An EC 1.4.3.* (oxidoreductase acting on donor CH-NH2 group, oxygen as acceptor) inhibitor that interferes with the action of monoamine oxidase (EC 1.4.3.4).
| Member | Definition | Class |
|---|
| 4-chloro-7-nitrobenzofurazan | A benzoxadiazole that is 2,1,3-benzoxadiazole which is substituted at position 4 by chlorine and at position 7 by a nitro group. | 4-chloro-7-nitrobenzofurazan |
| 4-cyanophenol | | 4-cyanophenol |
| 8-(3-chlorostyryl)caffeine | Caffeine substituted at its 8-position by an (E)-3-chlorostyryl group. | 8-(3-chlorostyryl)caffeine |
| amezinium | A pyridazinium ion that is pyridazin-1-ium which is substituted by a phenyl, amino and methoxy groups at positions 1, 4 and 6, respectively. | amezinium |
| clorgyline | An aromatic ether that is the 2,4-dichlorophenyl ether of 3-aminopropan-1-ol in which the nitrogen is substituted by a methyl group and a prop-1-yn-3-yl group. A monoamine oxidase inhibitor, it was formerly used as an antidepressant. | clorgyline |
| furazolidone | A member of the class of oxazolidines that is 1,3-oxazolidin-2-one in which the hydrogen attached to the nitrogen is replaced by an N-{[(5-nitro-2-furyl)methylene]amino} group. It has antibacterial and antiprotozoal properties, and is used in the treatment of giardiasis and cholera. | furazolidone |
| harmalol | A harmala alkaloid in which the harman skeleton is hydroxy-substituted at C-7 and has been reduced across the 3,4 bond. | harmalol |
| harman | An indole alkaloid fundamental parent with a structure of 9H-beta-carboline carrying a methyl substituent at C-1. It has been isolated from the bark of Sickingia rubra, Symplocus racemosa, Passiflora incarnata, Peganum harmala, Banisteriopsis caapi and Tribulus terrestris, as well as from tobacco smoke. It is a specific, reversible inhibitor of monoamine oxidase A. | harman |
| harmine | A harmala alkaloid in which the harman skeleton is methoxy-substituted at C-7. | harmine |
| isatin | An indoledione that is the 2,3-diketo derivative of indole. | isatin |
| isogentisin | A member of the class of xanthones that is 9H-xanthen-9-one substituted by hydroxy groups at positions 1 and 3 and a methoxy group at position 7. | isogentisin |
| licocoumarone | A member of the class of 1-benzofurans which consists of 1-benzofuran substituted by a hydroxy group at position 6, a methoxy group at position 4, a prenyl group at position 5 and a 2,4-dihydroxyphenyl group at position 2. It has been isolated from Glycyrrhiza uralensis. | licocoumarone |
| methylene blue | An organic chloride salt having 3,7-bis(dimethylamino)phenothiazin-5-ium as the counterion. A commonly used dye that also exhibits antioxidant, antimalarial, antidepressant and cardioprotective properties. | methylene blue |
| monocrotophos | An alkenyl phosphate that is the 4-(methylamino)-4-oxobut-2-en-2-yl ester of dimethyl phosphate. | monocrotophos |
| pimagedine | A one-carbon compound whose unique structure renders it capable of acting as a derivative of hydrazine, guanidine or formamide. | aminoguanidine |
| rasagiline | An indane that consists of 1-aminoindane bearing an N-propargyl substituent. A selective, irreversible monoamine oxidase-B inhibitor. | rasagiline |
| selegiline hydrochloride, (r)-isomer | | selegiline hydrochloride |
| tetrindole | A racemate composed of equimolar amounts of (R)- and (S)-tetrindole hydrochloride. | tetrindole hydrochloride |
| Protein | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Drugs |
|---|
| 15-hydroxyprostaglandin dehydrogenase [NAD(+)] isoform 1 | Homo sapiens (human) | Potency | 21.1705 | 1 | 12 |
| 67.9K protein | Vaccinia virus | Potency | 18.6649 | 2 | 3 |
| acetylcholinesterase | Homo sapiens (human) | Potency | 14.7177 | 4 | 11 |
| activating transcription factor 6 | Homo sapiens (human) | Potency | 0.4364 | 1 | 1 |
| aldehyde dehydrogenase 1 family, member A1 | Homo sapiens (human) | Potency | 19.3223 | 1 | 15 |
| alpha-galactosidase | Homo sapiens (human) | Potency | 4.8022 | 1 | 2 |
| Alpha-synuclein | Homo sapiens (human) | Potency | 15.8489 | 1 | 1 |
| AR protein | Homo sapiens (human) | Potency | 3.3117 | 7 | 11 |
| aryl hydrocarbon receptor | Homo sapiens (human) | Potency | 12.6568 | 2 | 6 |
| arylsulfatase A | Homo sapiens (human) | Potency | 12.7181 | 1 | 2 |
| ATAD5 protein, partial | Homo sapiens (human) | Potency | 10.1715 | 2 | 3 |
| Ataxin-2 | Homo sapiens (human) | Potency | 14.9601 | 1 | 1 |
| ATP-dependent phosphofructokinase | Trypanosoma brucei brucei TREU927 | Potency | 19.3450 | 2 | 2 |
| ATPase family AAA domain-containing protein 5 | Homo sapiens (human) | Potency | 14.9601 | 1 | 1 |
| Bloom syndrome protein isoform 1 | Homo sapiens (human) | Potency | 23.9274 | 2 | 5 |
| bromodomain adjacent to zinc finger domain 2B | Homo sapiens (human) | Potency | 39.8107 | 1 | 1 |
| caspase 7, apoptosis-related cysteine protease | Homo sapiens (human) | Potency | 10.8707 | 1 | 1 |
| caspase-1 isoform alpha precursor | Homo sapiens (human) | Potency | 15.8489 | 1 | 1 |
