Assay ID | Title | Year | Journal | Article |
AID1803485 | ChEMBL_158305 (CHEMBL763190) from Article 10.1016/j.bmc.2016.05.029: \\Anion inhibition profiles of a-, u00DF- and u00BF-carbonic anhydrases from the pathogenic bacterium Vibrio cholerae.\\ | 2016 | Bioorganic & medicinal chemistry, 08-15, Volume: 24, Issue:16
| Anion inhibition profiles of α-, β- and γ-carbonic anhydrases from the pathogenic bacterium Vibrio cholerae. |
AID1798763 | CA Inhibition Assay from Article 10.1016/j.bmcl.2008.12.082: \\Carbonic anhydrase inhibitors: the membrane-associated isoform XV is highly inhibited by inorganic anions.\\ | 2009 | Bioorganic & medicinal chemistry letters, Feb-15, Volume: 19, Issue:4
| Carbonic anhydrase inhibitors: the membrane-associated isoform XV is highly inhibited by inorganic anions. |
AID1803491 | ChEMBL_158311 (CHEMBL763368) from Article 10.1016/j.bmc.2016.05.029: \\Anion inhibition profiles of a-, u00DF- and u00BF-carbonic anhydrases from the pathogenic bacterium Vibrio cholerae.\\ | 2016 | Bioorganic & medicinal chemistry, 08-15, Volume: 24, Issue:16
| Anion inhibition profiles of α-, β- and γ-carbonic anhydrases from the pathogenic bacterium Vibrio cholerae. |
AID1803493 | ChEMBL_158313 (CHEMBL763370) from Article 10.1016/j.bmc.2016.05.029: \\Anion inhibition profiles of a-, u00DF- and u00BF-carbonic anhydrases from the pathogenic bacterium Vibrio cholerae.\\ | 2016 | Bioorganic & medicinal chemistry, 08-15, Volume: 24, Issue:16
| Anion inhibition profiles of α-, β- and γ-carbonic anhydrases from the pathogenic bacterium Vibrio cholerae. |
AID1803487 | ChEMBL_158307 (CHEMBL763192) from Article 10.1016/j.bmc.2016.05.029: \\Anion inhibition profiles of a-, u00DF- and u00BF-carbonic anhydrases from the pathogenic bacterium Vibrio cholerae.\\ | 2016 | Bioorganic & medicinal chemistry, 08-15, Volume: 24, Issue:16
| Anion inhibition profiles of α-, β- and γ-carbonic anhydrases from the pathogenic bacterium Vibrio cholerae. |
AID1803254 | CA Inhibition Assay from Article 10.3109/14756366.2011.649268: \\Inhibition of the alpha- and beta-carbonic anhydrases from the gastric pathogen Helycobacter pylori with anions.\\ | 2013 | Journal of enzyme inhibition and medicinal chemistry, Apr, Volume: 28, Issue:2
| Inhibition of the alpha- and beta-carbonic anhydrases from the gastric pathogen Helycobacter pylori with anions. |
AID1803484 | ChEMBL_158304 (CHEMBL763189) from Article 10.1016/j.bmc.2016.05.029: \\Anion inhibition profiles of a-, u00DF- and u00BF-carbonic anhydrases from the pathogenic bacterium Vibrio cholerae.\\ | 2016 | Bioorganic & medicinal chemistry, 08-15, Volume: 24, Issue:16
| Anion inhibition profiles of α-, β- and γ-carbonic anhydrases from the pathogenic bacterium Vibrio cholerae. |
AID1803486 | ChEMBL_158306 (CHEMBL763191) from Article 10.1016/j.bmc.2016.05.029: \\Anion inhibition profiles of a-, u00DF- and u00BF-carbonic anhydrases from the pathogenic bacterium Vibrio cholerae.\\ | 2016 | Bioorganic & medicinal chemistry, 08-15, Volume: 24, Issue:16
| Anion inhibition profiles of α-, β- and γ-carbonic anhydrases from the pathogenic bacterium Vibrio cholerae. |
AID1278741 | Inhibition of Vibrio cholerae alpha-carbonic anhydrase preincubated for 15 mins by stopped-flow CO2 hydration assay | 2016 | Bioorganic & medicinal chemistry letters, Mar-01, Volume: 26, Issue:5
| Anion inhibition studies of the β-carbonic anhydrase from the pathogenic bacterium Vibrio cholerae. |
AID1430528 | Inhibition of Burkholderia pseudomallei recombinant His-tagged carbonic anhydrase beta (256 residues) expressed in Escherichia coli BL21 (DE3) incubated for 15 mins prior to testing by stopped flow CO2 hydration method | | | |
AID484158 | Inhibition of full length human carbonic anhydrase 5a preincubated for 15 mins by CO2 hydration stopped-flow assay | 2010 | Bioorganic & medicinal chemistry letters, Jun-15, Volume: 20, Issue:12
| Carbonic anhydrase inhibitors: crystallographic and solution binding studies for the interaction of a boron-containing aromatic sulfamide with mammalian isoforms I-XV. |
AID484163 | Inhibition of human carbonic anhydrase 12 catalytic domain preincubated for 15 mins by CO2 hydration stopped-flow assay | 2010 | Bioorganic & medicinal chemistry letters, Jun-15, Volume: 20, Issue:12
| Carbonic anhydrase inhibitors: crystallographic and solution binding studies for the interaction of a boron-containing aromatic sulfamide with mammalian isoforms I-XV. |
AID1161951 | Inhibition of Porphyromonas gingivalis gamma-carbonic anhydrase preincubated for 15 mins by stopped flow CO2 hydration method | 2014 | Bioorganic & medicinal chemistry letters, Sep-15, Volume: 24, Issue:18
| Anion inhibition study of the β-class carbonic anhydrase (PgiCAb) from the oral pathogen Porphyromonas gingivalis. |
AID1237484 | Induction of growth delay of Pseudomonas aeruginosa PAO1 assessed as growth delay time | 2015 | Bioorganic & medicinal chemistry, Aug-01, Volume: 23, Issue:15
| Structure and inhibition studies of a type II beta-carbonic anhydrase psCA3 from Pseudomonas aeruginosa. |
AID411399 | Inhibition of Candida albicans carbonic anhydrase overexpressed in Escherichia coli BL21 (DE3) by CO2 hydration stopped-flow assay | 2008 | Bioorganic & medicinal chemistry letters, Dec-15, Volume: 18, Issue:24
| Carbonic anhydrase inhibitors. Inhibition of the beta-class enzyme from the yeast Saccharomyces cerevisiae with anions. |
AID1235242 | Inhibition of archaeon Methanosarcina thermophila gamma-CA after 15 mins by stopped-flow/Co2 hydration assay | 2015 | Bioorganic & medicinal chemistry, Aug-01, Volume: 23, Issue:15
| Cloning, characterization and anion inhibition studies of a new γ-carbonic anhydrase from the Antarctic bacterium Pseudoalteromonas haloplanktis. |
AID1336557 | Inhibition of human recombinant carbonic anhydrase 2 assessed as inhibition of CO2 hydration preincubated for 15 mins by Lineweaver-burk plot method | | | |
AID238653 | Inhibitory constant against carbonic anhydrase IV; nt= not tested | 2004 | Bioorganic & medicinal chemistry letters, Sep-06, Volume: 14, Issue:17
| Carbonic anhydrase inhibitors. Inhibition of the beta-class enzyme from the methanoarchaeon Methanobacterium thermoautotrophicum (Cab) with anions. |
AID239250 | Inhibitory activity against beta carbonic anhydrase (Cab) from Methanobacterium thermoautotrophicum | 2004 | Bioorganic & medicinal chemistry letters, Dec-20, Volume: 14, Issue:24
| Carbonic anhydrase inhibitors. Inhibition of the prokariotic beta and gamma-class enzymes from Archaea with sulfonamides. |
AID552130 | Inhibition of Stylophora pistillata carbonic anhydrase by stopped-flow CO2 hydration assay | 2011 | Bioorganic & medicinal chemistry letters, Jan-15, Volume: 21, Issue:2
