Protein | Potency Measurements | Inhibition Measurements | Activation Measurements | Drugs |
interleukin 8 | 2 | 0 | 0 | 2 |
TDP1 protein | 6 | 0 | 0 | 6 |
AR protein | 5 | 0 | 0 | 5 |
thyroid stimulating hormone receptor | 2 | 0 | 0 | 2 |
estrogen receptor 2 (ER beta) | 2 | 0 | 0 | 2 |
progesterone receptor | 4 | 0 | 0 | 4 |
glucocorticoid receptor [Homo sapiens] | 5 | 0 | 0 | 5 |
estrogen-related nuclear receptor alpha | 6 | 0 | 0 | 6 |
estrogen nuclear receptor alpha | 6 | 0 | 0 | 6 |
IDH1 | 2 | 0 | 0 | 2 |
euchromatic histone-lysine N-methyltransferase 2 | 2 | 0 | 0 | 2 |
Bloom syndrome protein isoform 1 | 1 | 0 | 0 | 1 |
transcriptional regulator ERG isoform 3 | 1 | 0 | 0 | 1 |
thyroid hormone receptor beta isoform 2 | 5 | 0 | 0 | 5 |
ras-related protein Rab-9A | 1 | 0 | 0 | 1 |
nuclear factor erythroid 2-related factor 2 isoform 1 | 3 | 0 | 0 | 3 |
geminin | 4 | 0 | 0 | 4 |
survival motor neuron protein isoform d | 2 | 0 | 0 | 2 |
lamin isoform A-delta10 | 3 | 0 | 0 | 3 |
ATP-binding cassette sub-family C member 3 | 0 | 6 | 0 | 6 |
Multidrug resistance-associated protein 4 | 0 | 6 | 0 | 6 |
Polyphenol oxidase 2 | 0 | 1 | 0 | 1 |
Voltage-dependent calcium channel gamma-2 subunit | 3 | 0 | 0 | 3 |
Bile salt export pump | 0 | 7 | 0 | 7 |
Hypoxanthine-guanine phosphoribosyltransferase | 0 | 0 | 0 | 1 |
Cellular tumor antigen p53 | 5 | 0 | 0 | 5 |
Glutamate receptor 2 | 3 | 0 | 0 | 3 |
Xanthine dehydrogenase/oxidase [Includes: Xanthine dehydrogenase | 0 | 1 | 0 | 1 |
Adenosine receptor A2a | 0 | 1 | 1 | 2 |
Xanthine dehydrogenase/oxidase | 0 | 2 | 0 | 2 |
Nuclear receptor ROR-gamma | 0 | 1 | 0 | 1 |
Xanthine dehydrogenase/oxidase | 0 | 2 | 1 | 4 |
Purine nucleoside phosphorylase | 0 | 0 | 1 | 1 |
TAR DNA-binding protein 43 | 1 | 0 | 0 | 1 |
Canalicular multispecific organic anion transporter 1 | 0 | 6 | 0 | 6 |
Shiga toxin subunit A | 0 | 1 | 0 | 1 |
Histamine H3 receptor | 0 | 1 | 0 | 1 |
Chain A, Beta-lactamase | 3 | 0 | 0 | 3 |
Motilin receptor | 0 | 0 | 1 | 1 |
acid sphingomyelinase | 1 | 0 | 0 | 1 |
GLI family zinc finger 3 | 4 | 0 | 0 | 4 |
low molecular weight phosphotyrosine protein phosphatase isoform c | 0 | 1 | 0 | 1 |
serine/threonine-protein kinase PLK1 | 1 | 0 | 0 | 1 |
streptokinase A precursor | 0 | 0 | 1 | 1 |
Motilin receptor | 0 | 1 | 1 | 2 |
Rap guanine nucleotide exchange factor 3 | 2 | 0 | 0 | 2 |
30S ribosomal protein S6 | 0 | 2 | 1 | 3 |
30S ribosomal protein S7 | 0 | 2 | 1 | 3 |
50S ribosomal protein L15 | 0 | 2 | 1 | 3 |
Albumin | 0 | 0 | 2 | 2 |
