A protein that is a translation product of the LOC100009551 gene in rabbit. [PRO:DNx, UniProtKB:P12337]
EC 3.1.1.1;
Acyl-coenzyme A:cholesterol acyltransferase
Timeframe | Studies on this Protein(%) | All Drugs % |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 0 (0.00) | 18.2507 |
2000's | 2 (66.67) | 29.6817 |
2010's | 1 (33.33) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
---|---|---|---|---|---|
diacetyl | Oryctolagus cuniculus (rabbit) | Ki | 100.0000 | 3 | 8 |
6,7-dichloroquinoxaline-2,3-dione | Oryctolagus cuniculus (rabbit) | Ki | 100.0000 | 2 | 6 |
benzophenone | Oryctolagus cuniculus (rabbit) | Ki | 100.0000 | 2 | 6 |
quinone | Oryctolagus cuniculus (rabbit) | Ki | 71.8579 | 2 | 7 |
5-bromoisatin | Oryctolagus cuniculus (rabbit) | Ki | 43.2700 | 1 | 6 |
isatin | Oryctolagus cuniculus (rabbit) | Ki | 100.0000 | 1 | 5 |
chloranil | Oryctolagus cuniculus (rabbit) | Ki | 0.1137 | 2 | 6 |
benzoin | Oryctolagus cuniculus (rabbit) | Ki | 68.2450 | 2 | 6 |
dibenzoylmethane | Oryctolagus cuniculus (rabbit) | Ki | 55.6500 | 2 | 6 |
benzil | Oryctolagus cuniculus (rabbit) | Ki | 20.0670 | 6 | 10 |
1,3-cyclohexanedione | Oryctolagus cuniculus (rabbit) | Ki | 100.0000 | 2 | 7 |
dibromsalicil | Oryctolagus cuniculus (rabbit) | Ki | 50.0300 | 2 | 6 |
1-acetylisatin | Oryctolagus cuniculus (rabbit) | Ki | 87.2000 | 1 | 5 |
1-phenyl-1,2-propanedione | Oryctolagus cuniculus (rabbit) | Ki | 31.7000 | 3 | 7 |
2,3-pentanedione | Oryctolagus cuniculus (rabbit) | Ki | 100.0000 | 2 | 6 |
5-methylisatin | Oryctolagus cuniculus (rabbit) | Ki | 85.2400 | 1 | 5 |
1,2-cyclohexanedione | Oryctolagus cuniculus (rabbit) | Ki | 100.0000 | 1 | 1 |
n-methylisatin | Oryctolagus cuniculus (rabbit) | Ki | 68.7160 | 1 | 5 |
acetylacetone | Oryctolagus cuniculus (rabbit) | Ki | 100.0000 | 2 | 6 |
5-Methoxyisatin | Oryctolagus cuniculus (rabbit) | Ki | 85.3400 | 1 | 5 |
3-methyl-1,2-cyclopentanedione | Oryctolagus cuniculus (rabbit) | Ki | 71.9000 | 2 | 6 |
4-benzoylbenzoic acid | Oryctolagus cuniculus (rabbit) | Ki | 100.0000 | 2 | 6 |
2-chloranil | Oryctolagus cuniculus (rabbit) | Ki | 2.2092 | 2 | 6 |
3,5-di-tert-butyl-1,2-benzoquinone | Oryctolagus cuniculus (rabbit) | Ki | 33.8184 | 2 | 6 |
5-Chloro-1H-indole-2,3-dione | Oryctolagus cuniculus (rabbit) | Ki | 44.0980 | 1 | 5 |
5-iodoisatin | Oryctolagus cuniculus (rabbit) | Ki | 50.1720 | 1 | 5 |
2,2-dimethoxy-2-phenylacetophenone | Oryctolagus cuniculus (rabbit) | Ki | 85.8833 | 2 | 6 |
anisoin | Oryctolagus cuniculus (rabbit) | Ki | 71.3000 | 2 | 6 |
hydrobenzoin | Oryctolagus cuniculus (rabbit) | Ki | 100.0000 | 2 | 6 |
5-Fluoroisatin | Oryctolagus cuniculus (rabbit) | Ki | 100.0000 | 1 | 6 |
1-[(3,4-dichlorophenyl)methyl]indole-2,3-dione | Oryctolagus cuniculus (rabbit) | Ki | 12.1926 | 1 | 5 |
5-Nitroisatin | Oryctolagus cuniculus (rabbit) | Ki | 81.2860 | 1 | 5 |