| Carbonic anhydrase inhibitors. Inhibition studies with anions and sulfonamides of a new cytosolic enzyme from the scleractinian coral Stylophora pistillata. |
AID238688 | Inhibitory activity against human carbonic anhydrase V expressed in Escherichia coli | 2004 | Bioorganic & medicinal chemistry letters, Nov-01, Volume: 14, Issue:21
| Carbonic anhydrase inhibitors. Inhibition of the newly isolated murine isozyme XIII with anions. |
AID1278739 | Inhibition of human carbonic anhydrase 1 preincubated for 15 mins by stopped-flow CO2 hydration assay | 2016 | Bioorganic & medicinal chemistry letters, Mar-01, Volume: 26, Issue:5
| Anion inhibition studies of the β-carbonic anhydrase from the pathogenic bacterium Vibrio cholerae. |
AID484164 | Inhibition of full length mouse carbonic anhydrase 13 preincubated for 15 mins by CO2 hydration stopped-flow assay | 2010 | Bioorganic & medicinal chemistry letters, Jun-15, Volume: 20, Issue:12
| Carbonic anhydrase inhibitors: crystallographic and solution binding studies for the interaction of a boron-containing aromatic sulfamide with mammalian isoforms I-XV. |
AID239145 | Inhibitory activity against alpha carbonic anhydrase (Co-Cam) from Methanosarcina thermophila | 2004 | Bioorganic & medicinal chemistry letters, Dec-20, Volume: 14, Issue:24
| Carbonic anhydrase inhibitors. Inhibition of the prokariotic beta and gamma-class enzymes from Archaea with sulfonamides. |
AID724719 | Inhibition of human recombinant CA10 mutant after 15 mins by stopped-flow CO2 hydration method | 2013 | Bioorganic & medicinal chemistry letters, Jan-01, Volume: 23, Issue:1
| Restoring catalytic activity to the human carbonic anhydrase (CA) related proteins VIII, X and XI affords isoforms with high catalytic efficiency and susceptibility to anion inhibition. |
AID238986 | Inhibitory activity against human carbonic anhydrase II at 0.01 uM | 2004 | Bioorganic & medicinal chemistry letters, Dec-20, Volume: 14, Issue:24
| Carbonic anhydrase inhibitors. Inhibition of the prokariotic beta and gamma-class enzymes from Archaea with sulfonamides. |
AID1312218 | Inhibition of Plasmodium falciparum full length recombinant His-fused Eta-carbonic anhydrase domain preincubated for 15 mins by stopped-flow CO2 hydrase assay | 2016 | Bioorganic & medicinal chemistry, 09-15, Volume: 24, Issue:18
| Anion inhibition profiles of the complete domain of the η-carbonic anhydrase from Plasmodium falciparum. |
AID47903 | Inhibitory activity against human cloned carbonic anhydrase II (hCA II) | 2003 | Bioorganic & medicinal chemistry letters, Mar-10, Volume: 13, Issue:5
| Carbonic anhydrase inhibitors: SAR and X-ray crystallographic study for the interaction of sugar sulfamates/sulfamides with isozymes I, II and IV. |
AID265737 | Inhibition of human recombinant CA7 | 2006 | Bioorganic & medicinal chemistry letters, Jun-15, Volume: 16, Issue:12
| Carbonic anhydrase inhibitors: inhibition of the cytosolic human isozyme VII with anions. |
AID552131 | Inhibition of Stylophora pistillata carbonic anhydrase 2 by stopped-flow CO2 hydration assay | 2011 | Bioorganic & medicinal chemistry letters, Jan-15, Volume: 21, Issue:2
| Carbonic anhydrase inhibitors. Inhibition studies with anions and sulfonamides of a new cytosolic enzyme from the scleractinian coral Stylophora pistillata. |
AID48125 | Inhibitory activity against carbonic anhydrase isolated from bovine lung microsome (bCA IV); nt is not tested | 2003 | Bioorganic & medicinal chemistry letters, Mar-10, Volume: 13, Issue:5
| Carbonic anhydrase inhibitors: SAR and X-ray crystallographic study for the interaction of sugar sulfamates/sulfamides with isozymes I, II and IV. |
AID392570 | Inhibition of human recombinant carbonic anhydrase 4 by CO2 hydration reaction | 2009 | Bioorganic & medicinal chemistry letters, Feb-15, Volume: 19, Issue:4
| Carbonic anhydrase inhibitors: the membrane-associated isoform XV is highly inhibited by inorganic anions. |
AID1161930 | Inhibition of human carbonic anhydrase 1 preincubated for 15 mins by stopped flow CO2 hydration method | 2014 | Bioorganic & medicinal chemistry letters, Sep-15, Volume: 24, Issue:18
| Discovery of a new family of carbonic anhydrases in the malaria pathogen Plasmodium falciparum--the η-carbonic anhydrases. |
AID647373 | Inhibition of Astrosclera willeyana recombinant GST-tagged astrosclerin 3 expressed in Escherichia coli BL21-DE3-RIPL cells preincubated for 15 mins measured for 10 to 100 secs by stopped flow CO2 hydration assay | 2012 | Bioorganic & medicinal chemistry letters, Feb-01, Volume: 22, Issue:3
| Anion inhibition studies of an α-carbonic anhydrase from the living fossil Astrosclera willeyana. |
AID1461935 | Inhibition of Burkholderia pseudomallei beta-CA incubated for 15 mins by stopped-flow CO2 hydration assay | | | |
AID411398 | Inhibition of human carbonic anhydrase 2 by CO2 hydration stopped-flow assay | 2008 | Bioorganic & medicinal chemistry letters, Dec-15, Volume: 18, Issue:24
| Carbonic anhydrase inhibitors. Inhibition of the beta-class enzyme from the yeast Saccharomyces cerevisiae with anions. |
AID1306524 | Inhibition of human carbonic anhydrase 2 preincubated for 15 mins by stopped-flow CO2 hydrase assay | 2016 | Bioorganic & medicinal chemistry, 08-15, Volume: 24, Issue:16
| Anion inhibition profiles of α-, β- and γ-carbonic anhydrases from the pathogenic bacterium Vibrio cholerae. |
AID730753 | Inhibition of human carbonic anhydrase 2 preincubated for 15 mins by stopped flow CO2 hydration assay | 2013 | Bioorganic & medicinal chemistry letters, Mar-15, Volume: 23, Issue:6
| Anion inhibition studies of the α-carbonic anhydrase from the pathogenic bacterium Vibrio cholerae. |
AID1336561 | Inhibition of Pseudoalteromonas haloplanktis recombinant carbonic anhydrase gamma assessed as inhibition of CO2 hydration preincubated for 15 mins by Lineweaver-burk plot method | | | |
AID763567 | Inhibition of Brucella suis beta carbonic anhydrase-1 at 20 degC by stopped-flow CO2 hydrase assay | 2013 | Bioorganic & medicinal chemistry, Aug-01, Volume: 21, Issue:15
| Anion inhibition studies of the α-carbonic anhydrase from the protozoan pathogen Trypanosoma cruzi, the causative agent of Chagas disease. |
AID433253 | Inhibition of Candida glabrata carbonic anhydrase by stopped flow CO2 hydration assay | 2009 | Bioorganic & medicinal chemistry letters, Aug-15, Volume: 19, Issue:16
| Carbonic anhydrase inhibitors. Inhibition of the beta-class enzyme from the pathogenic yeast Candida glabrata with anions. |
AID50356 | Inhibitory activity against human cloned isoenzyme carbonic anhydrase I (hCA I), by esterase method. | 2003 | Bioorganic & medicinal chemistry letters, Mar-10, Volume: 13, Issue:5
| Carbonic anhydrase inhibitors: inhibition of cytosolic isozymes I and II with sulfamide derivatives. |
