| Assay ID | Title | Year | Journal | Article |
|---|
| AID448893 | Inhibition of MMP2 after 10 to 15 mins by fluorescence assay | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID448224 | Inhibition of caspase 10 assessed as residual activity at 10 uM after 10 to 15 mins by fluorescence assay relative to control | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID448915 | Immunomodulatory activity in CD4+ human T cells assessed as inhibition of monocyte-derived dendritic cell presented tetanus toxin C-fragment-induced cell proliferation after 5 days by autologous mixed lymphocyte reaction assay | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID448896 | Inhibition of MMP8 catalytic domain after 10 to 15 mins by fluorescence assay | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID448184 | Inhibition of cathepsin E in human MCF7 cells by fluorescence assay | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID448235 | Inhibition of ACE1 assessed as residual activity at 10 uM after 10 to 15 mins by fluorescence assay relative to control | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID448211 | Inhibition of tryptase beta2 assessed as residual activity at 10 uM after 10 to 15 mins by fluorescence assay relative to control | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID448213 | Inhibition of urokinase assessed as residual activity at 10 uM after 10 to 15 mins by fluorescence assay relative to control | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID674497 | Inhibition of MHC class 2-dependent antigen processing in DO11.10 TCR transgenic mouse spleen CD11+ dendritic cells assessed as inhibition of whole ovalbumin-induced CD4+ T cell proliferation incubated for 1 hr prior to whole ovalbumin-challenge measured | 2012 | Bioorganic & medicinal chemistry, Aug-01, Volume: 20, Issue:15
| Total synthesis of grassystatin A, a probe for cathepsin E function. |
| AID448838 | Inhibition of MMP7 assessed as residual activity at 10 uM after 10 to 15 mins by fluorescence assay relative to control | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID448911 | Inhibition of human lung tryptase gamma1 after 10 to 15 mins by fluorescence assay | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID448236 | Inhibition of MMP1 assessed as residual activity at 10 uM after 10 to 15 mins by fluorescence assay relative to control | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID448884 | Inhibition of DPP8 after 10 to 15 mins by fluorescence assay | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID448847 | Inhibition of ADAM10 assessed as residual activity at 10 uM after 10 to 15 mins by fluorescence assay relative to control | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID448204 | Inhibition of kallikrein 4 assessed as residual activity at 10 uM after 10 to 15 mins by fluorescence assay relative to control | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID448843 | Inhibition of MMP12 assessed as residual activity at 10 uM after 10 to 15 mins by fluorescence assay relative to control | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID448887 | Inhibition of factor 10a after 10 to 15 mins by fluorescence assay | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID448228 | Inhibition of caspase 14 assessed as residual activity at 10 uM after 10 to 15 mins by fluorescence assay relative to control | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID448872 | Inhibition of cathepsin C after 10 to 15 mins by fluorescence assay | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID448898 | Inhibition of MMP10 catalytic domain after 10 to 15 mins by fluorescence assay | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID448866 | Inhibition of caspase 8 after 10 to 15 mins by fluorescence assay | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID448855 | Inhibition of ADAM9 after 10 to 15 mins by fluorescence assay | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID674498 | Inhibition of MHC class 2-dependent antigen processing in DO11.10 TCR transgenic mouse spleen CD11+ dendritic cells assessed as inhibition of ovalbumin 323 to 339-induced CD4+ T cell proliferation incubated for 1 hr prior to ovalbumin 323 to 339 challenge | 2012 | Bioorganic & medicinal chemistry, Aug-01, Volume: 20, Issue:15
| Total synthesis of grassystatin A, a probe for cathepsin E function. |
| AID448231 | Inhibition of cathepsin V assessed as residual activity at 10 uM after 10 to 15 mins by fluorescence assay relative to control | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID448851 | Inhibition of cathepsin E assessed as residual activity at 10 uM after 10 to 15 mins by fluorescence assay relative to control | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID448889 | Inhibition of kallikrein 4 after 10 to 15 mins by fluorescence assay | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID448217 | Inhibition of caspase 3 assessed as residual activity at 10 uM after 10 to 15 mins by fluorescence assay relative to control | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID448180 | Inhibition of TACE | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID448858 | Inhibition of calpain 1 after 10 to 15 mins by fluorescence assay | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID448845 | Inhibition of MMP14 assessed as residual activity at 10 uM after 10 to 15 mins by fluorescence assay relative to control | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID448218 | Inhibition of caspase 4 assessed as residual activity at 10 uM after 10 to 15 mins by fluorescence assay relative to control | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID448841 | Inhibition of MMP10 assessed as residual activity at 10 uM after 10 to 15 mins by fluorescence assay relative to control | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID448865 | Inhibition of caspase 7 after 10 to 15 mins by fluorescence assay | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID448918 | Immunomodulatory activity in CD4+ human T cells assessed as inhibition of allogenic activated monocyte-derived dendritic cell-stimulated cell proliferation at 10 uM after 5 days by allogenic mixed lymphocyte reaction assay | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID448194 | Inhibition of DPP4 assessed as residual activity at 10 uM after 10 to 15 mins by fluorescence assay relative to control | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID448203 | Inhibition of factor 11a assessed as residual activity at 10 uM after 10 to 15 mins by fluorescence assay relative to control | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID448849 | Inhibition of BACE1 assessed as residual activity at 10 uM after 10 to 15 mins by fluorescence assay relative to control | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID448214 | Inhibition of calpain 1 assessed as residual activity at 10 uM after 10 to 15 mins by fluorescence assay relative to control | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID448198 | Inhibition of activated protein C assessed as residual activity at 10 uM after 10 to 15 mins by fluorescence assay in presence of 50% glycine relative to control | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID448186 | Selectivity ratio of IC50 for cathepsin E in human MCF7 cells to IC50 for cathepsin E | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID448202 | Inhibition of factor 10a assessed as residual activity at 10 uM after 10 to 15 mins by fluorescence assay relative to control | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID448857 | Inhibition of BACE1 after 10 to 15 mins by fluorescence assay | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID448859 | Inhibition of caspase 1 after 10 to 15 mins by fluorescence assay | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID448219 | Inhibition of caspase 5 assessed as residual activity at 10 uM after 10 to 15 mins by fluorescence assay relative to control | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID448906 | Inhibition of human renin after 10 to 15 mins by fluorescence assay | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID448220 | Inhibition of caspase 6 assessed as residual activity at 10 uM after 10 to 15 mins by fluorescence assay relative to control | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID448199 | Inhibition of chymase assessed as residual activity at 10 uM after 10 to 15 mins by fluorescence assay relative to control | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID448179 | Inhibition of ADAM10 | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID448901 | Inhibition of MMP13 catalytic domain after 10 to 15 mins by fluorescence assay | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID448891 | Inhibition of kallikrein 8 after 10 to 15 mins by fluorescence assay | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID711205 | Selectivity index, ratio of IC50 for cathepsin D to IC50 for cathepsin E | 2012 | Journal of medicinal chemistry, Dec-13, Volume: 55, Issue:23
| Cyanobacterial peptides as a prototype for the design of potent β-secretase inhibitors and the development of selective chemical probes for other aspartic proteases. |
| AID448848 | Inhibition of TACE assessed as residual activity at 10 uM after 10 to 15 mins by fluorescence assay relative to control | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID448873 | Inhibition of cathepsin D after 10 to 15 mins by fluorescence assay | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID674499 | Inhibition of cathepsin D using MCA-KPILFFRLK(Dnp)-D-R-NH2 as substrate incubated for 10 to 15 mins prior to substrate addition measured every 5 min for 2 hrs by fluorometry | 2012 | Bioorganic & medicinal chemistry, Aug-01, Volume: 20, Issue:15
| Total synthesis of grassystatin A, a probe for cathepsin E function. |
| AID448188 | Inhibition of cathepsin D in human MCF7 cells treated for 1 hr measured after washout and trypsin treatment by fluorescence assay | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID448850 | Inhibition of cathepsin D assessed as residual activity at 10 uM after 10 to 15 mins by fluorescence assay relative to control | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID448913 | Immunomodulatory activity in human T cells assessed as inhibition of tetanus toxin C-fragment-induced cell proliferation at 10 uM after 3 mins by FACS analysis | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID1493089 | Selectivity ratio of IC50 for human liver cathepsin D to IC50 for recombinant human C-terminal His10-tagged cathepsin E (Gln18 to Pro396 residues) | 2017 | Journal of natural products, 11-22, Volume: 80, Issue:11
| Grassystatins D-F, Potent Aspartic Protease Inhibitors from Marine Cyanobacteria as Potential Antimetastatic Agents Targeting Invasive Breast Cancer. |
