An antiviral agent that destroys or inhibits the replication of the human immunodeficiency virus.
| Member | Definition | Class |
|---|
| 1-deoxynojirimycin | An optically active form of 2-(hydroxymethyl)piperidine-3,4,5-triol having 2R,3R,4R,5S-configuration. | duvoglustat |
| 16beta,17-dihydroxy-ent-kaurane-19-oic acid | A ent-kaurane diterpenoid that is ent-kaurane-19-oic acid substituted by hydroxy groups at positions 16 and 17 (the 16beta stereoisomer). It is isolated from Helianthus sp. and Annona squamosa and exhibits anti-HIV activity. | 16beta,17-dihydroxy-ent-kaurane-19-oic acid |
| andrographolide | A labdane diterpenoid isolated from the leaves and roots of Andrographis paniculata that exhibits anti-HIV, anti-inflammatory and antineoplastic properties. | andrographolide |
| betulinic acid | A pentacyclic triterpenoid that is lupane having a double bond at position 20(29) as well as 3beta-hydroxy and 28-carboxy substituents. It is found in the bark and other plant parts of several species of plants including Syzygium claviflorum. It exhibits anti-HIV, antimalarial, antineoplastic and anti-inflammatory properties. | betulinic acid |
| boromycin | A boron-containing macrolide antibiotic that is isolated from Streptomyces antibioticus. | boromycin |
| bromophycolide a | A diterpenoid that is a macrolide isolated from the Fijian red alga Callophycus serratus. It has been found to exhibit moderate cytotoxicity against several human tumour cell lines via specific apotopic cell death. It also displays anti-HIV, antibacterial, antifungal and antimalarial activity. | bromophycolide A |
| cenicriviroc | A member of the class of benzazocines that is (5Z)-1,2,3,4-tetrahydro-1-benzazocine which is substituted by a 2-methylpropyl, N-{4-[(S)-(1-propyl-1H-imidazol-5-yl)methanesulfinyl]phenyl}carboxamide and 4-(2-butoxyethoxy)phenyl groups at positions 1, 5 and 8, respectively. It is a potent chemokine 2 and 5 receptor antagonist currently in development for the treatment of liver fibrosis in adults with nonalcoholic steatohepatitis (NASH). | cenicriviroc |
| cidofovir anhydrous | Cytosine substituted at the 1 position by a 3-hydroxy-2-(phosphonomethoxy)propyl group (S configuration). A nucleoside analogue, it is an injectable antiviral used for the treatment of cytomegalovirus (CMV) retinitis in AIDS patients. | cidofovir anhydrous |
| colforsin | A labdane diterpenoid isolated from the Indian Coleus plant. | forskolin |
| dihydrobetulinic acid | A pentacyclic triterpenoid that is lupane having a 3beta-hydroxy and 28-carboxy substituents. Isolated from the leaves of Syzygium claviflorum, it exhibits anti-HIV and antileishmanial activity. | dihydrobetulinic acid |
| dmp 323 | A 1,3-diazepanone ring with two 4-(hydroxymethyl)benzyl groups as substituents at positions N-1 and N-4, two benzyl groups at C-4 and C-7, and two hydroxy groups at C-5 and C-6 respectively. | (4R,5S,6S,7R)-4,7-dibenzyl-5,6-dihydroxy-1,3-bis[4-(hydroxymethyl)benzyl]-1,3-diazepan-2-one |
| drymaritin | An indole alkaloid that is canthin-6-one substituted by a methoxy group at position 4. Isolated from the whole plants of Drymaria diandra, it exhibits anti-HIV activity. | drymaritin |
| harman | An indole alkaloid fundamental parent with a structure of 9H-beta-carboline carrying a methyl substituent at C-1. It has been isolated from the bark of Sickingia rubra, Symplocus racemosa, Passiflora incarnata, Peganum harmala, Banisteriopsis caapi and Tribulus terrestris, as well as from tobacco smoke. It is a specific, reversible inhibitor of monoamine oxidase A. | harman |
| harmine | A harmala alkaloid in which the harman skeleton is methoxy-substituted at C-7. | harmine |
| interiotherin b | A lignan with a dibenzocyclooctadiene skeleton attached to a fatty acid ester side chain. It is isolated from Kadsura interior and has been shown to exhibit anti-HIV activity. | interiotherin B |
| L-cycloserine | A 4-amino-1,2-oxazolidin-3-one that has S configuration. An antibiotic isolated from Erwinia uredovora. | L-cycloserine |
| lancifodilactone g | A triterpenoid that is a nortriterpenoid isolated from Schisandra lancifolia and has been shown to exhibit anti-HIV activity. | lancifodilactone G |
| macluraxanthone b | A member of the class of xanthones that is 9H-xanthen-9-one substituted by hydroxy groups at positions 1, 3, 6 and 7, a dimethylallyl group at position 2 and a prenyl group at position 4. Isolated from Maclura tinctoria and Cudrania tricuspidata, it exhibits anti-HIV and antineoplastic activity. | macluraxanthone B |
| miglustat | A hydroxypiperidine that is deoxynojirimycin in which the amino hydrogen is replaced by a butyl group. | miglustat |
| mor-14 | A hydroxypiperidine that is duvoglustat in which the amino hydrogen is replaced by a methyl group. It is an inhibitor of alpha-glucosidase, an agonist of the glucose sensor SGLT3 and exhibits anti-HIV activity. | N-methyl-1-deoxynojirimycin |
| moronic acid | A pentacyclic triterpenoid that is olean-18-ene substituted at position 3 by an oxo group and position 28 by a carboxy group. | moronic acid |
