Page last updated: 2024-08-05 15:22:01

gout suppressant

A drug that increases uric acid excretion by the kidney (uricosuric drug), decreases uric acid production (antihyperuricemic), or alleviates the pain and inflammation of acute attacks of gout.

ChEBI ID: 35845

Members (6)

MemberDefinitionClass
allopurinolA bicyclic structure comprising a pyrazole ring fused to a hydroxy-substituted pyrimidine ring.allopurinol
colchicineA colchicine that has (S)-configuration. It is a secondary metabolite, has anti-inflammatory properties and is used to treat gout, crystal-induced joint inflammation, familial Mediterranean fever, and many other conditions.(S)-colchicine
indomethacinA member of the class of indole-3-acetic acids that is indole-3-acetic acid in which the indole ring is substituted at positions 1, 2 and 5 by p-chlorobenzoyl, methyl, and methoxy groups, respectively. A non-steroidal anti-inflammatory drug, it is used in the treatment of musculoskeletal and joint disorders including osteoarthritis, rheumatoid arthritis, gout, bursitis and tendinitis.indometacin
naproxenA methoxynaphthalene that is 2-methoxynaphthalene substituted by a carboxy ethyl group at position 6. Naproxen is a non-steroidal anti-inflammatory drug commonly used for the reduction of pain, fever, inflammation and stiffness caused by conditions such as osteoarthritis, kidney stones, rheumatoid arthritis, psoriatic arthritis, gout, ankylosing spondylitis, menstrual cramps, tendinitis, bursitis, and for the treatment of primary dysmenorrhea. It works by inhibiting both the COX-1 and COX-2 enzymes.naproxen
oxyphenbutazoneA metabolite of phenylbutazone obtained by hydroxylation at position 4 of one of the phenyl rings. Commonly used (as its hydrate) to treat pain, swelling and stiffness associated with arthritis and gout, it was withdrawn from the market 1984 following association with blood dyscrasis and Stevens-Johnson syndrome.oxyphenbutazone
sarsasapogenin, (3beta,5alpha,25r)-isomerA widely used steroidal sapogenin isolated from several plant species and used for synthesizing steroid drugs.tigogenin

Research

Studies (61,267)

TimeframeStudies, Drugs with This Role(%)All Drugs %
pre-199025,675 (41.91)18.7374
1990's13,628 (22.24)18.2507
2000's10,007 (16.33)29.6817
2010's8,985 (14.67)24.3611
2020's2,972 (4.85)2.80

Study Types

Publication TypeStudies, Drugs with this Role (%)All Drugs (%)
Trials4,190 (6.36%)5.53%
Reviews3,601 (5.47%)6.00%
Case Studies4,180 (6.34%)4.05%
Observational92 (0.14%)0.25%
Other53,826 (81.69%)84.16%

Protein Targets (270)