| caspase-3 | Homo sapiens (human) | Potency | 10.8707 | 1 | 1 |
| Caspase-7 | Homo sapiens (human) | Potency | 12.5893 | 1 | 1 |
| Cellular tumor antigen p53 | Homo sapiens (human) | Potency | 11.9895 | 2 | 3 |
| Chain A, 2-oxoglutarate Oxygenase | Homo sapiens (human) | Potency | 23.9580 | 1 | 12 |
| Chain A, ATP-DEPENDENT DNA HELICASE Q1 | Homo sapiens (human) | Potency | 26.3648 | 2 | 3 |
| Chain A, Breast cancer type 1 susceptibility protein | Homo sapiens (human) | Potency | 31.6228 | 1 | 1 |
| Chain A, Cruzipain | Trypanosoma cruzi | Potency | 28.7994 | 2 | 8 |
| Chain A, Ferritin light chain | Equus caballus (horse) | Potency | 30.7246 | 2 | 6 |
| Chain A, HADH2 protein | Homo sapiens (human) | Potency | 20.3246 | 2 | 9 |
| Chain A, JmjC domain-containing histone demethylation protein 3A | Homo sapiens (human) | Potency | 44.6684 | 1 | 1 |
| Chain A, MAJOR APURINIC/APYRIMIDINIC ENDONUCLEASE | Homo sapiens (human) | Potency | 26.2529 | 2 | 12 |
| Chain A, Putative fructose-1,6-bisphosphate aldolase | Giardia intestinalis | Potency | 22.3342 | 1 | 1 |
| Chain A, TYROSYL-DNA PHOSPHODIESTERASE | Homo sapiens (human) | Potency | 29.2756 | 2 | 3 |
| Chain B, HADH2 protein | Homo sapiens (human) | Potency | 20.3246 | 2 | 9 |
| chaperonin-containing TCP-1 beta subunit homolog | Homo sapiens (human) | Potency | 22.3872 | 1 | 1 |
| chromobox protein homolog 1 | Homo sapiens (human) | Potency | 92.7501 | 2 | 3 |
| cytochrome P450 2C19 precursor | Homo sapiens (human) | Potency | 3.7619 | 1 | 2 |
| cytochrome P450 2C9, partial | Homo sapiens (human) | Potency | 0.6918 | 1 | 1 |
| cytochrome P450 2D6 | Homo sapiens (human) | Potency | 7.0960 | 1 | 2 |
| cytochrome P450 2D6 isoform 1 | Homo sapiens (human) | Potency | 13.3689 | 1 | 7 |
| cytochrome P450 3A4 isoform 1 | Homo sapiens (human) | Potency | 18.6516 | 2 | 14 |
| cytochrome P450 family 3 subfamily A polypeptide 4 | Homo sapiens (human) | Potency | 0.4897 | 1 | 1 |
| cytochrome P450, family 19, subfamily A, polypeptide 1, isoform CRA_a | Homo sapiens (human) | Potency | 4.9354 | 1 | 2 |
| DNA dC->dU-editing enzyme APOBEC-3G isoform 1 | Homo sapiens (human) | Potency | 21.1360 | 1 | 1 |
| DNA polymerase beta | Homo sapiens (human) | Potency | 25.1189 | 1 | 1 |
| DNA polymerase eta isoform 1 | Homo sapiens (human) | Potency | 56.2341 | 1 | 1 |
| DNA polymerase iota isoform a (long) | Homo sapiens (human) | Potency | 64.5194 | 1 | 3 |
| DNA polymerase kappa isoform 1 | Homo sapiens (human) | Potency | 12.5893 | 1 | 1 |
| dual specificity protein kinase CLK4 | Homo sapiens (human) | Potency | 0.0671 | 1 | 1 |
| estrogen nuclear receptor alpha | Homo sapiens (human) | Potency | 30.7609 | 8 | 15 |
| estrogen receptor 2 (ER beta) | Homo sapiens (human) | Potency | 14.5560 | 2 | 2 |
| estrogen-related nuclear receptor alpha | Homo sapiens (human) | Potency | 6.7374 | 9 | 17 |
| euchromatic histone-lysine N-methyltransferase 2 | Homo sapiens (human) | Potency | 45.0766 | 1 | 4 |
| farnesoid X nuclear receptor | Homo sapiens (human) | Potency | 15.1422 | 1 | 2 |
| flap endonuclease 1 | Homo sapiens (human) | Potency | 25.4461 | 1 | 3 |
| Fumarate hydratase | Homo sapiens (human) | Potency | 17.7828 | 1 | 1 |
| G | Vesicular stomatitis virus | Potency | 0.6918 | 1 | 1 |
| GABA theta subunit | Rattus norvegicus (Norway rat) | Potency | 18.6516 | 1 | 7 |
| Gamma-aminobutyric acid receptor subunit alpha-1 | Rattus norvegicus (Norway rat) | Potency | 18.6516 | 1 | 7 |
| Gamma-aminobutyric acid receptor subunit alpha-2 | Rattus norvegicus (Norway rat) | Potency | 18.6516 | 1 | 7 |
| Gamma-aminobutyric acid receptor subunit alpha-3 | Rattus norvegicus (Norway rat) | Potency | 18.6516 | 1 | 7 |
| Gamma-aminobutyric acid receptor subunit alpha-4 | Rattus norvegicus (Norway rat) | Potency | 18.6516 | 1 | 7 |
| Gamma-aminobutyric acid receptor subunit alpha-5 | Rattus norvegicus (Norway rat) | Potency | 18.6516 | 1 | 7 |
| Gamma-aminobutyric acid receptor subunit alpha-6 | Rattus norvegicus (Norway rat) | Potency | 18.6516 | 1 | 7 |
| Gamma-aminobutyric acid receptor subunit beta-1 | Rattus norvegicus (Norway rat) | Potency | 18.6516 | 1 | 7 |
| Gamma-aminobutyric acid receptor subunit beta-2 | Rattus norvegicus (Norway rat) | Potency | 18.6516 | 1 | 7 |
| Gamma-aminobutyric acid receptor subunit beta-3 | Rattus norvegicus (Norway rat) | Potency | 18.6516 | 1 | 7 |
| Gamma-aminobutyric acid receptor subunit delta | Rattus norvegicus (Norway rat) | Potency | 18.6516 | 1 | 7 |
| Gamma-aminobutyric acid receptor subunit epsilon | Rattus norvegicus (Norway rat) | Potency | 18.6516 | 1 | 7 |
| Gamma-aminobutyric acid receptor subunit gamma-1 | Rattus norvegicus (Norway rat) | Potency | 18.6516 | 1 | 7 |
| Gamma-aminobutyric acid receptor subunit gamma-2 | Rattus norvegicus (Norway rat) | Potency | 18.6516 | 1 | 7 |
| Gamma-aminobutyric acid receptor subunit gamma-3 | Rattus norvegicus (Norway rat) | Potency | 18.6516 | 1 | 7 |