| N-ethylharmine | A member of the class of beta-carbolines that is 9H-beta-carboline substituted by a ethyl group at position 9, methoxy group at position 7 and a methyl group at position 1. It is semisynthetic derivative of harmine and has been shown to exhibit significant anti-HIV activity. | N-ethylharmine |
| oxetanocin a | A nucleoside analogue found in Bacillus megaterium in which an adenine moiety is attached to position 2 of a of an oxetane ring which is substituted at positions 3 and 4 by hydroxymethyl groups. | oxetanocin A |
| platanic acid | A pentacyclic triterpenoid that is 30-norlupan-28-oic acid substituted by a 3beta-hydroxy and an oxo group at position 20. It is isolated from the leaves of Syzygium claviflorum and exhibits anti-HIV activity. | platanic acid |
| plerixafor | An azamacrocycle consisting of two cyclam rings connected by a 1,4-phenylenebis(methylene) linker. It is a CXCR4 chemokine receptor antagonist and a hematopoietic stem cell mobilizer. It is used in combination with grulocyte-colony stimulating factor (G-CSF) to mobilize hematopoietic stem cells to the perpheral blood for collection and subsequent autologous transplantation in patients with non-Hodgkin's lymphoma and multiple myeloma. | plerixafor |
| proanthocyanidin a2 | A proanthocyanidin obtained by the condensation of (-)-epicatechin units. | proanthocyanidin A2 |
| Protein | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Drugs |
|---|
| 15-hydroxyprostaglandin dehydrogenase [NAD(+)] isoform 1 | Homo sapiens (human) | Potency | 22.5585 | 1 | 9 |
| 67.9K protein | Vaccinia virus | Potency | 19.0832 | 2 | 7 |
| aldehyde dehydrogenase 1 family, member A1 | Homo sapiens (human) | Potency | 21.9559 | 1 | 11 |
| alpha-galactosidase | Homo sapiens (human) | Potency | 39.8107 | 1 | 1 |
| apical membrane antigen 1, AMA1 | Plasmodium falciparum 3D7 | Potency | 14.1254 | 1 | 1 |
| AR protein | Homo sapiens (human) | Potency | 14.9023 | 6 | 15 |
| aryl hydrocarbon receptor | Homo sapiens (human) | Potency | 19.7364 | 2 | 2 |
| ATAD5 protein, partial | Homo sapiens (human) | Potency | 13.7763 | 2 | 2 |
| Ataxin-2 | Homo sapiens (human) | Potency | 0.1940 | 1 | 2 |
| ATP-dependent phosphofructokinase | Trypanosoma brucei brucei TREU927 | Potency | 0.7569 | 1 | 1 |
| ATPase family AAA domain-containing protein 5 | Homo sapiens (human) | Potency | 0.2301 | 2 | 4 |
| Bloom syndrome protein isoform 1 | Homo sapiens (human) | Potency | 14.9422 | 2 | 4 |
| bromodomain adjacent to zinc finger domain 2B | Homo sapiens (human) | Potency | 0.6310 | 1 | 1 |
| Cellular tumor antigen p53 | Homo sapiens (human) | Potency | 19.0318 | 1 | 2 |
| Chain A, 2-oxoglutarate Oxygenase | Homo sapiens (human) | Potency | 22.7602 | 1 | 9 |
| Chain A, Cruzipain | Trypanosoma cruzi | Potency | 34.9134 | 2 | 6 |
| Chain A, Ferritin light chain | Equus caballus (horse) | Potency | 23.6612 | 2 | 3 |
| Chain A, HADH2 protein | Homo sapiens (human) | Potency | 21.6095 | 2 | 7 |
| Chain A, MAJOR APURINIC/APYRIMIDINIC ENDONUCLEASE | Homo sapiens (human) | Potency | 25.1703 | 2 | 11 |
| Chain A, TYROSYL-DNA PHOSPHODIESTERASE | Homo sapiens (human) | Potency | 31.6228 | 1 | 1 |
| Chain B, HADH2 protein | Homo sapiens (human) | Potency | 21.6095 | 2 | 7 |
| chromobox protein homolog 1 | Homo sapiens (human) | Potency | 89.1251 | 1 | 3 |
| cytochrome P450 2C9, partial | Homo sapiens (human) | Potency | 31.6925 | 1 | 3 |
| cytochrome P450 2D6 isoform 1 | Homo sapiens (human) | Potency | 14.8915 | 1 | 4 |
| cytochrome P450 3A4 isoform 1 | Homo sapiens (human) | Potency | 17.4102 | 2 | 8 |
| cytochrome P450 family 3 subfamily A polypeptide 4 | Homo sapiens (human) | Potency | 14.5100 | 2 | 6 |
| cytochrome P450, family 19, subfamily A, polypeptide 1, isoform CRA_a | Homo sapiens (human) | Potency | 1.0786 | 1 | 2 |
| DNA dC->dU-editing enzyme APOBEC-3F isoform a | Homo sapiens (human) | Potency | 6.3096 | 1 | 1 |
| DNA polymerase beta | Homo sapiens (human) | Potency | 3.1623 | 1 | 1 |
| DNA polymerase iota isoform a (long) | Homo sapiens (human) | Potency | 100.0000 | 1 | 1 |
| dopamine D1 receptor | Homo sapiens (human) | Potency | 4.6109 | 1 | 1 |
| dual specificity protein kinase CLK4 | Homo sapiens (human) | Potency | 0.0671 | 1 | 1 |
| endonuclease IV | Escherichia coli | Potency | 0.8913 | 1 | 1 |
| estrogen nuclear receptor alpha | Homo sapiens (human) | Potency | 11.0586 | 10 | 21 |
| estrogen receptor 2 (ER beta) | Homo sapiens (human) | Potency | 42.1660 | 2 | 2 |
| estrogen-related nuclear receptor alpha | Homo sapiens (human) | Potency | 7.7861 | 9 | 12 |
| euchromatic histone-lysine N-methyltransferase 2 | Homo sapiens (human) | Potency | 10.6074 | 1 | 2 |
| EWS/FLI fusion protein | Homo sapiens (human) | Potency | 4.6859 | 1 | 1 |
| farnesoid X nuclear receptor | Homo sapiens (human) | Potency | 34.2300 | 2 | 2 |
| flap endonuclease 1 | Homo sapiens (human) | Potency | 50.1187 | 1 | 1 |
| Fumarate hydratase | Homo sapiens (human) | Potency | 0.4176 | 1 | 1 |
| G | Vesicular stomatitis virus | Potency | 31.6925 | 1 | 3 |
| GABA theta subunit | Rattus norvegicus (Norway rat) | Potency | 17.4102 | 1 | 4 |