Potency Measurements

ProteinTaxonomyMeasurementAverage (mM)Bioassay(s)Drugs
15-hydroxyprostaglandin dehydrogenase [NAD(+)] isoform 1Homo sapiens (human)Potency39.810711
67.9K proteinVaccinia virusPotency2.025123
activating transcription factor 6Homo sapiens (human)Potency0.293913
aldehyde dehydrogenase 1 family, member A1Homo sapiens (human)Potency39.810711
AR proteinHomo sapiens (human)Potency10.65231042
aryl hydrocarbon receptorHomo sapiens (human)Potency17.821124
ATAD5 protein, partialHomo sapiens (human)Potency14.923134
Ataxin-2Homo sapiens (human)Potency0.122813
ATP-dependent phosphofructokinaseTrypanosoma brucei brucei TREU927Potency0.037911
ATPase family AAA domain-containing protein 5Homo sapiens (human)Potency0.135926
atrial natriuretic peptide receptor 2 precursorHomo sapiens (human)Potency1.849311
Bloom syndrome protein isoform 1Homo sapiens (human)Potency0.398122
bromodomain adjacent to zinc finger domain 2BHomo sapiens (human)Potency100.000011
caspase-1 isoform alpha precursorHomo sapiens (human)Potency39.810711
caspase-3Cricetulus griseus (Chinese hamster)Potency3.757811
Caspase-7Cricetulus griseus (Chinese hamster)Potency3.757811
Cellular tumor antigen p53Homo sapiens (human)Potency12.133835
cellular tumor antigen p53 isoform aHomo sapiens (human)Potency16.603812
Chain A, 2-oxoglutarate OxygenaseHomo sapiens (human)Potency10.000011
Chain A, Beta-lactamaseEscherichia coli K-12Potency24.840112
Chain A, CruzipainTrypanosoma cruziPotency39.810712
Chain A, Ferritin light chainEquus caballus (horse)Potency35.481311
Chain A, JmjC domain-containing histone demethylation protein 3AHomo sapiens (human)Potency56.234111
Chain A, MAJOR APURINIC/APYRIMIDINIC ENDONUCLEASEHomo sapiens (human)Potency23.953516
Chain A, Putative fructose-1,6-bisphosphate aldolaseGiardia intestinalisPotency25.157413
chromobox protein homolog 1Homo sapiens (human)Potency19.907222
CREB-binding proteinHomo sapiens (human)Potency5.011922
cytochrome P450 2C19 precursorHomo sapiens (human)Potency12.589311
cytochrome P450 2C9 precursorHomo sapiens (human)Potency20.975213
cytochrome P450 2C9, partialHomo sapiens (human)Potency9.836512
cytochrome P450 2D6Homo sapiens (human)Potency34.671311
cytochrome P450 2D6 isoform 1Homo sapiens (human)Potency8.321612
cytochrome P450 3A4 isoform 1Homo sapiens (human)Potency17.067424
cytochrome P450 family 3 subfamily A polypeptide 4Homo sapiens (human)Potency14.971124
cytochrome P450, family 19, subfamily A, polypeptide 1, isoform CRA_aHomo sapiens (human)Potency32.351312
DNA dC->dU-editing enzyme APOBEC-3G isoform 1Homo sapiens (human)Potency3.162311
DNA polymerase iota isoform a (long)Homo sapiens (human)Potency40.439212
DNA polymerase kappa isoform 1Homo sapiens (human)Potency7.519311
endonuclease IVEscherichia coliPotency2.511911
estrogen nuclear receptor alphaHomo sapiens (human)Potency9.75191140
estrogen receptor 2 (ER beta)Homo sapiens (human)Potency32.786838
estrogen-related nuclear receptor alphaHomo sapiens (human)Potency29.9688736
euchromatic histone-lysine N-methyltransferase 2Homo sapiens (human)Potency3.988815
EWS/FLI fusion proteinHomo sapiens (human)Potency15.475433
farnesoid X nuclear receptorHomo sapiens (human)Potency10.5422411
flap endonuclease 1Homo sapiens (human)Potency6.701611
Fumarate hydrataseHomo sapiens (human)Potency1.992412
GVesicular stomatitis virusPotency9.836512
GABA theta subunitRattus norvegicus (Norway rat)Potency17.067412
Gamma-aminobutyric acid receptor subunit alpha-1Rattus norvegicus (Norway rat)Potency17.067412
Gamma-aminobutyric acid receptor subunit alpha-2Rattus norvegicus (Norway rat)Potency17.067412
Gamma-aminobutyric acid receptor subunit alpha-3Rattus norvegicus (Norway rat)Potency17.067412
Gamma-aminobutyric acid receptor subunit alpha-4Rattus norvegicus (Norway rat)Potency17.067412
Gamma-aminobutyric acid receptor subunit alpha-5Rattus norvegicus (Norway rat)Potency17.067412
Gamma-aminobutyric acid receptor subunit alpha-6Rattus norvegicus (Norway rat)Potency17.067412
Gamma-aminobutyric acid receptor subunit beta-1Rattus norvegicus (Norway rat)Potency17.067412
Gamma-aminobutyric acid receptor subunit beta-2Rattus norvegicus (Norway rat)Potency17.067412
Gamma-aminobutyric acid receptor subunit beta-3Rattus norvegicus (Norway rat)Potency17.067412
Gamma-aminobutyric acid receptor subunit deltaRattus norvegicus (Norway rat)Potency17.067412
Gamma-aminobutyric acid receptor subunit epsilonRattus norvegicus (Norway rat)Potency17.067412
Gamma-aminobutyric acid receptor subunit gamma-1Rattus norvegicus (Norway rat)Potency17.067412
Gamma-aminobutyric acid receptor subunit gamma-2Rattus norvegicus (Norway rat)Potency17.067412
Gamma-aminobutyric acid receptor subunit gamma-3Rattus norvegicus (Norway rat)Potency17.067412
Gamma-aminobutyric acid receptor subunit piRattus norvegicus (Norway rat)Potency17.067412
gemininHomo sapiens (human)Potency1.317549
GLI family zinc finger 3Homo sapiens (human)Potency1.717228
glp-1 receptor, partialHomo sapiens (human)Potency12.589311
glucocerebrosidaseHomo sapiens (human)Potency20.220812