| Gamma-aminobutyric acid receptor subunit pi | Rattus norvegicus (Norway rat) | Potency | 18.6516 | 1 | 7 |
| geminin | Homo sapiens (human) | Potency | 11.9675 | 1 | 3 |
| GLI family zinc finger 3 | Homo sapiens (human) | Potency | 6.5276 | 2 | 6 |
| glp-1 receptor, partial | Homo sapiens (human) | Potency | 6.3096 | 1 | 1 |
| glucocorticoid receptor [Homo sapiens] | Homo sapiens (human) | Potency | 13.8062 | 2 | 2 |
| Glutamate receptor 2 | Rattus norvegicus (Norway rat) | Potency | 28.5776 | 1 | 2 |
| Glycoprotein hormones alpha chain | Homo sapiens (human) | Potency | 0.5012 | 1 | 1 |
| Guanine nucleotide-binding protein G | Homo sapiens (human) | Potency | 22.7406 | 1 | 2 |
| heat shock protein beta-1 | Homo sapiens (human) | Potency | 58.2929 | 2 | 2 |
| Histamine H2 receptor | Cavia porcellus (domestic guinea pig) | Potency | 15.8489 | 1 | 4 |
| histone acetyltransferase KAT2A isoform 1 | Homo sapiens (human) | Potency | 15.8489 | 1 | 1 |
| histone deacetylase 9 isoform 3 | Homo sapiens (human) | Potency | 12.3066 | 2 | 4 |
| Histone H2A.x | Cricetulus griseus (Chinese hamster) | Potency | 34.5673 | 2 | 5 |
| histone-lysine N-methyltransferase 2A isoform 2 precursor | Homo sapiens (human) | Potency | 19.9526 | 1 | 1 |
| HLA class I histocompatibility antigen, B alpha chain | Homo sapiens (human) | Potency | 0.6918 | 1 | 1 |
| huntingtin isoform 2 | Homo sapiens (human) | Potency | 12.5893 | 1 | 1 |
| hypothetical protein, conserved | Trypanosoma brucei | Potency | 19.9526 | 1 | 1 |
| hypoxia-inducible factor 1 alpha subunit | Homo sapiens (human) | Potency | 42.2707 | 2 | 3 |
| hypoxia-inducible factor 1, alpha subunit (basic helix-loop-helix transcription factor) | Homo sapiens (human) | Potency | 15.7142 | 2 | 4 |
| IDH1 | Homo sapiens (human) | Potency | 7.3078 | 1 | 1 |
| Inositol hexakisphosphate kinase 1 | Homo sapiens (human) | Potency | 0.6918 | 1 | 2 |
| Inositol monophosphatase 1 | Rattus norvegicus (Norway rat) | Potency | 15.9145 | 2 | 3 |
| Interferon beta | Homo sapiens (human) | Potency | 17.9313 | 3 | 5 |
| isocitrate dehydrogenase 1, partial | Homo sapiens (human) | Potency | 52.1194 | 1 | 1 |
| lethal factor (plasmid) | Bacillus anthracis str. A2012 | Potency | 16.9382 | 1 | 4 |
| Luciferase | Photinus pyralis (common eastern firefly) | Potency | 17.4943 | 2 | 3 |
| luciferase | Photuris pensylvanica (Pennsylania firefly) | Potency | 10.0000 | 1 | 1 |
| luteinizing hormone receptor | Homo sapiens (human) | Potency | 84.9214 | 1 | 1 |
| Microtubule-associated protein tau | Homo sapiens (human) | Potency | 6.6416 | 2 | 5 |
| mitogen-activated protein kinase 1 | Homo sapiens (human) | Potency | 29.2714 | 2 | 4 |
| muscarinic acetylcholine receptor M1 | Rattus norvegicus (Norway rat) | Potency | 19.0090 | 2 | 3 |
| muscleblind-like protein 1 isoform 1 | Homo sapiens (human) | Potency | 2.8184 | 1 | 1 |
| neuropeptide S receptor isoform A | Homo sapiens (human) | Potency | 3.6398 | 3 | 4 |
| NFKB1 protein, partial | Homo sapiens (human) | Potency | 0.9994 | 2 | 4 |
| NPC intracellular cholesterol transporter 1 precursor | Homo sapiens (human) | Potency | 16.3601 | 1 | 1 |
| nuclear factor erythroid 2-related factor 2 isoform 1 | Homo sapiens (human) | Potency | 10.6486 | 3 | 7 |
| nuclear factor erythroid 2-related factor 2 isoform 2 | Homo sapiens (human) | Potency | 17.3457 | 1 | 2 |
| nuclear factor of kappa light polypeptide gene enhancer in B-cells 1 (p105), isoform CRA_a | Homo sapiens (human) | Potency | 54.9410 | 1 | 1 |
| nuclear receptor ROR-gamma isoform 1 | Mus musculus (house mouse) | Potency | 17.8657 | 2 | 4 |
| nuclear receptor subfamily 1, group I, member 3 | Homo sapiens (human) | Potency | 13.8112 | 3 | 9 |
| parathyroid hormone/parathyroid hormone-related peptide receptor precursor | Homo sapiens (human) | Potency | 19.9526 | 1 | 1 |
| Parkin | Homo sapiens (human) | Potency | 9.2000 | 1 | 1 |
| peptidyl-prolyl cis-trans isomerase NIMA-interacting 1 | Homo sapiens (human) | Potency | 29.3138 | 2 | 2 |
| peripheral myelin protein 22 isoform 1 | Homo sapiens (human) | Potency | 95.2834 | 1 | 1 |
| peroxisome proliferator activated receptor gamma | Homo sapiens (human) | Potency | 43.6412 | 1 | 1 |
| peroxisome proliferator-activated receptor delta | Homo sapiens (human) | Potency | 36.7195 | 1 | 1 |
| phosphoglycerate kinase | Trypanosoma brucei brucei TREU927 | Potency | 17.7828 | 1 | 1 |
| phosphopantetheinyl transferase | Bacillus subtilis | Potency | 79.1397 | 3 | 4 |
| plasminogen precursor | Mus musculus (house mouse) | Potency | 2.2387 | 1 | 1 |
| polyprotein | Zika virus | Potency | 17.7828 | 1 | 1 |
| Polyunsaturated fatty acid lipoxygenase ALOX15B | Homo sapiens (human) | Potency | 15.8489 | 1 | 2 |
| potassium voltage-gated channel subfamily H member 2 isoform d | Homo sapiens (human) | Potency | 11.2202 | 1 | 1 |
| PPM1D protein | Homo sapiens (human) | Potency | 18.5569 | 1 | 2 |
| pregnane X nuclear receptor | Homo sapiens (human) | Potency | 24.8561 | 3 | 3 |
