Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
2-(4-amino-5-iodo-7-pyrrolo[2,3-d]pyrimidinyl)-5-(hydroxymethyl)oxolane-3,4-diol | Homo sapiens (human) | Potency | 0.0116 | 1 | 0 |
erlotinib | Homo sapiens (human) | Potency | 20.6665 | 1 | 0 |
tg 003 | Homo sapiens (human) | Potency | 0.0400 | 2 | 0 |
ml106 | Homo sapiens (human) | Potency | 0.0531 | 5 | 0 |
6-(1,3-benzodioxol-5-yl)-N-(2-furanylmethyl)-N-methyl-4-quinazolinamine | Homo sapiens (human) | Potency | 0.0461 | 3 | 0 |
N-(2-furanylmethyl)-6-(3-methoxyphenyl)-N-methyl-4-quinazolinamine | Homo sapiens (human) | Potency | 0.9226 | 6 | 0 |
6-(1,3-benzodioxol-5-yl)-N-[(3-methylphenyl)methyl]-4-quinazolinamine | Homo sapiens (human) | Potency | 0.1081 | 3 | 0 |
6-(2-chlorophenyl)-N-(3-pyridinylmethyl)-4-quinazolinamine | Homo sapiens (human) | Potency | 11.0665 | 6 | 0 |
6-(3-furanyl)-N-[(3-methylphenyl)methyl]-4-quinazolinamine | Homo sapiens (human) | Potency | 0.2442 | 3 | 0 |
6-(3-pyridinyl)-N-(3-pyridinylmethyl)-4-quinazolinamine | Homo sapiens (human) | Potency | 9.4920 | 3 | 0 |
6-(3-furanyl)-N-(thiophen-2-ylmethyl)-4-quinazolinamine | Homo sapiens (human) | Potency | 0.2192 | 6 | 0 |
6-(3-methoxyphenyl)-N-(3-pyridinylmethyl)-4-quinazolinamine | Homo sapiens (human) | Potency | 2.6022 | 6 | 0 |
6-(2-chlorophenyl)-N-(2-furanylmethyl)-N-methyl-4-quinazolinamine | Homo sapiens (human) | Potency | 11.8593 | 6 | 0 |
6-(3-methoxyphenyl)-N-(thiophen-2-ylmethyl)-4-quinazolinamine | Homo sapiens (human) | Potency | 0.8804 | 3 | 0 |
6-(3-furanyl)-N-(3-pyridinylmethyl)-4-quinazolinamine | Homo sapiens (human) | Potency | 1.2318 | 6 | 0 |
N-[(3-methylphenyl)methyl]-6-(3-pyridinyl)-4-quinazolinamine | Homo sapiens (human) | Potency | 3.7928 | 3 | 0 |
harmine | Homo sapiens (human) | Potency | 0.0671 | 1 | 0 |
N-(2-furanylmethyl)-N-methyl-6-(1-methyl-5-indolyl)-4-quinazolinamine | Homo sapiens (human) | Potency | 17.2779 | 3 | 0 |
6-(2-chlorophenyl)-N-[(3-methylphenyl)methyl]-4-quinazolinamine | Homo sapiens (human) | Potency | 9.8150 | 3 | 0 |
6-(3-methoxyphenyl)-N-[(3-methylphenyl)methyl]-4-quinazolinamine | Homo sapiens (human) | Potency | 1.3095 | 3 | 0 |
6-(2,3-dihydro-1,4-benzodioxin-6-yl)-N-[(3-methylphenyl)methyl]-4-quinazolinamine | Homo sapiens (human) | Potency | 0.5905 | 3 | 0 |
6-(2-chlorophenyl)-N-(thiophen-2-ylmethyl)-4-quinazolinamine | Homo sapiens (human) | Potency | 7.1108 | 3 | 0 |
6-(3-chlorophenyl)-N-(thiophen-2-ylmethyl)-4-quinazolinamine | Homo sapiens (human) | Potency | 6.6226 | 3 | 0 |
6-(3-pyridinyl)-N-(thiophen-2-ylmethyl)-4-quinazolinamine | Homo sapiens (human) | Potency | 4.7410 | 3 | 0 |