glucocorticoid receptor [Homo sapiens]Homo sapiens (human)Potency7.7478411
Glutamate receptor 2Rattus norvegicus (Norway rat)Potency21.243016
Guanine nucleotide-binding protein GHomo sapiens (human)Potency10.266312
heat shock 70kDa protein 5 (glucose-regulated protein, 78kDa)Homo sapiens (human)Potency14.125411
heat shock protein beta-1Homo sapiens (human)Potency16.240023
Histamine H2 receptorCavia porcellus (domestic guinea pig)Potency20.975219
histone deacetylase 9 isoform 3Homo sapiens (human)Potency25.156622
HLA class I histocompatibility antigen, B alpha chain Homo sapiens (human)Potency9.836512
hypothetical protein, conservedTrypanosoma bruceiPotency14.125411
hypoxia-inducible factor 1 alpha subunitHomo sapiens (human)Potency42.735112
hypoxia-inducible factor 1, alpha subunit (basic helix-loop-helix transcription factor)Homo sapiens (human)Potency7.539726
IDH1Homo sapiens (human)Potency9.615213
Inositol hexakisphosphate kinase 1Homo sapiens (human)Potency9.836514
Interferon betaHomo sapiens (human)Potency3.962625
interleukin 8Homo sapiens (human)Potency35.475614
lamin isoform A-delta10Homo sapiens (human)Potency3.547125
lethal factor (plasmid)Bacillus anthracis str. A2012Potency10.591013
LuciferasePhotinus pyralis (common eastern firefly)Potency40.601123
M-phase phosphoprotein 8Homo sapiens (human)Potency0.794311
Microtubule-associated protein tauHomo sapiens (human)Potency17.216823
muscarinic acetylcholine receptor M1Rattus norvegicus (Norway rat)Potency0.891311
muscleblind-like protein 1 isoform 1Homo sapiens (human)Potency14.219112
neuropeptide S receptor isoform AHomo sapiens (human)Potency2.048412
Nrf2Homo sapiens (human)Potency8.500322
nuclear factor erythroid 2-related factor 2 isoform 1Homo sapiens (human)Potency17.5889314
nuclear factor erythroid 2-related factor 2 isoform 2Homo sapiens (human)Potency12.993512
nuclear factor of kappa light polypeptide gene enhancer in B-cells 1 (p105), isoform CRA_aHomo sapiens (human)Potency35.627813
Nuclear receptor ROR-gammaHomo sapiens (human)Potency3.297613
nuclear receptor ROR-gamma isoform 1Mus musculus (house mouse)Potency7.559823
nuclear receptor subfamily 1, group I, member 2Rattus norvegicus (Norway rat)Potency17.782811
nuclear receptor subfamily 1, group I, member 3Homo sapiens (human)Potency6.683239
parathyroid hormone/parathyroid hormone-related peptide receptor precursorHomo sapiens (human)Potency17.782811
ParkinHomo sapiens (human)Potency20.596211
peripheral myelin protein 22Rattus norvegicus (Norway rat)Potency0.095522
peripheral myelin protein 22 isoform 1Homo sapiens (human)Potency84.921411
peroxisome proliferator activated receptor gammaHomo sapiens (human)Potency6.5440514
peroxisome proliferator-activated receptor deltaHomo sapiens (human)Potency10.9345516
plasminogen precursorMus musculus (house mouse)Potency0.891311
polyproteinZika virusPotency1.992412
PPM1D proteinHomo sapiens (human)Potency0.046612
pregnane X nuclear receptorHomo sapiens (human)Potency2.306437
pregnane X receptorRattus norvegicus (Norway rat)Potency6.339613
progesterone receptorHomo sapiens (human)Potency22.712325
RAR-related orphan receptor gammaMus musculus (house mouse)Potency16.2807214
ras-related protein Rab-9AHomo sapiens (human)Potency119.218715
retinoic acid nuclear receptor alpha variant 1Homo sapiens (human)Potency1.470239
retinoid X nuclear receptor alphaHomo sapiens (human)Potency7.6510419
serine/threonine-protein kinase mTOR isoform 1Homo sapiens (human)Potency4.645111
serine/threonine-protein kinase PLK1Homo sapiens (human)Potency23.778111
SMAD family member 2Homo sapiens (human)Potency15.553728
SMAD family member 3Homo sapiens (human)Potency15.553728
Smad3Homo sapiens (human)Potency3.372712
Spike glycoproteinSevere acute respiratory syndrome-related coronavirusPotency19.731212
survival motor neuron protein isoform dHomo sapiens (human)Potency1.000011
TAR DNA-binding protein 43Homo sapiens (human)Potency18.240612
TDP1 proteinHomo sapiens (human)Potency6.5308215
thioredoxin glutathione reductaseSchistosoma mansoniPotency10.000011
thioredoxin reductaseRattus norvegicus (Norway rat)Potency9.806435
ThrombopoietinHomo sapiens (human)Potency0.501222
thyroid hormone receptor beta isoform 2Rattus norvegicus (Norway rat)Potency6.7740211
thyroid hormone receptor beta isoform aHomo sapiens (human)Potency15.688514
thyroid stimulating hormone receptorHomo sapiens (human)Potency7.016629
transcriptional regulator ERG isoform 3Homo sapiens (human)Potency0.794311
urokinase plasminogen activator surface receptor precursorMus musculus (house mouse)Potency0.891311
urokinase-type plasminogen activator precursorMus musculus (house mouse)Potency0.891311
USP1 protein, partialHomo sapiens (human)Potency36.512323
v-jun sarcoma virus 17 oncogene homolog (avian)Homo sapiens (human)Potency2.380228
vitamin D (1,25- dihydroxyvitamin D3) receptorHomo sapiens (human)Potency8.9546514
vitamin D3 receptor isoform VDRAHomo sapiens (human)Potency22.285257
Voltage-dependent calcium channel gamma-2 subunitMus musculus (house mouse)Potency21.243016

