nootropic agent

Any compound that improves mental functions such as cognition, memory, intelligence, motivation, attention, and concentration.

ChEBI ID: 66980

Members (9)

Member	Definition	Class
((5z)5-(1,3-benzodioxol-5-yl)methylene-2-phenylamino-3,5-dihydro-4h-imidazol-4-one)	A member of the class of benzodioxoles that is 1,3-benzodioxole substituted by a (2-anilino-5-oxo-1,5-dihydro-4H-imidazol-4-ylidene)methyl group at position 5. It is an inhibitor of DYRK1A, DYRK2, CLK1, and CLK3 (IC50s = 0.04, 0.035, 0.015, and 4.5 muM, respectively).	leucettine L41
aminooxyacetic acid	A member of the class of hydroxylamines that is acetic acid substituted at postion 2 by an aminooxy group. It is a compound which inhibits aminobutyrate aminotransferase activity in vivo, resulting in increased levels of gamma-aminobutyric acid in tissues.	(aminooxy)acetic acid
donepezil	A racemate comprising equimolar amounts of (R)- and (S)-donepezil. A centrally acting reversible acetylcholinesterase inhibitor, its main therapeutic use is in the treatment of Alzheimer's disease where it is used to increase cortical acetylcholine.	2-[(1-benzylpiperidin-4-yl)methyl]-5,6-dimethoxyindan-1-one; donepezil
fasudil	An isoquinoline substituted by a (1,4-diazepan-1-yl)sulfonyl group at position 5. It is a Rho-kinase inhibitor and its hydrochloride hydrate form is approved for the treatment of cerebral vasospasm and cerebral ischemia.	fasudil
fasudil hydrochloride	A hydrochloride obtained by reaction of fasudil with one equivalent of hydrochloric acid.	fasudil hydrochloride
huperzine a	A sesquiterpene alkaloid isolated from a club moss Huperzia serrata that has been shown to exhibit neuroprotective activity. It is also an effective inhibitor of acetylcholinesterase and has attracted interest as a therapeutic candidate for Alzheimer's disease.	huperzine A
levocarnitine	The (R)-enantiomer of carnitine.	(R)-carnitine
ta 0910	An oligopeptide comprising of (4S)-1-methyl-2,6-dioxohexahydropyrimidine-4-carboxylic acid, L-histidine and L-prolinamide joined in sequence by peptide linkages. It is a thyrotropin-releasing hormone (TRH) analog. Its tetrahydrate form is approved in Japan for the treatment of spinal muscular atrophy.	taltirelin
tramiprosate	An amino sulfonic acid that is the 3-amino derivative of propanesulfonic acid.	3-aminopropanesulfonic acid zwitterion; 3-aminopropanesulfonic acid

Research

Studies (5,055)

Timeframe	Studies, Drugs with This Role(%)	All Drugs %
pre-1990	558 (11.04)	18.7374
1990's	465 (9.20)	18.2507
2000's	1,535 (30.37)	29.6817
2010's	1,879 (37.17)	24.3611
2020's	618 (12.23)	2.80

Study Types

Publication Type	Studies, Drugs with this Role (%)	All Drugs (%)
Trials	615 (11.51%)	5.53%
Reviews	549 (10.28%)	6.00%
Case Studies	269 (5.03%)	4.05%
Observational	22 (0.41%)	0.25%
Other	3,888 (72.77%)	84.16%

Protein Targets (462)