| progesterone receptor | Homo sapiens (human) | Potency | 51.0406 | 1 | 2 |
| pyruvate kinase PKM isoform a | Homo sapiens (human) | Potency | 39.8107 | 2 | 2 |
| RAR-related orphan receptor gamma | Mus musculus (house mouse) | Potency | 15.5180 | 2 | 4 |
| ras-related protein Rab-9A | Homo sapiens (human) | Potency | 20.5962 | 1 | 1 |
| regulator of G-protein signaling 4 | Homo sapiens (human) | Potency | 10.6860 | 1 | 5 |
| retinoic acid nuclear receptor alpha variant 1 | Homo sapiens (human) | Potency | 19.7060 | 3 | 7 |
| retinoid X nuclear receptor alpha | Homo sapiens (human) | Potency | 32.7859 | 2 | 3 |
| serine-protein kinase ATM isoform a | Homo sapiens (human) | Potency | 13.0258 | 4 | 4 |
| SMAD family member 2 | Homo sapiens (human) | Potency | 6.7400 | 1 | 1 |
| SMAD family member 3 | Homo sapiens (human) | Potency | 6.7400 | 1 | 1 |
| Smad3 | Homo sapiens (human) | Potency | 22.7406 | 1 | 2 |
| Spike glycoprotein | Severe acute respiratory syndrome-related coronavirus | Potency | 25.5154 | 1 | 2 |
| survival motor neuron protein isoform d | Homo sapiens (human) | Potency | 6.6776 | 1 | 4 |
| T cell receptor, partial | Homo sapiens (human) | Potency | 6.2841 | 1 | 1 |
| TAR DNA-binding protein 43 | Homo sapiens (human) | Potency | 15.8489 | 1 | 1 |
| TDP1 protein | Homo sapiens (human) | Potency | 12.3505 | 2 | 22 |
| thioredoxin glutathione reductase | Schistosoma mansoni | Potency | 31.6228 | 1 | 1 |
| thioredoxin reductase | Rattus norvegicus (Norway rat) | Potency | 34.9784 | 4 | 13 |
| Thrombopoietin | Homo sapiens (human) | Potency | 3.9811 | 2 | 2 |
| thyroid hormone receptor beta isoform 2 | Rattus norvegicus (Norway rat) | Potency | 20.0220 | 2 | 5 |
| thyroid hormone receptor beta isoform a | Homo sapiens (human) | Potency | 42.2395 | 2 | 2 |
| thyroid stimulating hormone receptor | Homo sapiens (human) | Potency | 12.1225 | 7 | 16 |
| TSHR protein | Homo sapiens (human) | Potency | 15.5035 | 2 | 2 |
| urokinase plasminogen activator surface receptor precursor | Mus musculus (house mouse) | Potency | 2.2387 | 1 | 1 |
| urokinase-type plasminogen activator precursor | Mus musculus (house mouse) | Potency | 2.2387 | 1 | 1 |
| USP1 protein, partial | Homo sapiens (human) | Potency | 56.8072 | 1 | 2 |
| v-jun sarcoma virus 17 oncogene homolog (avian) | Homo sapiens (human) | Potency | 8.1966 | 2 | 4 |
| vitamin D (1,25- dihydroxyvitamin D3) receptor | Homo sapiens (human) | Potency | 0.3890 | 1 | 1 |
| Voltage-dependent calcium channel gamma-2 subunit | Mus musculus (house mouse) | Potency | 28.5776 | 1 | 2 |
| Vpr | Human immunodeficiency virus 1 | Potency | 39.8107 | 1 | 1 |
| Protein | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Drugs |
|---|
| [Tau protein] kinase | Sus scrofa (pig) | IC50 | 12.2500 | 4 | 4 |
| 10 kDa chaperonin | Escherichia coli | IC50 | 58.0000 | 2 | 2 |
| 10 kDa heat shock protein, mitochondrial | Homo sapiens (human) | IC50 | 100.0000 | 1 | 1 |
| 5-hydroxytryptamine receptor 1A | Homo sapiens (human) | Ki | 10.0000 | 1 | 1 |
| 5-hydroxytryptamine receptor 1B | Homo sapiens (human) | Ki | 10.0000 | 1 | 1 |
| 5-hydroxytryptamine receptor 1D | Homo sapiens (human) | Ki | 10.0000 | 1 | 1 |
| 5-hydroxytryptamine receptor 2A | Rattus norvegicus (Norway rat) | Ki | 7.7900 | 1 | 1 |
| 5-hydroxytryptamine receptor 2C | Homo sapiens (human) | Ki | 9.3400 | 1 | 1 |
| 5-hydroxytryptamine receptor 3A | Homo sapiens (human) | Ki | 10.0000 | 1 | 1 |
| 5-hydroxytryptamine receptor 3B | Homo sapiens (human) | Ki | 10.0000 | 1 | 1 |
| 5-hydroxytryptamine receptor 3C | Homo sapiens (human) | Ki | 10.0000 | 1 | 1 |
| 5-hydroxytryptamine receptor 3D | Homo sapiens (human) | Ki | 10.0000 | 1 | 1 |
| 5-hydroxytryptamine receptor 3E | Homo sapiens (human) | Ki | 10.0000 | 1 | 1 |
| 5-hydroxytryptamine receptor 5A | Homo sapiens (human) | Ki | 10.0000 | 2 | 3 |
| 5-hydroxytryptamine receptor 6 | Homo sapiens (human) | Ki | 0.7407 | 2 | 2 |
| 5-hydroxytryptamine receptor 7 | Homo sapiens (human) | Ki | 5.5000 | 1 | 1 |
| 60 kDa chaperonin | Escherichia coli K-12 | IC50 | 250.0000 | 1 | 1 |
| 60 kDa chaperonin | Escherichia coli | IC50 | 58.0000 | 2 | 2 |
| 60 kDa heat shock protein, mitochondrial | Homo sapiens (human) | IC50 | 100.0000 | 1 | 1 |
| Acetylcholinesterase | Electrophorus electricus (electric eel) | IC50 | 260.8633 | 4 | 6 |
| Acetylcholinesterase | Homo sapiens (human) | IC50 | 250.0095 | 2 | 2 |
| Acetylcholinesterase | Homo sapiens (human) | Ki | 100.0000 | 2 | 6 |
| Adenosine receptor A1 | Rattus norvegicus (Norway rat) | IC50 | 0.0385 | 1 | 1 |
| Adenosine receptor A1 | Homo sapiens (human) | Ki | 10.0000 | 1 | 1 |
| Adenosine receptor A1 | Rattus norvegicus (Norway rat) | Ki | 28.1333 | 2 | 3 |
| Adenosine receptor A2a | Homo sapiens (human) | Ki | 0.0928 | 3 | 3 |
| Adenosine receptor A2a | Rattus norvegicus (Norway rat) | Ki | 0.2793 | 4 | 4 |
| Adenosine receptor A2b | Homo sapiens (human) | Ki | 4.6000 | 2 | 2 |