Inhibition Measurements

ProteinTaxonomyMeasurementAverage (mM)Bioassay(s)Drugs
3',5'-cyclic-AMP phosphodiesterase Sus scrofa (pig)IC501,000.000011
Adenosine receptor A1Rattus norvegicus (Norway rat)IC50589.500012
Adenosine receptor A2aRattus norvegicus (Norway rat)IC50589.500012
AlbuminHomo sapiens (human)Ki15,135,600,000.000011
Aldo-keto reductase family 1 member B1Bos taurus (cattle)IC505.000012
Aldo-keto reductase family 1 member B1Homo sapiens (human)IC506.000011
Aldo-keto reductase family 1 member C1Homo sapiens (human)IC50106.500034
Aldo-keto reductase family 1 member C2 Homo sapiens (human)IC5043.294367
Aldo-keto reductase family 1 member C3Homo sapiens (human)IC502.5900910
Aldo-keto reductase family 1 member C3Homo sapiens (human)Ki1.185022
Aldo-keto reductase family 1 member C4Homo sapiens (human)IC5084.666723
ATP-binding cassette sub-family C member 3Homo sapiens (human)IC50116.250014
ATP-dependent translocase ABCB1Homo sapiens (human)IC5042.000045
ATP-dependent translocase ABCB1Mus musculus (house mouse)IC5050.000044
Beta lactamase (plasmid)Pseudomonas aeruginosaIC5043.545011
Bifunctional epoxide hydrolase 2Homo sapiens (human)IC501.000011
Bile salt export pumpHomo sapiens (human)IC50200.0927411
C-X-C chemokine receptor type 3Homo sapiens (human)IC500.050011
Canalicular multispecific organic anion transporter 1Homo sapiens (human)IC50158.500024
caspase recruitment domain family, member 15Homo sapiens (human)IC506.633011
Caspase-1Homo sapiens (human)IC5028.666716
Caspase-3Homo sapiens (human)IC5028.666716
Caspase-4Homo sapiens (human)IC5028.666716
Caspase-5Homo sapiens (human)IC5028.666716
Caspase-9Homo sapiens (human)IC5028.666716
Chain A, membrane-associated prostaglandin E synthase-2Macaca fascicularis (crab-eating macaque)IC501,000.000011
Cytochrome c oxidase subunit 2Homo sapiens (human)IC500.340022
Cytochrome P450 2C9 Homo sapiens (human)IC5050.000011
Cytochrome P450 2J2Homo sapiens (human)IC5050.000011
Cytochrome P450 3A4Homo sapiens (human)IC5050.000011
Cytosolic phospholipase A2 gammaHomo sapiens (human)IC50100.000011
Dehydrogenase/reductase SDR family member 9Homo sapiens (human)IC5014.000011
Dihydrofolate reductaseHomo sapiens (human)Ki7,000.000011
Epidermal growth factor receptorHomo sapiens (human)IC5010.000011
glucose-6-phosphate 1-dehydrogenase isoform bHomo sapiens (human)IC5080.000011
glucose-6-phosphate dehydrogenase-6-phosphogluconolactonasePlasmodium bergheiIC5063.125034
Histamine H3 receptorCavia porcellus (domestic guinea pig)IC508.690011
Hormone-sensitive lipaseRattus norvegicus (Norway rat)IC501.200011
Indoleamine 2,3-dioxygenase 1Mus musculus (house mouse)IC500.082012
Interleukin-8Homo sapiens (human)IC500.050011
Lactoylglutathione lyaseHomo sapiens (human)Ki22.166733
Multidrug and toxin extrusion protein 1Homo sapiens (human)IC50500.000011
Multidrug resistance-associated protein 1 Homo sapiens (human)IC5012.300022
Multidrug resistance-associated protein 4Homo sapiens (human)IC50101.200014
Neuronal acetylcholine receptor subunit alpha-4Rattus norvegicus (Norway rat)IC500.004011
Neuronal acetylcholine receptor subunit beta-2Rattus norvegicus (Norway rat)IC500.004011
Nicotinate phosphoribosyltransferaseHomo sapiens (human)Ki0.000212
Nitric oxide synthase, inducibleMus musculus (house mouse)IC5024.350055