Potency Measurements

Protein	Taxonomy	Measurement	Average (mM)	Bioassay(s)	Drugs
acetylcholinesterase	Homo sapiens (human)	Potency	0.3647	4	4
AR protein	Homo sapiens (human)	Potency	26.4049	4	4
arylsulfatase A	Homo sapiens (human)	Potency	0.0601	1	1
ATAD5 protein, partial	Homo sapiens (human)	Potency	19.9971	2	3
Ataxin-2	Homo sapiens (human)	Potency	18.8336	1	1
ATPase family AAA domain-containing protein 5	Homo sapiens (human)	Potency	18.8336	1	1
atrial natriuretic peptide receptor 1 precursor	Homo sapiens (human)	Potency	0.8492	1	1
Chain A, Beta-lactamase	Escherichia coli K-12	Potency	11.8998	2	2
Chain A, JmjC domain-containing histone demethylation protein 3A	Homo sapiens (human)	Potency	89.1251	1	1
Chain A, MAJOR APURINIC/APYRIMIDINIC ENDONUCLEASE	Homo sapiens (human)	Potency	50.1187	1	1
cytochrome P450 2D6	Homo sapiens (human)	Potency	0.8709	1	1
cytochrome P450 2D6 isoform 1	Homo sapiens (human)	Potency	0.1995	1	1
cytochrome P450 3A4 isoform 1	Homo sapiens (human)	Potency	12.5893	2	2
cytochrome P450 family 3 subfamily A polypeptide 4	Homo sapiens (human)	Potency	27.5404	1	1
cytochrome P450, family 19, subfamily A, polypeptide 1, isoform CRA_a	Homo sapiens (human)	Potency	13.3332	1	1
D(1A) dopamine receptor	Homo sapiens (human)	Potency	0.1458	1	1
dopamine D1 receptor	Homo sapiens (human)	Potency	5.8048	1	1
estrogen nuclear receptor alpha	Homo sapiens (human)	Potency	8.6200	5	5
estrogen-related nuclear receptor alpha	Homo sapiens (human)	Potency	27.9136	6	6
euchromatic histone-lysine N-methyltransferase 2	Homo sapiens (human)	Potency	33.8025	1	3
EWS/FLI fusion protein	Homo sapiens (human)	Potency	13.1812	2	2
farnesoid X nuclear receptor	Homo sapiens (human)	Potency	13.3322	1	1
GABA theta subunit	Rattus norvegicus (Norway rat)	Potency	12.5893	1	1
GALC protein	Homo sapiens (human)	Potency	0.7079	1	2
Gamma-aminobutyric acid receptor subunit alpha-1	Rattus norvegicus (Norway rat)	Potency	12.5893	1	1
Gamma-aminobutyric acid receptor subunit alpha-2	Rattus norvegicus (Norway rat)	Potency	12.5893	1	1
Gamma-aminobutyric acid receptor subunit alpha-3	Rattus norvegicus (Norway rat)	Potency	12.5893	1	1
Gamma-aminobutyric acid receptor subunit alpha-4	Rattus norvegicus (Norway rat)	Potency	12.5893	1	1
Gamma-aminobutyric acid receptor subunit alpha-5	Rattus norvegicus (Norway rat)	Potency	12.5893	1	1
Gamma-aminobutyric acid receptor subunit alpha-6	Rattus norvegicus (Norway rat)	Potency	12.5893	1	1
Gamma-aminobutyric acid receptor subunit beta-1	Rattus norvegicus (Norway rat)	Potency	12.5893	1	1
Gamma-aminobutyric acid receptor subunit beta-2	Rattus norvegicus (Norway rat)	Potency	12.5893	1	1
Gamma-aminobutyric acid receptor subunit beta-3	Rattus norvegicus (Norway rat)	Potency	12.5893	1	1
Gamma-aminobutyric acid receptor subunit delta	Rattus norvegicus (Norway rat)	Potency	12.5893	1	1
Gamma-aminobutyric acid receptor subunit epsilon	Rattus norvegicus (Norway rat)	Potency	12.5893	1	1
Gamma-aminobutyric acid receptor subunit gamma-1	Rattus norvegicus (Norway rat)	Potency	12.5893	1	1
Gamma-aminobutyric acid receptor subunit gamma-2	Rattus norvegicus (Norway rat)	Potency	12.5893	1	1
Gamma-aminobutyric acid receptor subunit gamma-3	Rattus norvegicus (Norway rat)	Potency	12.5893	1	1
Gamma-aminobutyric acid receptor subunit pi	Rattus norvegicus (Norway rat)	Potency	12.5893	1	1
geminin	Homo sapiens (human)	Potency	24.5634	2	3
GLI family zinc finger 3	Homo sapiens (human)	Potency	19.9826	2	2
glucocorticoid receptor [Homo sapiens]	Homo sapiens (human)	Potency	9.5205	1	1
Glutamate receptor 2	Rattus norvegicus (Norway rat)	Potency	6.6824	1	1
histone acetyltransferase KAT2A isoform 1	Homo sapiens (human)	Potency	39.8107	1	1
huntingtin isoform 2	Homo sapiens (human)	Potency	12.5893	1	1
IDH1	Homo sapiens (human)	Potency	16.3601	1	1
Interferon beta	Homo sapiens (human)	Potency	33.2940	1	1
lethal factor (plasmid)	Bacillus anthracis str. A2012	Potency	12.5893	1	1
muscarinic acetylcholine receptor M1	Rattus norvegicus (Norway rat)	Potency	2.2387	1	1
nuclear factor erythroid 2-related factor 2 isoform 1	Homo sapiens (human)	Potency	10.5901	2	2
nuclear receptor subfamily 1, group I, member 3	Homo sapiens (human)	Potency	13.0822	2	2
parathyroid hormone/parathyroid hormone-related peptide receptor precursor	Homo sapiens (human)	Potency	44.6684	1	1
peripheral myelin protein 22	Rattus norvegicus (Norway rat)	Potency	10.1815	1	1
peroxisome proliferator activated receptor gamma	Homo sapiens (human)	Potency	26.8325	1	1
pregnane X nuclear receptor	Homo sapiens (human)	Potency	33.4915	1	1
RAR-related orphan receptor gamma	Mus musculus (house mouse)	Potency	26.6032	1	1
regulator of G-protein signaling 4	Homo sapiens (human)	Potency	0.7512	1	1
retinoic acid nuclear receptor alpha variant 1	Homo sapiens (human)	Potency	29.8493	2	2
Smad3	Homo sapiens (human)	Potency	2.8184	1	1
Spike glycoprotein	Severe acute respiratory syndrome-related coronavirus	Potency	39.8107	1	3
survival motor neuron protein isoform d	Homo sapiens (human)	Potency	17.7828	1	1
TAR DNA-binding protein 43	Homo sapiens (human)	Potency	35.4813	1	1
TDP1 protein	Homo sapiens (human)	Potency	21.8651	2	8
thioredoxin reductase	Rattus norvegicus (Norway rat)	Potency	3.2336	2	2
Thrombopoietin	Homo sapiens (human)	Potency	5.0119	2	2
thyroid stimulating hormone receptor	Homo sapiens (human)	Potency	31.6228	2	2
Voltage-dependent calcium channel gamma-2 subunit	Mus musculus (house mouse)	Potency	6.6824	1	1

