Protein | Potency Measurements | Inhibition Measurements | Activation Measurements | Drugs |
Sodium/glucose cotransporter 1 | 0 | 0 | 1 | 1 |
Sodium/glucose cotransporter 2 | 0 | 1 | 1 | 2 |
Glycogen phosphorylase, muscle form | 0 | 1 | 0 | 1 |
Asialoglycoprotein receptor 1 | 0 | 1 | 1 | 2 |
Chain A, Glutamine Binding Protein | 0 | 0 | 1 | 1 |
thioredoxin reductase | 2 | 0 | 0 | 2 |
15-lipoxygenase, partial | 1 | 0 | 0 | 1 |
GLS protein | 1 | 0 | 0 | 1 |
arylsulfatase A | 2 | 0 | 0 | 2 |
euchromatic histone-lysine N-methyltransferase 2 | 3 | 0 | 0 | 3 |
Bloom syndrome protein isoform 1 | 1 | 0 | 0 | 1 |
peripheral myelin protein 22 isoform 1 | 1 | 0 | 0 | 1 |
flap endonuclease 1 | 2 | 0 | 0 | 2 |
histone-lysine N-methyltransferase 2A isoform 2 precursor | 1 | 0 | 0 | 1 |
Carbonic anhydrase 1 | 0 | 0 | 0 | 3 |
Carbonic anhydrase 2 | 0 | 1 | 0 | 4 |
Neutral amino acid transporter A | 0 | 1 | 0 | 1 |
Asc-type amino acid transporter 1 | 0 | 1 | 0 | 1 |
Neutral amino acid transporter B(0) | 0 | 1 | 0 | 1 |
Carbonic anhydrase-like protein, putative | 0 | 0 | 0 | 2 |
Amino acid transporter | 0 | 1 | 0 | 1 |
ATP-dependent phosphofructokinase | 1 | 0 | 0 | 1 |
Chain A, HISTIDINE-BINDING PROTEIN | 0 | 0 | 1 | 1 |
Chain E, LYSINE, ARGININE, ORNITHINE-BINDING PROTEIN | 0 | 0 | 1 | 1 |
Chain E, LYSINE, ARGININE, ORNITHINE-BINDING PROTEIN | 0 | 0 | 1 | 1 |
Chain E, LYSINE, ARGININE, ORNITHINE-BINDING PROTEIN | 0 | 0 | 1 | 1 |
ATAD5 protein, partial | 1 | 0 | 0 | 1 |
cytochrome P450 3A4 isoform 1 | 1 | 0 | 0 | 1 |
histone acetyltransferase KAT2A isoform 1 | 1 | 0 | 0 | 1 |
Gamma-aminobutyric acid receptor subunit pi | 1 | 1 | 1 | 3 |
Carbonic anhydrase 12 | 0 | 0 | 0 | 1 |
Plasma kallikrein | 0 | 0 | 0 | 1 |
Carbonic anhydrase 3 | 0 | 0 | 0 | 1 |
Histidine-binding periplasmic protein | 0 | 0 | 1 | 1 |
Gamma-aminobutyric acid receptor subunit beta-1 | 1 | 1 | 1 | 3 |
Gamma-aminobutyric acid receptor subunit delta | 1 | 1 | 1 | 3 |
Gamma-aminobutyric acid receptor subunit gamma-2 | 1 | 1 | 1 | 3 |
Gamma-aminobutyric acid receptor subunit alpha-5 | 1 | 1 | 1 | 3 |
Gamma-aminobutyric acid receptor subunit alpha-3 | 1 | 1 | 1 | 3 |
Carbonic anhydrase 4 | 0 | 0 | 0 | 1 |
Carbonic anhydrase 6 | 0 | 0 | 0 | 1 |
Gamma-aminobutyric acid receptor subunit gamma-1 | 1 | 1 | 1 | 3 |
Gamma-aminobutyric acid receptor subunit alpha-2 | 1 | 1 | 1 | 3 |
Adenosine receptor A1 | 0 | 0 | 0 | 1 |
5-hydroxytryptamine receptor 1D | 0 | 0 | 0 | 1 |
Gamma-aminobutyric acid receptor subunit alpha-4 | 1 | 1 | 1 | 3 |