Nuclear receptor ROR-gammaMus musculus (house mouse)IC5011.100011
nuclear receptor subfamily 0 group B member 1Homo sapiens (human)IC5067.568011
P2Y purinoceptor 12Rattus norvegicus (Norway rat)IC500.960011
Phospholipase A2, major isoenzymeSus scrofa (pig)IC501,000.000011
Polyphenol oxidase 2Agaricus bisporusIC501,000.000011
Polyunsaturated fatty acid 5-lipoxygenaseRattus norvegicus (Norway rat)IC50645.666756
Potassium voltage-gated channel subfamily H member 2Homo sapiens (human)IC50301.995011
Procathepsin LHomo sapiens (human)IC5011.800011
Prostaglandin D2 receptor Mus musculus (house mouse)IC5010.000011
Prostaglandin D2 receptor Mus musculus (house mouse)Ki10.000022
Prostaglandin D2 receptor 2Homo sapiens (human)Ki4.025022
Prostaglandin E synthaseHomo sapiens (human)IC5040.600011
Prostaglandin E2 receptor EP1 subtypeMus musculus (house mouse)Ki10.000022
Prostaglandin E2 receptor EP2 subtypeMus musculus (house mouse)Ki10.000022
Prostaglandin E2 receptor EP3 subtypeMus musculus (house mouse)Ki10.000022
Prostaglandin E2 receptor EP4 subtypeMus musculus (house mouse)Ki10.000022
Prostaglandin G/H synthase 1Homo sapiens (human)IC501.62835968
Prostaglandin G/H synthase 1Mus musculus (house mouse)IC500.011022
Prostaglandin G/H synthase 1Ovis aries (sheep)IC502.466880101
Prostaglandin G/H synthase 1Ovis aries (sheep)Ki7.900011
Prostaglandin G/H synthase 1 Bos taurus (cattle)IC5075.18701116
Prostaglandin G/H synthase 1 Rattus norvegicus (Norway rat)IC500.485488
Prostaglandin G/H synthase 2Homo sapiens (human)IC5017.050999119
Prostaglandin G/H synthase 2Mus musculus (house mouse)IC501.26531322
Prostaglandin G/H synthase 2Ovis aries (sheep)IC50102.76052630
Prostaglandin G/H synthase 2Homo sapiens (human)Ki1.500011
Prostaglandin G/H synthase 2Ovis aries (sheep)Ki9.860011
Prostaglandin G/H synthase 2 Bos taurus (cattle)IC500.776469
Prostaglandin G/H synthase 2 Rattus norvegicus (Norway rat)IC500.489188
Prostaglandin-H2 D-isomeraseMus musculus (house mouse)IC501.100022
receptor-interacting serine/threonine-protein kinase 2 isoform 1Homo sapiens (human)IC506.633011
Rho-associated protein kinase 2Rattus norvegicus (Norway rat)IC507.700012
Serine/threonine-protein kinase pim-1Homo sapiens (human)IC504.300011
Serum paraoxonase/arylesterase 1Homo sapiens (human)Ki97.000011
Shiga toxin subunit AShigella dysenteriaeIC5023.900011
Sigma intracellular receptor 2Rattus norvegicus (Norway rat)IC500.490011
Similar to alpha-tubulin isoform 1 Bos taurus (cattle)IC503.53162038
Sodium- and chloride-dependent betaine transporterRattus norvegicus (Norway rat)IC500.200011
Sodium- and chloride-dependent GABA transporter 1Rattus norvegicus (Norway rat)IC500.200011
Sodium- and chloride-dependent GABA transporter 2Rattus norvegicus (Norway rat)IC500.200011
Sodium- and chloride-dependent GABA transporter 3Rattus norvegicus (Norway rat)IC500.200011
Sodium-dependent dopamine transporterRattus norvegicus (Norway rat)IC5014.000011
Solute carrier family 22 member 3Homo sapiens (human)Ki0.120011
Solute carrier family 22 member 6Homo sapiens (human)IC504.400012
Solute carrier family 22 member 6Rattus norvegicus (Norway rat)Ki12.050024
Solute carrier family 22 member 8Homo sapiens (human)Ki5.950011