Inhibition Measurements

Protein	Taxonomy	Measurement	Average (mM)	Bioassay(s)	Drugs
[Tau protein] kinase	Sus scrofa (pig)	IC50	2.9350	4	4
5-hydroxytryptamine receptor 1A	Rattus norvegicus (Norway rat)	IC50	7.4200	1	1
Acetylcholine receptor subunit epsilon	Homo sapiens (human)	IC50	0.0324	1	1
Acetylcholinesterase	Electrophorus electricus (electric eel)	IC50	0.8976	144	155
Acetylcholinesterase	Homo sapiens (human)	IC50	1.0700	140	146
Acetylcholinesterase	Mus musculus (house mouse)	IC50	5.8826	5	6
Acetylcholinesterase	Rattus norvegicus (Norway rat)	IC50	0.0285	29	30
Acetylcholinesterase	Tetronarce californica (Pacific electric ray)	IC50	0.0265	4	4
Acetylcholinesterase	Electrophorus electricus (electric eel)	Ki	0.0287	4	4
Acetylcholinesterase	Homo sapiens (human)	Ki	0.5949	10	12
Acetylcholinesterase	Bos taurus (cattle)	IC50	0.1552	6	7
Acetylcholinesterase	Bos taurus (cattle)	Ki	0.0029	2	2
Acyl-CoA:cholesterol acyltransferase	Oryctolagus cuniculus (rabbit)	IC50	0.0080	1	1
Amine oxidase [flavin-containing] A	Homo sapiens (human)	IC50	925.0000	2	2
Amine oxidase [flavin-containing] A	Bos taurus (cattle)	IC50	828.0000	1	1
Amine oxidase [flavin-containing] A	Rattus norvegicus (Norway rat)	IC50	286.2833	3	6
Amine oxidase [flavin-containing] B	Homo sapiens (human)	IC50	17.7333	3	3
Amine oxidase [flavin-containing] B	Rattus norvegicus (Norway rat)	IC50	174.1000	4	5
Amyloid-beta precursor protein	Homo sapiens (human)	IC50	50.0110	2	2
ATP-binding cassette sub-family C member 3	Homo sapiens (human)	IC50	133.0000	1	1
ATP-dependent translocase ABCB1	Homo sapiens (human)	IC50	34.8500	1	1
Beta-secretase 1	Homo sapiens (human)	IC50	0.8666	5	5
Bile salt export pump	Homo sapiens (human)	IC50	143.1000	3	3
Bile salt export pump	Rattus norvegicus (Norway rat)	IC50	519.3000	1	1
C-C chemokine receptor type 2	Homo sapiens (human)	IC50	35.0000	2	2
C-C motif chemokine 2	Homo sapiens (human)	IC50	6.9183	1	1
cAMP-dependent protein kinase catalytic subunit alpha	Bos taurus (cattle)	IC50	1.8042	1	12
cAMP-dependent protein kinase catalytic subunit alpha	Homo sapiens (human)	IC50	4.5800	1	1
cAMP-dependent protein kinase catalytic subunit alpha	Homo sapiens (human)	Ki	0.4600	1	1
cAMP-dependent protein kinase catalytic subunit alpha	Mus musculus (house mouse)	Ki	0.4950	1	2
cAMP-dependent protein kinase catalytic subunit beta	Homo sapiens (human)	IC50	4.5800	1	1
cAMP-dependent protein kinase catalytic subunit beta	Homo sapiens (human)	Ki	0.4600	1	1
cAMP-dependent protein kinase catalytic subunit gamma	Homo sapiens (human)	IC50	4.5800	1	1
cAMP-dependent protein kinase catalytic subunit gamma	Homo sapiens (human)	Ki	0.4600	1	1
cAMP-specific 3',5'-cyclic phosphodiesterase 4D	Homo sapiens (human)	IC50	36.0000	1	1
Canalicular multispecific organic anion transporter 1	Homo sapiens (human)	IC50	133.0000	1	1
Cannabinoid receptor 1	Homo sapiens (human)	IC50	0.3140	1	1
Carboxylic ester hydrolase	Equus caballus (horse)	IC50	4.5551	3	3
Carboxylic ester hydrolase	Rattus norvegicus (Norway rat)	IC50	24.3044	14	15
Carboxylic ester hydrolase	Equus caballus (horse)	Ki	0.6400	2	2
Carnitine O-palmitoyltransferase 1, muscle isoform	Rattus norvegicus (Norway rat)	Ki	100.0000	1	1
Carnitine O-palmitoyltransferase 2, mitochondrial	Rattus norvegicus (Norway rat)	Ki	100.0000	1	1
Casein kinase II subunit alpha	Homo sapiens (human)	IC50	0.4150	2	2
Casein kinase II subunit alpha 3	Homo sapiens (human)	IC50	0.5100	1	1
Casein kinase II subunit alpha'	Homo sapiens (human)	IC50	0.4150	2	2
Casein kinase II subunit beta	Homo sapiens (human)	IC50	0.4150	2	2
Cell division control protein 42 homolog	Homo sapiens (human)	IC50	6.5000	2	2
cGMP-specific 3',5'-cyclic phosphodiesterase	Homo sapiens (human)	IC50	100.0000	1	1
Chain A, Acetylcholinesterase	Tetronarce californica (Pacific electric ray)	Ki	0.2500	1	1
Chain A, cAMP-dependent protein kinase, alpha-catalytic subunit	Bos taurus (cattle)	IC50	2.2800	1	5
Chain A, Rho-associated protein kinase 1	Homo sapiens (human)	Ki	0.5300	1	3
Chain B, Rho-associated protein kinase 1	Homo sapiens (human)	Ki	0.5300	1	1
Chain E, cAMP-dependent protein kinase, alpha-catalytic subunit	Mus musculus (house mouse)	Ki	0.5300	1	1
Chain I, cAMP-dependent protein kinase inhibitor alpha	synthetic construct	IC50	2.2800	1	2
Chain I, cAMP-dependent protein kinase inhibitor, alpha form	synthetic construct	Ki	0.5300	1	1
Choline O-acetyltransferase	Rattus norvegicus (Norway rat)	IC50	0.0053	1	1
Cholinesterase	Canis lupus familiaris (dog)	IC50	10,000.0000	1	1
Cholinesterase	Equus caballus (horse)	IC50	4.3817	110	110