ATP-dependent translocase ABCB1 | 0 | 2 | 0 | 2 |
ATP-dependent translocase ABCB1 | 0 | 2 | 0 | 2 |
Cytochrome P450 3A4 | 0 | 1 | 0 | 1 |
60 kDa chaperonin | 0 | 1 | 0 | 1 |
50S ribosomal protein L10 | 0 | 2 | 1 | 3 |
50S ribosomal protein L11 | 0 | 2 | 1 | 3 |
50S ribosomal protein L7/L12 | 0 | 2 | 1 | 3 |
50S ribosomal protein L19 | 0 | 2 | 1 | 3 |
50S ribosomal protein L1 | 0 | 2 | 1 | 3 |
50S ribosomal protein L20 | 0 | 2 | 1 | 3 |
50S ribosomal protein L27 | 0 | 2 | 1 | 3 |
50S ribosomal protein L28 | 0 | 2 | 1 | 3 |
50S ribosomal protein L29 | 0 | 2 | 1 | 3 |
50S ribosomal protein L31 | 0 | 2 | 1 | 3 |
50S ribosomal protein L31 type B | 0 | 2 | 1 | 3 |
50S ribosomal protein L32 | 0 | 2 | 1 | 3 |
50S ribosomal protein L33 | 0 | 2 | 1 | 3 |
50S ribosomal protein L34 | 0 | 2 | 1 | 3 |
50S ribosomal protein L35 | 0 | 2 | 1 | 3 |
50S ribosomal protein L36 | 0 | 2 | 1 | 3 |
30S ribosomal protein S10 | 0 | 2 | 1 | 3 |
30S ribosomal protein S11 | 0 | 2 | 1 | 3 |
30S ribosomal protein S12 | 0 | 2 | 1 | 3 |
30S ribosomal protein S13 | 0 | 2 | 1 | 3 |
30S ribosomal protein S16 | 0 | 2 | 1 | 3 |
30S ribosomal protein S18 | 0 | 2 | 1 | 3 |
30S ribosomal protein S19 | 0 | 2 | 1 | 3 |
30S ribosomal protein S20 | 0 | 2 | 1 | 3 |
30S ribosomal protein S2 | 0 | 2 | 1 | 3 |
30S ribosomal protein S3 | 0 | 2 | 1 | 3 |
30S ribosomal protein S4 | 0 | 2 | 1 | 3 |
30S ribosomal protein S5 | 0 | 2 | 1 | 3 |
30S ribosomal protein S8 | 0 | 2 | 1 | 3 |
30S ribosomal protein S9 | 0 | 2 | 1 | 3 |
50S ribosomal protein L13 | 0 | 2 | 1 | 3 |
50S ribosomal protein L14 | 0 | 2 | 1 | 3 |
50S ribosomal protein L16 | 0 | 2 | 1 | 3 |
50S ribosomal protein L23 | 0 | 2 | 1 | 3 |
30S ribosomal protein S15 | 0 | 2 | 1 | 3 |
50S ribosomal protein L17 | 0 | 2 | 1 | 3 |
50S ribosomal protein L21 | 0 | 2 | 1 | 3 |
50S ribosomal protein L30 | 0 | 2 | 1 | 3 |
50S ribosomal protein L6 | 0 | 2 | 1 | 3 |
30S ribosomal protein S14 | 0 | 2 | 1 | 3 |
30S ribosomal protein S17 | 0 | 2 | 1 | 3 |
30S ribosomal protein S1 | 0 | 2 | 1 | 3 |
50S ribosomal protein L18 | 0 | 2 | 1 | 3 |
60 kDa heat shock protein, mitochondrial | 0 | 1 | 0 | 1 |
Cytochrome P450 2C9 | 0 | 3 | 0 | 3 |
Chitinase B | 0 | 1 | 0 | 1 |
ATP-dependent translocase ABCB1 | 0 | 2 | 0 | 2 |
Low molecular weight phosphotyrosine protein phosphatase | 0 | 1 | 0 | 1 |
Cytochrome P450 2J2 | 0 | 2 | 0 | 2 |
50S ribosomal protein L2 | 0 | 2 | 1 | 3 |
50S ribosomal protein L3 | 0 | 2 | 1 | 3 |
50S ribosomal protein L24 | 0 | 2 | 1 | 3 |
50S ribosomal protein L4 | 0 | 2 | 1 | 3 |