| Adenosine receptor A3 | Homo sapiens (human) | Ki | 1.0000 | 1 | 1 |
| Aldehyde oxidase | Homo sapiens (human) | IC50 | 0.0300 | 1 | 1 |
| Aldo-keto reductase family 1 member B1 | Rattus norvegicus (Norway rat) | IC50 | 30.0000 | 1 | 1 |
| Alpha-1A adrenergic receptor | Rattus norvegicus (Norway rat) | IC50 | 0.5000 | 1 | 1 |
| Alpha-1A adrenergic receptor | Homo sapiens (human) | Ki | 3.8733 | 2 | 3 |
| Alpha-1B adrenergic receptor | Rattus norvegicus (Norway rat) | IC50 | 0.5000 | 1 | 1 |
| Alpha-1B adrenergic receptor | Homo sapiens (human) | Ki | 5.4050 | 2 | 2 |
| Alpha-1D adrenergic receptor | Rattus norvegicus (Norway rat) | IC50 | 0.5000 | 1 | 1 |
| Alpha-1D adrenergic receptor | Homo sapiens (human) | Ki | 0.8100 | 1 | 1 |
| Alpha-2A adrenergic receptor | Homo sapiens (human) | Ki | 6.2700 | 2 | 2 |
| Alpha-2A adrenergic receptor | Mus musculus (house mouse) | Ki | 10.0000 | 1 | 1 |
| Alpha-2B adrenergic receptor | Homo sapiens (human) | Ki | 1.1300 | 1 | 1 |
| Alpha-2B adrenergic receptor | Mus musculus (house mouse) | Ki | 10.0000 | 1 | 1 |
| Alpha-2C adrenergic receptor | Homo sapiens (human) | Ki | 0.8100 | 1 | 1 |
| Alpha-2C adrenergic receptor | Mus musculus (house mouse) | Ki | 10.0000 | 1 | 1 |
| Amine oxidase [flavin-containing] A | Homo sapiens (human) | IC50 | 21.5961 | 130 | 165 |
| Amine oxidase [flavin-containing] A | Homo sapiens (human) | Ki | 5.2482 | 15 | 21 |
| Amine oxidase [flavin-containing] A | Bos taurus (cattle) | IC50 | 0.0032 | 4 | 4 |
| Amine oxidase [flavin-containing] A | Rattus norvegicus (Norway rat) | IC50 | 146.6231 | 11 | 13 |
| Amine oxidase [flavin-containing] A | Bos taurus (cattle) | Ki | 9.7117 | 5 | 6 |
| Amine oxidase [flavin-containing] A | Rattus norvegicus (Norway rat) | Ki | 0.0142 | 1 | 1 |
| Amine oxidase [flavin-containing] B | Bos taurus (cattle) | IC50 | 2,634.0000 | 4 | 4 |
| Amine oxidase [flavin-containing] B | Homo sapiens (human) | IC50 | 96.2010 | 111 | 155 |
| Amine oxidase [flavin-containing] B | Rattus norvegicus (Norway rat) | IC50 | 76.4085 | 12 | 12 |
| Amine oxidase [flavin-containing] B | Bos taurus (cattle) | Ki | 28.6413 | 6 | 11 |
| Amine oxidase [flavin-containing] B | Homo sapiens (human) | Ki | 6.8592 | 18 | 27 |
| Amine oxidase [flavin-containing] B | Mus musculus (house mouse) | Ki | 4.1833 | 2 | 6 |
| Amine oxidase [flavin-containing] B | Rattus norvegicus (Norway rat) | Ki | 3.1540 | 3 | 8 |
| Amyloid-beta precursor protein | Homo sapiens (human) | IC50 | 0.5000 | 1 | 1 |
| Apoptotic peptidase activating factor 1 | Homo sapiens (human) | IC50 | 57.7500 | 2 | 2 |
| ATP-binding cassette sub-family C member 3 | Homo sapiens (human) | IC50 | 133.0000 | 1 | 1 |
| Beta-1 adrenergic receptor | Homo sapiens (human) | Ki | 10.0000 | 1 | 1 |
| Beta-2 adrenergic receptor | Homo sapiens (human) | Ki | 10.0000 | 1 | 1 |
| Bile salt export pump | Homo sapiens (human) | IC50 | 134.0000 | 2 | 2 |
| Broad substrate specificity ATP-binding cassette transporter ABCG2 | Homo sapiens (human) | GI50 | 1.6700 | 3 | 3 |
| Broad substrate specificity ATP-binding cassette transporter ABCG2 | Homo sapiens (human) | IC50 | 5.0800 | 1 | 1 |
| Canalicular multispecific organic anion transporter 1 | Homo sapiens (human) | IC50 | 133.0000 | 1 | 1 |
| Carbonic anhydrase 1 | Homo sapiens (human) | Ki | 206.4539 | 3 | 15 |
| Carbonic anhydrase 12 | Homo sapiens (human) | Ki | 203.1434 | 2 | 14 |
| Carbonic anhydrase 13 | Mus musculus (house mouse) | Ki | 205.7006 | 2 | 14 |
| Carbonic anhydrase 14 | Homo sapiens (human) | Ki | 204.5649 | 2 | 14 |
| Carbonic anhydrase 15 | Mus musculus (house mouse) | Ki | 434.0000 | 1 | 1 |
| Carbonic anhydrase 2 | Homo sapiens (human) | Ki | 189.0016 | 3 | 15 |
| Carbonic anhydrase 3 | Homo sapiens (human) | Ki | 202.9649 | 2 | 14 |
| Carbonic anhydrase 4 | Homo sapiens (human) | Ki | 247.7720 | 2 | 14 |
| Carbonic anhydrase 5A, mitochondrial | Homo sapiens (human) | Ki | 239.6291 | 2 | 14 |
| Carbonic anhydrase 5B, mitochondrial | Homo sapiens (human) | Ki | 242.2720 | 2 | 14 |
| Carbonic anhydrase 6 | Homo sapiens (human) | Ki | 203.4649 | 2 | 14 |
| Carbonic anhydrase 7 | Homo sapiens (human) | Ki | 257.9863 | 2 | 14 |
| Carbonic anhydrase 9 | Homo sapiens (human) | Ki | 206.4863 | 2 | 14 |
| Casein kinase I isoform delta | Homo sapiens (human) | IC50 | 1.5000 | 2 | 2 |
| Casein kinase I isoform epsilon | Homo sapiens (human) | IC50 | 1.5000 | 1 | 1 |
| caspase-3 isoform a preproprotein | Homo sapiens (human) | IC50 | 17.0000 | 1 | 1 |
| caspase-9 isoform alpha precursor | Homo sapiens (human) | IC50 | 17.0000 | 1 | 1 |
| Chain A, Dual specificity tyrosine-phosphorylation-regulated kinase 1A | Homo sapiens (human) | IC50 | 0.3500 | 1 | 1 |
| Chain E, Fibrin beta chain | Homo sapiens (human) | IC50 | 46.2655 | 2 | 2 |
| Cholinesterase | Equus caballus (horse) | IC50 | 504.5333 | 3 | 3 |
| Cholinesterase | Homo sapiens (human) | IC50 | 168.2577 | 3 | 3 |
| Cholinesterase | Homo sapiens (human) | Ki | 100.0000 | 2 | 6 |
