Page last updated: 2024-08-07 16:22:06
Dipeptidyl peptidase 4
A dipeptidyl peptidase 4 that is encoded in the genome of mouse. [OMA:P28843, PRO:DNx]
Synonyms
EC 3.4.14.5;
Dipeptidyl peptidase IV;
DPP IV;
T-cell activation antigen CD26;
Thymocyte-activating molecule;
THAM
Research
Bioassay Publications (6)
Timeframe | Studies on this Protein(%) | All Drugs % |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 0 (0.00) | 18.2507 |
2000's | 4 (66.67) | 29.6817 |
2010's | 2 (33.33) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Compounds (7)
Drugs with Inhibition Measurements
Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
---|---|---|---|---|---|
sitagliptin | Mus musculus (house mouse) | IC50 | 50.0230 | 2 | 2 |
2-ethyl-5-methoxy-n,n-dimethyltryptamine | Mus musculus (house mouse) | Ki | 0.0160 | 1 | 1 |
vildagliptin | Mus musculus (house mouse) | IC50 | 0.0510 | 1 | 1 |
ms-245 | Mus musculus (house mouse) | Ki | 0.0021 | 1 | 1 |
nvp-dpp728 | Mus musculus (house mouse) | IC50 | 0.0530 | 1 | 1 |
mk-3102 | Mus musculus (house mouse) | IC50 | 30.0000 | 1 | 1 |
Drugs with Activation Measurements
Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
---|---|---|---|---|---|
quinpirole | Mus musculus (house mouse) | EC50 | 0.0034 | 1 | 1 |