Cholinesterase	Homo sapiens (human)	IC50	121.4321	83	87
Cholinesterase	Mus musculus (house mouse)	IC50	1.9920	1	1
Cholinesterase	Equus caballus (horse)	Ki	2.1400	1	1
Cholinesterase	Homo sapiens (human)	Ki	4.7266	3	4
Cyclin-A1	Homo sapiens (human)	IC50	30.0000	1	1
Cyclin-A2	Homo sapiens (human)	IC50	20.0000	2	2
Cyclin-dependent kinase 2	Homo sapiens (human)	IC50	20.0000	2	2
Cyclin-dependent kinase 5 activator 1	Homo sapiens (human)	IC50	13.4700	3	3
Cyclin-dependent kinase 7	Homo sapiens (human)	IC50	10.0000	1	1
Cyclin-dependent kinase 9	Homo sapiens (human)	IC50	14.0000	2	2
Cyclin-dependent-like kinase 5	Homo sapiens (human)	IC50	13.4700	3	3
Cyclin-H	Homo sapiens (human)	IC50	10.0000	1	1
Cyclin-T1	Homo sapiens (human)	IC50	14.0000	2	2
Cystathionine beta-synthase	Homo sapiens (human)	IC50	5.2750	4	4
Cystathionine gamma-lyase	Homo sapiens (human)	IC50	2.2850	2	2
Cytochrome P450 1B1	Homo sapiens (human)	IC50	15.2400	1	1
Cytochrome P450 3A4	Homo sapiens (human)	IC50	18.2903	3	3
Dual specificity protein kinase CLK1	Homo sapiens (human)	IC50	0.0710	1	1
Dual specificity protein kinase CLK1	Mus musculus (house mouse)	IC50	0.0360	4	4
Dual specificity protein kinase CLK2	Mus musculus (house mouse)	IC50	0.3900	3	3
Dual specificity protein kinase CLK3	Mus musculus (house mouse)	IC50	6.0500	4	4
Dual specificity protein kinase CLK4	Mus musculus (house mouse)	IC50	0.0393	3	3
Dual specificity tyrosine-phosphorylation-regulated kinase 1A	Homo sapiens (human)	IC50	0.0371	6	6
Dual specificity tyrosine-phosphorylation-regulated kinase 1A	Rattus norvegicus (Norway rat)	IC50	0.0300	3	3
Dual specificity tyrosine-phosphorylation-regulated kinase 1B	Homo sapiens (human)	IC50	0.0550	4	4
Dual specificity tyrosine-phosphorylation-regulated kinase 2	Homo sapiens (human)	IC50	0.0855	4	4
Dual specificity tyrosine-phosphorylation-regulated kinase 3	Homo sapiens (human)	IC50	0.4167	3	3
Dual specificity tyrosine-phosphorylation-regulated kinase 4	Homo sapiens (human)	IC50	0.5200	1	1
Glycogen synthase kinase-3 alpha	Homo sapiens (human)	IC50	0.2100	1	1
Glycogen synthase kinase-3 beta	Homo sapiens (human)	IC50	27.8450	4	4
Glycogen synthase kinase-3 beta	Sus scrofa (pig)	IC50	2.9350	4	4
Histamine H3 receptor	Homo sapiens (human)	IC50	0.3500	1	1
Kappa-type opioid receptor	Cavia porcellus (domestic guinea pig)	IC50	5.0355	2	2
Liver carboxylesterase 1	Homo sapiens (human)	IC50	100.0000	1	1
Mitogen-activated protein kinase 1	Rattus norvegicus (Norway rat)	IC50	30.0000	1	1
MO15-related protein kinase Pfmrk	Plasmodium falciparum (malaria parasite P. falciparum)	IC50	500.0000	1	1
Multidrug resistance-associated protein 4	Homo sapiens (human)	IC50	72.9000	1	1
Myosin light chain kinase, smooth muscle	Homo sapiens (human)	IC50	12.6000	2	2
Myosin light chain kinase, smooth muscle	Homo sapiens (human)	Ki	36.0000	1	1
Myotonin-protein kinase	Homo sapiens (human)	IC50	8.0000	1	1
Potassium voltage-gated channel subfamily H member 2	Homo sapiens (human)	IC50	3.7844	3	3
Potassium voltage-gated channel subfamily H member 2	Homo sapiens (human)	Ki	25.1189	1	1
Protein kinase C epsilon type	Homo sapiens (human)	IC50	3.0000	2	2
Proton-coupled amino acid transporter 1	Homo sapiens (human)	Ki	7,100.0000	1	1
Rho-associated protein kinase 1	Homo sapiens (human)	IC50	1.0502	10	10
Rho-associated protein kinase 1	Homo sapiens (human)	Ki	0.4300	6	7
Rho-associated protein kinase 2	Bos taurus (cattle)	IC50	1.8043	1	12
Rho-associated protein kinase 2	Homo sapiens (human)	IC50	1.3060	14	14
Rho-associated protein kinase 2	Rattus norvegicus (Norway rat)	IC50	1.9000	1	1
Rho-associated protein kinase 2	Homo sapiens (human)	Ki	0.3300	1	1
Ribosomal protein S6 kinase alpha-5	Homo sapiens (human)	IC50	5.0000	1	1
Serine/threonine-protein kinase N1	Homo sapiens (human)	IC50	1.7000	1	1
Serine/threonine-protein kinase N2	Homo sapiens (human)	IC50	1.8533	3	3
Serine/threonine-protein kinase pim-1	Homo sapiens (human)	IC50	2.0600	3	3
Sigma non-opioid intracellular receptor 1	Cavia porcellus (domestic guinea pig)	Ki	0.0146	2	2
Sigma non-opioid intracellular receptor 1	Homo sapiens (human)	Ki	0.0146	2	2
Sodium-dependent serotonin transporter	Homo sapiens (human)	IC50	1,000.0000	1	1
Voltage-dependent L-type calcium channel subunit alpha-1C	Homo sapiens (human)	IC50	34.3000	1	1
Voltage-dependent L-type calcium channel subunit alpha-1D	Homo sapiens (human)	IC50	34.3000	1	1
Voltage-dependent L-type calcium channel subunit alpha-1F	Homo sapiens (human)	IC50	34.3000	1	1
Voltage-dependent L-type calcium channel subunit alpha-1S	Homo sapiens (human)	IC50	34.3000	1	1