| Coagulation factor XII | Homo sapiens (human) | Ki | 100.0000 | 1 | 5 |
| Collagenase 3 | Homo sapiens (human) | IC50 | 72.0000 | 1 | 1 |
| Complement C1s subcomponent | Homo sapiens (human) | Ki | 18,100.0000 | 1 | 1 |
| Cruzipain | Trypanosoma cruzi | IC50 | 40.0000 | 4 | 4 |
| Cyclin-A1 | Homo sapiens (human) | IC50 | 32.5000 | 2 | 2 |
| Cyclin-A2 | Homo sapiens (human) | IC50 | 25.0000 | 3 | 3 |
| Cyclin-dependent kinase 1 | Homo sapiens (human) | IC50 | 18.0000 | 1 | 1 |
| Cyclin-dependent kinase 2 | Homo sapiens (human) | IC50 | 25.0000 | 3 | 3 |
| Cyclin-dependent kinase 5 activator 1 | Homo sapiens (human) | IC50 | 11.4000 | 5 | 5 |
| Cyclin-dependent kinase 7 | Homo sapiens (human) | IC50 | 10.0000 | 1 | 1 |
| Cyclin-dependent kinase 9 | Homo sapiens (human) | IC50 | 0.7200 | 1 | 1 |
| Cyclin-dependent-like kinase 5 | Homo sapiens (human) | IC50 | 11.4000 | 5 | 5 |
| Cyclin-H | Homo sapiens (human) | IC50 | 10.0000 | 1 | 1 |
| Cyclin-T1 | Homo sapiens (human) | IC50 | 0.7200 | 1 | 1 |
| Cytochrome P450 2B1 | Rattus norvegicus (Norway rat) | Ki | 1.5000 | 1 | 1 |
| D(1A) dopamine receptor | Homo sapiens (human) | Ki | 10.0000 | 1 | 1 |
| D(1B) dopamine receptor | Homo sapiens (human) | Ki | 10.0000 | 1 | 1 |
| D(2) dopamine receptor | Homo sapiens (human) | Ki | 10.0000 | 1 | 1 |
| D(3) dopamine receptor | Homo sapiens (human) | Ki | 10.0000 | 1 | 1 |
| D(4) dopamine receptor | Homo sapiens (human) | Ki | 10.0000 | 1 | 1 |
| Dihydrolipoyl dehydrogenase | Plasmodium falciparum (malaria parasite P. falciparum) | IC50 | 1,000.0000 | 1 | 1 |
| Dihydrolipoyl dehydrogenase, mitochondrial | Sus scrofa (pig) | IC50 | 1,000.0000 | 1 | 1 |
| Dual specificity protein kinase CLK1 | Homo sapiens (human) | IC50 | 0.0860 | 4 | 4 |
| Dual specificity protein kinase CLK1 | Mus musculus (house mouse) | IC50 | 0.0720 | 1 | 1 |
| Dual specificity protein kinase CLK2 | Mus musculus (house mouse) | IC50 | 0.2800 | 1 | 1 |
| Dual specificity protein kinase CLK3 | Mus musculus (house mouse) | IC50 | 10.0000 | 1 | 1 |
| Dual specificity protein kinase CLK4 | Mus musculus (house mouse) | IC50 | 0.0500 | 1 | 1 |
| Dual specificity tyrosine-phosphorylation-regulated kinase 1A | Homo sapiens (human) | IC50 | 0.5073 | 30 | 30 |
| Dual specificity tyrosine-phosphorylation-regulated kinase 1A | Rattus norvegicus (Norway rat) | IC50 | 0.0397 | 3 | 3 |
| Dual specificity tyrosine-phosphorylation-regulated kinase 1A | Homo sapiens (human) | Ki | 0.0330 | 1 | 1 |
| Dual specificity tyrosine-phosphorylation-regulated kinase 1B | Homo sapiens (human) | IC50 | 0.1183 | 5 | 5 |
| Dual specificity tyrosine-phosphorylation-regulated kinase 1B | Homo sapiens (human) | Ki | 0.1660 | 1 | 1 |
| Dual specificity tyrosine-phosphorylation-regulated kinase 2 | Homo sapiens (human) | IC50 | 1.3138 | 8 | 8 |
| Dual specificity tyrosine-phosphorylation-regulated kinase 3 | Homo sapiens (human) | IC50 | 0.6040 | 5 | 5 |
| Dual specificity tyrosine-phosphorylation-regulated kinase 4 | Homo sapiens (human) | IC50 | 54.5000 | 3 | 3 |
| G2/mitotic-specific cyclin-B1 | Homo sapiens (human) | IC50 | 18.0000 | 1 | 1 |
| G2/mitotic-specific cyclin-B2 | Homo sapiens (human) | IC50 | 18.0000 | 1 | 1 |
| G2/mitotic-specific cyclin-B3 | Homo sapiens (human) | IC50 | 18.0000 | 1 | 1 |
| GABA theta subunit | Rattus norvegicus (Norway rat) | IC50 | 12.3920 | 3 | 3 |
| GABA theta subunit | Rattus norvegicus (Norway rat) | Ki | 10.8000 | 2 | 3 |
| Gamma-aminobutyric acid receptor subunit alpha-1 | Homo sapiens (human) | IC50 | 12.3027 | 1 | 1 |
| Gamma-aminobutyric acid receptor subunit alpha-1 | Rattus norvegicus (Norway rat) | IC50 | 12.3920 | 3 | 3 |
| Gamma-aminobutyric acid receptor subunit alpha-1 | Rattus norvegicus (Norway rat) | Ki | 10.8000 | 2 | 3 |
| Gamma-aminobutyric acid receptor subunit alpha-2 | Homo sapiens (human) | IC50 | 12.3027 | 1 | 1 |
| Gamma-aminobutyric acid receptor subunit alpha-2 | Rattus norvegicus (Norway rat) | IC50 | 12.3920 | 3 | 3 |
| Gamma-aminobutyric acid receptor subunit alpha-2 | Rattus norvegicus (Norway rat) | Ki | 10.8000 | 2 | 3 |
| Gamma-aminobutyric acid receptor subunit alpha-3 | Homo sapiens (human) | IC50 | 12.3027 | 1 | 1 |
| Gamma-aminobutyric acid receptor subunit alpha-3 | Rattus norvegicus (Norway rat) | IC50 | 12.3920 | 3 | 3 |
| Gamma-aminobutyric acid receptor subunit alpha-3 | Rattus norvegicus (Norway rat) | Ki | 10.8000 | 2 | 3 |
| Gamma-aminobutyric acid receptor subunit alpha-4 | Homo sapiens (human) | IC50 | 12.3027 | 1 | 1 |
| Gamma-aminobutyric acid receptor subunit alpha-4 | Rattus norvegicus (Norway rat) | IC50 | 12.3920 | 3 | 3 |
| Gamma-aminobutyric acid receptor subunit alpha-4 | Rattus norvegicus (Norway rat) | Ki | 10.8000 | 2 | 3 |
| Gamma-aminobutyric acid receptor subunit alpha-5 | Homo sapiens (human) | IC50 | 12.3027 | 1 | 1 |
| Gamma-aminobutyric acid receptor subunit alpha-5 | Rattus norvegicus (Norway rat) | IC50 | 12.3920 | 3 | 3 |
| Gamma-aminobutyric acid receptor subunit alpha-5 | Rattus norvegicus (Norway rat) | Ki | 10.8000 | 2 | 3 |