| Gamma-aminobutyric acid receptor subunit alpha-1 | Rattus norvegicus (Norway rat) | Potency | 17.4102 | 1 | 4 |
| Gamma-aminobutyric acid receptor subunit alpha-2 | Rattus norvegicus (Norway rat) | Potency | 17.4102 | 1 | 4 |
| Gamma-aminobutyric acid receptor subunit alpha-3 | Rattus norvegicus (Norway rat) | Potency | 17.4102 | 1 | 4 |
| Gamma-aminobutyric acid receptor subunit alpha-4 | Rattus norvegicus (Norway rat) | Potency | 17.4102 | 1 | 4 |
| Gamma-aminobutyric acid receptor subunit alpha-5 | Rattus norvegicus (Norway rat) | Potency | 17.4102 | 1 | 4 |
| Gamma-aminobutyric acid receptor subunit alpha-6 | Rattus norvegicus (Norway rat) | Potency | 17.4102 | 1 | 4 |
| Gamma-aminobutyric acid receptor subunit beta-1 | Rattus norvegicus (Norway rat) | Potency | 17.4102 | 1 | 4 |
| Gamma-aminobutyric acid receptor subunit beta-2 | Rattus norvegicus (Norway rat) | Potency | 17.4102 | 1 | 4 |
| Gamma-aminobutyric acid receptor subunit beta-3 | Rattus norvegicus (Norway rat) | Potency | 17.4102 | 1 | 4 |
| Gamma-aminobutyric acid receptor subunit delta | Rattus norvegicus (Norway rat) | Potency | 17.4102 | 1 | 4 |
| Gamma-aminobutyric acid receptor subunit epsilon | Rattus norvegicus (Norway rat) | Potency | 17.4102 | 1 | 4 |
| Gamma-aminobutyric acid receptor subunit gamma-1 | Rattus norvegicus (Norway rat) | Potency | 17.4102 | 1 | 4 |
| Gamma-aminobutyric acid receptor subunit gamma-2 | Rattus norvegicus (Norway rat) | Potency | 17.4102 | 1 | 4 |
| Gamma-aminobutyric acid receptor subunit gamma-3 | Rattus norvegicus (Norway rat) | Potency | 17.4102 | 1 | 4 |
| Gamma-aminobutyric acid receptor subunit pi | Rattus norvegicus (Norway rat) | Potency | 17.4102 | 1 | 4 |
| geminin | Homo sapiens (human) | Potency | 12.0147 | 2 | 2 |
| GLI family zinc finger 3 | Homo sapiens (human) | Potency | 4.3783 | 2 | 6 |
| glp-1 receptor, partial | Homo sapiens (human) | Potency | 1.6966 | 2 | 3 |
| glucocerebrosidase | Homo sapiens (human) | Potency | 12.5893 | 1 | 1 |
| glucocorticoid receptor [Homo sapiens] | Homo sapiens (human) | Potency | 0.5468 | 1 | 2 |
| Glutamate receptor 2 | Rattus norvegicus (Norway rat) | Potency | 11.4265 | 1 | 2 |
| Histamine H2 receptor | Cavia porcellus (domestic guinea pig) | Potency | 15.8489 | 1 | 4 |
| histone acetyltransferase KAT2A isoform 1 | Homo sapiens (human) | Potency | 27.8298 | 1 | 2 |
| histone-lysine N-methyltransferase 2A isoform 2 precursor | Homo sapiens (human) | Potency | 10.0000 | 1 | 1 |
| HLA class I histocompatibility antigen, B alpha chain | Homo sapiens (human) | Potency | 31.6925 | 1 | 3 |
| hypoxia-inducible factor 1, alpha subunit (basic helix-loop-helix transcription factor) | Homo sapiens (human) | Potency | 6.3096 | 2 | 2 |
| Inositol hexakisphosphate kinase 1 | Homo sapiens (human) | Potency | 31.6925 | 1 | 6 |
| Interferon beta | Homo sapiens (human) | Potency | 21.7006 | 2 | 6 |
| lamin isoform A-delta10 | Homo sapiens (human) | Potency | 0.0112 | 1 | 1 |
| lethal factor (plasmid) | Bacillus anthracis str. A2012 | Potency | 1.9953 | 1 | 1 |
| lysosomal alpha-glucosidase preproprotein | Homo sapiens (human) | Potency | 0.0580 | 5 | 5 |
| Microtubule-associated protein tau | Homo sapiens (human) | Potency | 0.5623 | 1 | 1 |
| mitogen-activated protein kinase 1 | Homo sapiens (human) | Potency | 100.0000 | 1 | 1 |
| muscarinic acetylcholine receptor M1 | Rattus norvegicus (Norway rat) | Potency | 25.1189 | 1 | 1 |
| neuropeptide S receptor isoform A | Homo sapiens (human) | Potency | 7.5060 | 1 | 2 |
| NFKB1 protein, partial | Homo sapiens (human) | Potency | 1.9953 | 2 | 2 |
| nuclear factor erythroid 2-related factor 2 isoform 1 | Homo sapiens (human) | Potency | 30.6421 | 2 | 2 |
| nuclear factor erythroid 2-related factor 2 isoform 2 | Homo sapiens (human) | Potency | 23.1093 | 1 | 1 |
| nuclear receptor ROR-gamma isoform 1 | Mus musculus (house mouse) | Potency | 20.0809 | 2 | 3 |
| nuclear receptor subfamily 1, group I, member 2 | Rattus norvegicus (Norway rat) | Potency | 5.0119 | 1 | 1 |
| nuclear receptor subfamily 1, group I, member 3 | Homo sapiens (human) | Potency | 25.6653 | 2 | 3 |
| parathyroid hormone/parathyroid hormone-related peptide receptor precursor | Homo sapiens (human) | Potency | 25.8740 | 1 | 2 |
| peripheral myelin protein 22 | Rattus norvegicus (Norway rat) | Potency | 0.5344 | 2 | 2 |
| peroxisome proliferator activated receptor gamma | Homo sapiens (human) | Potency | 13.4792 | 2 | 2 |
| peroxisome proliferator-activated receptor delta | Homo sapiens (human) | Potency | 5.0077 | 2 | 2 |
| polyprotein | Zika virus | Potency | 0.4176 | 1 | 1 |
| Polyunsaturated fatty acid lipoxygenase ALOX15B | Homo sapiens (human) | Potency | 15.8489 | 1 | 2 |
| PPM1D protein | Homo sapiens (human) | Potency | 11.7086 | 1 | 2 |
| pregnane X nuclear receptor | Homo sapiens (human) | Potency | 14.7594 | 3 | 4 |
| pregnane X receptor | Rattus norvegicus (Norway rat) | Potency | 7.9433 | 1 | 1 |
| progesterone receptor | Homo sapiens (human) | Potency | 0.2169 | 1 | 1 |
| Rap guanine nucleotide exchange factor 3 | Homo sapiens (human) | Potency | 100.0000 | 1 | 1 |