Activation Measurements

Protein	Taxonomy	Measurement	Average (mM)	Bioassay(s)	Drugs
26S proteasome regulatory subunit 6B	Homo sapiens (human)	Kd	30.0000	1	1
5'-AMP-activated protein kinase catalytic subunit alpha-1	Homo sapiens (human)	Kd	30.0000	1	1
5'-AMP-activated protein kinase subunit gamma-1	Homo sapiens (human)	Kd	30.0000	1	1
5'-AMP-activated protein kinase subunit gamma-2	Homo sapiens (human)	Kd	30.0000	1	1
AarF domain-containing protein kinase 1	Homo sapiens (human)	Kd	30.0000	1	1
Acetylcholinesterase	Homo sapiens (human)	EC50	0.0430	1	1
Acetylcholinesterase	Homo sapiens (human)	Kd	0.0125	1	2
Actin-related protein 2	Homo sapiens (human)	Kd	30.0000	1	1
Actin-related protein 3	Homo sapiens (human)	Kd	30.0000	1	1
Activated CDC42 kinase 1	Homo sapiens (human)	Kd	30.0000	1	1
Activin receptor type-1	Homo sapiens (human)	Kd	30.0000	1	1
Activin receptor type-1B	Homo sapiens (human)	Kd	30.0000	1	1
Activin receptor type-2B	Homo sapiens (human)	Kd	30.0000	1	1
Acyl-CoA dehydrogenase family member 10	Homo sapiens (human)	Kd	30.0000	1	1
Acyl-CoA dehydrogenase family member 11	Homo sapiens (human)	Kd	30.0000	1	1
Adenine phosphoribosyltransferase	Homo sapiens (human)	Kd	30.0000	1	1
Adenosine kinase	Homo sapiens (human)	Kd	30.0000	1	1
Adenylate kinase 2, mitochondrial	Homo sapiens (human)	Kd	30.0000	1	1
ADP/ATP translocase 2	Homo sapiens (human)	Kd	30.0000	1	1
ADP/ATP translocase 3	Homo sapiens (human)	Kd	30.0000	1	1
AP2-associated protein kinase 1	Homo sapiens (human)	Kd	30.0000	1	1
ATP-dependent 6-phosphofructokinase, platelet type	Homo sapiens (human)	Kd	30.0000	1	1
ATP-dependent RNA helicase DDX1	Homo sapiens (human)	Kd	30.0000	1	1
ATP-dependent RNA helicase DDX3X	Homo sapiens (human)	Kd	30.0000	1	1
ATP-dependent RNA helicase DDX42	Homo sapiens (human)	Kd	30.0000	1	1
ATP-dependent RNA helicase DHX30	Homo sapiens (human)	Kd	30.0000	1	2
Atypical kinase COQ8A, mitochondrial	Homo sapiens (human)	Kd	30.0000	1	1
Aurora kinase A	Homo sapiens (human)	Kd	30.0000	1	1
Aurora kinase B	Homo sapiens (human)	Kd	30.0000	1	1
Beta-adrenergic receptor kinase 1	Homo sapiens (human)	Kd	30.0000	1	1
BMP-2-inducible protein kinase	Homo sapiens (human)	Kd	33.7880	1	1
Bone morphogenetic protein receptor type-1A	Homo sapiens (human)	Kd	30.0000	1	1
Bone morphogenetic protein receptor type-1B	Homo sapiens (human)	Kd	30.0000	1	1
Bone morphogenetic protein receptor type-2	Homo sapiens (human)	Kd	30.0000	1	1
Breakpoint cluster region protein	Homo sapiens (human)	Kd	30.0000	1	1
Calcium/calmodulin-dependent protein kinase kinase 2	Homo sapiens (human)	Kd	30.0000	1	1
Calcium/calmodulin-dependent protein kinase type II subunit delta	Homo sapiens (human)	Kd	30.0000	1	1
Calcium/calmodulin-dependent protein kinase type II subunit gamma	Homo sapiens (human)	Kd	30.0000	1	1
Calcium/calmodulin-dependent protein kinase type IV	Homo sapiens (human)	Kd	30.0000	1	2
cAMP-dependent protein kinase catalytic subunit alpha	Homo sapiens (human)	Kd	30.0000	1	1
cAMP-dependent protein kinase catalytic subunit beta	Homo sapiens (human)	Kd	30.0000	1	1
cAMP-dependent protein kinase catalytic subunit gamma	Homo sapiens (human)	Kd	30.0000	1	1
cAMP-dependent protein kinase type II-alpha regulatory subunit	Homo sapiens (human)	Kd	30.0000	1	1
Casein kinase I isoform alpha	Homo sapiens (human)	Kd	30.0000	1	1
Casein kinase I isoform delta	Homo sapiens (human)	Kd	30.0000	1	1
Casein kinase I isoform epsilon	Homo sapiens (human)	Kd	30.0000	1	1
Casein kinase I isoform gamma-1	Homo sapiens (human)	Kd	30.0000	1	1
Casein kinase I isoform gamma-2	Homo sapiens (human)	Kd	30.0000	1	1
Casein kinase I isoform gamma-3	Homo sapiens (human)	Kd	30.0000	1	1
Casein kinase II subunit alpha'	Homo sapiens (human)	Kd	30.0000	1	1
Cell division cycle 7-related protein kinase	Homo sapiens (human)	Kd	30.0000	1	1
cGMP-dependent protein kinase 1	Homo sapiens (human)	Kd	30.0000	1	1
Choline-phosphate cytidylyltransferase A	Homo sapiens (human)	Kd	30.0000	1	1
Chromodomain-helicase-DNA-binding protein 4	Homo sapiens (human)	Kd	30.0000	1	1
Citron Rho-interacting kinase	Homo sapiens (human)	Kd	48.8760	1	1
Cyclin-dependent kinase 1	Homo sapiens (human)	Kd	30.0000	1	1
Cyclin-dependent kinase 12	Homo sapiens (human)	Kd	3.4800	1	1
Cyclin-dependent kinase 13	Homo sapiens (human)	Kd	4.5180	1	1
Cyclin-dependent kinase 16	Homo sapiens (human)	Kd	30.0000	1	2
Cyclin-dependent kinase 17	Homo sapiens (human)	Kd	30.0000	1	1
Cyclin-dependent kinase 2	Homo sapiens (human)	Kd	30.0000	1	1
Cyclin-dependent kinase 3	Homo sapiens (human)	Kd	30.0000	1	1
Cyclin-dependent kinase 4	Homo sapiens (human)	Kd	30.0000	1	1
Cyclin-dependent kinase 6	Homo sapiens (human)	Kd	30.0000	1	1
Cyclin-dependent kinase 7	Homo sapiens (human)	Kd	30.0000	1	1
Cyclin-dependent kinase 9	Homo sapiens (human)	Kd	4.2510	1	1
Cyclin-dependent-like kinase 5	Homo sapiens (human)	Kd	30.0000	1	1
Cyclin-G-associated kinase	Homo sapiens (human)	Kd	30.0000	1	1
Cysteine--tRNA ligase, cytoplasmic	Homo sapiens (human)	Kd	30.0000	1	1
Cytochrome c1, heme protein, mitochondrial	Homo sapiens (human)	Kd	30.0000	1	1
dCTP pyrophosphatase 1	Homo sapiens (human)	Kd	30.0000	1	2
Delta(24)-sterol reductase	Homo sapiens (human)	Kd	30.0000	1	1
Deoxycytidine kinase	Homo sapiens (human)	Kd	30.0000	1	1
Discoidin domain-containing receptor 2	Homo sapiens (human)	Kd	30.0000	1	1
DNA replication licensing factor MCM4	Homo sapiens (human)	Kd	30.0000	1	1
DNA topoisomerase 2-alpha	Homo sapiens (human)	Kd	30.0000	1	1
DNA topoisomerase 2-beta	Homo sapiens (human)	Kd	30.0000	1	1
DnaJ homolog subfamily A member 1	Homo sapiens (human)	Kd	30.0000	1	1
Dual specificity mitogen-activated protein kinase kinase 1	Homo sapiens (human)	Kd	30.0000	1	1
