Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
mandelic acid | Homo sapiens (human) | IC50 | 100.0000 | 2 | 0 |
5,8,11,14-eicosatetraynoic acid | Homo sapiens (human) | IC50 | 17.7000 | 2 | 0 |
hydroflumethiazide | Homo sapiens (human) | IC50 | 100.0000 | 1 | 0 |
2-naphthoxyacetic acid | Homo sapiens (human) | IC50 | 88.6750 | 3 | 0 |
rhein | Homo sapiens (human) | IC50 | 19.6200 | 1 | 0 |
mandelic acid, (r)-isomer | Homo sapiens (human) | IC50 | 100.0000 | 2 | 0 |
N'-methyl-N,N-diphenylurea | Homo sapiens (human) | IC50 | 100.0000 | 1 | 0 |
src-820 r | Homo sapiens (human) | IC50 | 79.4000 | 1 | 0 |
toxoflavin | Homo sapiens (human) | IC50 | 1.2400 | 1 | 0 |
mandelic acid, (s)-isomer | Homo sapiens (human) | IC50 | 100.0000 | 2 | 0 |
1,3,6-trimethylpyrimido[5,4-e][1,2,4]triazine-5,7-dione | Homo sapiens (human) | IC50 | 1.2400 | 1 | 0 |
4,5-diphenyl-1,2,3-triazole | Homo sapiens (human) | IC50 | 100.0000 | 1 | 0 |
N-(5-ethyl-1,3,4-thiadiazol-2-yl)-2-[[5-(2-methyl-3-furanyl)-4-(2-methylpropyl)-1,2,4-triazol-3-yl]thio]acetamide | Homo sapiens (human) | IC50 | 100.0000 | 1 | 0 |
5-[4-morpholinyl(oxo)methyl]-2-pyranone | Homo sapiens (human) | IC50 | 0.9900 | 1 | 0 |
(3aR,6aS)-3-(2-chlorophenyl)-5-(2,5-dimethoxyphenyl)-3a,6a-dihydropyrrolo[3,4-d]isoxazole-4,6-dione | Homo sapiens (human) | IC50 | 8.2500 | 1 | 0 |
4,7-dimethoxy-1-methyl-2-quinolinone | Homo sapiens (human) | IC50 | 79.4000 | 1 | 0 |
[3-(4-chlorophenyl)-5-(methylthio)-1,2,4-triazol-1-yl]-(2-furanyl)methanone | Homo sapiens (human) | IC50 | 79.4000 | 1 | 0 |
1-[[(1,3-dimethyl-4-pyrazolyl)-oxomethyl]amino]-3-(4-methylphenyl)thiourea | Homo sapiens (human) | IC50 | 100.0000 | 1 | 0 |
[4-amino-3-(4-methylphenyl)-2-sulfanylidene-5-thiazolyl]-(4-morpholinyl)methanone | Homo sapiens (human) | IC50 | 100.0000 | 1 | 0 |
1-cyclopropyl-3-(4-sulfamoylphenyl)thiourea | Homo sapiens (human) | IC50 | 35.6970 | 4 | 0 |
1-[[(5-bromo-2-furanyl)-oxomethyl]amino]-3-(2,5-dimethylphenyl)thiourea | Homo sapiens (human) | IC50 | 100.0000 | 1 | 0 |
2-(4-methylphenoxy)-N-[4-(2-oxazolo[4,5-b]pyridinyl)phenyl]acetamide | Homo sapiens (human) | IC50 | 100.0000 | 1 | 0 |
2-(4-methoxyphenyl)-N-[4-[5-(4-methylphenyl)-1,3,4-oxadiazol-2-yl]phenyl]acetamide | Homo sapiens (human) | IC50 | 100.0000 | 1 | 0 |
[1-(2-phenoxyethyl)-3-indolyl]-(1-pyrrolidinyl)methanethione | Homo sapiens (human) | IC50 | 0.5680 | 2 | 0 |
2-(2-furanyl)-4-quinolinecarboxylic acid [2-[4-amino-1-methyl-3-(2-methylpropyl)-2,6-dioxo-5-pyrimidinyl]-2-oxoethyl] ester | Homo sapiens (human) | IC50 | 5.2700 | 1 | 0 |
4-[2-[[3-(4-methylphenyl)-5-triazolo[1,5-a]quinazolinyl]amino]ethyl]benzenesulfonamide | Homo sapiens (human) | IC50 | 0.8190 | 1 | 0 |
2-[[4-amino-6-(2-methylanilino)-1,3,5-triazin-2-yl]methyl-methylamino]-N-(2-ethylphenyl)acetamide | Homo sapiens (human) | IC50 | 100.0000 | 1 | 0 |
6-[(3,4-difluoroanilino)-oxomethyl]-1-cyclohex-3-enecarboxylic acid | Homo sapiens (human) | IC50 | 100.0000 | 1 | 0 |
4-(diethylamino)benzoic acid [2-oxo-2-(4-phenyl-1-piperazinyl)ethyl] ester | Homo sapiens (human) | IC50 | 100.0000 | 1 | 0 |
5,6-dihydro-4H-cyclopenta[b]thiophene-2-carboxylic acid [2-[(1,1-dioxo-3-thiolanyl)-(2-methylpropyl)amino]-2-oxoethyl] ester | Homo sapiens (human) | IC50 | 1.2100 | 1 | 0 |
benzoic acid [5-(6-benzamido-9-purinyl)-3-fluoro-4-hydroxy-2-oxolanyl]methyl ester | Homo sapiens (human) | IC50 | 100.0000 | 1 | 0 |
3-[(4-phenyl-1-piperazinyl)sulfonyl]benzoic acid [2-(2-furanylmethylamino)-2-oxoethyl] ester | Homo sapiens (human) | IC50 | 4.9700 | 1 | 0 |
N-[2,2,2-trichloro-1-[[(2,6-dichloroanilino)-sulfanylidenemethyl]amino]ethyl]carbamic acid (phenylmethyl) ester | Homo sapiens (human) | IC50 | 63.0000 | 1 | 0 |
1,6-dimethyl-3-propylpyrimido[5,4-e][1,2,4]triazine-5,7-dione | Homo sapiens (human) | IC50 | 1.2400 | 1 | 0 |
3-chloro-N-(5-chloro-2-pyridinyl)-4-ethoxybenzamide | Homo sapiens (human) | IC50 | 79.4000 | 1 | 0 |
2-(3-methylanilino)-[1,3,4]thiadiazolo[2,3-b]quinazolin-5-one | Homo sapiens (human) | IC50 | 2.7400 | 1 | 0 |
4-amino-3-(3,4-dimethylphenyl)-N-(2-fluorophenyl)-2-sulfanylidene-5-thiazolecarboxamide | Homo sapiens (human) | IC50 | 50.5000 | 1 | 0 |
prostaglandin a2 | Homo sapiens (human) | IC50 | 13.7000 | 1 | 0 |
cefamandole nafate | Homo sapiens (human) | IC50 | 0.1000 | 1 | 0 |
sodium cephalothin | Homo sapiens (human) | IC50 | 0.9200 | 1 | 0 |
tetracycline | Homo sapiens (human) | IC50 | 8.3300 | 1 | 0 |