| Rap guanine nucleotide exchange factor 4 | Homo sapiens (human) | Potency | 100.0000 | 1 | 1 |
| RAR-related orphan receptor gamma | Mus musculus (house mouse) | Potency | 31.8828 | 2 | 5 |
| regulator of G-protein signaling 4 | Homo sapiens (human) | Potency | 15.0030 | 1 | 1 |
| relaxin receptor 1 isoform 1 | Homo sapiens (human) | Potency | 0.0388 | 1 | 1 |
| relaxin receptor 2 isoform 1 | Homo sapiens (human) | Potency | 0.0488 | 1 | 1 |
| retinoic acid nuclear receptor alpha variant 1 | Homo sapiens (human) | Potency | 34.0811 | 2 | 2 |
| retinoid X nuclear receptor alpha | Homo sapiens (human) | Potency | 16.8068 | 1 | 2 |
| serine/threonine-protein kinase PLK1 | Homo sapiens (human) | Potency | 33.5875 | 1 | 1 |
| Smad3 | Homo sapiens (human) | Potency | 35.4813 | 1 | 1 |
| Spike glycoprotein | Severe acute respiratory syndrome-related coronavirus | Potency | 3.9811 | 1 | 1 |
| survival motor neuron protein isoform d | Homo sapiens (human) | Potency | 3.9074 | 1 | 3 |
| TDP1 protein | Homo sapiens (human) | Potency | 11.6935 | 2 | 24 |
| thioredoxin reductase | Rattus norvegicus (Norway rat) | Potency | 42.7231 | 3 | 9 |
| thyroid hormone receptor beta isoform 2 | Rattus norvegicus (Norway rat) | Potency | 7.2378 | 2 | 6 |
| thyroid stimulating hormone receptor | Homo sapiens (human) | Potency | 5.6318 | 6 | 9 |
| vitamin D (1,25- dihydroxyvitamin D3) receptor | Homo sapiens (human) | Potency | 0.0044 | 1 | 1 |
| Voltage-dependent calcium channel gamma-2 subunit | Mus musculus (house mouse) | Potency | 11.4265 | 1 | 2 |
| Protein | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Drugs |
|---|
| [Tau protein] kinase | Sus scrofa (pig) | IC50 | 12.2500 | 4 | 4 |
| 5-hydroxytryptamine receptor 1A | Homo sapiens (human) | IC50 | 0.0410 | 1 | 1 |
| 5-hydroxytryptamine receptor 1A | Homo sapiens (human) | Ki | 10.0000 | 1 | 1 |
| 5-hydroxytryptamine receptor 1B | Homo sapiens (human) | Ki | 10.0000 | 1 | 1 |
| 5-hydroxytryptamine receptor 1D | Homo sapiens (human) | Ki | 10.0000 | 1 | 1 |
| 5-hydroxytryptamine receptor 2A | Rattus norvegicus (Norway rat) | Ki | 7.7900 | 1 | 1 |
| 5-hydroxytryptamine receptor 2C | Homo sapiens (human) | Ki | 9.3400 | 1 | 1 |
| 5-hydroxytryptamine receptor 3A | Homo sapiens (human) | Ki | 10.0000 | 1 | 1 |
| 5-hydroxytryptamine receptor 3B | Homo sapiens (human) | Ki | 10.0000 | 1 | 1 |
| 5-hydroxytryptamine receptor 3C | Homo sapiens (human) | Ki | 10.0000 | 1 | 1 |
| 5-hydroxytryptamine receptor 3D | Homo sapiens (human) | Ki | 10.0000 | 1 | 1 |
| 5-hydroxytryptamine receptor 3E | Homo sapiens (human) | Ki | 10.0000 | 1 | 1 |
| 5-hydroxytryptamine receptor 5A | Homo sapiens (human) | Ki | 10.0000 | 2 | 2 |
| 5-hydroxytryptamine receptor 6 | Homo sapiens (human) | Ki | 1.4800 | 1 | 1 |
| 5-hydroxytryptamine receptor 7 | Homo sapiens (human) | Ki | 5.5000 | 1 | 1 |
| 5'-nucleotidase | Homo sapiens (human) | IC50 | 7.2800 | 1 | 1 |
| 5'-nucleotidase | Mus musculus (house mouse) | IC50 | 68.7900 | 1 | 1 |
| Acetylcholinesterase | Electrophorus electricus (electric eel) | IC50 | 17.9667 | 2 | 3 |
| Acetylcholinesterase | Electrophorus electricus (electric eel) | Ki | 34.2500 | 2 | 2 |
| Adenylate cyclase type 1 | Homo sapiens (human) | IC50 | 0.0955 | 2 | 2 |
| Aldehyde oxidase | Homo sapiens (human) | IC50 | 0.0300 | 1 | 1 |
| Aldo-keto reductase family 1 member B1 | Homo sapiens (human) | IC50 | 11.0000 | 1 | 1 |
| Aldo-keto reductase family 1 member B10 | Homo sapiens (human) | IC50 | 2.0000 | 1 | 1 |
| Alpha-1A adrenergic receptor | Rattus norvegicus (Norway rat) | IC50 | 1.3000 | 1 | 1 |
| Alpha-1A adrenergic receptor | Homo sapiens (human) | Ki | 3.8733 | 2 | 3 |
| Alpha-1B adrenergic receptor | Rattus norvegicus (Norway rat) | IC50 | 1.3000 | 1 | 1 |
| Alpha-1B adrenergic receptor | Homo sapiens (human) | Ki | 5.4050 | 2 | 2 |
| Alpha-1D adrenergic receptor | Rattus norvegicus (Norway rat) | IC50 | 1.3000 | 1 | 1 |
| Alpha-1D adrenergic receptor | Homo sapiens (human) | Ki | 0.8100 | 1 | 1 |
| Alpha-2A adrenergic receptor | Homo sapiens (human) | Ki | 6.2700 | 2 | 2 |
| Alpha-2A adrenergic receptor | Mus musculus (house mouse) | Ki | 10.0000 | 1 | 1 |
| Alpha-2B adrenergic receptor | Homo sapiens (human) | Ki | 1.1300 | 1 | 1 |
| Alpha-2B adrenergic receptor | Mus musculus (house mouse) | Ki | 10.0000 | 1 | 1 |
| Alpha-2C adrenergic receptor | Homo sapiens (human) | Ki | 0.8100 | 1 | 1 |
| Alpha-2C adrenergic receptor | Mus musculus (house mouse) | Ki | 10.0000 | 1 | 1 |
| Alpha-amylase | Geobacillus stearothermophilus | IC50 | 1.6700 | 1 | 1 |
| Alpha-galactosidase A | Homo sapiens (human) | Ki | 18.0000 | 1 | 1 |
| Alpha-glucosidase MAL12 | Saccharomyces cerevisiae S288C | IC50 | 278.0000 | 1 | 1 |
| Alpha-glucosidase MAL12 | Saccharomyces cerevisiae S288C | Ki | 18.0000 | 1 | 1 |
| Alpha-glucosidase MAL32 | Saccharomyces cerevisiae S288C | IC50 | 175.0000 | 1 | 2 |
| Alpha-glucosidase MAL62 | Saccharomyces cerevisiae (brewer's yeast) | IC50 | 212,855.0000 | 2 | 2 |
| Alpha-mannosidase | Canavalia ensiformis (jack bean) | Ki | 270.0000 | 1 | 1 |
| Alpha-mannosidase 2 | Rattus norvegicus (Norway rat) | Ki | 50.0000 | 1 | 3 |