| Gamma-aminobutyric acid receptor subunit alpha-6 | Homo sapiens (human) | IC50 | 12.3027 | 1 | 1 |
| Gamma-aminobutyric acid receptor subunit alpha-6 | Rattus norvegicus (Norway rat) | IC50 | 12.3920 | 3 | 3 |
| Gamma-aminobutyric acid receptor subunit alpha-6 | Rattus norvegicus (Norway rat) | Ki | 10.8000 | 2 | 3 |
| Gamma-aminobutyric acid receptor subunit beta-1 | Homo sapiens (human) | IC50 | 12.3027 | 1 | 1 |
| Gamma-aminobutyric acid receptor subunit beta-1 | Rattus norvegicus (Norway rat) | IC50 | 12.3920 | 3 | 3 |
| Gamma-aminobutyric acid receptor subunit beta-1 | Rattus norvegicus (Norway rat) | Ki | 10.8000 | 2 | 3 |
| Gamma-aminobutyric acid receptor subunit beta-2 | Homo sapiens (human) | IC50 | 12.3027 | 1 | 1 |
| Gamma-aminobutyric acid receptor subunit beta-2 | Rattus norvegicus (Norway rat) | IC50 | 12.3920 | 3 | 3 |
| Gamma-aminobutyric acid receptor subunit beta-2 | Rattus norvegicus (Norway rat) | Ki | 10.8000 | 2 | 3 |
| Gamma-aminobutyric acid receptor subunit beta-3 | Homo sapiens (human) | IC50 | 12.3027 | 1 | 1 |
| Gamma-aminobutyric acid receptor subunit beta-3 | Rattus norvegicus (Norway rat) | IC50 | 12.3920 | 3 | 3 |
| Gamma-aminobutyric acid receptor subunit beta-3 | Rattus norvegicus (Norway rat) | Ki | 10.8000 | 2 | 3 |
| Gamma-aminobutyric acid receptor subunit delta | Homo sapiens (human) | IC50 | 12.3027 | 1 | 1 |
| Gamma-aminobutyric acid receptor subunit delta | Rattus norvegicus (Norway rat) | IC50 | 12.3920 | 3 | 3 |
| Gamma-aminobutyric acid receptor subunit delta | Rattus norvegicus (Norway rat) | Ki | 10.8000 | 2 | 3 |
| Gamma-aminobutyric acid receptor subunit epsilon | Homo sapiens (human) | IC50 | 12.3027 | 1 | 1 |
| Gamma-aminobutyric acid receptor subunit epsilon | Rattus norvegicus (Norway rat) | IC50 | 12.3920 | 3 | 3 |
| Gamma-aminobutyric acid receptor subunit epsilon | Rattus norvegicus (Norway rat) | Ki | 10.8000 | 2 | 3 |
| Gamma-aminobutyric acid receptor subunit gamma-1 | Homo sapiens (human) | IC50 | 12.3027 | 1 | 1 |
| Gamma-aminobutyric acid receptor subunit gamma-1 | Rattus norvegicus (Norway rat) | IC50 | 12.3920 | 3 | 3 |
| Gamma-aminobutyric acid receptor subunit gamma-1 | Rattus norvegicus (Norway rat) | Ki | 10.8000 | 2 | 3 |
| Gamma-aminobutyric acid receptor subunit gamma-2 | Homo sapiens (human) | IC50 | 12.3027 | 1 | 1 |
| Gamma-aminobutyric acid receptor subunit gamma-2 | Rattus norvegicus (Norway rat) | IC50 | 12.3920 | 3 | 3 |
| Gamma-aminobutyric acid receptor subunit gamma-2 | Rattus norvegicus (Norway rat) | Ki | 10.8000 | 2 | 3 |
| Gamma-aminobutyric acid receptor subunit gamma-3 | Homo sapiens (human) | IC50 | 12.3027 | 1 | 1 |
| Gamma-aminobutyric acid receptor subunit gamma-3 | Rattus norvegicus (Norway rat) | IC50 | 12.3920 | 3 | 3 |
| Gamma-aminobutyric acid receptor subunit gamma-3 | Rattus norvegicus (Norway rat) | Ki | 10.8000 | 2 | 3 |
| Gamma-aminobutyric acid receptor subunit pi | Homo sapiens (human) | IC50 | 12.3027 | 1 | 1 |
| Gamma-aminobutyric acid receptor subunit pi | Rattus norvegicus (Norway rat) | IC50 | 12.3920 | 3 | 3 |
| Gamma-aminobutyric acid receptor subunit pi | Rattus norvegicus (Norway rat) | Ki | 10.8000 | 2 | 3 |
| Gamma-aminobutyric acid receptor subunit theta | Homo sapiens (human) | IC50 | 12.3027 | 1 | 1 |
| Glutathione reductase | Plasmodium falciparum 3D7 | IC50 | 6.4000 | 1 | 1 |
| Glutathione reductase, mitochondrial | Homo sapiens (human) | IC50 | 16.2000 | 2 | 2 |
| Glycogen synthase kinase-3 alpha | Homo sapiens (human) | IC50 | 10.0000 | 3 | 3 |
| Glycogen synthase kinase-3 beta | Homo sapiens (human) | IC50 | 24.0333 | 6 | 6 |
| Glycogen synthase kinase-3 beta | Sus scrofa (pig) | IC50 | 12.2500 | 4 | 4 |
| Histone deacetylase 1 | Homo sapiens (human) | IC50 | 5.5000 | 6 | 6 |
| Histone deacetylase 11 | Homo sapiens (human) | IC50 | 10.0000 | 3 | 3 |
| Histone deacetylase 2 | Homo sapiens (human) | IC50 | 10.0000 | 3 | 3 |
| Histone deacetylase 3 | Homo sapiens (human) | IC50 | 10.0000 | 3 | 3 |
| Histone deacetylase 4 | Homo sapiens (human) | IC50 | 10.0000 | 3 | 3 |
| Histone deacetylase 5 | Homo sapiens (human) | IC50 | 10.0000 | 3 | 3 |
| Histone deacetylase 6 | Homo sapiens (human) | IC50 | 10.0000 | 3 | 3 |
| Histone deacetylase 7 | Homo sapiens (human) | IC50 | 10.0000 | 3 | 3 |
| Histone deacetylase 8 | Homo sapiens (human) | IC50 | 10.0000 | 3 | 3 |
| Histone deacetylase 9 | Homo sapiens (human) | IC50 | 10.0000 | 3 | 3 |
| integrase, partial | Human immunodeficiency virus 1 | IC50 | 19.2405 | 2 | 2 |
| Kappa-type opioid receptor | Cavia porcellus (domestic guinea pig) | IC50 | 5.0360 | 2 | 2 |
| lens epithelium-derived growth factor p75 | Homo sapiens (human) | IC50 | 19.2405 | 2 | 2 |
| Liver carboxylesterase 1 | Homo sapiens (human) | Ki | 100.0000 | 2 | 6 |
| Liver carboxylesterase 1 | Oryctolagus cuniculus (rabbit) | Ki | 100.0000 | 1 | 5 |
| Metabotropic glutamate receptor 1 | Rattus norvegicus (Norway rat) | Ki | 10.0000 | 1 | 1 |