AID238715 | Inhibitory activity against human carbonic anhydrase II expressed in Escherichia coli | 2004 | Bioorganic & medicinal chemistry letters, Nov-01, Volume: 14, Issue:21
| Carbonic anhydrase inhibitors. Inhibition of the newly isolated murine isozyme XIII with anions. |
AID1161952 | Inhibition of Porphyromonas gingivalis beta-carbonic anhydrase preincubated for 15 mins by stopped flow CO2 hydration method | 2014 | Bioorganic & medicinal chemistry letters, Sep-15, Volume: 24, Issue:18
| Anion inhibition study of the β-class carbonic anhydrase (PgiCAb) from the oral pathogen Porphyromonas gingivalis. |
AID411397 | Inhibition of human carbonic anhydrase 1 by CO2 hydration stopped-flow assay | 2008 | Bioorganic & medicinal chemistry letters, Dec-15, Volume: 18, Issue:24
| Carbonic anhydrase inhibitors. Inhibition of the beta-class enzyme from the yeast Saccharomyces cerevisiae with anions. |
AID1161932 | Inhibition of recombinant Plasmodium falciparum eta-carbonic anhydrase preincubated for 15 mins by stopped flow CO2 hydration method | 2014 | Bioorganic & medicinal chemistry letters, Sep-15, Volume: 24, Issue:18
| Discovery of a new family of carbonic anhydrases in the malaria pathogen Plasmodium falciparum--the η-carbonic anhydrases. |
AID1461938 | Inhibition of recombinant His6-tagged Francisella tularensis beta-CA (227 residues) expressed in Escherichia coli BL21(DE3) incubated for 15 mins by stopped-flow CO2 hydration assay | | | |
AID749809 | Inhibition of human carbonic anhydrase-2 preincubated for 15 mins by stopped-flow CO2 hydration assay | 2013 | Bioorganic & medicinal chemistry, Jun-01, Volume: 21, Issue:11
| Synthesis and carbonic anhydrase inhibitory properties of sulfamides structurally related to dopamine. |
AID484159 | Inhibition of full length human carbonic anhydrase 5b preincubated for 15 mins by CO2 hydration stopped-flow assay | 2010 | Bioorganic & medicinal chemistry letters, Jun-15, Volume: 20, Issue:12
| Carbonic anhydrase inhibitors: crystallographic and solution binding studies for the interaction of a boron-containing aromatic sulfamide with mammalian isoforms I-XV. |
AID387188 | Inhibition of human carbonic anhydrase 2 at 20 degC by CO2 hydration method | 2008 | Bioorganic & medicinal chemistry letters, Sep-15, Volume: 18, Issue:18
| Carbonic anhydrase inhibitors: inhibition of the beta-class enzymes from the fungal pathogens Candida albicans and Cryptococcus neoformans with simple anions. |
AID295046 | Inhibition of human recombinant carbonic anhydrase 1 | 2007 | Bioorganic & medicinal chemistry letters, May-15, Volume: 17, Issue:10
| Carbonic anhydrase inhibitors: the X-ray crystal structure of the adduct of N-hydroxysulfamide with isozyme II explains why this new zinc binding function is effective in the design of potent inhibitors. |
AID392568 | Inhibition of human recombinant carbonic anhydrase 2 by CO2 hydration reaction | 2009 | Bioorganic & medicinal chemistry letters, Feb-15, Volume: 19, Issue:4
| Carbonic anhydrase inhibitors: the membrane-associated isoform XV is highly inhibited by inorganic anions. |
AID1235244 | Inhibition of Nostoc commune CA after 15 mins by stopped-flow/Co2 hydration assay | 2015 | Bioorganic & medicinal chemistry, Aug-01, Volume: 23, Issue:15
| Cloning, characterization and anion inhibition studies of a new γ-carbonic anhydrase from the Antarctic bacterium Pseudoalteromonas haloplanktis. |
AID587130 | Inhibition of human carbonic anhydrase 1 after 15 mins by CO2 hydrase assay at pH 7.5 | 2011 | Bioorganic & medicinal chemistry, Mar-15, Volume: 19, Issue:6
| Purification and inhibition studies with anions and sulfonamides of an α-carbonic anhydrase from the Antarctic seal Leptonychotes weddellii. |
AID730752 | Inhibition of Helicobacter pylori alpha carbonic anhydrase preincubated for 15 mins by stopped flow CO2 hydration assay | 2013 | Bioorganic & medicinal chemistry letters, Mar-15, Volume: 23, Issue:6
| Anion inhibition studies of the α-carbonic anhydrase from the pathogenic bacterium Vibrio cholerae. |
AID732714 | Inhibition of human erythrocytes esterase activity of carbonic anhydrase-2 using 4-nitrophenylacetate as substrate after 3 mins by Lineweaver-Burk plot analysis | 2013 | Bioorganic & medicinal chemistry, Mar-15, Volume: 21, Issue:6
| Novel sulfamides as potential carbonic anhydrase isoenzymes inhibitors. |
AID677271 | Inhibition of Helicobacter pylori alpha-carbonic anhydrase-catalyzed CO2 hydration reaction preincubated for 15 mins by stopped flow CO2 hydrase assay | 2012 | Bioorganic & medicinal chemistry letters, Sep-01, Volume: 22, Issue:17
| Anion inhibition studies of an α-carbonic anhydrase from the thermophilic bacterium Sulfurihydrogenibium yellowstonense YO3AOP1. |
AID1235245 | Inhibition of Pseudoalteromonas haloplanktis gamma-CA after 15 mins by stopped-flow/Co2 hydration assay | 2015 | Bioorganic & medicinal chemistry, Aug-01, Volume: 23, Issue:15
| Cloning, characterization and anion inhibition studies of a new γ-carbonic anhydrase from the Antarctic bacterium Pseudoalteromonas haloplanktis. |
AID484162 | Inhibition of human carbonic anhydrase 9 catalytic domain preincubated for 15 mins by CO2 hydration stopped-flow assay | 2010 | Bioorganic & medicinal chemistry letters, Jun-15, Volume: 20, Issue:12
| Carbonic anhydrase inhibitors: crystallographic and solution binding studies for the interaction of a boron-containing aromatic sulfamide with mammalian isoforms I-XV. |
AID730373 | Inhibition of human cytosolic carbonic anhydrase-2 preincubated for 15 mins by stopped flow CO2 hydration assay | 2013 | Bioorganic & medicinal chemistry letters, Mar-15, Volume: 23, Issue:6
| Kinetic and anion inhibition studies of a β-carbonic anhydrase (FbiCA 1) from the C4 plant Flaveria bidentis. |
AID1336562 | Inhibition of Burkholderia pseudomallei recombinant His-tagged carbonic anhydrase gamma expressed in Escherichia coli BL21 (DE3) assessed as inhibition of CO2 hydration preincubated for 15 mins by Lineweaver-burk plot method | | | |
AID305488 | Inhibition of full length human recombinant full length CA6 expressed in Escherichia coli BL21 by CO2 hydration method | 2007 | Bioorganic & medicinal chemistry letters, Feb-15, Volume: 17, Issue:4
| Carbonic anhydrase inhibitors. Inhibition studies of the human secretory isoform VI with anions. |
AID47904 | Inhibitory activity against human cloned isoenzyme carbonic anhydrase II (hCA II), by esterase method. | 2003 | Bioorganic & medicinal chemistry letters, Mar-10, Volume: 13, Issue:5
| Carbonic anhydrase inhibitors: inhibition of cytosolic isozymes I and II with sulfamide derivatives. |