50S ribosomal protein L22 | 0 | 2 | 1 | 3 |
10 kDa heat shock protein, mitochondrial | 0 | 1 | 0 | 1 |
50S ribosomal protein L5 | 0 | 2 | 1 | 3 |
30S ribosomal protein S21 | 0 | 2 | 1 | 3 |
50S ribosomal protein L25 | 0 | 2 | 1 | 3 |
Potassium voltage-gated channel subfamily H member 2 | 0 | 2 | 0 | 2 |
Cytochrome P450 1B1 | 0 | 1 | 0 | 1 |
Thiosulfate sulfurtransferase | 0 | 1 | 0 | 1 |
Lanosterol 14-alpha demethylase | 0 | 1 | 0 | 1 |
50S ribosomal protein L36 2 | 0 | 2 | 1 | 3 |
60 kDa chaperonin | 0 | 1 | 0 | 1 |
10 kDa chaperonin | 0 | 1 | 0 | 1 |
Multidrug and toxin extrusion protein 1 | 0 | 2 | 0 | 2 |
Chain A, MAJOR APURINIC/APYRIMIDINIC ENDONUCLEASE | 1 | 0 | 0 | 1 |
thioredoxin reductase | 1 | 0 | 0 | 1 |
RAR-related orphan receptor gamma | 4 | 0 | 0 | 4 |
GLS protein | 1 | 0 | 0 | 1 |
Microtubule-associated protein tau | 1 | 0 | 0 | 1 |
aldehyde dehydrogenase 1 family, member A1 | 4 | 0 | 0 | 4 |
vitamin D (1,25- dihydroxyvitamin D3) receptor | 2 | 0 | 0 | 2 |
chromobox protein homolog 1 | 2 | 0 | 0 | 2 |
mitogen-activated protein kinase 1 | 1 | 0 | 0 | 1 |
flap endonuclease 1 | 1 | 0 | 0 | 1 |
cytochrome P450 3A4 isoform 1 | 2 | 0 | 0 | 2 |
muscarinic acetylcholine receptor M1 | 2 | 0 | 0 | 2 |
Gamma-aminobutyric acid receptor subunit pi | 2 | 0 | 0 | 2 |
Potassium channel subfamily K member 3 | 0 | 1 | 0 | 1 |
Potassium channel subfamily K member 2 | 0 | 1 | 0 | 1 |
Sodium channel protein type 1 subunit alpha | 0 | 1 | 0 | 1 |
Sodium channel protein type 2 subunit alpha | 0 | 1 | 0 | 1 |
Sodium channel protein type 3 subunit alpha | 0 | 1 | 0 | 1 |
Gamma-aminobutyric acid receptor subunit beta-1 | 2 | 0 | 0 | 2 |
Gamma-aminobutyric acid receptor subunit delta | 2 | 0 | 0 | 2 |
Gamma-aminobutyric acid receptor subunit gamma-2 | 2 | 0 | 0 | 2 |
Gamma-aminobutyric acid receptor subunit alpha-5 | 2 | 0 | 0 | 2 |
Gamma-aminobutyric acid receptor subunit alpha-3 | 2 | 0 | 0 | 2 |
Potassium voltage-gated channel subfamily A member 5 | 0 | 1 | 0 | 1 |
Gamma-aminobutyric acid receptor subunit gamma-1 | 2 | 0 | 0 | 2 |
Gamma-aminobutyric acid receptor subunit alpha-2 | 2 | 0 | 0 | 2 |
Gamma-aminobutyric acid receptor subunit alpha-4 | 2 | 0 | 0 | 2 |
Gamma-aminobutyric acid receptor subunit gamma-3 | 2 | 0 | 0 | 2 |
Gamma-aminobutyric acid receptor subunit alpha-6 | 2 | 0 | 0 | 2 |
Sodium channel protein type 4 subunit alpha | 0 | 1 | 0 | 1 |
Gamma-aminobutyric acid receptor subunit alpha-1 | 2 | 0 | 0 | 2 |
Gamma-aminobutyric acid receptor subunit beta-3 | 2 | 0 | 0 | 2 |