| AID448862 | Inhibition of caspase 4 after 10 to 15 mins by fluorescence assay | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID448234 | Inhibition of cathepsin Z assessed as residual activity at 10 uM after 10 to 15 mins by fluorescence assay relative to control | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID448233 | Inhibition of cathepsin X assessed as residual activity at 10 uM after 10 to 15 mins by fluorescence assay relative to control | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID448853 | Inhibition of activated protein C after 10 to 15 mins by fluorescence assay in presence of 50% glycine | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID448916 | Antiinflammatory activity in CD4+ human T cells assessed as inhibition of autologous activated monocyte-derived dendritic cell-induced IL17 upregulation at 0.1 to 10 uM after 5 days by FACS analysis | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID448864 | Inhibition of caspase 6 after 10 to 15 mins by fluorescence assay | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID448209 | Inhibition of thrombin alpha assessed as residual activity at 10 uM after 10 to 15 mins by fluorescence assay relative to control | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID448875 | Inhibition of cathepsin H after 10 to 15 mins by fluorescence assay | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID448890 | Inhibition of kallikrein 5 after 10 to 15 mins by fluorescence assay | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID448237 | Inhibition of MMP2 assessed as residual activity at 10 uM after 10 to 15 mins by fluorescence assay relative to control | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID448226 | Inhibition of cathepsin B assessed as residual activity at 10 uM after 10 to 15 mins by fluorescence assay relative to control | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID448899 | Inhibition of MMP11 catalytic domain after 10 to 15 mins by fluorescence assay | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID448840 | Inhibition of MMP9 assessed as residual activity at 10 uM after 10 to 15 mins by fluorescence assay relative to control | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID448882 | Inhibition of chymotrypsin after 10 to 15 mins by fluorescence assay | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID448886 | Inhibition of porcine pancreatic elastase after 10 to 15 mins by fluorescence assay | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID1493087 | Inhibition of human liver cathepsin D using Mca-Gly-Lys-Pro-Ile-Leu-PhePhe-Arg-Leu-Lys-(Dnp)-D-Arg-NH2 as substrate pretreated for 15 mins followed by substrate addition measured at 5 mins interval for 120 mins by fluorescence assay | 2017 | Journal of natural products, 11-22, Volume: 80, Issue:11
| Grassystatins D-F, Potent Aspartic Protease Inhibitors from Marine Cyanobacteria as Potential Antimetastatic Agents Targeting Invasive Breast Cancer. |
| AID448894 | Inhibition of MMP3 after 10 to 15 mins by fluorescence assay | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID448854 | Inhibition of ACE1 after 10 to 15 mins by fluorescence assay | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID448895 | Inhibition of MMP7 after 10 to 15 mins by fluorescence assay | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID448844 | Inhibition of MMP13 assessed as residual activity at 10 uM after 10 to 15 mins by fluorescence assay relative to control | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID448879 | Inhibition of cathepsin X after 10 to 15 mins by fluorescence assay | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID448207 | Inhibition of plasma kallikrein assessed as residual activity at 10 uM after 10 to 15 mins by fluorescence assay relative to control | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID448903 | Inhibition of papaya papain after 10 to 15 mins by fluorescence assay | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID448190 | Selectivity ratio of IC50 for cathepsin D in human MCF7 cells treated for 1 hr measured after washout and trypsin treatment to IC50 for cathepsin D | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID448907 | Inhibition of TACE after 10 to 15 mins by fluorescence assay | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID448210 | Inhibition of bovine pancreatic trypsin assessed as residual activity at 10 uM after 10 to 15 mins by fluorescence assay relative to control | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID448208 | Inhibition of human plasmin assessed as residual activity at 10 uM after 10 to 15 mins by fluorescence assay relative to control | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID448215 | Inhibition of caspase 1 assessed as residual activity at 10 uM after 10 to 15 mins by fluorescence assay relative to control | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID448881 | Inhibition of chymase after 10 to 15 mins by fluorescence assay | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID448229 | Inhibition of cathepsin K assessed as residual activity at 10 uM after 10 to 15 mins by fluorescence assay relative to control | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID448230 | Inhibition of cathepsin S assessed as residual activity at 10 uM after 10 to 15 mins by fluorescence assay relative to control | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID448222 | Inhibition of caspase 8 assessed as residual activity at 10 uM after 10 to 15 mins by fluorescence assay relative to control | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID448880 | Inhibition of cathepsin Z after 10 to 15 mins by fluorescence assay | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID448195 | Inhibition of DPP8 assessed as residual activity at 10 uM after 10 to 15 mins by fluorescence assay relative to control | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID448878 | Inhibition of cathepsin V after 10 to 15 mins by fluorescence assay | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID448842 | Inhibition of MMP11 assessed as residual activity at 10 uM after 10 to 15 mins by fluorescence assay relative to control | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID448871 | Inhibition of cathepsin B after 10 to 15 mins by fluorescence assay | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID711208 | Inhibition of BACE1 by fluorescence assay | 2012 | Journal of medicinal chemistry, Dec-13, Volume: 55, Issue:23