AID387190 | Inhibition of Cryptococcus neoformans Can2 at 20 degC by CO2 hydration method | 2008 | Bioorganic & medicinal chemistry letters, Sep-15, Volume: 18, Issue:18
| Carbonic anhydrase inhibitors: inhibition of the beta-class enzymes from the fungal pathogens Candida albicans and Cryptococcus neoformans with simple anions. |
AID238222 | Inhibitory constant against human Carbonic anhydrase II | 2005 | Bioorganic & medicinal chemistry letters, May-02, Volume: 15, Issue:9
| Carbonic anhydrase inhibitors: synthesis and inhibition of cytosolic/tumor-associated carbonic anhydrase isozymes I, II, IX, and XII with N-hydroxysulfamides--a new zinc-binding function in the design of inhibitors. |
AID598731 | Inhibition of Salmonella Typhimurium carbonic anhydrase 1 after 15 mins by stopped flow CO2 hydration assay at pH 8.3 | 2011 | Bioorganic & medicinal chemistry letters, Jun-15, Volume: 21, Issue:12
| Inhibition studies with anions and small molecules of two novel β-carbonic anhydrases from the bacterial pathogen Salmonella enterica serovar Typhimurium. |
AID552785 | Inhibition of Streptococcus pneumoniae beta-carbonic anhydrase after 15 mins by stopped flow CO2 hydration assay | 2011 | Bioorganic & medicinal chemistry, Jan-01, Volume: 19, Issue:1
| Inhibition of the β-carbonic anhydrase from Streptococcus pneumoniae by inorganic anions and small molecules: Toward innovative drug design of antiinfectives? |
AID552127 | Inhibition of human recombinant CA1 by stopped-flow CO2 hydration assay | 2011 | Bioorganic & medicinal chemistry letters, Jan-15, Volume: 21, Issue:2
| Carbonic anhydrase inhibitors. Inhibition studies with anions and sulfonamides of a new cytosolic enzyme from the scleractinian coral Stylophora pistillata. |
AID238327 | Inhibitory constant against carbonic anhydrase II | 2004 | Bioorganic & medicinal chemistry letters, Sep-06, Volume: 14, Issue:17
| Carbonic anhydrase inhibitors. Inhibition of the beta-class enzyme from the methanoarchaeon Methanobacterium thermoautotrophicum (Cab) with anions. |
AID1058389 | Inhibition of Clostridium perfringens carbonic anhydrase preincubated for 15 mins by stopped flow CO2 hydration assay | 2013 | Bioorganic & medicinal chemistry letters, Dec-15, Volume: 23, Issue:24
| Anion inhibition studies of a β-carbonic anhydrase from Clostridium perfringens. |
AID1336560 | Inhibition of Nostoc commune recombinant carbonic anhydrase gamma assessed as inhibition of CO2 hydration preincubated for 15 mins by Lineweaver-burk plot method | | | |
AID724718 | Inhibition of human recombinant CA11 mutant after 15 mins by stopped-flow CO2 hydration method | 2013 | Bioorganic & medicinal chemistry letters, Jan-01, Volume: 23, Issue:1
| Restoring catalytic activity to the human carbonic anhydrase (CA) related proteins VIII, X and XI affords isoforms with high catalytic efficiency and susceptibility to anion inhibition. |
AID295047 | Inhibition of human recombinant carbonic anhydrase 2 | 2007 | Bioorganic & medicinal chemistry letters, May-15, Volume: 17, Issue:10
| Carbonic anhydrase inhibitors: the X-ray crystal structure of the adduct of N-hydroxysulfamide with isozyme II explains why this new zinc binding function is effective in the design of potent inhibitors. |
AID730754 | Inhibition of human carbonic anhydrase 1 preincubated for 15 mins by stopped flow CO2 hydration assay | 2013 | Bioorganic & medicinal chemistry letters, Mar-15, Volume: 23, Issue:6
| Anion inhibition studies of the α-carbonic anhydrase from the pathogenic bacterium Vibrio cholerae. |
AID724721 | Inhibition of human recombinant wild type CA2 by stopped-flow CO2 hydration method | 2013 | Bioorganic & medicinal chemistry letters, Jan-01, Volume: 23, Issue:1
| Restoring catalytic activity to the human carbonic anhydrase (CA) related proteins VIII, X and XI affords isoforms with high catalytic efficiency and susceptibility to anion inhibition. |
AID238687 | Inhibitory activity against human carbonic anhydrase I expressed in Escherichia coli | 2004 | Bioorganic & medicinal chemistry letters, Nov-01, Volume: 14, Issue:21
| Carbonic anhydrase inhibitors. Inhibition of the newly isolated murine isozyme XIII with anions. |
AID484154 | Inhibition of full length human carbonic anhydrase 1 preincubated for 15 mins by CO2 hydration stopped-flow assay | 2010 | Bioorganic & medicinal chemistry letters, Jun-15, Volume: 20, Issue:12
| Carbonic anhydrase inhibitors: crystallographic and solution binding studies for the interaction of a boron-containing aromatic sulfamide with mammalian isoforms I-XV. |
AID1306530 | Inhibition of Vibrio cholerae carbonic anhydrase beta preincubated for 15 mins by stopped-flow CO2 hydrase assay | 2016 | Bioorganic & medicinal chemistry, 08-15, Volume: 24, Issue:16
| Anion inhibition profiles of α-, β- and γ-carbonic anhydrases from the pathogenic bacterium Vibrio cholerae. |
AID1306525 | Inhibition of Helicobacter pylori alpha carbonic anhydrase preincubated for 15 mins by stopped-flow CO2 hydrase assay | 2016 | Bioorganic & medicinal chemistry, 08-15, Volume: 24, Issue:16
| Anion inhibition profiles of α-, β- and γ-carbonic anhydrases from the pathogenic bacterium Vibrio cholerae. |
AID758952 | Inhibition of human recombinant CA2 by CO2 hydration assay | 2013 | Bioorganic & medicinal chemistry letters, Jul-15, Volume: 23, Issue:14
| A highly catalytically active γ-carbonic anhydrase from the pathogenic anaerobe Porphyromonas gingivalis and its inhibition profile with anions and small molecules. |
AID1430527 | Inhibition of Burkholderia pseudomallei recombinant carbonic anhydrase gamma incubated for 15 mins prior to testing by stopped flow CO2 hydration method | | | |
AID677270 | Inhibition of Sulfurihydrogenibium yellowstonense YO3AOP1 alpha-carbonic anhydrase-catalyzed CO2 hydration reaction preincubated for 15 mins by stopped flow CO2 hydrase assay | 2012 | Bioorganic & medicinal chemistry letters, Sep-01, Volume: 22, Issue:17
| Anion inhibition studies of an α-carbonic anhydrase from the thermophilic bacterium Sulfurihydrogenibium yellowstonense YO3AOP1. |
AID1306532 | Inhibition of Vibrio cholerae recombinant carbonic anhydrase gamma expressed in Escherichia coli DE3 cells preincubated for 15 mins by stopped-flow CO2 hydrase assay | 2016 | Bioorganic & medicinal chemistry, 08-15, Volume: 24, Issue:16
| Anion inhibition profiles of α-, β- and γ-carbonic anhydrases from the pathogenic bacterium Vibrio cholerae. |
AID763566 | Inhibition of Brucella suis beta carbonic anhydrase-2 at 20 degC by stopped-flow CO2 hydrase assay | 2013 | Bioorganic & medicinal chemistry, Aug-01, Volume: 21, Issue:15
| Anion inhibition studies of the α-carbonic anhydrase from the protozoan pathogen Trypanosoma cruzi, the causative agent of Chagas disease. |
AID1461934 | Inhibition of human CA2 incubated for 15 mins by stopped-flow CO2 hydration assay | | | |