Gamma-aminobutyric acid receptor subunit beta-2 | 2 | 0 | 0 | 2 |
Sodium channel protein type 5 subunit alpha | 0 | 1 | 0 | 1 |
Sodium channel protein type 9 subunit alpha | 0 | 1 | 0 | 1 |
Potassium voltage-gated channel subfamily D member 2 | 0 | 1 | 0 | 1 |
Potassium channel subfamily K member 18 | 0 | 1 | 0 | 1 |
GABA theta subunit | 2 | 0 | 0 | 2 |
Gamma-aminobutyric acid receptor subunit epsilon | 2 | 0 | 0 | 2 |
Sodium channel protein type 3 subunit alpha | 0 | 1 | 0 | 1 |
Carbonic anhydrase 1 | 0 | 1 | 0 | 1 |
Carbonic anhydrase 2 | 0 | 1 | 0 | 1 |
Carbonic anhydrase 4 | 0 | 1 | 0 | 1 |
Carbonic anhydrase 5A, mitochondrial | 0 | 1 | 0 | 1 |
Carbonic anhydrase 9 | 0 | 1 | 0 | 1 |
Epidermal growth factor receptor | 0 | 1 | 0 | 1 |
Tyrosine-protein kinase Fyn | 0 | 1 | 0 | 1 |
Beta-2 adrenergic receptor | 0 | 2 | 0 | 2 |
Aldo-keto reductase family 1 member B1 | 0 | 2 | 0 | 2 |
Alpha-2A adrenergic receptor | 0 | 2 | 0 | 2 |
Adenosine receptor A3 | 0 | 3 | 0 | 3 |
Cytochrome P450 2C8 | 0 | 1 | 0 | 1 |
Muscarinic acetylcholine receptor M1 | 0 | 2 | 0 | 2 |
Beta-3 adrenergic receptor | 0 | 2 | 0 | 2 |
Alpha-1B adrenergic receptor | 0 | 3 | 0 | 3 |
Alpha-2C adrenergic receptor | 0 | 2 | 0 | 2 |
Muscarinic acetylcholine receptor M3 | 0 | 2 | 0 | 2 |
Substance-K receptor | 0 | 2 | 0 | 2 |
Sodium-dependent noradrenaline transporter | 0 | 2 | 0 | 2 |
Thromboxane-A synthase | 0 | 1 | 0 | 1 |
D(3) dopamine receptor | 0 | 2 | 0 | 2 |
Delta-type opioid receptor | 0 | 2 | 0 | 2 |
5-hydroxytryptamine receptor 2B | 0 | 2 | 0 | 2 |
Alpha-1A adrenergic receptor | 0 | 3 | 0 | 3 |
Sodium-dependent dopamine transporter | 0 | 2 | 0 | 2 |
Uracil nucleotide/cysteinyl leukotriene receptor | 0 | 1 | 0 | 1 |
Mitogen-activated protein kinase 14 | 0 | 1 | 0 | 1 |
Leukotriene C4 synthase | 0 | 1 | 0 | 1 |
Cysteinyl leukotriene receptor 1 | 0 | 1 | 0 | 1 |
Cysteinyl leukotriene receptor 2 | 0 | 1 | 0 | 1 |
Cysteinyl leukotriene receptor 1 | 0 | 2 | 1 | 3 |
luciferase | 0 | 0 | 0 | 1 |
hypoxia-inducible factor 1 alpha subunit | 1 | 0 | 0 | 1 |
cytochrome P450 family 3 subfamily A polypeptide 4 | 2 | 0 | 0 | 2 |
retinoic acid nuclear receptor alpha variant 1 | 4 | 0 | 0 | 4 |
pregnane X nuclear receptor | 4 | 0 | 0 | 4 |
aryl hydrocarbon receptor | 1 | 0 | 0 | 1 |
cytochrome P450, family 19, subfamily A, polypeptide 1, isoform CRA_a | 3 | 0 | 0 | 3 |
v-jun sarcoma virus 17 oncogene homolog (avian) | 2 | 0 | 0 | 2 |
nuclear receptor subfamily 1, group I, member 2 | 1 | 0 | 0 | 1 |