| Amine oxidase [flavin-containing] A | Homo sapiens (human) | IC50 | 0.0044 | 3 | 3 |
| Amine oxidase [flavin-containing] A | Homo sapiens (human) | Ki | 0.0152 | 4 | 4 |
| Amine oxidase [flavin-containing] B | Homo sapiens (human) | Ki | 60.4110 | 2 | 2 |
| ATP-binding cassette sub-family C member 3 | Homo sapiens (human) | IC50 | 133.0000 | 1 | 2 |
| ATP-dependent translocase ABCB1 | Homo sapiens (human) | IC50 | 134.2000 | 2 | 2 |
| Beta-1 adrenergic receptor | Homo sapiens (human) | Ki | 10.0000 | 1 | 1 |
| Beta-2 adrenergic receptor | Homo sapiens (human) | Ki | 10.0000 | 1 | 1 |
| Beta-galactosidase | Mus musculus (house mouse) | IC50 | 750.0000 | 1 | 1 |
| Beta-glucosidase | Agrobacterium tumefaciens | Ki | 12.0000 | 2 | 2 |
| Beta-glucosidase | Prunus avium (sweet cherry) | IC50 | 81.0000 | 1 | 1 |
| Beta-glucosidase A | Caldicellulosiruptor saccharolyticus | IC50 | 218.3333 | 3 | 3 |
| Bile acid receptor | Homo sapiens (human) | IC50 | 9.7000 | 2 | 2 |
| Bile salt export pump | Homo sapiens (human) | IC50 | 133.0000 | 1 | 2 |
| Botulinum neurotoxin type A | Clostridium botulinum | IC50 | 20.0000 | 1 | 1 |
| Botulinum neurotoxin type A | Clostridium botulinum | Ki | 14.3000 | 1 | 1 |
| Broad substrate specificity ATP-binding cassette transporter ABCG2 | Homo sapiens (human) | GI50 | 1.6700 | 3 | 3 |
| Broad substrate specificity ATP-binding cassette transporter ABCG2 | Homo sapiens (human) | IC50 | 5.0800 | 1 | 1 |
| C-C chemokine receptor type 2 | Homo sapiens (human) | IC50 | 0.0030 | 4 | 4 |
| C-C chemokine receptor type 5 | Homo sapiens (human) | IC50 | 0.0030 | 1 | 1 |
| C-C chemokine receptor type 5 | Mus musculus (house mouse) | IC50 | 0.0002 | 1 | 1 |
| C-C chemokine receptor type 7 | Homo sapiens (human) | IC50 | 0.0031 | 1 | 1 |
| C-X-C chemokine receptor type 4 | Homo sapiens (human) | IC50 | 0.8234 | 37 | 37 |
| C-X-C chemokine receptor type 4 | Rattus norvegicus (Norway rat) | IC50 | 0.1080 | 1 | 1 |
| C-X-C chemokine receptor type 4 | Homo sapiens (human) | Ki | 6.1137 | 43 | 43 |
| Canalicular multispecific organic anion transporter 1 | Homo sapiens (human) | IC50 | 133.0000 | 1 | 2 |
| Casein kinase I isoform delta | Homo sapiens (human) | IC50 | 1.5000 | 2 | 2 |
| Casein kinase I isoform epsilon | Homo sapiens (human) | IC50 | 1.5000 | 1 | 1 |
| Ceramide glucosyltransferase | Homo sapiens (human) | IC50 | 43.8000 | 4 | 5 |
| Ceramide glucosyltransferase | Mus musculus (house mouse) | IC50 | 40.9667 | 3 | 3 |
| Chain A, Dual specificity tyrosine-phosphorylation-regulated kinase 1A | Homo sapiens (human) | IC50 | 0.3500 | 1 | 1 |
| Chain A, HIV-1 PROTEASE | Human immunodeficiency virus 1 | Ki | 0.2462 | 1 | 10 |
| Chain B, HIV-1 PROTEASE | Human immunodeficiency virus 1 | Ki | 0.2462 | 1 | 10 |
| Cholinesterase | Equus caballus (horse) | IC50 | 13.6000 | 1 | 1 |
| Cholinesterase | Equus caballus (horse) | Ki | 50.0000 | 1 | 1 |
| Cyclin-A1 | Homo sapiens (human) | IC50 | 32.5000 | 2 | 2 |
| Cyclin-A2 | Homo sapiens (human) | IC50 | 25.0000 | 3 | 3 |
| Cyclin-dependent kinase 1 | Homo sapiens (human) | IC50 | 18.0000 | 1 | 1 |
| Cyclin-dependent kinase 2 | Homo sapiens (human) | IC50 | 25.0000 | 3 | 3 |
| Cyclin-dependent kinase 5 activator 1 | Homo sapiens (human) | IC50 | 11.4000 | 5 | 5 |
| Cyclin-dependent kinase 7 | Homo sapiens (human) | IC50 | 10.0000 | 1 | 1 |
| Cyclin-dependent kinase 9 | Homo sapiens (human) | IC50 | 0.7200 | 1 | 1 |
| Cyclin-dependent-like kinase 5 | Homo sapiens (human) | IC50 | 11.4000 | 5 | 5 |
| Cyclin-H | Homo sapiens (human) | IC50 | 10.0000 | 1 | 1 |
| Cyclin-T1 | Homo sapiens (human) | IC50 | 0.7200 | 1 | 1 |
| Cytochrome P450 3A4 | Homo sapiens (human) | IC50 | 22.0000 | 1 | 1 |
| Cytosolic beta-glucosidase | Homo sapiens (human) | IC50 | 160.0000 | 2 | 2 |
| D(1A) dopamine receptor | Homo sapiens (human) | Ki | 10.0000 | 1 | 1 |
| D(1B) dopamine receptor | Homo sapiens (human) | Ki | 10.0000 | 1 | 1 |
| D(2) dopamine receptor | Homo sapiens (human) | Ki | 10.0000 | 1 | 1 |
| D(3) dopamine receptor | Homo sapiens (human) | Ki | 10.0000 | 1 | 1 |
| D(4) dopamine receptor | Homo sapiens (human) | Ki | 10.0000 | 1 | 1 |
| DNA polymerase beta | Homo sapiens (human) | IC50 | 41.1833 | 3 | 3 |
| DNA polymerase beta | Rattus norvegicus (Norway rat) | IC50 | 10.2500 | 2 | 2 |
| Dual specificity protein kinase CLK1 | Homo sapiens (human) | IC50 | 0.0860 | 4 | 4 |
| Dual specificity protein kinase CLK1 | Mus musculus (house mouse) | IC50 | 0.0720 | 1 | 1 |
| Dual specificity protein kinase CLK2 | Mus musculus (house mouse) | IC50 | 0.2800 | 1 | 1 |
| Dual specificity protein kinase CLK3 | Mus musculus (house mouse) | IC50 | 10.0000 | 1 | 1 |
| Dual specificity protein kinase CLK4 | Mus musculus (house mouse) | IC50 | 0.0500 | 1 | 1 |
| Dual specificity tyrosine-phosphorylation-regulated kinase 1A | Homo sapiens (human) | IC50 | 0.1020 | 29 | 30 |
| Dual specificity tyrosine-phosphorylation-regulated kinase 1A | Rattus norvegicus (Norway rat) | IC50 | 0.0397 | 3 | 3 |
| Dual specificity tyrosine-phosphorylation-regulated kinase 1A | Homo sapiens (human) | Ki | 0.0330 | 1 | 1 |