| Cyanobacterial peptides as a prototype for the design of potent β-secretase inhibitors and the development of selective chemical probes for other aspartic proteases. |
| AID448227 | Inhibition of cathepsin H assessed as residual activity at 10 uM after 10 to 15 mins by fluorescence assay relative to control | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID448860 | Inhibition of caspase 2 after 10 to 15 mins by fluorescence assay | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID448839 | Inhibition of MMP8 assessed as residual activity at 10 uM after 10 to 15 mins by fluorescence assay relative to control | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID448201 | Inhibition of porcine pancreatic elastase assessed as residual activity at 10 uM after 10 to 15 mins by fluorescence assay relative to control | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID448856 | Inhibition of ADAM10 after 10 to 15 mins by fluorescence assay | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID448223 | Inhibition of caspase 9 assessed as residual activity at 10 uM after 10 to 15 mins by fluorescence assay relative to control | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID711207 | Inhibition of cathepsin D by fluorescence assay | 2012 | Journal of medicinal chemistry, Dec-13, Volume: 55, Issue:23
| Cyanobacterial peptides as a prototype for the design of potent β-secretase inhibitors and the development of selective chemical probes for other aspartic proteases. |
| AID448178 | Inhibition of ADAM9 | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID448905 | Inhibition of human plasmin after 10 to 15 mins by fluorescence assay | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID448876 | Inhibition of cathepsin K after 10 to 15 mins by fluorescence assay | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID448885 | Inhibition of DPP9 after 10 to 15 mins by fluorescence assay | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID448177 | Inhibition of cathepsin E | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID448917 | Antiinflammatory activity in CD4+ human T cells assessed as inhibition of autologous activated monocyte-derived dendritic cell-induced IFN-gamma upregulation at 0.1 to 10 uM after 5 days by FACS analysis | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID448225 | Inhibition of mouse caspase 11 assessed as residual activity at 10 uM after 10 to 15 mins by fluorescence assay relative to control | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID448908 | Inhibition of thrombin alpha after 10 to 15 mins by fluorescence assay | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID448837 | Inhibition of MMP3 assessed as residual activity at 10 uM after 10 to 15 mins by fluorescence assay relative to control | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID448206 | Inhibition of kallikrein 8 assessed as residual activity at 10 uM after 10 to 15 mins by fluorescence assay relative to control | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID448914 | Cytotoxicity against human T cells at 10 uM after 30 mins by FACS | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID448909 | Inhibition of bovine pancreatic trypsin after 10 to 15 mins by fluorescence assay | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID448183 | Inhibition of cathepsin D in human MCF7 cells by fluorescence assay | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID448897 | Inhibition of MMP9 catalytic domain after 10 to 15 mins by fluorescence assay | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID674496 | Inhibition of cathepsin E using MCA-KPILFFRLK(Dnp)-D-R-NH2 as substrate incubated for 10 to 15 mins prior to substrate addition measured every 5 min for 2 hrs by fluorometry | 2012 | Bioorganic & medicinal chemistry, Aug-01, Volume: 20, Issue:15
| Total synthesis of grassystatin A, a probe for cathepsin E function. |
| AID448197 | Inhibition of cathepsin C assessed as residual activity at 10 uM after 10 to 15 mins by fluorescence assay relative to control | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID448892 | Inhibition of MMP1 after 10 to 15 mins by fluorescence assay | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID448232 | Inhibition of papaya papain assessed as residual activity at 10 uM after 10 to 15 mins by fluorescence assay relative to control | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID448221 | Inhibition of caspase 7 assessed as residual activity at 10 uM after 10 to 15 mins by fluorescence assay relative to control | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID448216 | Inhibition of caspase 2 assessed as residual activity at 10 uM after 10 to 15 mins by fluorescence assay relative to control | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID448200 | Inhibition of chymotrypsin assessed as residual activity at 10 uM after 10 to 15 mins by fluorescence assay relative to control | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID448912 | Inhibition of urokinase after 10 to 15 mins by fluorescence assay | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID448869 | Inhibition of mouse caspase 11 after 10 to 15 mins by fluorescence assay | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID448176 | Inhibition of cathepsin D | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID447677 | Antiinflammatory activity in CD4+ human T cells assessed as inhibition of allogenic activated monocyte-derived dendritic cell-induced IL17 upregulation at 0.1 to 10 uM after 5 days by FACS analysis | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID448868 | Inhibition of caspase 10 after 10 to 15 mins by fluorescence assay | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID448187 | Selectivity ratio of IC50 for cathepsin D to IC50 for cathepsin E | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID448846 | Inhibition of ADAM9 assessed as residual activity at 10 uM after 10 to 15 mins by fluorescence assay relative to control | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID448888 | Inhibition of factor 11a after 10 to 15 mins by fluorescence assay | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID448192 | Selectivity ratio of IC50 for cathepsin D in human MCF7 cells treated for 1 hr measured after washout and trypsin treatment to IC50 for cathepsin D in human MCF7 cells | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID448910 | Inhibition of tryptase beta2 after 10 to 15 mins by fluorescence assay | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID1493088 | Inhibition of recombinant human C-terminal His10-tagged cathepsin E (Gln18 to Pro396 residues) using Mca-Gly-Lys-Pro-Ile-Leu-PhePhe-Arg-Leu-Lys-(Dnp)-D-Arg-NH2 as substrate pretreated for 15 mins followed by substrate addition measured at 5 mins interval | 2017 | Journal of natural products, 11-22, Volume: 80, Issue:11
| Grassystatins D-F, Potent Aspartic Protease Inhibitors from Marine Cyanobacteria as Potential Antimetastatic Agents Targeting Invasive Breast Cancer. |
| AID448181 | Inhibition of cathepsin E at 5.08 to 100000 nM | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID447678 | Antiinflammatory activity in CD4+ human T cells assessed as inhibition of allogenic activated monocyte-derived dendritic cell-induced IFN-gamma upregulation at 0.1 to 10 uM after 5 days by FACS analysis | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID448877 | Inhibition of cathepsin S after 10 to 15 mins by fluorescence assay | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID448852 | Inhibition of human renin assessed as residual activity at 10 uM after 10 to 15 mins by fluorescence assay relative to control | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID448189 | Inhibition of cathepsin E in human MCF7 cells treated for 1 hr measured after washout and trypsin treatment by fluorescence assay | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID448870 | Inhibition of caspase 14 after 10 to 15 mins by fluorescence assay | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID448212 | Inhibition of human lung tryptase gamma1 assessed as residual activity at 10 uM after 10 to 15 mins by fluorescence assay relative to control | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID711206 | Inhibition of cathepsin E by fluorescence assay | 2012 | Journal of medicinal chemistry, Dec-13, Volume: 55, Issue:23
| Cyanobacterial peptides as a prototype for the design of potent β-secretase inhibitors and the development of selective chemical probes for other aspartic proteases. |
| AID448904 | Inhibition of plasma kallikrein after 10 to 15 mins by fluorescence assay | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID447679 | Immunomodulatory activity in CD4+ human T cells assessed as inhibition of monocyte-derived dendritic cell presented PMA-induced cell proliferation after 5 days by autologous mixed lymphocyte reaction assay | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID448861 | Inhibition of caspase 3 after 10 to 15 mins by fluorescence assay | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID448902 | Inhibition of MMP14 catalytic domain after 10 to 15 mins by fluorescence assay | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID448196 | Inhibition of DPP9 assessed as residual activity at 10 uM after 10 to 15 mins by fluorescence assay relative to control | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID448867 | Inhibition of caspase 9 after 10 to 15 mins by fluorescence assay | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID448883 | Inhibition of DPP4 after 10 to 15 mins by fluorescence assay | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID448863 | Inhibition of caspase 5 after 10 to 15 mins by fluorescence assay | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID448185 | Selectivity ratio of IC50 for cathepsin D in human MCF7 cells to IC50 for cathepsin D | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID448874 | Inhibition of cathepsin E after 10 to 15 mins by fluorescence assay | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID448182 | Inhibition of TACE at 5.08 to 100000 nM | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID448900 | Inhibition of MMP12 catalytic domain after 10 to 15 mins by fluorescence assay | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID448205 | Inhibition of kallikrein 5 assessed as residual activity at 10 uM after 10 to 15 mins by fluorescence assay relative to control | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID1345892 | Human cathepsin D (A1: Pepsin) | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| AID1345444 | Human Caspase 14 (C14: Caspase) | 2009 | Journal of medicinal chemistry, Sep-24, Volume: 52, Issue:18
| Grassystatins A-C from marine cyanobacteria, potent cathepsin E inhibitors that reduce antigen presentation. |
| [information is prepared from bioassay data collected from National Library of Medicine (NLM), extracted Dec-2023] |