Gamma-aminobutyric acid receptor subunit gamma-3 | 1 | 1 | 1 | 3 |
Gamma-aminobutyric acid receptor subunit alpha-6 | 1 | 1 | 1 | 3 |
Adenosine receptor A2a | 0 | 0 | 0 | 1 |
Carbonic anhydrase 5A, mitochondrial | 0 | 0 | 0 | 1 |
Glutamate receptor ionotropic, NMDA 1 | 0 | 0 | 0 | 1 |
Carbonic anhydrase | 0 | 0 | 0 | 1 |
Carbonic anhydrase 7 | 0 | 0 | 0 | 1 |
Carbonic anhydrase | 0 | 0 | 0 | 1 |
Gamma-aminobutyric acid receptor subunit alpha-1 | 1 | 1 | 1 | 3 |
Gamma-aminobutyric acid receptor subunit beta-3 | 1 | 1 | 1 | 3 |
Gamma-aminobutyric acid receptor subunit beta-2 | 1 | 1 | 1 | 3 |
Glutamate receptor ionotropic, NMDA 2A | 0 | 0 | 0 | 1 |
Glutamate receptor ionotropic, NMDA 2B | 0 | 0 | 0 | 1 |
Glutamate receptor ionotropic, NMDA 2C | 0 | 0 | 0 | 1 |
Large neutral amino acids transporter small subunit 1 | 0 | 1 | 0 | 1 |
Glutaminyl-peptide cyclotransferase | 0 | 1 | 0 | 1 |
Carbonic anhydrase 9 | 0 | 0 | 0 | 1 |
Carbonic anhydrase | 0 | 0 | 0 | 1 |
Carbonic anhydrase | 0 | 0 | 0 | 1 |
Carbonic anhydrase | 0 | 0 | 0 | 1 |
Glutamate receptor ionotropic, NMDA 2D | 0 | 0 | 0 | 1 |
Carbonic anhydrase | 0 | 0 | 0 | 1 |
Carbonic anhydrase 13 | 0 | 0 | 0 | 1 |
Glutamate receptor ionotropic, NMDA 3B | 0 | 0 | 0 | 1 |
GABA theta subunit | 1 | 1 | 1 | 3 |
Carbonic anhydrase 4 | 0 | 0 | 0 | 1 |
Carbonic anhydrase 15 | 0 | 0 | 0 | 1 |
Carbonic anhydrase 13 | 0 | 0 | 0 | 1 |
Gamma-aminobutyric acid receptor subunit epsilon | 1 | 1 | 1 | 3 |
Glutamate receptor ionotropic, NMDA 3A | 0 | 0 | 0 | 1 |
Carbonic anhydrase 14 | 0 | 0 | 0 | 1 |
Carbonic anhydrase 5B, mitochondrial | 0 | 0 | 0 | 1 |
Chain A, MAJOR APURINIC/APYRIMIDINIC ENDONUCLEASE | 1 | 0 | 0 | 1 |
TDP1 protein | 2 | 0 | 0 | 2 |
aldehyde dehydrogenase 1 family, member A1 | 1 | 0 | 0 | 1 |
EWS/FLI fusion protein | 1 | 0 | 0 | 1 |
CDGSH iron-sulfur domain-containing protein 1 | 0 | 1 | 0 | 1 |
tyrosine-protein kinase Yes | 1 | 0 | 0 | 1 |
Free fatty acid receptor 1 | 0 | 0 | 1 | 1 |
ATP-binding cassette sub-family C member 3 | 0 | 3 | 0 | 3 |
Multidrug resistance-associated protein 4 | 0 | 3 | 0 | 3 |
Bile salt export pump | 0 | 2 | 0 | 2 |
Peroxisome proliferator-activated receptor gamma | 0 | 1 | 0 | 1 |
Bile salt export pump | 0 | 3 | 0 | 3 |
Muscarinic acetylcholine receptor M1 | 0 | 0 | 1 | 1 |
Muscarinic acetylcholine receptor M3 | 0 | 0 | 1 | 1 |
Muscarinic acetylcholine receptor M4 | 0 | 0 | 1 | 1 |
Steryl-sulfatase | 0 | 1 | 0 | 1 |
Muscarinic acetylcholine receptor M5 | 0 | 0 | 1 | 1 |
Muscarinic acetylcholine receptor M2 | 0 | 0 | 1 | 1 |
