Page last updated: 2024-08-07 12:27:51
Motilin receptor
[no definition available]
Synonyms
Research
Bioassay Publications (4)
| Timeframe | Studies on this Protein(%) | All Drugs % |
|---|
| pre-1990 | 0 (0.00) | 18.7374 |
| 1990's | 0 (0.00) | 18.2507 |
| 2000's | 2 (50.00) | 29.6817 |
| 2010's | 2 (50.00) | 24.3611 |
| 2020's | 0 (0.00) | 2.80 |
Compounds (2)
Drugs with Inhibition Measurements
| Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
|---|
| gm 109 | Oryctolagus cuniculus (rabbit) | IC50 | 0.0100 | 1 | 1 |
Drugs with Activation Measurements
| Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
|---|
| erythromycin | Oryctolagus cuniculus (rabbit) | EC50 | 1.2000 | 3 | 3 |
The role of the 4''-hydroxyl on motilin agonist potency in the 9-dihydroerythromycin series.Bioorganic & medicinal chemistry letters, , Jun-15, Volume: 21, Issue:12, 2011
9-Dihydroerythromycins as non-antibiotic motilin receptor agonists.Bioorganic & medicinal chemistry letters, , Oct-01, Volume: 20, Issue:19, 2010
Structure-activity relationships of 9-substituted-9-dihydroerythromycin-based motilin agonists: optimizing for potency and safety.Journal of medicinal chemistry, , Nov-12, Volume: 52, Issue:21, 2009