| Dual specificity tyrosine-phosphorylation-regulated kinase 1B | Homo sapiens (human) | IC50 | 0.1183 | 5 | 5 |
| Dual specificity tyrosine-phosphorylation-regulated kinase 1B | Homo sapiens (human) | Ki | 0.1660 | 1 | 1 |
| Dual specificity tyrosine-phosphorylation-regulated kinase 2 | Homo sapiens (human) | IC50 | 1.3138 | 8 | 8 |
| Dual specificity tyrosine-phosphorylation-regulated kinase 3 | Homo sapiens (human) | IC50 | 0.6040 | 5 | 5 |
| Dual specificity tyrosine-phosphorylation-regulated kinase 4 | Homo sapiens (human) | IC50 | 54.5000 | 3 | 3 |
| G2/mitotic-specific cyclin-B1 | Homo sapiens (human) | IC50 | 18.0000 | 1 | 1 |
| G2/mitotic-specific cyclin-B2 | Homo sapiens (human) | IC50 | 18.0000 | 1 | 1 |
| G2/mitotic-specific cyclin-B3 | Homo sapiens (human) | IC50 | 18.0000 | 1 | 1 |
| GABA theta subunit | Rattus norvegicus (Norway rat) | IC50 | 12.3920 | 3 | 3 |
| GABA theta subunit | Rattus norvegicus (Norway rat) | Ki | 10.8000 | 2 | 3 |
| Gag-Pol polyprotein | Human immunodeficiency virus type 1 (BRU ISOLATE) | Ki | 0.0003 | 1 | 1 |
| Gag-Pol polyprotein | Human immunodeficiency virus type 1 (NEW YORK-5 ISOLATE) | Ki | 0.0010 | 1 | 1 |
| Gamma-aminobutyric acid receptor subunit alpha-1 | Homo sapiens (human) | IC50 | 12.3027 | 1 | 1 |
| Gamma-aminobutyric acid receptor subunit alpha-1 | Rattus norvegicus (Norway rat) | IC50 | 12.3920 | 3 | 3 |
| Gamma-aminobutyric acid receptor subunit alpha-1 | Rattus norvegicus (Norway rat) | Ki | 10.8000 | 2 | 3 |
| Gamma-aminobutyric acid receptor subunit alpha-2 | Homo sapiens (human) | IC50 | 12.3027 | 1 | 1 |
| Gamma-aminobutyric acid receptor subunit alpha-2 | Rattus norvegicus (Norway rat) | IC50 | 12.3920 | 3 | 3 |
| Gamma-aminobutyric acid receptor subunit alpha-2 | Rattus norvegicus (Norway rat) | Ki | 10.8000 | 2 | 3 |
| Gamma-aminobutyric acid receptor subunit alpha-3 | Homo sapiens (human) | IC50 | 12.3027 | 1 | 1 |
| Gamma-aminobutyric acid receptor subunit alpha-3 | Rattus norvegicus (Norway rat) | IC50 | 12.3920 | 3 | 3 |
| Gamma-aminobutyric acid receptor subunit alpha-3 | Rattus norvegicus (Norway rat) | Ki | 10.8000 | 2 | 3 |
| Gamma-aminobutyric acid receptor subunit alpha-4 | Homo sapiens (human) | IC50 | 12.3027 | 1 | 1 |
| Gamma-aminobutyric acid receptor subunit alpha-4 | Rattus norvegicus (Norway rat) | IC50 | 12.3920 | 3 | 3 |
| Gamma-aminobutyric acid receptor subunit alpha-4 | Rattus norvegicus (Norway rat) | Ki | 10.8000 | 2 | 3 |
| Gamma-aminobutyric acid receptor subunit alpha-5 | Homo sapiens (human) | IC50 | 12.3027 | 1 | 1 |
| Gamma-aminobutyric acid receptor subunit alpha-5 | Rattus norvegicus (Norway rat) | IC50 | 12.3920 | 3 | 3 |
| Gamma-aminobutyric acid receptor subunit alpha-5 | Rattus norvegicus (Norway rat) | Ki | 10.8000 | 2 | 3 |
| Gamma-aminobutyric acid receptor subunit alpha-6 | Homo sapiens (human) | IC50 | 12.3027 | 1 | 1 |
| Gamma-aminobutyric acid receptor subunit alpha-6 | Rattus norvegicus (Norway rat) | IC50 | 12.3920 | 3 | 3 |
| Gamma-aminobutyric acid receptor subunit alpha-6 | Rattus norvegicus (Norway rat) | Ki | 10.8000 | 2 | 3 |
| Gamma-aminobutyric acid receptor subunit beta-1 | Homo sapiens (human) | IC50 | 12.3027 | 1 | 1 |
| Gamma-aminobutyric acid receptor subunit beta-1 | Rattus norvegicus (Norway rat) | IC50 | 12.3920 | 3 | 3 |
| Gamma-aminobutyric acid receptor subunit beta-1 | Rattus norvegicus (Norway rat) | Ki | 10.8000 | 2 | 3 |
| Gamma-aminobutyric acid receptor subunit beta-2 | Homo sapiens (human) | IC50 | 12.3027 | 1 | 1 |
| Gamma-aminobutyric acid receptor subunit beta-2 | Rattus norvegicus (Norway rat) | IC50 | 12.3920 | 3 | 3 |
| Gamma-aminobutyric acid receptor subunit beta-2 | Rattus norvegicus (Norway rat) | Ki | 10.8000 | 2 | 3 |
| Gamma-aminobutyric acid receptor subunit beta-3 | Homo sapiens (human) | IC50 | 12.3027 | 1 | 1 |
| Gamma-aminobutyric acid receptor subunit beta-3 | Rattus norvegicus (Norway rat) | IC50 | 12.3920 | 3 | 3 |
| Gamma-aminobutyric acid receptor subunit beta-3 | Rattus norvegicus (Norway rat) | Ki | 10.8000 | 2 | 3 |
| Gamma-aminobutyric acid receptor subunit delta | Homo sapiens (human) | IC50 | 12.3027 | 1 | 1 |
| Gamma-aminobutyric acid receptor subunit delta | Rattus norvegicus (Norway rat) | IC50 | 12.3920 | 3 | 3 |
| Gamma-aminobutyric acid receptor subunit delta | Rattus norvegicus (Norway rat) | Ki | 10.8000 | 2 | 3 |
| Gamma-aminobutyric acid receptor subunit epsilon | Homo sapiens (human) | IC50 | 12.3027 | 1 | 1 |
| Gamma-aminobutyric acid receptor subunit epsilon | Rattus norvegicus (Norway rat) | IC50 | 12.3920 | 3 | 3 |
| Gamma-aminobutyric acid receptor subunit epsilon | Rattus norvegicus (Norway rat) | Ki | 10.8000 | 2 | 3 |
| Gamma-aminobutyric acid receptor subunit gamma-1 | Homo sapiens (human) | IC50 | 12.3027 | 1 | 1 |
| Gamma-aminobutyric acid receptor subunit gamma-1 | Rattus norvegicus (Norway rat) | IC50 | 12.3920 | 3 | 3 |
| Gamma-aminobutyric acid receptor subunit gamma-1 | Rattus norvegicus (Norway rat) | Ki | 10.8000 | 2 | 3 |
| Gamma-aminobutyric acid receptor subunit gamma-2 | Homo sapiens (human) | IC50 | 12.3027 | 1 | 1 |
| Gamma-aminobutyric acid receptor subunit gamma-2 | Rattus norvegicus (Norway rat) | IC50 | 12.3920 | 3 | 3 |