Tyrosine-protein phosphatase non-receptor type 1 | 0 | 1 | 0 | 1 |
Carnitine O-palmitoyltransferase 2, mitochondrial | 0 | 1 | 0 | 1 |
Amine oxidase [flavin-containing] B | 0 | 1 | 0 | 1 |
Amine oxidase [flavin-containing] A | 0 | 1 | 0 | 1 |
Amine oxidase [flavin-containing] A | 0 | 1 | 0 | 1 |
Peroxisome proliferator-activated receptor alpha | 0 | 1 | 0 | 1 |
Carnitine O-palmitoyltransferase 2, mitochondrial | 0 | 1 | 0 | 1 |
Amine oxidase [flavin-containing] B | 0 | 2 | 0 | 2 |
Peroxisome proliferator-activated receptor gamma | 0 | 2 | 2 | 5 |
Peroxisome proliferator-activated receptor gamma | 0 | 1 | 1 | 2 |
Carnitine O-palmitoyltransferase 1, liver isoform | 0 | 1 | 0 | 1 |
Peroxisome proliferator-activated receptor alpha | 0 | 1 | 1 | 2 |
Enoyl-[acyl-carrier-protein] reductase [NADH] | 0 | 1 | 0 | 1 |
CDGSH iron-sulfur domain-containing protein 2 | 0 | 1 | 0 | 1 |
CDGSH iron-sulfur domain-containing protein 1 | 0 | 2 | 0 | 2 |
Beta-1 adrenergic receptor | 0 | 1 | 1 | 3 |
D(1A) dopamine receptor | 1 | 0 | 0 | 1 |
Solute carrier family 22 member 1 | 0 | 1 | 0 | 1 |
Voltage-dependent L-type calcium channel subunit alpha-1C | 0 | 1 | 0 | 1 |
5-hydroxytryptamine receptor 4 | 0 | 2 | 0 | 2 |
Albumin | 0 | 0 | 1 | 1 |
Cytochrome P450 1A2 | 0 | 1 | 0 | 1 |
Beta-2 adrenergic receptor | 0 | 2 | 1 | 3 |
Muscarinic acetylcholine receptor M2 | 0 | 1 | 1 | 2 |
ATP-dependent translocase ABCB1 | 0 | 2 | 0 | 2 |
Beta-1 adrenergic receptor | 0 | 2 | 1 | 3 |
Cytochrome P450 3A4 | 0 | 1 | 0 | 1 |
5-hydroxytryptamine receptor 1A | 0 | 1 | 0 | 1 |
Alpha-2A adrenergic receptor | 0 | 1 | 2 | 4 |
Adenosine receptor A3 | 0 | 1 | 1 | 2 |
Beta-2 adrenergic receptor | 0 | 2 | 0 | 3 |
Cytochrome P450 2C8 | 0 | 1 | 0 | 1 |
Cytochrome P450 2D6 | 0 | 1 | 0 | 1 |
Muscarinic acetylcholine receptor M1 | 0 | 1 | 1 | 2 |
Cytochrome P450 2C9 | 0 | 1 | 0 | 1 |
Beta-3 adrenergic receptor | 0 | 2 | 1 | 3 |
D(2) dopamine receptor | 0 | 1 | 1 | 2 |
Alpha-1B adrenergic receptor | 0 | 1 | 1 | 2 |
Alpha-2B adrenergic receptor | 0 | 0 | 1 | 2 |
Beta-1 adrenergic receptor | 0 | 2 | 1 | 4 |
Alpha-2C adrenergic receptor | 0 | 1 | 2 | 4 |
D(3) dopamine receptor | 0 | 1 | 0 | 1 |
5-hydroxytryptamine receptor 1A | 0 | 2 | 1 | 4 |
Alpha-2B adrenergic receptor | 0 | 0 | 1 | 1 |
Muscarinic acetylcholine receptor M3 | 0 | 1 | 1 | 2 |
D(1A) dopamine receptor | 0 | 1 | 1 | 2 |
Voltage-dependent L-type calcium channel subunit alpha-1C | 0 | 1 | 0 | 1 |
Alpha-2C adrenergic receptor | 0 | 0 | 1 | 1 |
