Page last updated: 2024-08-07 15:19:55

dual specificity protein kinase CLK4

[no definition available]

Synonyms

Research

Bioassay Publications (0)

TimeframeStudies on this Protein(%)All Drugs %
pre-19900 (0)18.7374
1990's0 (0)18.2507
2000's0 (0)29.6817
2010's0 (0)24.3611
2020's0 (0)2.80

Compounds (46)

Drugs with Potency Measurements

DrugTaxonomyMeasurementAverage (mM)Bioassay(s)Publication(s)
2-(4-amino-5-iodo-7-pyrrolo[2,3-d]pyrimidinyl)-5-(hydroxymethyl)oxolane-3,4-diolHomo sapiens (human)Potency0.011610
erlotinibHomo sapiens (human)Potency20.666510
tg 003Homo sapiens (human)Potency0.040020
ml106Homo sapiens (human)Potency0.053150
6-(1,3-benzodioxol-5-yl)-N-(2-furanylmethyl)-N-methyl-4-quinazolinamineHomo sapiens (human)Potency0.046130
N-(2-furanylmethyl)-6-(3-methoxyphenyl)-N-methyl-4-quinazolinamineHomo sapiens (human)Potency0.922660
6-(1,3-benzodioxol-5-yl)-N-[(3-methylphenyl)methyl]-4-quinazolinamineHomo sapiens (human)Potency0.108130
6-(2-chlorophenyl)-N-(3-pyridinylmethyl)-4-quinazolinamineHomo sapiens (human)Potency11.066560
6-(3-furanyl)-N-[(3-methylphenyl)methyl]-4-quinazolinamineHomo sapiens (human)Potency0.244230
6-(3-pyridinyl)-N-(3-pyridinylmethyl)-4-quinazolinamineHomo sapiens (human)Potency9.492030
6-(3-furanyl)-N-(thiophen-2-ylmethyl)-4-quinazolinamineHomo sapiens (human)Potency0.219260
6-(3-methoxyphenyl)-N-(3-pyridinylmethyl)-4-quinazolinamineHomo sapiens (human)Potency2.602260
6-(2-chlorophenyl)-N-(2-furanylmethyl)-N-methyl-4-quinazolinamineHomo sapiens (human)Potency11.859360
6-(3-methoxyphenyl)-N-(thiophen-2-ylmethyl)-4-quinazolinamineHomo sapiens (human)Potency0.880430
6-(3-furanyl)-N-(3-pyridinylmethyl)-4-quinazolinamineHomo sapiens (human)Potency1.231860
N-[(3-methylphenyl)methyl]-6-(3-pyridinyl)-4-quinazolinamineHomo sapiens (human)Potency3.792830
harmineHomo sapiens (human)Potency0.067110
N-(2-furanylmethyl)-N-methyl-6-(1-methyl-5-indolyl)-4-quinazolinamineHomo sapiens (human)Potency17.277930
6-(2-chlorophenyl)-N-[(3-methylphenyl)methyl]-4-quinazolinamineHomo sapiens (human)Potency9.815030
6-(3-methoxyphenyl)-N-[(3-methylphenyl)methyl]-4-quinazolinamineHomo sapiens (human)Potency1.309530
6-(2,3-dihydro-1,4-benzodioxin-6-yl)-N-[(3-methylphenyl)methyl]-4-quinazolinamineHomo sapiens (human)Potency0.590530
6-(2-chlorophenyl)-N-(thiophen-2-ylmethyl)-4-quinazolinamineHomo sapiens (human)Potency7.110830
6-(3-chlorophenyl)-N-(thiophen-2-ylmethyl)-4-quinazolinamineHomo sapiens (human)Potency6.622630
6-(3-pyridinyl)-N-(thiophen-2-ylmethyl)-4-quinazolinamineHomo sapiens (human)Potency4.741030
6-(3-methylphenyl)-N-(thiophen-2-ylmethyl)-4-quinazolinamineHomo sapiens (human)Potency10.290630
6-(1-methyl-5-indolyl)-N-(thiophen-2-ylmethyl)-4-quinazolinamineHomo sapiens (human)Potency24.644030
6-(2,3-dihydro-1,4-benzodioxin-6-yl)-N-(thiophen-2-ylmethyl)-4-quinazolinamineHomo sapiens (human)Potency0.137330
N-(1,3-benzodioxol-5-ylmethyl)-6-(2,3-dihydro-1,4-benzodioxin-6-yl)-4-quinazolinamineHomo sapiens (human)Potency2.085230
6-(2,3-dihydro-1,4-benzodioxin-6-yl)-N-(3-pyridinylmethyl)-4-quinazolinamineHomo sapiens (human)Potency0.517630
6-(1,3-benzodioxol-5-yl)-N-[(3-fluorophenyl)methyl]-4-quinazolinamineHomo sapiens (human)Potency0.110130
6-(3-chlorophenyl)-N-(3-pyridinylmethyl)-4-quinazolinamineHomo sapiens (human)Potency3.815230
6-(3-methylphenyl)-N-(3-pyridinylmethyl)-4-quinazolinamineHomo sapiens (human)Potency7.796430
6-(1,3-benzodioxol-5-yl)-N-(3-pyridinylmethyl)-4-quinazolinamineHomo sapiens (human)Potency0.105030
N-(1,3-benzodioxol-5-ylmethyl)-6-(2-chlorophenyl)-4-quinazolinamineHomo sapiens (human)Potency11.034420
N-(1,3-benzodioxol-5-ylmethyl)-6-(3-methoxyphenyl)-4-quinazolinamineHomo sapiens (human)Potency1.636730
N-(1,3-benzodioxol-5-ylmethyl)-6-(3-pyridinyl)-4-quinazolinamineHomo sapiens (human)Potency8.203130
N-(1,3-benzodioxol-5-ylmethyl)-6-(3-furanyl)-4-quinazolinamineHomo sapiens (human)Potency0.743430
6-(2-chlorophenyl)-N-[(4-methyl-2-thiophenyl)methyl]-4-quinazolinamineHomo sapiens (human)Potency10.044230
6-(3-chlorophenyl)-N-[(4-methyl-2-thiophenyl)methyl]-4-quinazolinamineHomo sapiens (human)Potency9.492030
6-(3-methoxyphenyl)-N-[(4-methyl-2-thiophenyl)methyl]-4-quinazolinamineHomo sapiens (human)Potency0.981530
N-[(4-methyl-2-thiophenyl)methyl]-6-(3-pyridinyl)-4-quinazolinamineHomo sapiens (human)Potency6.717930
6-(1,3-benzodioxol-5-yl)-N-[(4-methyl-2-thiophenyl)methyl]-4-quinazolinamineHomo sapiens (human)Potency0.152830
6-(2,3-dihydro-1,4-benzodioxin-6-yl)-N-[(4-methyl-2-thiophenyl)methyl]-4-quinazolinamineHomo sapiens (human)Potency0.485230
6-(3-furanyl)-N-[(4-methyl-2-thiophenyl)methyl]-4-quinazolinamineHomo sapiens (human)Potency0.493130
6-(1,3-benzodioxol-5-yl)-N-methyl-N-(thiophen-2-ylmethyl)-4-quinazolinamineHomo sapiens (human)Potency0.021020
[5-[4-[(5-methyl-2-furanyl)methylamino]-6-quinazolinyl]-2-furanyl]methanolHomo sapiens (human)Potency0.186330