Dual specificity mitogen-activated protein kinase kinase 2	Homo sapiens (human)	Kd	30.0000	1	1
Dual specificity mitogen-activated protein kinase kinase 3	Homo sapiens (human)	Kd	30.0000	1	1
Dual specificity mitogen-activated protein kinase kinase 5	Homo sapiens (human)	Kd	30.0000	1	1
Dual specificity mitogen-activated protein kinase kinase 6	Homo sapiens (human)	Kd	30.0000	1	1
Dual specificity protein kinase CLK1	Homo sapiens (human)	Kd	0.1135	2	2
Dual specificity protein kinase CLK2	Homo sapiens (human)	Kd	15.1800	2	2
Dual specificity protein kinase CLK3	Homo sapiens (human)	Kd	15.5500	2	2
Dual specificity protein kinase CLK4	Homo sapiens (human)	Kd	15.0350	2	2
Dual specificity protein kinase TTK	Homo sapiens (human)	Kd	30.0000	1	2
Dual specificity testis-specific protein kinase 1	Homo sapiens (human)	Kd	30.0000	1	1
Dual specificity testis-specific protein kinase 2	Homo sapiens (human)	Kd	30.0000	1	1
Dual specificity tyrosine-phosphorylation-regulated kinase 1A	Homo sapiens (human)	Kd	15.0039	2	2
Dual specificity tyrosine-phosphorylation-regulated kinase 1B	Homo sapiens (human)	Kd	0.1400	1	1
Dual specificity tyrosine-phosphorylation-regulated kinase 2	Homo sapiens (human)	Kd	0.4500	1	1
Dynamin-like 120 kDa protein, mitochondrial	Homo sapiens (human)	Kd	30.0000	1	1
EKC/KEOPS complex subunit TP53RK	Homo sapiens (human)	Kd	30.0000	1	1
Electron transfer flavoprotein subunit beta	Homo sapiens (human)	Kd	30.0000	1	1
Elongation factor Tu, mitochondrial	Homo sapiens (human)	Kd	30.0000	1	1
Ephrin type-A receptor 1	Homo sapiens (human)	Kd	30.0000	1	1
Ephrin type-A receptor 2	Homo sapiens (human)	Kd	30.0000	1	1
Ephrin type-A receptor 4	Homo sapiens (human)	Kd	30.0000	1	1
Ephrin type-A receptor 5	Homo sapiens (human)	Kd	30.0000	1	1
Ephrin type-A receptor 7	Homo sapiens (human)	Kd	30.0000	1	1
Ephrin type-B receptor 2	Homo sapiens (human)	Kd	30.0000	1	1
Ephrin type-B receptor 3	Homo sapiens (human)	Kd	30.0000	1	2
Ephrin type-B receptor 4	Homo sapiens (human)	Kd	30.0000	1	1
Ephrin type-B receptor 6	Homo sapiens (human)	Kd	30.0000	1	1
Epidermal growth factor receptor	Homo sapiens (human)	Kd	30.0000	1	1
Epithelial discoidin domain-containing receptor 1	Homo sapiens (human)	Kd	30.0000	1	1
Eukaryotic peptide chain release factor GTP-binding subunit ERF3B	Homo sapiens (human)	Kd	30.0000	1	1
Eukaryotic translation initiation factor 2-alpha kinase 1	Homo sapiens (human)	Kd	30.0000	1	1
Eukaryotic translation initiation factor 5B	Homo sapiens (human)	Kd	30.0000	1	1
Exosome RNA helicase MTR4	Homo sapiens (human)	Kd	30.0000	1	1
Ferrochelatase, mitochondrial	Homo sapiens (human)	Kd	30.0000	1	1
Fibroblast growth factor receptor 1	Homo sapiens (human)	Kd	30.0000	1	1
Focal adhesion kinase 1	Homo sapiens (human)	Kd	30.0000	1	1
G protein-coupled receptor kinase 6	Homo sapiens (human)	Kd	30.0000	1	1
General transcription and DNA repair factor IIH helicase subunit XPD	Homo sapiens (human)	Kd	30.0000	1	1
Glycine--tRNA ligase	Homo sapiens (human)	Kd	30.0000	1	1
Glycogen phosphorylase, brain form	Homo sapiens (human)	Kd	30.0000	1	1
Glycogen phosphorylase, liver form	Homo sapiens (human)	Kd	30.0000	1	1
Glycogen synthase kinase-3 alpha	Homo sapiens (human)	Kd	15.2750	2	2
Glycogen synthase kinase-3 beta	Homo sapiens (human)	Kd	30.0000	1	1
GTP-binding nuclear protein Ran	Homo sapiens (human)	Kd	30.0000	1	1
Guanine nucleotide-binding protein G(i) subunit alpha-2	Homo sapiens (human)	Kd	30.0000	1	1
Heme oxygenase 2	Homo sapiens (human)	Kd	30.0000	1	1
Hepatocyte growth factor receptor	Homo sapiens (human)	Kd	30.0000	1	1
High affinity nerve growth factor receptor	Homo sapiens (human)	Kd	30.0000	1	1
Homeodomain-interacting protein kinase 1	Homo sapiens (human)	Kd	0.3200	1	1
Homeodomain-interacting protein kinase 3	Homo sapiens (human)	Kd	0.2300	1	1
Inhibitor of nuclear factor kappa-B kinase subunit epsilon	Homo sapiens (human)	Kd	30.0000	1	1
Inosine-5'-monophosphate dehydrogenase 2	Homo sapiens (human)	Kd	30.0000	1	1
Insulin receptor	Homo sapiens (human)	Kd	30.0000	1	1
Insulin-like growth factor 1 receptor	Homo sapiens (human)	Kd	30.0000	1	1
Integrin-linked protein kinase	Homo sapiens (human)	Kd	30.0000	1	1
Interleukin-1 receptor-associated kinase 1	Homo sapiens (human)	Kd	15.4650	2	2
Interleukin-1 receptor-associated kinase 3	Homo sapiens (human)	Kd	30.0000	1	1
Interleukin-1 receptor-associated kinase 4	Homo sapiens (human)	Kd	30.0000	1	1
LIM domain kinase 1	Homo sapiens (human)	Kd	30.0000	1	1
LIM domain kinase 2	Homo sapiens (human)	Kd	30.0000	1	2
Long-chain-fatty-acid--CoA ligase 5	Homo sapiens (human)	Kd	30.0000	1	1
Macrophage-stimulating protein receptor	Homo sapiens (human)	Kd	30.0000	1	2
MAP kinase-activated protein kinase 2	Homo sapiens (human)	Kd	30.0000	1	1
MAP kinase-activated protein kinase 5	Homo sapiens (human)	Kd	30.0000	1	1
MAP/microtubule affinity-regulating kinase 3	Homo sapiens (human)	Kd	30.0000	1	1
MAP/microtubule affinity-regulating kinase 4	Homo sapiens (human)	Kd	30.0000	1	1
Maternal embryonic leucine zipper kinase	Homo sapiens (human)	Kd	1.9220	1	1
Membrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinase	Homo sapiens (human)	Kd	30.0000	1	1
Midasin	Homo sapiens (human)	Kd	30.0000	1	2
Mitogen-activated protein kinase 1	Homo sapiens (human)	Kd	30.0000	1	2
Mitogen-activated protein kinase 10	Homo sapiens (human)	Kd	30.0000	1	1
Mitogen-activated protein kinase 11	Homo sapiens (human)	Kd	30.0000	1	1
Mitogen-activated protein kinase 14	Homo sapiens (human)	Kd	30.0000	1	1
Mitogen-activated protein kinase 15	Homo sapiens (human)	Kd	30.0000	1	1
Mitogen-activated protein kinase 3	Homo sapiens (human)	Kd	30.0000	1	1
Mitogen-activated protein kinase 7	Homo sapiens (human)	Kd	30.0000	1	1
