Page last updated: 2024-08-07 16:50:56
Beta-2 adrenergic receptor
A beta-2 adrenergic receptor that is encoded in the genome of dog. [OMA:P54833, PRO:DNx]
Synonyms
Beta-2 adrenoreceptor;
Beta-2 adrenoceptor
Research
Bioassay Publications (8)
| Timeframe | Studies on this Protein(%) | All Drugs % |
|---|---|---|
| pre-1990 | 1 (12.50) | 18.7374 |
| 1990's | 4 (50.00) | 18.2507 |
| 2000's | 3 (37.50) | 29.6817 |
| 2010's | 0 (0.00) | 24.3611 |
| 2020's | 0 (0.00) | 2.80 |
Compounds (17)
Drugs with Inhibition Measurements
| Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
|---|---|---|---|---|---|
| 1-(2-methoxyphenyl)piperazine | Canis lupus familiaris (dog) | IC50 | 34.0000 | 1 | 1 |
| 1-(3-chlorophenyl)piperazine | Canis lupus familiaris (dog) | IC50 | 18.0000 | 1 | 1 |
| 6-fluoronorepinephrine | Canis lupus familiaris (dog) | Ki | 58.0000 | 1 | 1 |
| isoproterenol | Canis lupus familiaris (dog) | IC50 | 0.6667 | 2 | 3 |
| naftopidil | Canis lupus familiaris (dog) | Ki | 1.0000 | 1 | 1 |
| propranolol | Canis lupus familiaris (dog) | IC50 | 0.0170 | 1 | 1 |
| sotalol | Canis lupus familiaris (dog) | IC50 | 5.0667 | 3 | 3 |
| phenylpiperazine | Canis lupus familiaris (dog) | IC50 | 100.0000 | 1 | 1 |
| 1-(4-nitrophenyl)piperazine | Canis lupus familiaris (dog) | IC50 | 56.0000 | 1 | 1 |
| 1-(4-chlorophenyl)piperazine | Canis lupus familiaris (dog) | IC50 | 70.0000 | 1 | 1 |
| 5-fluorodopamine | Canis lupus familiaris (dog) | Ki | 130.0000 | 1 | 1 |
| ersentilide | Canis lupus familiaris (dog) | IC50 | 46.5000 | 1 | 1 |
| 3-fluoronorepinephrine | Canis lupus familiaris (dog) | Ki | 0.1400 | 1 | 1 |
| 2-fluorodopamine | Canis lupus familiaris (dog) | Ki | 70.0000 | 1 | 1 |
| epitrate | Canis lupus familiaris (dog) | Ki | 3.7000 | 1 | 1 |
| 1-(4-methoxyphenyl)piperazine | Canis lupus familiaris (dog) | IC50 | 100.0000 | 1 | 1 |
Drugs with Activation Measurements
| Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
|---|---|---|---|---|---|
| practolol | Canis lupus familiaris (dog) | Kd | 0.1862 | 1 | 1 |