| Gamma-aminobutyric acid receptor subunit gamma-2 | Rattus norvegicus (Norway rat) | Ki | 10.8000 | 2 | 3 |
| Gamma-aminobutyric acid receptor subunit gamma-3 | Homo sapiens (human) | IC50 | 12.3027 | 1 | 1 |
| Gamma-aminobutyric acid receptor subunit gamma-3 | Rattus norvegicus (Norway rat) | IC50 | 12.3920 | 3 | 3 |
| Gamma-aminobutyric acid receptor subunit gamma-3 | Rattus norvegicus (Norway rat) | Ki | 10.8000 | 2 | 3 |
| Gamma-aminobutyric acid receptor subunit pi | Homo sapiens (human) | IC50 | 12.3027 | 1 | 1 |
| Gamma-aminobutyric acid receptor subunit pi | Rattus norvegicus (Norway rat) | IC50 | 12.3920 | 3 | 3 |
| Gamma-aminobutyric acid receptor subunit pi | Rattus norvegicus (Norway rat) | Ki | 10.8000 | 2 | 3 |
| Gamma-aminobutyric acid receptor subunit theta | Homo sapiens (human) | IC50 | 12.3027 | 1 | 1 |
| Glycogen debranching enzyme | Homo sapiens (human) | IC50 | 10.0000 | 1 | 2 |
| Glycogen debranching enzyme | Oryctolagus cuniculus (rabbit) | IC50 | 0.1900 | 1 | 1 |
| Glycogen phosphorylase, muscle form | Oryctolagus cuniculus (rabbit) | IC50 | 42.9145 | 3 | 4 |
| Glycogen synthase kinase-3 alpha | Homo sapiens (human) | IC50 | 10.0000 | 3 | 3 |
| Glycogen synthase kinase-3 beta | Homo sapiens (human) | IC50 | 24.0333 | 6 | 6 |
| Glycogen synthase kinase-3 beta | Sus scrofa (pig) | IC50 | 12.2500 | 4 | 4 |
| Hexokinase-2 | Homo sapiens (human) | IC50 | 50.0000 | 1 | 1 |
| Histone deacetylase 1 | Homo sapiens (human) | IC50 | 5.5000 | 6 | 6 |
| Histone deacetylase 11 | Homo sapiens (human) | IC50 | 10.0000 | 3 | 3 |
| Histone deacetylase 2 | Homo sapiens (human) | IC50 | 10.0000 | 3 | 3 |
| Histone deacetylase 3 | Homo sapiens (human) | IC50 | 10.0000 | 3 | 3 |
| Histone deacetylase 4 | Homo sapiens (human) | IC50 | 10.0000 | 3 | 3 |
| Histone deacetylase 5 | Homo sapiens (human) | IC50 | 10.0000 | 3 | 3 |
| Histone deacetylase 6 | Homo sapiens (human) | IC50 | 10.0000 | 3 | 3 |
| Histone deacetylase 7 | Homo sapiens (human) | IC50 | 10.0000 | 3 | 3 |
| Histone deacetylase 8 | Homo sapiens (human) | IC50 | 10.0000 | 3 | 3 |
| Histone deacetylase 9 | Homo sapiens (human) | IC50 | 10.0000 | 3 | 3 |
| Kappa-type opioid receptor | Cavia porcellus (domestic guinea pig) | IC50 | 5.0360 | 2 | 2 |
| Lactase-phlorizin hydrolase | Homo sapiens (human) | IC50 | 81.0000 | 1 | 2 |
| Lactase-phlorizin hydrolase | Rattus norvegicus (Norway rat) | IC50 | 231.2333 | 3 | 6 |
| Low molecular weight phosphotyrosine protein phosphatase | Homo sapiens (human) | IC50 | 24.0000 | 2 | 2 |
| Lysosomal acid glucosylceramidase | Bos taurus (cattle) | IC50 | 210.0000 | 1 | 1 |
| Lysosomal acid glucosylceramidase | Homo sapiens (human) | IC50 | 244.9412 | 12 | 17 |
| Lysosomal acid glucosylceramidase | Homo sapiens (human) | Ki | 80.2500 | 3 | 4 |
| Lysosomal alpha-glucosidase | Homo sapiens (human) | IC50 | 43.7511 | 7 | 9 |
| Lysosomal alpha-glucosidase | Mus musculus (house mouse) | IC50 | 9.0000 | 1 | 1 |
| Lysosomal alpha-glucosidase | Rattus norvegicus (Norway rat) | IC50 | 1.4417 | 5 | 6 |
| Lysosomal alpha-glucosidase | Homo sapiens (human) | Ki | 6.3295 | 2 | 4 |
| Maltase-glucoamylase, intestinal | Homo sapiens (human) | IC50 | 25.4550 | 8 | 10 |
| Metabotropic glutamate receptor 1 | Rattus norvegicus (Norway rat) | Ki | 10.0000 | 1 | 1 |
| Metabotropic glutamate receptor 2 | Rattus norvegicus (Norway rat) | Ki | 10.0000 | 1 | 1 |
| Metabotropic glutamate receptor 3 | Rattus norvegicus (Norway rat) | Ki | 10.0000 | 1 | 1 |
| Metabotropic glutamate receptor 4 | Rattus norvegicus (Norway rat) | Ki | 10.0000 | 1 | 1 |
| Metabotropic glutamate receptor 5 | Rattus norvegicus (Norway rat) | Ki | 10.0000 | 1 | 1 |
| Metabotropic glutamate receptor 6 | Rattus norvegicus (Norway rat) | Ki | 10.0000 | 1 | 1 |
| Metabotropic glutamate receptor 7 | Rattus norvegicus (Norway rat) | Ki | 10.0000 | 1 | 1 |
| Metabotropic glutamate receptor 8 | Rattus norvegicus (Norway rat) | Ki | 10.0000 | 1 | 1 |
| Mitogen-activated protein kinase 1 | Rattus norvegicus (Norway rat) | IC50 | 30.0000 | 1 | 1 |
| Multidrug resistance-associated protein 4 | Homo sapiens (human) | IC50 | 133.0000 | 1 | 2 |
| Muscarinic acetylcholine receptor M1 | Homo sapiens (human) | Ki | 10.0000 | 1 | 1 |
| Muscarinic acetylcholine receptor M2 | Homo sapiens (human) | Ki | 10.0000 | 1 | 1 |
| Muscarinic acetylcholine receptor M3 | Homo sapiens (human) | Ki | 10.0000 | 1 | 1 |
| Muscarinic acetylcholine receptor M4 | Homo sapiens (human) | Ki | 10.0000 | 1 | 1 |
| Muscarinic acetylcholine receptor M5 | Homo sapiens (human) | Ki | 10.0000 | 1 | 1 |
| Neuromedin-B receptor | Homo sapiens (human) | Ki | 10.0000 | 1 | 1 |
| Neutral alpha-glucosidase AB | Homo sapiens (human) | IC50 | 472.8250 | 3 | 4 |
| Neutral alpha-glucosidase AB | Homo sapiens (human) | Ki | 410.0000 | 1 | 1 |
| Nischarin | Homo sapiens (human) | Ki | 6.9110 | 2 | 2 |
| Non-lysosomal glucosylceramidase | Homo sapiens (human) | IC50 | 25.5485 | 8 | 11 |
| Non-lysosomal glucosylceramidase | Mus musculus (house mouse) | IC50 | 11.5200 | 2 | 2 |
| Non-structural protein 1 | Dengue virus | IC50 | 1.7000 | 1 | 1 |