Solute carrier organic anion transporter family member 1A3Rattus norvegicus (Norway rat)Ki1,000.000011
Solute carrier organic anion transporter family member 1B1Homo sapiens (human)IC5012.000011
Solute carrier organic anion transporter family member 1B1Homo sapiens (human)Ki11.000011
Solute carrier organic anion transporter family member 1B3Homo sapiens (human)IC5041.000011
Solute carrier organic anion transporter family member 1B3Homo sapiens (human)Ki38.000011
Solute carrier organic anion transporter family member 2B1 Homo sapiens (human)IC50140.000011
Solute carrier organic anion transporter family member 2B1 Homo sapiens (human)Ki130.000011
steroidogenic factor 1Homo sapiens (human)IC5067.568011
Substance-P receptorCavia porcellus (domestic guinea pig)IC505.700011
Thromboxane-A synthase Homo sapiens (human)IC5050.050022
Tubulin alpha-1A chainHomo sapiens (human)IC5022.88383939
Tubulin alpha-1A chainSus scrofa (pig)IC504.67592828
Tubulin alpha-1A chainHomo sapiens (human)Ki2.400011
Tubulin alpha-1A chainSus scrofa (pig)Ki5.750011
Tubulin alpha-1B chainHomo sapiens (human)IC5022.88383939
Tubulin alpha-1B chainHomo sapiens (human)Ki2.400011
Tubulin alpha-1C chainHomo sapiens (human)IC5022.88383939
Tubulin alpha-1C chainHomo sapiens (human)Ki2.400011
Tubulin alpha-3C chainHomo sapiens (human)IC5022.88383939
Tubulin alpha-3C chainHomo sapiens (human)Ki2.400011
Tubulin alpha-3E chainHomo sapiens (human)IC5022.88383939
Tubulin alpha-3E chainHomo sapiens (human)Ki2.400011
Tubulin alpha-4A chainHomo sapiens (human)IC5022.88383939
Tubulin alpha-4A chainHomo sapiens (human)Ki2.400011
Tubulin beta chainHomo sapiens (human)IC5021.70714242
Tubulin beta chainSus scrofa (pig)IC504.84452626
Tubulin beta chainHomo sapiens (human)Ki2.400011
Tubulin beta chainSus scrofa (pig)Ki5.750011
Tubulin beta-1 chainHomo sapiens (human)IC5022.88383939
Tubulin beta-1 chainHomo sapiens (human)Ki2.400011
Tubulin beta-2A chainHomo sapiens (human)IC5022.88383939
Tubulin beta-2A chainHomo sapiens (human)Ki2.400011
Tubulin beta-2B chainBos taurus (cattle)IC50469.72332424
Tubulin beta-2B chainHomo sapiens (human)IC5022.88383939
Tubulin beta-2B chainBos taurus (cattle)Ki0.780011
Tubulin beta-2B chainHomo sapiens (human)Ki2.400011
Tubulin beta-3 chainHomo sapiens (human)IC5022.88383939
Tubulin beta-3 chainHomo sapiens (human)Ki2.400011
Tubulin beta-4A chainHomo sapiens (human)IC5022.88383939
Tubulin beta-4A chainHomo sapiens (human)Ki2.400011
Tubulin beta-4B chainHomo sapiens (human)IC5022.88383939
Tubulin beta-4B chainHomo sapiens (human)Ki2.400011
Tubulin beta-6 chainHomo sapiens (human)IC5022.88383939
Tubulin beta-6 chainHomo sapiens (human)Ki2.400011
Tubulin beta-8 chainHomo sapiens (human)IC5022.88383939
Tubulin beta-8 chainHomo sapiens (human)Ki2.400011
Uracil nucleotide/cysteinyl leukotriene receptorHomo sapiens (human)IC5028.800022
Vesicular acetylcholine transporterTetronarce californica (Pacific electric ray)IC502.620011
Xanthine dehydrogenase/oxidaseBos taurus (cattle)IC5013.75204242
Xanthine dehydrogenase/oxidaseHomo sapiens (human)IC5010.99684040
Xanthine dehydrogenase/oxidaseBos taurus (cattle)Ki1.800022
Xanthine dehydrogenase/oxidaseHomo sapiens (human)Ki2.891766
Xanthine dehydrogenase/oxidase [Includes: Xanthine dehydrogenase Rattus norvegicus (Norway rat)IC509.317733