Mitogen-activated protein kinase 8	Homo sapiens (human)	Kd	30.0000	1	1
Mitogen-activated protein kinase 9	Homo sapiens (human)	Kd	30.0000	1	1
Mitogen-activated protein kinase kinase kinase 1	Homo sapiens (human)	Kd	30.0000	1	1
Mitogen-activated protein kinase kinase kinase 11	Homo sapiens (human)	Kd	30.0000	1	1
Mitogen-activated protein kinase kinase kinase 2	Homo sapiens (human)	Kd	30.0000	1	1
Mitogen-activated protein kinase kinase kinase 20	Homo sapiens (human)	Kd	30.0000	1	1
Mitogen-activated protein kinase kinase kinase 3	Homo sapiens (human)	Kd	30.0000	1	1
Mitogen-activated protein kinase kinase kinase 4	Homo sapiens (human)	Kd	30.0000	1	1
Mitogen-activated protein kinase kinase kinase 5	Homo sapiens (human)	Kd	30.0000	1	2
Mitogen-activated protein kinase kinase kinase 6	Homo sapiens (human)	Kd	30.0000	1	1
Mitogen-activated protein kinase kinase kinase kinase 1	Homo sapiens (human)	Kd	30.0000	1	1
Mitogen-activated protein kinase kinase kinase kinase 2	Homo sapiens (human)	Kd	30.0000	1	1
Mitogen-activated protein kinase kinase kinase kinase 3	Homo sapiens (human)	Kd	30.0000	1	1
Mitogen-activated protein kinase kinase kinase kinase 4	Homo sapiens (human)	Kd	30.0000	1	1
Mitogen-activated protein kinase kinase kinase kinase 5	Homo sapiens (human)	Kd	30.0000	1	1
Mitotic checkpoint serine/threonine-protein kinase BUB1	Homo sapiens (human)	Kd	30.0000	1	1
Multifunctional protein ADE2	Homo sapiens (human)	Kd	30.0000	1	1
Myosin light chain kinase 3	Homo sapiens (human)	Kd	30.0000	1	1
Myosin light chain kinase, smooth muscle	Homo sapiens (human)	Kd	30.0000	1	1
Myosin-10	Homo sapiens (human)	Kd	30.0000	1	1
Myosin-14	Homo sapiens (human)	Kd	30.0000	1	1
NADH dehydrogenase [ubiquinone] 1 alpha subcomplex subunit 13	Homo sapiens (human)	Kd	30.0000	1	1
Non-receptor tyrosine-protein kinase TNK1	Homo sapiens (human)	Kd	30.0000	1	1
Non-receptor tyrosine-protein kinase TYK2	Homo sapiens (human)	Kd	30.0000	1	1
NUAK family SNF1-like kinase 2	Homo sapiens (human)	Kd	30.0000	1	1
Nucleolar GTP-binding protein 1	Homo sapiens (human)	Kd	30.0000	1	2
Obg-like ATPase 1	Homo sapiens (human)	Kd	30.0000	1	1
PAS domain-containing serine/threonine-protein kinase	Homo sapiens (human)	Kd	30.0000	1	1
Peroxisomal acyl-coenzyme A oxidase 1	Homo sapiens (human)	Kd	30.0000	1	1
Peroxisomal acyl-coenzyme A oxidase 3	Homo sapiens (human)	Kd	30.0000	1	1
Phenylalanine--tRNA ligase beta subunit	Homo sapiens (human)	Kd	30.0000	1	1
Phosphatidylethanolamine-binding protein 1	Homo sapiens (human)	Kd	30.0000	1	1
Phosphatidylinositol 5-phosphate 4-kinase type-2 alpha	Homo sapiens (human)	Kd	30.0000	1	1
Phosphatidylinositol 5-phosphate 4-kinase type-2 gamma	Homo sapiens (human)	Kd	30.0000	1	1
Phosphorylase b kinase gamma catalytic chain, liver/testis isoform	Homo sapiens (human)	Kd	30.0000	1	1
Platelet-derived growth factor receptor beta	Homo sapiens (human)	Kd	30.0000	1	1
Probable ATP-dependent RNA helicase DDX6	Homo sapiens (human)	Kd	30.0000	1	1
Protein kinase C alpha type	Homo sapiens (human)	Kd	30.0000	1	1
Protein kinase C beta type	Homo sapiens (human)	Kd	30.0000	1	1
Protein kinase C delta type	Homo sapiens (human)	Kd	4.7890	1	1
Protein kinase C iota type	Homo sapiens (human)	Kd	30.0000	1	1
Protein kinase C theta type	Homo sapiens (human)	Kd	30.0000	1	1
Protein kinase C zeta type	Homo sapiens (human)	Kd	30.0000	1	1
Protein-tyrosine kinase 2-beta	Homo sapiens (human)	Kd	30.0000	1	1
Protein-tyrosine kinase 6	Homo sapiens (human)	Kd	30.0000	1	1
Proto-oncogene tyrosine-protein kinase receptor Ret	Homo sapiens (human)	Kd	30.0000	1	1
Proto-oncogene tyrosine-protein kinase Src	Homo sapiens (human)	Kd	30.0000	1	1
Putative heat shock protein HSP 90-beta 2	Homo sapiens (human)	Kd	30.0000	1	1
Pyridoxal kinase	Homo sapiens (human)	Kd	30.0000	1	2
RAC-alpha serine/threonine-protein kinase	Homo sapiens (human)	Kd	30.0000	1	1
RAC-beta serine/threonine-protein kinase	Homo sapiens (human)	Kd	30.0000	1	1
RAC-gamma serine/threonine-protein kinase	Homo sapiens (human)	Kd	30.0000	1	1
Ras-related C3 botulinum toxin substrate 1	Homo sapiens (human)	Kd	30.0000	1	1
Ras-related protein Rab-10	Homo sapiens (human)	Kd	30.0000	1	2
Ras-related protein Rab-27A	Homo sapiens (human)	Kd	30.0000	1	1
Ras-related protein Rab-6A	Homo sapiens (human)	Kd	30.0000	1	1
Receptor-interacting serine/threonine-protein kinase 2	Homo sapiens (human)	Kd	30.0000	1	1
Receptor-interacting serine/threonine-protein kinase 3	Homo sapiens (human)	Kd	30.0000	1	1
Receptor-type tyrosine-protein kinase FLT3	Homo sapiens (human)	Kd	30.0000	1	1
Rho-associated protein kinase 1	Homo sapiens (human)	Kd	0.9060	1	1
Rho-associated protein kinase 2	Homo sapiens (human)	Kd	0.5105	2	2
Ribosomal protein S6 kinase alpha-1	Homo sapiens (human)	Kd	30.0000	1	1
Ribosomal protein S6 kinase alpha-3	Homo sapiens (human)	Kd	30.0000	1	1
Ribosomal protein S6 kinase alpha-4	Homo sapiens (human)	Kd	30.0000	1	1
Ribosomal protein S6 kinase alpha-5	Homo sapiens (human)	Kd	30.0000	1	1
Ribosomal protein S6 kinase alpha-6	Homo sapiens (human)	Kd	30.0000	1	1
Ribosomal protein S6 kinase beta-1	Homo sapiens (human)	Kd	30.0000	1	1
Ribosyldihydronicotinamide dehydrogenase [quinone]	Homo sapiens (human)	Kd	2.4510	1	1
RNA cytidine acetyltransferase	Homo sapiens (human)	Kd	30.0000	1	1
S-adenosylmethionine synthase isoform type-2	Homo sapiens (human)	Kd	30.0000	1	1
Septin-9	Homo sapiens (human)	Kd	30.0000	1	1
Serine/threonine-protein kinase 10	Homo sapiens (human)	Kd	30.0000	1	1
Serine/threonine-protein kinase 16	Homo sapiens (human)	Kd	30.0000	1	1
Serine/threonine-protein kinase 26	Homo sapiens (human)	Kd	30.0000	1	1
Serine/threonine-protein kinase 3	Homo sapiens (human)	Kd	30.0000	1	1
serine/threonine-protein kinase 33 isoform a	Homo sapiens (human)	EC50	9.5830	1	1