| Nuclear factor NF-kappa-B p105 subunit | Homo sapiens (human) | IC50 | 49.6000 | 1 | 1 |
| nuclear receptor subfamily 0 group B member 1 | Homo sapiens (human) | IC50 | 1.7290 | 1 | 1 |
| nucleotide-binding oligomerization domain-containing protein 2 isoform 1 | Homo sapiens (human) | IC50 | 8.0770 | 1 | 1 |
| Oligo-1,6-glucosidase IMA1 | Saccharomyces cerevisiae S288C | IC50 | 330.0000 | 1 | 1 |
| Oxysterols receptor LXR-alpha | Homo sapiens (human) | IC50 | 137.5000 | 3 | 4 |
| Oxysterols receptor LXR-beta | Homo sapiens (human) | IC50 | 150.0000 | 2 | 3 |
| Pancreatic alpha-amylase | Sus scrofa (pig) | IC50 | 200.0000 | 1 | 1 |
| Phosphodiesterase isozyme 4 | Homo sapiens (human) | IC50 | 125.0000 | 1 | 1 |
| Polyamine deacetylase HDAC10 | Homo sapiens (human) | IC50 | 10.0000 | 3 | 3 |
| Probable maltase-glucoamylase 2 | Homo sapiens (human) | IC50 | 115.7500 | 2 | 2 |
| Protease | Human immunodeficiency virus 1 | IC50 | 73.0417 | 3 | 3 |
| Protease | Human immunodeficiency virus 1 | Ki | 0.0003 | 13 | 13 |
| Protein kinase C alpha type | Homo sapiens (human) | IC50 | 250.0000 | 1 | 1 |
| Protein kinase C beta type | Homo sapiens (human) | IC50 | 183.3333 | 2 | 3 |
| Protein kinase C delta type | Homo sapiens (human) | IC50 | 250.0000 | 1 | 1 |
| Protein kinase C epsilon type | Homo sapiens (human) | IC50 | 183.3333 | 2 | 3 |
| Protein kinase C eta type | Homo sapiens (human) | IC50 | 250.0000 | 1 | 1 |
| Protein kinase C gamma type | Homo sapiens (human) | IC50 | 250.0000 | 1 | 1 |
| Protein kinase C iota type | Homo sapiens (human) | IC50 | 250.0000 | 1 | 1 |
| Protein kinase C theta type | Homo sapiens (human) | IC50 | 250.0000 | 1 | 1 |
| Protein kinase C zeta type | Homo sapiens (human) | IC50 | 250.0000 | 1 | 1 |
| Protein-lysine 6-oxidase | Homo sapiens (human) | IC50 | 39.2500 | 1 | 4 |
| Protein-lysine 6-oxidase | Homo sapiens (human) | Ki | 97.5000 | 1 | 2 |
| Proton-coupled amino acid transporter 1 | Homo sapiens (human) | Ki | 7,400.0000 | 1 | 1 |
| Putative alpha-glucosidase | Oryza sativa Japonica Group (Japanese rice) | IC50 | 0.1667 | 2 | 3 |
| Receptor-type tyrosine-protein phosphatase F | Homo sapiens (human) | IC50 | 45.6000 | 1 | 1 |
| Replicase polyprotein 1ab | Severe acute respiratory syndrome coronavirus 2 | IC50 | 15.0000 | 1 | 1 |
| Serine/threonine-protein kinase D1 | Homo sapiens (human) | IC50 | 250.0000 | 1 | 1 |
| Serine/threonine-protein kinase D3 | Homo sapiens (human) | IC50 | 250.0000 | 1 | 1 |
| Serine/threonine-protein kinase haspin | Homo sapiens (human) | IC50 | 0.5900 | 1 | 1 |
| Serine/threonine-protein kinase pim-1 | Homo sapiens (human) | IC50 | 10.0000 | 1 | 1 |
| Serine/threonine-protein kinase pim-3 | Homo sapiens (human) | IC50 | 4.3000 | 1 | 1 |
| Sodium-dependent dopamine transporter | Bos taurus (cattle) | Ki | 10.0000 | 1 | 1 |
| Sodium-dependent noradrenaline transporter | Homo sapiens (human) | Ki | 3.2600 | 1 | 1 |
| Sodium-dependent serotonin transporter | Homo sapiens (human) | Ki | 10.0000 | 1 | 1 |
| Solute carrier family 22 member 6 | Homo sapiens (human) | IC50 | 60.0000 | 1 | 1 |
| steroidogenic factor 1 | Homo sapiens (human) | IC50 | 67.5470 | 1 | 1 |
| Sterol O-acyltransferase 1 | Homo sapiens (human) | IC50 | 96.0000 | 1 | 1 |
| Sterol O-acyltransferase 2 | Homo sapiens (human) | IC50 | 112.0000 | 1 | 1 |
| Sucrase-isomaltase | Mus musculus (house mouse) | IC50 | 1.0500 | 2 | 2 |
| Sucrase-isomaltase, intestinal | Homo sapiens (human) | IC50 | 58.5000 | 3 | 4 |
| Sucrase-isomaltase, intestinal | Rattus norvegicus (Norway rat) | IC50 | 5.9170 | 17 | 23 |
| SUMO-conjugating enzyme UBC9 | Homo sapiens (human) | IC50 | 11.2000 | 2 | 2 |
| SUMO1 activating enzyme subunit 1 | Homo sapiens (human) | IC50 | 11.2000 | 2 | 2 |
| Thymidine kinase | Macacine alphaherpesvirus 1 | IC50 | 900.0000 | 1 | 1 |
| Transcription factor p65 | Homo sapiens (human) | IC50 | 10.0000 | 1 | 1 |
| Translocator protein | Rattus norvegicus (Norway rat) | IC50 | 12.3880 | 1 | 1 |
| Transporter | Rattus norvegicus (Norway rat) | Ki | 3.2600 | 1 | 1 |
| Trehalase | Homo sapiens (human) | IC50 | 40.0000 | 1 | 1 |
| Trehalase | Rattus norvegicus (Norway rat) | IC50 | 34.0000 | 3 | 6 |
| Trehalase | Sus scrofa (pig) | IC50 | 39.3333 | 2 | 3 |
| Trehalose synthase/amylase TreS | Mycobacterium tuberculosis CDC1551 | Ki | 0.2500 | 1 | 1 |
| Tryptophan 2,3-dioxygenase | Homo sapiens (human) | IC50 | 6.3100 | 1 | 1 |
| tumor necrosis factor | Homo sapiens (human) | IC50 | 10.8800 | 1 | 1 |
| Tyrosine-protein kinase Fyn | Homo sapiens (human) | IC50 | 250.0000 | 1 | 1 |
| Tyrosine-protein kinase Lck | Homo sapiens (human) | IC50 | 250.0000 | 1 | 1 |
| Tyrosine-protein kinase Lyn | Homo sapiens (human) | IC50 | 250.0000 | 1 | 1 |
| Tyrosine-protein phosphatase non-receptor type 1 | Homo sapiens (human) | IC50 | 9.3000 | 3 | 3 |
| Tyrosine-protein phosphatase non-receptor type 1 | Homo sapiens (human) | Ki | 8.0000 | 1 | 1 |
| Ubiquitin-like modifier activating enzyme 2 | Homo sapiens (human) | IC50 | 11.2000 | 2 | 2 |
| Zinc finger protein GLI1 | Homo sapiens (human) | IC50 | 32.0000 | 2 | 2 |