6-(3-methylphenyl)-N-(thiophen-2-ylmethyl)-4-quinazolinamine | Homo sapiens (human) | Potency | 10.2906 | 3 | 0 |
6-(1-methyl-5-indolyl)-N-(thiophen-2-ylmethyl)-4-quinazolinamine | Homo sapiens (human) | Potency | 24.6440 | 3 | 0 |
6-(2,3-dihydro-1,4-benzodioxin-6-yl)-N-(thiophen-2-ylmethyl)-4-quinazolinamine | Homo sapiens (human) | Potency | 0.1373 | 3 | 0 |
N-(1,3-benzodioxol-5-ylmethyl)-6-(2,3-dihydro-1,4-benzodioxin-6-yl)-4-quinazolinamine | Homo sapiens (human) | Potency | 2.0852 | 3 | 0 |
6-(2,3-dihydro-1,4-benzodioxin-6-yl)-N-(3-pyridinylmethyl)-4-quinazolinamine | Homo sapiens (human) | Potency | 0.5176 | 3 | 0 |
6-(1,3-benzodioxol-5-yl)-N-[(3-fluorophenyl)methyl]-4-quinazolinamine | Homo sapiens (human) | Potency | 0.1101 | 3 | 0 |
6-(3-chlorophenyl)-N-(3-pyridinylmethyl)-4-quinazolinamine | Homo sapiens (human) | Potency | 3.8152 | 3 | 0 |
6-(3-methylphenyl)-N-(3-pyridinylmethyl)-4-quinazolinamine | Homo sapiens (human) | Potency | 7.7964 | 3 | 0 |
6-(1,3-benzodioxol-5-yl)-N-(3-pyridinylmethyl)-4-quinazolinamine | Homo sapiens (human) | Potency | 0.1050 | 3 | 0 |
N-(1,3-benzodioxol-5-ylmethyl)-6-(2-chlorophenyl)-4-quinazolinamine | Homo sapiens (human) | Potency | 11.0344 | 2 | 0 |
N-(1,3-benzodioxol-5-ylmethyl)-6-(3-methoxyphenyl)-4-quinazolinamine | Homo sapiens (human) | Potency | 1.6367 | 3 | 0 |
N-(1,3-benzodioxol-5-ylmethyl)-6-(3-pyridinyl)-4-quinazolinamine | Homo sapiens (human) | Potency | 8.2031 | 3 | 0 |
N-(1,3-benzodioxol-5-ylmethyl)-6-(3-furanyl)-4-quinazolinamine | Homo sapiens (human) | Potency | 0.7434 | 3 | 0 |
6-(2-chlorophenyl)-N-[(4-methyl-2-thiophenyl)methyl]-4-quinazolinamine | Homo sapiens (human) | Potency | 10.0442 | 3 | 0 |
6-(3-chlorophenyl)-N-[(4-methyl-2-thiophenyl)methyl]-4-quinazolinamine | Homo sapiens (human) | Potency | 9.4920 | 3 | 0 |
6-(3-methoxyphenyl)-N-[(4-methyl-2-thiophenyl)methyl]-4-quinazolinamine | Homo sapiens (human) | Potency | 0.9815 | 3 | 0 |
N-[(4-methyl-2-thiophenyl)methyl]-6-(3-pyridinyl)-4-quinazolinamine | Homo sapiens (human) | Potency | 6.7179 | 3 | 0 |
6-(1,3-benzodioxol-5-yl)-N-[(4-methyl-2-thiophenyl)methyl]-4-quinazolinamine | Homo sapiens (human) | Potency | 0.1528 | 3 | 0 |
6-(2,3-dihydro-1,4-benzodioxin-6-yl)-N-[(4-methyl-2-thiophenyl)methyl]-4-quinazolinamine | Homo sapiens (human) | Potency | 0.4852 | 3 | 0 |
6-(3-furanyl)-N-[(4-methyl-2-thiophenyl)methyl]-4-quinazolinamine | Homo sapiens (human) | Potency | 0.4931 | 3 | 0 |
6-(1,3-benzodioxol-5-yl)-N-methyl-N-(thiophen-2-ylmethyl)-4-quinazolinamine | Homo sapiens (human) | Potency | 0.0210 | 2 | 0 |
[5-[4-[(5-methyl-2-furanyl)methylamino]-6-quinazolinyl]-2-furanyl]methanol | Homo sapiens (human) | Potency | 0.1863 | 3 | 0 |