Serine/threonine-protein kinase 4	Homo sapiens (human)	Kd	30.0000	1	2
Serine/threonine-protein kinase A-Raf	Homo sapiens (human)	Kd	30.0000	1	1
Serine/threonine-protein kinase B-raf	Homo sapiens (human)	Kd	30.0000	1	1
Serine/threonine-protein kinase Chk1	Homo sapiens (human)	Kd	30.0000	1	1
Serine/threonine-protein kinase D2	Homo sapiens (human)	Kd	6.4160	1	1
Serine/threonine-protein kinase D3	Homo sapiens (human)	Kd	23.3410	1	1
Serine/threonine-protein kinase LATS1	Homo sapiens (human)	Kd	4.1700	1	1
Serine/threonine-protein kinase MARK2	Homo sapiens (human)	Kd	30.0000	1	1
Serine/threonine-protein kinase MRCK alpha	Homo sapiens (human)	Kd	30.0000	1	1
Serine/threonine-protein kinase MRCK beta	Homo sapiens (human)	Kd	30.0000	1	1
Serine/threonine-protein kinase MRCK gamma	Homo sapiens (human)	Kd	30.0000	1	1
Serine/threonine-protein kinase N1	Homo sapiens (human)	Kd	0.8410	1	1
Serine/threonine-protein kinase N2	Homo sapiens (human)	Kd	2.5990	1	1
Serine/threonine-protein kinase N3	Homo sapiens (human)	Kd	0.0990	1	1
Serine/threonine-protein kinase Nek1	Homo sapiens (human)	Kd	30.0000	1	1
Serine/threonine-protein kinase Nek2	Homo sapiens (human)	Kd	30.0000	1	1
Serine/threonine-protein kinase Nek3	Homo sapiens (human)	Kd	30.0000	1	1
Serine/threonine-protein kinase Nek7	Homo sapiens (human)	Kd	30.0000	1	1
Serine/threonine-protein kinase Nek9	Homo sapiens (human)	Kd	30.0000	1	1
Serine/threonine-protein kinase NLK	Homo sapiens (human)	Kd	30.0000	1	1
Serine/threonine-protein kinase PAK 2	Homo sapiens (human)	Kd	30.0000	1	1
Serine/threonine-protein kinase PAK 4	Homo sapiens (human)	Kd	30.0000	1	1
Serine/threonine-protein kinase pim-1	Homo sapiens (human)	Kd	30.0000	1	1
Serine/threonine-protein kinase PLK1	Homo sapiens (human)	Kd	30.0000	1	2
Serine/threonine-protein kinase PLK4	Homo sapiens (human)	Kd	30.0000	1	1
Serine/threonine-protein kinase SIK2	Homo sapiens (human)	Kd	30.0000	1	1
Serine/threonine-protein kinase SIK3	Homo sapiens (human)	Kd	30.0000	1	1
Serine/threonine-protein kinase STK11	Homo sapiens (human)	Kd	30.0000	1	1
Serine/threonine-protein kinase TAO1	Homo sapiens (human)	Kd	15.8500	2	2
Serine/threonine-protein kinase TAO2	Homo sapiens (human)	Kd	30.0000	1	1
Serine/threonine-protein kinase TAO3	Homo sapiens (human)	Kd	30.0000	1	1
Serine/threonine-protein kinase TBK1	Homo sapiens (human)	Kd	30.0000	1	1
Serine/threonine-protein kinase ULK1	Homo sapiens (human)	Kd	30.0000	1	1
Serine/threonine-protein kinase ULK3	Homo sapiens (human)	Kd	30.0000	1	1
Serine/threonine-protein kinase/endoribonuclease IRE1	Homo sapiens (human)	Kd	30.0000	1	1
Serine/threonine-protein kinase/endoribonuclease IRE2	Homo sapiens (human)	Kd	30.0000	1	1
Signal recognition particle receptor subunit alpha	Homo sapiens (human)	Kd	30.0000	1	1
STE20-like serine/threonine-protein kinase	Homo sapiens (human)	Kd	30.0000	1	1
STE20-related kinase adapter protein alpha	Homo sapiens (human)	Kd	30.0000	1	1
Structural maintenance of chromosomes protein 1A	Homo sapiens (human)	Kd	30.0000	1	1
Structural maintenance of chromosomes protein 2	Homo sapiens (human)	Kd	30.0000	1	1
Succinate--CoA ligase [ADP-forming] subunit beta, mitochondrial	Homo sapiens (human)	Kd	30.0000	1	2
TGF-beta receptor type-1	Homo sapiens (human)	Kd	30.0000	1	1
TGF-beta receptor type-2	Homo sapiens (human)	Kd	30.0000	1	1
Thyroid hormone receptor-associated protein 3	Homo sapiens (human)	Kd	30.0000	1	1
TRAF2 and NCK-interacting protein kinase	Homo sapiens (human)	Kd	30.0000	1	1
Tyrosine--tRNA ligase, cytoplasmic	Homo sapiens (human)	Kd	30.0000	1	1
Tyrosine-protein kinase ABL1	Homo sapiens (human)	Kd	30.0000	1	1
Tyrosine-protein kinase ABL2	Homo sapiens (human)	Kd	30.0000	1	2
Tyrosine-protein kinase BTK	Homo sapiens (human)	Kd	30.0000	1	1
Tyrosine-protein kinase CSK	Homo sapiens (human)	Kd	30.0000	1	1
Tyrosine-protein kinase Fer	Homo sapiens (human)	Kd	30.0000	1	1
Tyrosine-protein kinase Fes/Fps	Homo sapiens (human)	Kd	30.0000	1	1
Tyrosine-protein kinase Fgr	Homo sapiens (human)	Kd	30.0000	1	1
Tyrosine-protein kinase FRK	Homo sapiens (human)	Kd	30.0000	1	1
Tyrosine-protein kinase Fyn	Homo sapiens (human)	Kd	30.0000	1	2
Tyrosine-protein kinase HCK	Homo sapiens (human)	Kd	30.0000	1	1
Tyrosine-protein kinase JAK1	Homo sapiens (human)	Kd	30.0000	1	1
Tyrosine-protein kinase Lck	Homo sapiens (human)	Kd	30.0000	1	1
Tyrosine-protein kinase Lyn	Homo sapiens (human)	Kd	30.0000	1	2
Tyrosine-protein kinase SYK	Homo sapiens (human)	Kd	30.0000	1	1
Tyrosine-protein kinase Tec	Homo sapiens (human)	Kd	30.0000	1	1
Tyrosine-protein kinase Yes	Homo sapiens (human)	Kd	30.0000	1	1
U5 small nuclear ribonucleoprotein 200 kDa helicase	Homo sapiens (human)	Kd	30.0000	1	1
UMP-CMP kinase	Homo sapiens (human)	Kd	30.0000	1	1
Uncharacterized aarF domain-containing protein kinase 5	Homo sapiens (human)	Kd	30.0000	1	1
Uncharacterized protein FLJ45252	Homo sapiens (human)	Kd	30.0000	1	2
Very long-chain specific acyl-CoA dehydrogenase, mitochondrial	Homo sapiens (human)	Kd	30.0000	1	1
Wee1-like protein kinase	Homo sapiens (human)	Kd	30.0000	1	1

Other Measurements

Protein	Taxonomy	Measurement	Average (mM)	Bioassay(s)	Drugs
cAMP-dependent protein kinase catalytic subunit alpha isoform Calpha1	Homo sapiens (human)	AC50	1.1975	2	2
Cannabinoid receptor 1	Homo sapiens (human)	Kb	2.2000	1	1
Carnitine O-acetyltransferase	Homo sapiens (human)	Km	300.0000	1	1
Cytochrome P450 1A2	Homo sapiens (human)	INH	10.0000	1	1
Cytochrome P450 2D6	Homo sapiens (human)	INH	3.6000	1	1
Cytochrome P450 3A4	Homo sapiens (human)	INH	10.0000	1	1
serine/threonine-protein kinase 33 isoform a	Homo sapiens (human)	AC50	9.3400	2	3
Solute carrier family 22 member 8	Mus musculus (house mouse)	Km	0.0619	1	1