Activation Measurements

ProteinTaxonomyMeasurementAverage (mM)Bioassay(s)Drugs
Adenosine receptor A2aHomo sapiens (human)Kd77.000011
AlbuminHomo sapiens (human)Kd60.350022
Androgen receptorHomo sapiens (human)EC500.000111
Peroxisome proliferator-activated receptor gammaHomo sapiens (human)EC5050.000011
Prostaglandin D2 receptor 2Homo sapiens (human)EC500.389012
Prostaglandin G/H synthase 2Homo sapiens (human)Kd1.020011
Purine nucleoside phosphorylaseMycobacterium tuberculosis H37RvKd1,000.000011
Tubulin alpha-1A chainHomo sapiens (human)EC500.200011
Tubulin alpha-1A chainHomo sapiens (human)Kd5.679022
Tubulin alpha-1A chainSus scrofa (pig)Kd7.500022
Tubulin alpha-1B chainHomo sapiens (human)EC500.200011
Tubulin alpha-1B chainHomo sapiens (human)Kd5.679022
Tubulin alpha-1C chainHomo sapiens (human)EC500.200011
Tubulin alpha-1C chainHomo sapiens (human)Kd5.679022
Tubulin alpha-3C chainHomo sapiens (human)EC500.200011
Tubulin alpha-3C chainHomo sapiens (human)Kd5.679022
Tubulin alpha-3E chainHomo sapiens (human)EC500.200011
Tubulin alpha-3E chainHomo sapiens (human)Kd5.679022
Tubulin alpha-4A chainHomo sapiens (human)EC500.200011
Tubulin alpha-4A chainHomo sapiens (human)Kd5.679022
Tubulin beta chainHomo sapiens (human)EC500.200011
Tubulin beta chainHomo sapiens (human)Kd5.679022
Tubulin beta chainSus scrofa (pig)Kd7.500022
Tubulin beta-1 chainHomo sapiens (human)EC500.200011
Tubulin beta-1 chainHomo sapiens (human)Kd5.679022
Tubulin beta-2A chainHomo sapiens (human)EC500.200011
Tubulin beta-2A chainHomo sapiens (human)Kd5.679022
Tubulin beta-2B chainHomo sapiens (human)EC500.200011
Tubulin beta-2B chainHomo sapiens (human)Kd5.679022
Tubulin beta-3 chainHomo sapiens (human)EC500.200011
Tubulin beta-3 chainHomo sapiens (human)Kd5.679022
Tubulin beta-4A chainHomo sapiens (human)EC500.200011
Tubulin beta-4A chainHomo sapiens (human)Kd5.679022
Tubulin beta-4B chainHomo sapiens (human)EC500.200011
Tubulin beta-4B chainHomo sapiens (human)Kd5.679022
Tubulin beta-6 chainHomo sapiens (human)EC500.200011
Tubulin beta-6 chainHomo sapiens (human)Kd5.679022
Tubulin beta-8 chainHomo sapiens (human)EC500.200011
Tubulin beta-8 chainHomo sapiens (human)Kd5.679022
Tubulin polymerization-promoting proteinBos taurus (cattle)EC500.750011
Xanthine dehydrogenase/oxidaseBos taurus (cattle)Kd0.000511