nuclear factor erythroid 2-related factor 2 isoform 2 | 3 | 0 | 0 | 3 |
Interferon beta | 2 | 0 | 0 | 2 |
Fatty acid-binding protein, liver | 0 | 1 | 0 | 1 |
Estrogen receptor | 0 | 2 | 0 | 2 |
Glucocorticoid receptor | 0 | 4 | 2 | 11 |
Progesterone receptor | 0 | 2 | 0 | 3 |
Glucocorticoid receptor | 0 | 1 | 1 | 2 |
Glucocorticoid receptor | 0 | 0 | 1 | 1 |
Glycine receptor subunit alpha-1 | 0 | 4 | 0 | 4 |
Corticosteroid-binding globulin | 0 | 1 | 0 | 1 |
Mineralocorticoid receptor | 0 | 2 | 1 | 3 |
Androgen receptor | 0 | 2 | 0 | 2 |
Glutamine synthetase | 0 | 0 | 1 | 1 |
Androgen receptor | 0 | 1 | 0 | 1 |
Glycine receptor subunit beta | 0 | 4 | 0 | 4 |
Glycine receptor subunit alpha-2 | 0 | 4 | 0 | 4 |
Glycine receptor subunit alpha-3 | 0 | 4 | 0 | 4 |
Histamine H1 receptor | 0 | 0 | 1 | 1 |
Prostaglandin G/H synthase 2 | 0 | 1 | 0 | 1 |
Nociceptin receptor | 0 | 0 | 1 | 1 |
Estrogen receptor beta | 0 | 2 | 0 | 2 |
ATPase family AAA domain-containing protein 5 | 1 | 0 | 0 | 1 |
Ataxin-2 | 2 | 0 | 0 | 2 |
Chain A, TYROSYL-DNA PHOSPHODIESTERASE | 1 | 0 | 0 | 1 |
Chain A, HADH2 protein | 2 | 0 | 0 | 2 |
Chain B, HADH2 protein | 2 | 0 | 0 | 2 |
pregnane X receptor | 1 | 0 | 0 | 1 |
thioredoxin glutathione reductase | 1 | 0 | 0 | 1 |
hypoxia-inducible factor 1, alpha subunit (basic helix-loop-helix transcription factor) | 1 | 0 | 0 | 1 |
nuclear receptor subfamily 1, group I, member 3 | 2 | 0 | 0 | 2 |
vitamin D3 receptor isoform VDRA | 1 | 0 | 0 | 1 |
nuclear receptor ROR-gamma isoform 1 | 1 | 0 | 0 | 1 |
Nuclear receptor ROR-gamma | 2 | 0 | 0 | 2 |
NS5 | 0 | 0 | 1 | 1 |
Thrombopoietin | 1 | 0 | 0 | 1 |
farnesoid X nuclear receptor | 1 | 0 | 0 | 1 |
peroxisome proliferator activated receptor gamma | 3 | 0 | 0 | 3 |
arylsulfatase A | 1 | 0 | 0 | 1 |
alpha-galactosidase | 1 | 0 | 0 | 1 |
Histone H2A.x | 2 | 0 | 0 | 2 |
Spike glycoprotein | 0 | 0 | 1 | 1 |
Replicase polyprotein 1ab | 0 | 0 | 1 | 1 |
peripheral myelin protein 22 isoform 1 | 1 | 0 | 0 | 1 |
glycogen synthase kinase-3 beta isoform 1 | 0 | 0 | 1 | 1 |
urokinase-type plasminogen activator precursor | 1 | 0 | 0 | 1 |
plasminogen precursor | 1 | 0 | 0 | 1 |
urokinase plasminogen activator surface receptor precursor | 1 | 0 | 0 | 1 |
Transmembrane protease serine 2 | 0 | 0 | 1 | 1 |
Voltage-dependent L-type calcium channel subunit alpha-1F | 0 | 1 | 0 | 1 |
Polymerase basic protein 2 | 0 | 0 | 1 | 1 |
RNA-directed RNA polymerase catalytic subunit | 0 | 0 | 1 | 1 |
Polymerase acidic protein | 0 | 0 | 1 | 1 |
Procathepsin L | 0 | 0 | 1 | 1 |
