 13 | Microsphere-based flow cytometry protease assays for use in protease activity detection and high-throughput screening. |
AID588499 | High-throughput multiplex microsphere screening for inhibitors of toxin protease, specifically Botulinum neurotoxin light chain A protease, MLPCN compound set | 2006 | Cytometry. Part A : the journal of the International Society for Analytical Cytology, May, Volume: 69, Issue:5
| Microsphere-based protease assays and screening application for lethal factor and factor Xa. |
AID588499 | High-throughput multiplex microsphere screening for inhibitors of toxin protease, specifically Botulinum neurotoxin light chain A protease, MLPCN compound set | 2010 | Assay and drug development technologies, Feb, Volume: 8, Issue:1
| High-throughput multiplex flow cytometry screening for botulinum neurotoxin type a light chain protease inhibitors. |
AID588501 | High-throughput multiplex microsphere screening for inhibitors of toxin protease, specifically Lethal Factor Protease, MLPCN compound set | 2010 | Current protocols in cytometry, Oct, Volume: Chapter 13 | Microsphere-based flow cytometry protease assays for use in protease activity detection and high-throughput screening. |
AID588501 | High-throughput multiplex microsphere screening for inhibitors of toxin protease, specifically Lethal Factor Protease, MLPCN compound set | 2006 | Cytometry. Part A : the journal of the International Society for Analytical Cytology, May, Volume: 69, Issue:5
| Microsphere-based protease assays and screening application for lethal factor and factor Xa. |
AID588501 | High-throughput multiplex microsphere screening for inhibitors of toxin protease, specifically Lethal Factor Protease, MLPCN compound set | 2010 | Assay and drug development technologies, Feb, Volume: 8, Issue:1
| High-throughput multiplex flow cytometry screening for botulinum neurotoxin type a light chain protease inhibitors. |
[information is prepared from bioassay data collected from National Library of Medicine (NLM), extracted Dec-2023] |