AID310902 | Inhibition of human recombinant catalytic domain CA12 | 2007 | Bioorganic & medicinal chemistry letters, Mar-15, Volume: 17, Issue:6
| Carbonic anhydrase inhibitors. Inhibition of transmembrane isozymes XII (cancer-associated) and XIV with anions. |
AID1269931 | Inhibition of Colwellia psychrerythraea gamma carbonic anhydrase expressed in Escherichia coli incubated for 15 mins prior to testing by stopped flow CO2 hydration method | 2016 | Bioorganic & medicinal chemistry, Feb-15, Volume: 24, Issue:4
| Cloning, characterization and anion inhibition studies of a γ-carbonic anhydrase from the Antarctic bacterium Colwellia psychrerythraea. |
AID238210 | Inhibitory constant against human Carbonic anhydrase I | 2005 | Bioorganic & medicinal chemistry letters, May-02, Volume: 15, Issue:9
| Carbonic anhydrase inhibitors: synthesis and inhibition of cytosolic/tumor-associated carbonic anhydrase isozymes I, II, IX, and XII with N-hydroxysulfamides--a new zinc-binding function in the design of inhibitors. |
AID484166 | Inhibition of full length mouse carbonic anhydrase 15 preincubated for 15 mins by CO2 hydration stopped-flow assay | 2010 | Bioorganic & medicinal chemistry letters, Jun-15, Volume: 20, Issue:12
| Carbonic anhydrase inhibitors: crystallographic and solution binding studies for the interaction of a boron-containing aromatic sulfamide with mammalian isoforms I-XV. |
AID238604 | Inhibition constant against human carbonic anhydrase isozyme hCA II | 2004 | Bioorganic & medicinal chemistry letters, Dec-06, Volume: 14, Issue:23
| Carbonic anhydrase inhibitors: inhibition of the membrane-bound human isozyme IV with anions. |
AID295049 | Inhibition of human recombinant carbonic anhydrase 12 catalytic domain by CO2 hydrase method | 2007 | Bioorganic & medicinal chemistry letters, May-15, Volume: 17, Issue:10
| Carbonic anhydrase inhibitors: the X-ray crystal structure of the adduct of N-hydroxysulfamide with isozyme II explains why this new zinc binding function is effective in the design of potent inhibitors. |
AID587131 | Inhibition of human carbonic anhydrase 2 after 15 mins by CO2 hydrase assay at pH 7.5 | 2011 | Bioorganic & medicinal chemistry, Mar-15, Volume: 19, Issue:6
| Purification and inhibition studies with anions and sulfonamides of an α-carbonic anhydrase from the Antarctic seal Leptonychotes weddellii. |
AID484155 | Inhibition of full length human carbonic anhydrase 2 preincubated for 15 mins by CO2 hydration stopped-flow assay | 2010 | Bioorganic & medicinal chemistry letters, Jun-15, Volume: 20, Issue:12
| Carbonic anhydrase inhibitors: crystallographic and solution binding studies for the interaction of a boron-containing aromatic sulfamide with mammalian isoforms I-XV. |
AID484156 | Inhibition of human carbonic anhydrase 3 preincubated for 15 mins by CO2 hydration stopped-flow assay | 2010 | Bioorganic & medicinal chemistry letters, Jun-15, Volume: 20, Issue:12
| Carbonic anhydrase inhibitors: crystallographic and solution binding studies for the interaction of a boron-containing aromatic sulfamide with mammalian isoforms I-XV. |
AID1306526 | Inhibition of Vibrio cholerae alpha carbonic anhydrase preincubated for 15 mins by stopped-flow CO2 hydrase assay | 2016 | Bioorganic & medicinal chemistry, 08-15, Volume: 24, Issue:16
| Anion inhibition profiles of α-, β- and γ-carbonic anhydrases from the pathogenic bacterium Vibrio cholerae. |
AID238605 | Inhibition constant against human carbonic anhydrase isozyme hCA IV | 2004 | Bioorganic & medicinal chemistry letters, Dec-06, Volume: 14, Issue:23
| Carbonic anhydrase inhibitors: inhibition of the membrane-bound human isozyme IV with anions. |
AID367655 | Inhibition of human secreted carbonic anhydrase 4 measured by CO2 hydration reaction assay | 2009 | Bioorganic & medicinal chemistry letters, Feb-01, Volume: 19, Issue:3
| Carbonic anhydrase inhibitors: inhibition studies of a coral secretory isoform with inorganic anions. |
AID763569 | Inhibition of human carbonic anhydrase-1 at 20 degC preincubated for 15 mins by stopped-flow CO2 hydrase assay | 2013 | Bioorganic & medicinal chemistry, Aug-01, Volume: 21, Issue:15
| Anion inhibition studies of the α-carbonic anhydrase from the protozoan pathogen Trypanosoma cruzi, the causative agent of Chagas disease. |
AID484160 | Inhibition of human carbonic anhydrase 6 preincubated for 15 mins by CO2 hydration stopped-flow assay | 2010 | Bioorganic & medicinal chemistry letters, Jun-15, Volume: 20, Issue:12
| Carbonic anhydrase inhibitors: crystallographic and solution binding studies for the interaction of a boron-containing aromatic sulfamide with mammalian isoforms I-XV. |
AID301197 | Inhibition of human mitochondrial CA5B by CO2 hydration assay | 2007 | Bioorganic & medicinal chemistry, Nov-01, Volume: 15, Issue:21
| Carbonic anhydrase inhibitors: the inhibition profiles of the human mitochondrial isoforms VA and VB with anions are very different. |
AID1278742 | Inhibition of recombinant Vibrio cholerae beta-carbonic anhydrase expressed in competent Escherichia coli BL21(DE3) cells preincubated for 15 mins by stopped-flow CO2 hydration assay | 2016 | Bioorganic & medicinal chemistry letters, Mar-01, Volume: 26, Issue:5
| Anion inhibition studies of the β-carbonic anhydrase from the pathogenic bacterium Vibrio cholerae. |
AID238579 | Inhibition constant against human carbonic anhydrase isozyme hCA V | 2004 | Bioorganic & medicinal chemistry letters, Dec-06, Volume: 14, Issue:23
| Carbonic anhydrase inhibitors: inhibition of the membrane-bound human isozyme IV with anions. |
AID484157 | Inhibition of full length human carbonic anhydrase 4 preincubated for 15 mins by CO2 hydration stopped-flow assay | 2010 | Bioorganic & medicinal chemistry letters, Jun-15, Volume: 20, Issue:12
| Carbonic anhydrase inhibitors: crystallographic and solution binding studies for the interaction of a boron-containing aromatic sulfamide with mammalian isoforms I-XV. |
AID763565 | Inhibition of recombinant Trypanosoma cruzi CL Brener alpha carbonic anhydrase expressed in baculovirus infected SF9 cells at 20 degC preincubated for 15 mins by stopped-flow CO2 hydrase assay | 2013 | Bioorganic & medicinal chemistry, Aug-01, Volume: 21, Issue:15
| Anion inhibition studies of the α-carbonic anhydrase from the protozoan pathogen Trypanosoma cruzi, the causative agent of Chagas disease. |
AID238410 | Inhibitory activity against human Carbonic anhydrase I | 2005 | Bioorganic & medicinal chemistry letters, Feb-01, Volume: 15, Issue:3
| Carbonic anhydrase inhibitors. Inhibition of isozymes I, II, IV, V, and IX with anions isosteric and isoelectronic with sulfate, nitrate, and carbonate. |
