Page last updated: 2024-08-07 17:21:50

Acyl-CoA:cholesterol acyltransferase

[no definition available]

Synonyms

Research

Bioassay Publications (13)

TimeframeStudies on this Protein(%)All Drugs %
pre-19900 (0.00)18.7374
1990's9 (69.23)18.2507
2000's4 (30.77)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Compounds (18)

Drugs with Inhibition Measurements

DrugTaxonomyMeasurementAverage (mM)Bioassay(s)Publication(s)
tacrineOryctolagus cuniculus (rabbit)IC500.267011
donepezilOryctolagus cuniculus (rabbit)IC500.008011
physostigmineOryctolagus cuniculus (rabbit)IC500.018911
3,5-dichlorosalicylic acidOryctolagus cuniculus (rabbit)Ki24.000011
lovastatinOryctolagus cuniculus (rabbit)IC5016.800011
zileutonOryctolagus cuniculus (rabbit)IC5055.000011
pd 128042Oryctolagus cuniculus (rabbit)IC500.148834
ramatrobanOryctolagus cuniculus (rabbit)IC507.655522
cl 277082Oryctolagus cuniculus (rabbit)IC500.143334
n-(2,6-bis(1-methylethyl)phenyl)-n'-((1-(4-(dimethylamino)phenyl)cyclopentyl)methyl)urea hydrochlorideOryctolagus cuniculus (rabbit)IC500.052011
n-(2,6-bis(isopropyl)phenyl)-n'-((1-(4-(dimethylaminomethyl)phenyl)cyclopentyl)methyl)ureaOryctolagus cuniculus (rabbit)IC500.037011
e 5324Oryctolagus cuniculus (rabbit)IC500.088011
avasimibeOryctolagus cuniculus (rabbit)IC507.600011
pactimibeOryctolagus cuniculus (rabbit)IC506.333333
oleoylanilideOryctolagus cuniculus (rabbit)IC5026.000011
pd 138142-15Oryctolagus cuniculus (rabbit)IC504.000011
oc000459Oryctolagus cuniculus (rabbit)IC5015.003022
mk-7246Oryctolagus cuniculus (rabbit)IC502.503022