Alpha-2A adrenergic receptor | 0 | 0 | 1 | 1 |
Alpha-1D adrenergic receptor | 0 | 1 | 1 | 2 |
Alpha-1D adrenergic receptor | 0 | 0 | 1 | 2 |
Endothelin-1 receptor | 0 | 1 | 1 | 2 |
Beta-3 adrenergic receptor | 0 | 2 | 0 | 2 |
5-hydroxytryptamine receptor 1B | 0 | 2 | 1 | 3 |
5-hydroxytryptamine receptor 2A | 0 | 2 | 1 | 3 |
5-hydroxytryptamine receptor 2C | 0 | 2 | 1 | 3 |
5-hydroxytryptamine receptor 1B | 0 | 2 | 0 | 2 |
Adenosine receptor A2a | 0 | 1 | 1 | 2 |
Neuromedin-K receptor | 0 | 0 | 1 | 1 |
Type-1 angiotensin II receptor | 0 | 1 | 1 | 2 |
Sodium-dependent serotonin transporter | 0 | 2 | 0 | 2 |
Cholecystokinin receptor type A | 0 | 1 | 1 | 2 |
Cytochrome P450 2C19 | 0 | 1 | 0 | 1 |
5-hydroxytryptamine receptor 7 | 0 | 1 | 1 | 2 |
Beta-1 adrenergic receptor | 0 | 1 | 0 | 1 |
Alpha-1A adrenergic receptor | 0 | 1 | 2 | 4 |
Alpha-1B adrenergic receptor | 0 | 0 | 1 | 2 |
Mu-type opioid receptor | 0 | 1 | 1 | 2 |
Vasopressin V1a receptor | 0 | 1 | 1 | 2 |
Delta-type opioid receptor | 0 | 1 | 1 | 2 |
Kappa-type opioid receptor | 0 | 1 | 1 | 2 |
5-hydroxytryptamine receptor 2B | 0 | 2 | 1 | 3 |
Alpha-1A adrenergic receptor | 0 | 1 | 1 | 2 |
5-hydroxytryptamine receptor 6 | 0 | 2 | 1 | 3 |
5-hydroxytryptamine receptor 7 | 0 | 1 | 0 | 1 |
Cytochrome P450 2J2 | 0 | 1 | 0 | 1 |
Beta-2 adrenergic receptor | 0 | 1 | 0 | 1 |
Potassium voltage-gated channel subfamily H member 2 | 0 | 1 | 0 | 1 |
Voltage-dependent L-type calcium channel subunit alpha-1C | 0 | 1 | 0 | 1 |
Sodium channel protein type 5 subunit alpha | 0 | 1 | 0 | 1 |
Sodium/bile acid cotransporter | 0 | 1 | 0 | 1 |
Beta-2 adrenergic receptor | 0 | 1 | 1 | 3 |
Canalicular multispecific organic anion transporter 1 | 0 | 2 | 0 | 2 |
Ataxin-2 | 1 | 0 | 0 | 1 |
Sigma non-opioid intracellular receptor 1 | 0 | 2 | 0 | 2 |
Nuclear receptor subfamily 2 group E member 1 | 0 | 0 | 2 | 2 |
Dipeptidyl peptidase 9 | 0 | 1 | 0 | 1 |
Dipeptidyl peptidase IV | 0 | 2 | 0 | 2 |
Kynurenine 3-monooxygenase | 0 | 1 | 0 | 1 |
Heat shock protein HSP 90-beta | 0 | 1 | 0 | 1 |
Dipeptidyl peptidase 4 | 0 | 1 | 0 | 1 |
Dipeptidyl peptidase 4 | 0 | 2 | 1 | 3 |
Dipeptidyl peptidase 4 | 0 | 1 | 0 | 1 |
Prolyl endopeptidase | 0 | 1 | 0 | 1 |
Prolyl endopeptidase FAP | 0 | 1 | 0 | 1 |
Prolyl endopeptidase FAP | 0 | 1 | 0 | 1 |
Dipeptidyl peptidase 8 | 0 | 2 | 0 | 2 |
Dipeptidyl peptidase 9 | 0 | 2 | 0 | 2 |
Dipeptidyl peptidase 2 | 0 | 1 | 0 | 1 |
[prepared from compound, protein, and bioassay information from National Library of Medicine (NLM), extracted Dec-2023] |