AID367653 | Inhibition of human carbonic anhydrase 1 measured by CO2 hydration reaction assay | 2009 | Bioorganic & medicinal chemistry letters, Feb-01, Volume: 19, Issue:3
| Carbonic anhydrase inhibitors: inhibition studies of a coral secretory isoform with inorganic anions. |
AID1237486 | Growth inhibition of Pseudomonas aeruginosa PAO1 | 2015 | Bioorganic & medicinal chemistry, Aug-01, Volume: 23, Issue:15
| Structure and inhibition studies of a type II beta-carbonic anhydrase psCA3 from Pseudomonas aeruginosa. |
AID387434 | Inhibition of Candida albicans Nce103 at 20 degC by CO2 hydration method | 2008 | Bioorganic & medicinal chemistry letters, Sep-15, Volume: 18, Issue:18
| Carbonic anhydrase inhibitors: inhibition of the beta-class enzymes from the fungal pathogens Candida albicans and Cryptococcus neoformans with simple anions. |
AID730751 | Inhibition of Vibrio cholerae alpha carbonic anhydrase preincubated for 15 mins by stopped flow CO2 hydration assay | 2013 | Bioorganic & medicinal chemistry letters, Mar-15, Volume: 23, Issue:6
| Anion inhibition studies of the α-carbonic anhydrase from the pathogenic bacterium Vibrio cholerae. |
AID238957 | Inhibitory activity against human carbonic anhydrase I at 0.09 uM | 2004 | Bioorganic & medicinal chemistry letters, Dec-20, Volume: 14, Issue:24
| Carbonic anhydrase inhibitors. Inhibition of the prokariotic beta and gamma-class enzymes from Archaea with sulfonamides. |
AID239146 | Inhibitory activity against alpha carbonic anhydrase (Zn-Cam) from Methanosarcina thermophila | 2004 | Bioorganic & medicinal chemistry letters, Dec-20, Volume: 14, Issue:24
| Carbonic anhydrase inhibitors. Inhibition of the prokariotic beta and gamma-class enzymes from Archaea with sulfonamides. |
AID1336559 | Inhibition of Porphyromonas gingivalis recombinant carbonic anhydrase gamma assessed as inhibition of CO2 hydration preincubated for 15 mins by Lineweaver-burk plot method | | | |
AID392569 | Inhibition of human recombinant carbonic anhydrase 1 by CO2 hydration reaction | 2009 | Bioorganic & medicinal chemistry letters, Feb-15, Volume: 19, Issue:4
| Carbonic anhydrase inhibitors: the membrane-associated isoform XV is highly inhibited by inorganic anions. |
AID367654 | Inhibition of human carbonic anhydrase 2 measured by CO2 hydration reaction assay | 2009 | Bioorganic & medicinal chemistry letters, Feb-01, Volume: 19, Issue:3
| Carbonic anhydrase inhibitors: inhibition studies of a coral secretory isoform with inorganic anions. |
AID387189 | Inhibition of Methanobacterium thermoautotrophicum Cab at 20 degC by CO2 hydration method | 2008 | Bioorganic & medicinal chemistry letters, Sep-15, Volume: 18, Issue:18
| Carbonic anhydrase inhibitors: inhibition of the beta-class enzymes from the fungal pathogens Candida albicans and Cryptococcus neoformans with simple anions. |
AID50355 | Inhibitory activity against human cloned carbonic anhydrase I (hCA I) | 2003 | Bioorganic & medicinal chemistry letters, Mar-10, Volume: 13, Issue:5
| Carbonic anhydrase inhibitors: SAR and X-ray crystallographic study for the interaction of sugar sulfamates/sulfamides with isozymes I, II and IV. |
AID730368 | Inhibition of Helicobacter pylori beta-carbonic anhydrase preincubated for 15 mins by stopped flow CO2 hydration assay | 2013 | Bioorganic & medicinal chemistry letters, Mar-15, Volume: 23, Issue:6
| Kinetic and anion inhibition studies of a β-carbonic anhydrase (FbiCA 1) from the C4 plant Flaveria bidentis. |
AID310903 | Inhibition of human recombinant full length CA14 | 2007 | Bioorganic & medicinal chemistry letters, Mar-15, Volume: 17, Issue:6
| Carbonic anhydrase inhibitors. Inhibition of transmembrane isozymes XII (cancer-associated) and XIV with anions. |
AID552129 | Inhibition of human recombinant CA6 by stopped-flow CO2 hydration assay | 2011 | Bioorganic & medicinal chemistry letters, Jan-15, Volume: 21, Issue:2
| Carbonic anhydrase inhibitors. Inhibition studies with anions and sulfonamides of a new cytosolic enzyme from the scleractinian coral Stylophora pistillata. |
AID598728 | Inhibition of recombinant human carbonic anhydrase 2 after 15 mins by stopped flow CO2 hydration assay at pH 8.3 | 2011 | Bioorganic & medicinal chemistry letters, Jun-15, Volume: 21, Issue:12
| Inhibition studies with anions and small molecules of two novel β-carbonic anhydrases from the bacterial pathogen Salmonella enterica serovar Typhimurium. |
AID1262263 | Inhibition of human CA1 incubated for 15 mins prior to testing by stopped flow CO2 hydrase assay | 2015 | Bioorganic & medicinal chemistry letters, Dec-01, Volume: 25, Issue:23
| Anion and sulfonamide inhibition studies of an α-carbonic anhydrase from the Antarctic hemoglobinless fish Chionodraco hamatus. |
AID758948 | Inhibition of Porphyromonas gingivalis recombinant CA by CO2 hydration assay | 2013 | Bioorganic & medicinal chemistry letters, Jul-15, Volume: 23, Issue:14
| A highly catalytically active γ-carbonic anhydrase from the pathogenic anaerobe Porphyromonas gingivalis and its inhibition profile with anions and small molecules. |
AID238411 | Inhibitory activity against human Carbonic anhydrase V | 2005 | Bioorganic & medicinal chemistry letters, Feb-01, Volume: 15, Issue:3
| Carbonic anhydrase inhibitors. Inhibition of isozymes I, II, IV, V, and IX with anions isosteric and isoelectronic with sulfate, nitrate, and carbonate. |
AID724722 | Inhibition of human recombinant wild type CA1 by stopped-flow CO2 hydration method | 2013 | Bioorganic & medicinal chemistry letters, Jan-01, Volume: 23, Issue:1
| Restoring catalytic activity to the human carbonic anhydrase (CA) related proteins VIII, X and XI affords isoforms with high catalytic efficiency and susceptibility to anion inhibition. |
AID1262267 | Inhibition of Chionodraco hamatus alphaCA incubated for 15 mins prior to testing by stopped flow CO2 hydrase assay | 2015 | Bioorganic & medicinal chemistry letters, Dec-01, Volume: 25, Issue:23
| Anion and sulfonamide inhibition studies of an α-carbonic anhydrase from the Antarctic hemoglobinless fish Chionodraco hamatus. |
AID484161 | Inhibition of full length human carbonic anhydrase 7 preincubated for 15 mins by CO2 hydration stopped-flow assay | 2010 | Bioorganic & medicinal chemistry letters, Jun-15, Volume: 20, Issue:12
| Carbonic anhydrase inhibitors: crystallographic and solution binding studies for the interaction of a boron-containing aromatic sulfamide with mammalian isoforms I-XV. |
AID238441 | Inhibitory activity against human Carbonic anhydrase IV | 2005 | Bioorganic & medicinal chemistry letters, Feb-01, Volume: 15, Issue:3
| Carbonic anhydrase inhibitors. Inhibition of isozymes I, II, IV, V, and IX with anions isosteric and isoelectronic with sulfate, nitrate, and carbonate. |