Replicase polyprotein 1a | 0 | 0 | 1 | 1 |
Replicase polyprotein 1ab | 0 | 0 | 1 | 1 |
Replicase polyprotein 1ab | 0 | 0 | 1 | 1 |
Replicase polyprotein 1ab | 0 | 0 | 1 | 1 |
Adenosylhomocysteinase | 0 | 0 | 0 | 2 |
Adenosine receptor A1 | 0 | 1 | 0 | 1 |
Spike glycoprotein | 0 | 0 | 1 | 1 |
Voltage-dependent L-type calcium channel subunit alpha-1D | 0 | 1 | 0 | 1 |
Voltage-dependent L-type calcium channel subunit alpha-1S | 0 | 1 | 0 | 1 |
Voltage-dependent L-type calcium channel subunit alpha-1C | 0 | 1 | 0 | 1 |
Adenosine receptor A1 | 0 | 1 | 0 | 1 |
Genome polyprotein | 0 | 0 | 1 | 1 |
Angiotensin-converting enzyme 2 | 0 | 0 | 1 | 1 |
90-kda heat shock protein beta HSP90 beta, partial | 0 | 1 | 0 | 1 |
EWS/FLI fusion protein | 2 | 0 | 0 | 2 |
estrogen receptor beta isoform 1 | 0 | 1 | 0 | 1 |
heat shock protein HSP 90-alpha isoform 2 | 0 | 1 | 0 | 1 |
tyrosine-protein phosphatase non-receptor type 7 isoform 2 | 0 | 1 | 0 | 1 |
Dihydroxyacetone phosphate acyltransferase | 0 | 0 | 0 | 1 |
Tetracycline resistance protein, class B | 0 | 0 | 0 | 1 |
Muscarinic acetylcholine receptor M2 | 0 | 1 | 0 | 1 |
72 kDa type IV collagenase | 0 | 1 | 0 | 1 |
Stromelysin-1 | 0 | 1 | 0 | 1 |
Multidrug transporter MdfA | 0 | 1 | 0 | 1 |
Neutrophil collagenase | 0 | 1 | 0 | 1 |
Alpha-1D adrenergic receptor | 0 | 1 | 0 | 1 |
Alpha-synuclein | 0 | 1 | 0 | 1 |
Collagenase 3 | 0 | 1 | 0 | 1 |
Cannabinoid receptor 1 | 0 | 1 | 0 | 1 |
Integrase | 0 | 1 | 0 | 1 |
Solute carrier family 22 member 8 | 0 | 0 | 0 | 1 |
P2Y purinoceptor 12 | 0 | 1 | 0 | 1 |
Solute carrier family 22 member 11 | 0 | 0 | 0 | 1 |
Protein-arginine deiminase type-4 | 0 | 1 | 0 | 1 |
Solute carrier family 22 member 7 | 0 | 0 | 0 | 1 |
Chain A, Putative fructose-1,6-bisphosphate aldolase | 1 | 0 | 0 | 1 |
Chain A, 2-oxoglutarate Oxygenase | 1 | 0 | 0 | 1 |
PPM1D protein | 1 | 0 | 0 | 1 |
thyroid hormone receptor beta isoform a | 1 | 0 | 0 | 1 |
parathyroid hormone/parathyroid hormone-related peptide receptor precursor | 1 | 0 | 0 | 1 |
Albumin | 0 | 0 | 1 | 1 |
Proprotein convertase subtilisin/kexin type 7 | 0 | 1 | 0 | 1 |
Vitamin K epoxide reductase complex subunit 1-like protein 1 | 0 | 1 | 0 | 1 |
Vitamin K epoxide reductase complex subunit 1 | 0 | 1 | 0 | 1 |
Protease | 0 | 1 | 0 | 1 |
Vitamin K epoxide reductase complex subunit 1-like protein 1 | 0 | 1 | 0 | 1 |
Vitamin K epoxide reductase complex subunit 1 | 0 | 2 | 0 | 2 |
[prepared from compound, protein, and bioassay information from National Library of Medicine (NLM), extracted Dec-2023] |