| Metabotropic glutamate receptor 2 | Rattus norvegicus (Norway rat) | Ki | 10.0000 | 1 | 1 |
| Metabotropic glutamate receptor 3 | Rattus norvegicus (Norway rat) | Ki | 10.0000 | 1 | 1 |
| Metabotropic glutamate receptor 4 | Rattus norvegicus (Norway rat) | Ki | 10.0000 | 1 | 1 |
| Metabotropic glutamate receptor 5 | Rattus norvegicus (Norway rat) | Ki | 10.0000 | 1 | 1 |
| Metabotropic glutamate receptor 6 | Rattus norvegicus (Norway rat) | Ki | 10.0000 | 1 | 1 |
| Metabotropic glutamate receptor 7 | Rattus norvegicus (Norway rat) | Ki | 10.0000 | 1 | 1 |
| Metabotropic glutamate receptor 8 | Rattus norvegicus (Norway rat) | Ki | 10.0000 | 1 | 1 |
| Microtubule-associated protein tau | Homo sapiens (human) | IC50 | 9.4250 | 4 | 4 |
| Mitogen-activated protein kinase 1 | Rattus norvegicus (Norway rat) | IC50 | 30.0000 | 1 | 1 |
| Multidrug resistance-associated protein 4 | Homo sapiens (human) | IC50 | 133.0000 | 1 | 1 |
| Muscarinic acetylcholine receptor M1 | Homo sapiens (human) | Ki | 10.0000 | 1 | 1 |
| Muscarinic acetylcholine receptor M2 | Homo sapiens (human) | Ki | 10.0000 | 1 | 1 |
| Muscarinic acetylcholine receptor M3 | Homo sapiens (human) | Ki | 10.0000 | 1 | 1 |
| Muscarinic acetylcholine receptor M4 | Homo sapiens (human) | Ki | 10.0000 | 1 | 1 |
| Muscarinic acetylcholine receptor M5 | Homo sapiens (human) | Ki | 10.0000 | 1 | 1 |
| Neuromedin-B receptor | Homo sapiens (human) | Ki | 10.0000 | 1 | 1 |
| neutrophil cytosol factor 1 | Homo sapiens (human) | IC50 | 0.3900 | 1 | 1 |
| Neutrophil elastase | Homo sapiens (human) | IC50 | 72.0000 | 1 | 1 |
| Nischarin | Homo sapiens (human) | Ki | 6.9110 | 2 | 2 |
| Nitric oxide synthase, brain | Homo sapiens (human) | IC50 | 61.9500 | 2 | 2 |
| Nitric oxide synthase, brain | Homo sapiens (human) | Ki | 3.3000 | 1 | 1 |
| Nitric oxide synthase, endothelial | Homo sapiens (human) | IC50 | 224.0000 | 3 | 3 |
| Nitric oxide synthase, inducible | Homo sapiens (human) | IC50 | 275,027.3500 | 4 | 4 |
| Nitric oxide synthase, inducible | Mus musculus (house mouse) | IC50 | 27.5100 | 2 | 2 |
| Nitric oxide synthase, inducible | Rattus norvegicus (Norway rat) | IC50 | 132.0100 | 1 | 1 |
| Polyamine deacetylase HDAC10 | Homo sapiens (human) | IC50 | 10.0000 | 3 | 3 |
| Protein kinase C alpha type | Homo sapiens (human) | IC50 | 250.0000 | 1 | 1 |
| Protein kinase C beta type | Homo sapiens (human) | IC50 | 250.0000 | 1 | 1 |
| Protein kinase C delta type | Homo sapiens (human) | IC50 | 250.0000 | 1 | 1 |
| Protein kinase C epsilon type | Homo sapiens (human) | IC50 | 250.0000 | 1 | 1 |
| Protein kinase C eta type | Homo sapiens (human) | IC50 | 250.0000 | 1 | 1 |
| Protein kinase C gamma type | Homo sapiens (human) | IC50 | 250.0000 | 1 | 1 |
| Protein kinase C iota type | Homo sapiens (human) | IC50 | 250.0000 | 1 | 1 |
| Protein kinase C theta type | Homo sapiens (human) | IC50 | 250.0000 | 1 | 1 |
| Protein kinase C zeta type | Homo sapiens (human) | IC50 | 250.0000 | 1 | 1 |
| Protein-glutamine gamma-glutamyltransferase 2 | Homo sapiens (human) | IC50 | 250.0000 | 1 | 1 |
| Replicase polyprotein 1ab | Betacoronavirus England 1 | IC50 | 141.0000 | 1 | 1 |
| Secreted chorismate mutase | Mycobacterium tuberculosis H37Rv | IC50 | 1.0800 | 1 | 1 |
| Serine/threonine-protein kinase D1 | Homo sapiens (human) | IC50 | 250.0000 | 1 | 1 |
| Serine/threonine-protein kinase D3 | Homo sapiens (human) | IC50 | 250.0000 | 1 | 1 |
| Serine/threonine-protein kinase haspin | Homo sapiens (human) | IC50 | 0.5900 | 1 | 1 |
| Serine/threonine-protein kinase pim-1 | Homo sapiens (human) | IC50 | 10.0000 | 1 | 1 |
| Serine/threonine-protein kinase pim-3 | Homo sapiens (human) | IC50 | 4.3000 | 1 | 1 |
| Sigma intracellular receptor 2 | Mus musculus (house mouse) | Ki | 0.5050 | 1 | 1 |
| Sigma non-opioid intracellular receptor 1 | Mus musculus (house mouse) | Ki | 0.0029 | 1 | 1 |
| Sodium-dependent dopamine transporter | Bos taurus (cattle) | Ki | 10.0000 | 1 | 1 |
| Sodium-dependent noradrenaline transporter | Homo sapiens (human) | Ki | 3.2600 | 1 | 1 |
| Sodium-dependent serotonin transporter | Homo sapiens (human) | Ki | 10.0000 | 1 | 1 |
| Thioredoxin reductase 1, cytoplasmic | Homo sapiens (human) | IC50 | 30.0000 | 1 | 1 |
| Thiosulfate sulfurtransferase | Homo sapiens (human) | IC50 | 9.7000 | 1 | 1 |
| Translocator protein | Rattus norvegicus (Norway rat) | IC50 | 12.3880 | 1 | 1 |
| Transporter | Rattus norvegicus (Norway rat) | Ki | 3.2600 | 1 | 1 |
| Transthyretin | Homo sapiens (human) | IC50 | 50.0000 | 1 | 1 |
| Tryptophan 2,3-dioxygenase | Homo sapiens (human) | IC50 | 6.3100 | 1 | 1 |
| Tyrosine-protein kinase Fyn | Homo sapiens (human) | IC50 | 250.0000 | 1 | 1 |
| Tyrosine-protein kinase Lck | Homo sapiens (human) | IC50 | 250.0000 | 1 | 1 |
| Tyrosine-protein kinase Lyn | Homo sapiens (human) | IC50 | 250.0000 | 1 | 1 |
| Tyrosine-protein phosphatase non-receptor type 1 | Homo sapiens (human) | IC50 | 71.2000 | 1 | 1 |