AID392571 | Inhibition of mouse recombinant carbonic anhydrase 15 expressed in COS7 cells by CO2 hydration reaction | 2009 | Bioorganic & medicinal chemistry letters, Feb-15, Volume: 19, Issue:4
| Carbonic anhydrase inhibitors: the membrane-associated isoform XV is highly inhibited by inorganic anions. |
AID238853 | Inhibitory activity against mouse carbonic anhydrase XIII expressed in Escherichia coli TOP 10 | 2004 | Bioorganic & medicinal chemistry letters, Nov-01, Volume: 14, Issue:21
| Carbonic anhydrase inhibitors. Inhibition of the newly isolated murine isozyme XIII with anions. |
AID598732 | Inhibition of Salmonella Typhimurium carbonic anhydrase 2 after 15 mins by stopped flow CO2 hydration assay at pH 8.3 | 2011 | Bioorganic & medicinal chemistry letters, Jun-15, Volume: 21, Issue:12
| Inhibition studies with anions and small molecules of two novel β-carbonic anhydrases from the bacterial pathogen Salmonella enterica serovar Typhimurium. |
AID1161950 | Inhibition of human carbonic anhydrase 2 preincubated for 15 mins by stopped flow CO2 hydration method | 2014 | Bioorganic & medicinal chemistry letters, Sep-15, Volume: 24, Issue:18
| Anion inhibition study of the β-class carbonic anhydrase (PgiCAb) from the oral pathogen Porphyromonas gingivalis. |
AID1070021 | Inhibition of Legionella pneumophila carbonic anhydrase 2 preincubated for 15 mins by stopped-flow CO2 hydrase assay | 2014 | Bioorganic & medicinal chemistry letters, Feb-15, Volume: 24, Issue:4
| Anion inhibition studies of two new β-carbonic anhydrases from the bacterial pathogen Legionella pneumophila. |
AID238226 | Inhibitory constant against human tumor Carbonic anhydrases IX or XII | 2005 | Bioorganic & medicinal chemistry letters, May-02, Volume: 15, Issue:9
| Carbonic anhydrase inhibitors: synthesis and inhibition of cytosolic/tumor-associated carbonic anhydrase isozymes I, II, IX, and XII with N-hydroxysulfamides--a new zinc-binding function in the design of inhibitors. |
AID310901 | Inhibition of human recombinant catalytic domain CA9 | 2007 | Bioorganic & medicinal chemistry letters, Mar-15, Volume: 17, Issue:6
| Carbonic anhydrase inhibitors. Inhibition of transmembrane isozymes XII (cancer-associated) and XIV with anions. |
AID238607 | Inhibitory constant against Zn-Cam (Methanosarcina thermophila) | 2004 | Bioorganic & medicinal chemistry letters, Sep-06, Volume: 14, Issue:17
| Carbonic anhydrase inhibitors. Inhibition of the beta-class enzyme from the methanoarchaeon Methanobacterium thermoautotrophicum (Cab) with anions. |
AID763568 | Inhibition of human carbonic anhydrase-2 at 20 degC preincubated for 15 mins by stopped-flow CO2 hydrase assay | 2013 | Bioorganic & medicinal chemistry, Aug-01, Volume: 21, Issue:15
| Anion inhibition studies of the α-carbonic anhydrase from the protozoan pathogen Trypanosoma cruzi, the causative agent of Chagas disease. |
AID239224 | Inhibitory activity against human carbonic anhydrase IX at 0.09 uM; not tested | 2004 | Bioorganic & medicinal chemistry letters, Dec-20, Volume: 14, Issue:24
| Carbonic anhydrase inhibitors. Inhibition of the prokariotic beta and gamma-class enzymes from Archaea with sulfonamides. |
AID587132 | Inhibition of Leptonychotes weddellii alpha-carbonic anhydrase after 15 mins by CO2 hydrase assay at pH 7.5 | 2011 | Bioorganic & medicinal chemistry, Mar-15, Volume: 19, Issue:6
| Purification and inhibition studies with anions and sulfonamides of an α-carbonic anhydrase from the Antarctic seal Leptonychotes weddellii. |
AID1430526 | Inhibition of recombinant human carbonic anhydrase 2 assessed as inhibition of CO2 hydration incubated for 15 mins prior to testing by stopped flow CO2 hydration method | | | |
AID724720 | Inhibition of human recombinant CA8 mutant after 15 mins by stopped-flow CO2 hydration method | 2013 | Bioorganic & medicinal chemistry letters, Jan-01, Volume: 23, Issue:1
| Restoring catalytic activity to the human carbonic anhydrase (CA) related proteins VIII, X and XI affords isoforms with high catalytic efficiency and susceptibility to anion inhibition. |
AID411400 | Inhibition of Saccharomyces cerevisiae carbonic anhydrase overexpressed in Escherichia coli BL21 (DE3) by CO2 hydration stopped-flow assay | 2008 | Bioorganic & medicinal chemistry letters, Dec-15, Volume: 18, Issue:24
| Carbonic anhydrase inhibitors. Inhibition of the beta-class enzyme from the yeast Saccharomyces cerevisiae with anions. |
AID730372 | Inhibition of Flaveria bidentis beta-carbonic anhydrase-1 preincubated for 15 mins by stopped flow CO2 hydration assay | 2013 | Bioorganic & medicinal chemistry letters, Mar-15, Volume: 23, Issue:6
| Kinetic and anion inhibition studies of a β-carbonic anhydrase (FbiCA 1) from the C4 plant Flaveria bidentis. |
AID1235241 | Inhibition of human CA2 after 15 mins by stopped-flow/Co2 hydration assay | 2015 | Bioorganic & medicinal chemistry, Aug-01, Volume: 23, Issue:15
| Cloning, characterization and anion inhibition studies of a new γ-carbonic anhydrase from the Antarctic bacterium Pseudoalteromonas haloplanktis. |
AID598726 | Inhibition of recombinant human carbonic anhydrase 1 after 15 mins by stopped flow CO2 hydration assay at pH 8.3 | 2011 | Bioorganic & medicinal chemistry letters, Jun-15, Volume: 21, Issue:12
| Inhibition studies with anions and small molecules of two novel β-carbonic anhydrases from the bacterial pathogen Salmonella enterica serovar Typhimurium. |
AID238317 | Inhibitory constant against carbonic anhydrase I | 2004 | Bioorganic & medicinal chemistry letters, Sep-06, Volume: 14, Issue:17
| Carbonic anhydrase inhibitors. Inhibition of the beta-class enzyme from the methanoarchaeon Methanobacterium thermoautotrophicum (Cab) with anions. |
AID1070022 | Inhibition of Legionella pneumophila carbonic anhydrase 1 preincubated for 15 mins by stopped-flow CO2 hydrase assay | 2014 | Bioorganic & medicinal chemistry letters, Feb-15, Volume: 24, Issue:4
| Anion inhibition studies of two new β-carbonic anhydrases from the bacterial pathogen Legionella pneumophila. |
AID387187 | Inhibition of human carbonic anhydrase 1 at 20 degC by CO2 hydration method | 2008 | Bioorganic & medicinal chemistry letters, Sep-15, Volume: 18, Issue:18
| Carbonic anhydrase inhibitors: inhibition of the beta-class enzymes from the fungal pathogens Candida albicans and Cryptococcus neoformans with simple anions. |
AID238578 | Inhibition constant against human carbonic anhydrase isozyme hCA I | 2004 | Bioorganic & medicinal chemistry letters, Dec-06, Volume: 14, Issue:23
| Carbonic anhydrase inhibitors: inhibition of the membrane-bound human isozyme IV with anions. |
AID238440 | Inhibitory activity against human Carbonic anhydrase II | 2005 | Bioorganic & medicinal chemistry letters, Feb-01, Volume: 15, Issue:3