Other Measurements

ProteinTaxonomyMeasurementAverage (mM)Bioassay(s)Drugs
ATP-dependent translocase ABCB1Homo sapiens (human)Km23.165022
Caspase-1Homo sapiens (human)ID5030.000011
Hypoxanthine-guanine phosphoribosyltransferaseHomo sapiens (human)Km91.450022
Microphthalmia-associated transcription factorHomo sapiens (human)AC5035.000011
PAX8Homo sapiens (human)AC500.260011
Plasma kallikreinHomo sapiens (human)Activity1.060011
Polyunsaturated fatty acid 5-lipoxygenaseRattus norvegicus (Norway rat)Change100.000022
Polyunsaturated fatty acid 5-lipoxygenaseRattus norvegicus (Norway rat)ID5025.000011
Polyunsaturated fatty acid 5-lipoxygenaseRattus norvegicus (Norway rat)Inhibition20.000011
Prostaglandin G/H synthase 1Ovis aries (sheep)Kinact3.900011
Prostaglandin G/H synthase 1 Rattus norvegicus (Norway rat)Change0.200022
Prostaglandin G/H synthase 1 Bos taurus (cattle)ID500.430011
Prostaglandin G/H synthase 2Mus musculus (house mouse)Activity0.250011
Prostaglandin G/H synthase 2 Rattus norvegicus (Norway rat)Change0.200022
Prostaglandin G/H synthase 2 Bos taurus (cattle)ID500.430011
Solute carrier family 22 member 7Rattus norvegicus (Norway rat)Km0.366011
Tubulin alpha-1A chainHomo sapiens (human)Activity9.473399
Tubulin alpha-1B chainHomo sapiens (human)Activity9.473399
Tubulin alpha-1C chainHomo sapiens (human)Activity9.473399
Tubulin alpha-3C chainHomo sapiens (human)Activity9.473399
Tubulin alpha-3E chainHomo sapiens (human)Activity9.473399
Tubulin alpha-4A chainHomo sapiens (human)Activity9.473399
Tubulin beta chainHomo sapiens (human)Activity9.473399
Tubulin beta-1 chainHomo sapiens (human)Activity9.473399
Tubulin beta-2A chainHomo sapiens (human)Activity9.473399
Tubulin beta-2B chainHomo sapiens (human)Activity9.473399
Tubulin beta-3 chainHomo sapiens (human)Activity9.473399
Tubulin beta-4A chainHomo sapiens (human)Activity9.473399
Tubulin beta-4B chainHomo sapiens (human)Activity9.473399
Tubulin beta-6 chainHomo sapiens (human)Activity9.473399
Tubulin beta-8 chainHomo sapiens (human)Activity9.473399
UDP-glucuronosyltransferase 1A4Homo sapiens (human)Km7.000011
Xanthine dehydrogenase/oxidaseBos taurus (cattle)Km58.375044