| Carbonic anhydrase inhibitors. Inhibition of isozymes I, II, IV, V, and IX with anions isosteric and isoelectronic with sulfate, nitrate, and carbonate. |
AID1336558 | Inhibition of Methanosarcina thermophila recombinant carbonic anhydrase gamma assessed as inhibition of CO2 hydration preincubated for 15 mins by Lineweaver-burk plot method | | | |
AID238958 | Inhibitory constant against methanoarchaeon Methanobacterium thermoautotrophicum (Cab) | 2004 | Bioorganic & medicinal chemistry letters, Sep-06, Volume: 14, Issue:17
| Carbonic anhydrase inhibitors. Inhibition of the beta-class enzyme from the methanoarchaeon Methanobacterium thermoautotrophicum (Cab) with anions. |
AID310900 | Inhibition of human recombinant CA2 | 2007 | Bioorganic & medicinal chemistry letters, Mar-15, Volume: 17, Issue:6
| Carbonic anhydrase inhibitors. Inhibition of transmembrane isozymes XII (cancer-associated) and XIV with anions. |
AID758950 | Inhibition of Methanosarcina thermophila recombinant gamma-CA by CO2 hydration assay | 2013 | Bioorganic & medicinal chemistry letters, Jul-15, Volume: 23, Issue:14
| A highly catalytically active γ-carbonic anhydrase from the pathogenic anaerobe Porphyromonas gingivalis and its inhibition profile with anions and small molecules. |
AID1058395 | Inhibition of human cytosolic carbonic anhydrase 2 preincubated for 15 mins by stopped flow CO2 hydration assay | 2013 | Bioorganic & medicinal chemistry letters, Dec-15, Volume: 23, Issue:24
| Anion inhibition studies of a β-carbonic anhydrase from Clostridium perfringens. |
AID1161931 | Inhibition of human carbonic anhydrase 2 preincubated for 15 mins by stopped flow CO2 hydration method | 2014 | Bioorganic & medicinal chemistry letters, Sep-15, Volume: 24, Issue:18
| Discovery of a new family of carbonic anhydrases in the malaria pathogen Plasmodium falciparum--the η-carbonic anhydrases. |
AID1237475 | Inhibition of human carbonic anhydrase-2 by CO2 hydration reaction based colorimetric stopped-flow method | 2015 | Bioorganic & medicinal chemistry, Aug-01, Volume: 23, Issue:15
| Structure and inhibition studies of a type II beta-carbonic anhydrase psCA3 from Pseudomonas aeruginosa. |
AID1237477 | Inhibition of Pseudomonas aeruginosa PAO1 type-2 beta-carbonic anhydrase psCA3 expressed in Escherichia coli Tuner BL21 (DE3) cells pre-incubated for 15 mins at pH 8.3 and 293K by CO2 hydration reaction based colorimetric stopped-flow method | 2015 | Bioorganic & medicinal chemistry, Aug-01, Volume: 23, Issue:15
| Structure and inhibition studies of a type II beta-carbonic anhydrase psCA3 from Pseudomonas aeruginosa. |
AID1070020 | Inhibition of human carbonic anhydrase 2 by stopped-flow CO2 hydrase assay | 2014 | Bioorganic & medicinal chemistry letters, Feb-15, Volume: 24, Issue:4
| Anion inhibition studies of two new β-carbonic anhydrases from the bacterial pathogen Legionella pneumophila. |
AID484165 | Inhibition of full length human carbonic anhydrase 14 preincubated for 15 mins by CO2 hydration stopped-flow assay | 2010 | Bioorganic & medicinal chemistry letters, Jun-15, Volume: 20, Issue:12
| Carbonic anhydrase inhibitors: crystallographic and solution binding studies for the interaction of a boron-containing aromatic sulfamide with mammalian isoforms I-XV. |
AID1262264 | Inhibition of human CA2 incubated for 15 mins prior to testing by stopped flow CO2 hydrase assay | 2015 | Bioorganic & medicinal chemistry letters, Dec-01, Volume: 25, Issue:23
| Anion and sulfonamide inhibition studies of an α-carbonic anhydrase from the Antarctic hemoglobinless fish Chionodraco hamatus. |
AID1235243 | Inhibition of Porphyromonas gingivalis CA after 15 mins by stopped-flow/Co2 hydration assay | 2015 | Bioorganic & medicinal chemistry, Aug-01, Volume: 23, Issue:15
| Cloning, characterization and anion inhibition studies of a new γ-carbonic anhydrase from the Antarctic bacterium Pseudoalteromonas haloplanktis. |
AID310899 | Inhibition of human recombinant carbonic anhydrase 1 | 2007 | Bioorganic & medicinal chemistry letters, Mar-15, Volume: 17, Issue:6
| Carbonic anhydrase inhibitors. Inhibition of transmembrane isozymes XII (cancer-associated) and XIV with anions. |
AID1278740 | Inhibition of human carbonic anhydrase 2 preincubated for 15 mins by stopped-flow CO2 hydration assay | 2016 | Bioorganic & medicinal chemistry letters, Mar-01, Volume: 26, Issue:5
| Anion inhibition studies of the β-carbonic anhydrase from the pathogenic bacterium Vibrio cholerae. |
AID367656 | Inhibition of Stylophora pistillata carbonic anhydrase measured by CO2 hydration reaction assay | 2009 | Bioorganic & medicinal chemistry letters, Feb-01, Volume: 19, Issue:3
| Carbonic anhydrase inhibitors: inhibition studies of a coral secretory isoform with inorganic anions. |
AID238442 | Inhibitory activity against human Carbonic anhydrase IX | 2005 | Bioorganic & medicinal chemistry letters, Feb-01, Volume: 15, Issue:3
| Carbonic anhydrase inhibitors. Inhibition of isozymes I, II, IV, V, and IX with anions isosteric and isoelectronic with sulfate, nitrate, and carbonate. |
AID238606 | Inhibition constant against human carbonic anhydrase isozyme hCA IX | 2004 | Bioorganic & medicinal chemistry letters, Dec-06, Volume: 14, Issue:23
| Carbonic anhydrase inhibitors: inhibition of the membrane-bound human isozyme IV with anions. |
AID552128 | Inhibition of human recombinant CA2 by stopped-flow CO2 hydration assay | 2011 | Bioorganic & medicinal chemistry letters, Jan-15, Volume: 21, Issue:2
| Carbonic anhydrase inhibitors. Inhibition studies with anions and sulfonamides of a new cytosolic enzyme from the scleractinian coral Stylophora pistillata. |
AID295048 | Inhibition of human recombinant carbonic anhydrase 9 catalytic domain by CO2 hydrase method | 2007 | Bioorganic & medicinal chemistry letters, May-15, Volume: 17, Issue:10
| Carbonic anhydrase inhibitors: the X-ray crystal structure of the adduct of N-hydroxysulfamide with isozyme II explains why this new zinc binding function is effective in the design of potent inhibitors. |
AID1306523 | Inhibition of human carbonic anhydrase 1 preincubated for 15 mins by stopped-flow CO2 hydrase assay | 2016 | Bioorganic & medicinal chemistry, 08-15, Volume: 24, Issue:16
| Anion inhibition profiles of α-, β- and γ-carbonic anhydrases from the pathogenic bacterium Vibrio cholerae. |
AID1237485 | Induction of growth defect in Pseudomonas aeruginosa PAO1 up to 1 mM | 2015 | Bioorganic & medicinal chemistry, Aug-01, Volume: 23, Issue:15
| Structure and inhibition studies of a type II beta-carbonic anhydrase psCA3 from Pseudomonas aeruginosa. |
[information is prepared from bioassay data collected from National Library of Medicine (NLM), extracted Dec-2023] |