Assay ID | Title | Year | Journal | Article |
AID1347154 | Primary screen GU AMC qHTS for Zika virus inhibitors | 2020 | Proceedings of the National Academy of Sciences of the United States of America, 12-08, Volume: 117, Issue:49
| Therapeutic candidates for the Zika virus identified by a high-throughput screen for Zika protease inhibitors. |
AID1508630 | Primary qHTS for small molecule stabilizers of the endoplasmic reticulum resident proteome: Secreted ER Calcium Modulated Protein (SERCaMP) assay | 2021 | Cell reports, 04-27, Volume: 35, Issue:4
| A target-agnostic screen identifies approved drugs to stabilize the endoplasmic reticulum-resident proteome. |
AID1815474 | Activation of human carbonic anhydrase 1 by stopped flow assay | 2021 | European journal of medicinal chemistry, Dec-15, Volume: 226 | Binding site comparison for coumarin inhibitors and amine/amino acid activators of human carbonic anhydrases. |
AID691713 | Activity of human recombinant CA1 cytosolic isoform after 15 mins by phenol red staining based stopped flow CO2 hydration assay | 2012 | Bioorganic & medicinal chemistry letters, Oct-15, Volume: 22, Issue:20
| The first activation study of a bacterial carbonic anhydrase (CA). The thermostable α-CA from Sulfurihydrogenibium yellowstonense YO3AOP1 is highly activated by amino acids and amines. |
AID1815484 | Activation of human carbonic anhydrase 13 by stopped flow assay | 2021 | European journal of medicinal chemistry, Dec-15, Volume: 226 | Binding site comparison for coumarin inhibitors and amine/amino acid activators of human carbonic anhydrases. |
AID365577 | Activity of human recombinant CA2 at 10 uM stopped-flow CO2 hydration method | 2008 | Bioorganic & medicinal chemistry letters, Aug-01, Volume: 18, Issue:15
| Carbonic anhydrase activators: Activation of the human cytosolic isozyme III and membrane-associated isoform IV with amino acids and amines. |
AID1815485 | Activation of human carbonic anhydrase 14 by stopped flow CO2 hydrase assay | 2021 | European journal of medicinal chemistry, Dec-15, Volume: 226 | Binding site comparison for coumarin inhibitors and amine/amino acid activators of human carbonic anhydrases. |
AID1815483 | Activation of human carbonic anhydrase 12 by stopped flow assay | 2021 | European journal of medicinal chemistry, Dec-15, Volume: 226 | Binding site comparison for coumarin inhibitors and amine/amino acid activators of human carbonic anhydrases. |
AID1331204 | Activation of recombinant human carbonic anhydrase 2 at 10 uM incubated for 15 mins prior to testing by stopped flow CO2 hydration assay | 2017 | Bioorganic & medicinal chemistry letters, 01-01, Volume: 27, Issue:1
| Burkholderia pseudomallei γ-carbonic anhydrase is strongly activated by amino acids and amines. |
AID1815479 | Activation of human carbonic anhydrase 5B by stopped flow assay | 2021 | European journal of medicinal chemistry, Dec-15, Volume: 226 | Binding site comparison for coumarin inhibitors and amine/amino acid activators of human carbonic anhydrases. |
AID318345 | Activation of human recombinant CA9 catalytic domain by stopped-flow CO2 hydration method | 2008 | Bioorganic & medicinal chemistry, Apr-01, Volume: 16, Issue:7
| Carbonic anhydrase activators: activation of the human tumor-associated isozymes IX and XII with amino acids and amines. |
AID1397322 | Activation of Trypanosoma cruzi CA preincubated for 15 mins followed by CO2 addition by stopped-flow assay | | | |
AID365829 | Activation of human recombinant CA3 at 10 uM by stopped-flow CO2 hydration method | 2008 | Bioorganic & medicinal chemistry letters, Aug-01, Volume: 18, Issue:15
| Carbonic anhydrase activators: Activation of the human cytosolic isozyme III and membrane-associated isoform IV with amino acids and amines. |
AID458787 | Activation of Cryptococcus neoformans beta-carbonic anhydrase Can2 by stopped flow CO2 hydration assay | 2010 | Bioorganic & medicinal chemistry, Feb, Volume: 18, Issue:3
| Carbonic anhydrase activators: activation of the beta-carbonic anhydrases from the pathogenic fungi Candida albicans and Cryptococcus neoformans with amines and amino acids. |
AID725227 | Activation of Sulfurihydrogenibium yellowstonense recombinant CA by stopped flow CO2 hydrase method | 2013 | Bioorganic & medicinal chemistry letters, Feb-15, Volume: 23, Issue:4
| The extremo-α-carbonic anhydrase (CA) from Sulfurihydrogenibium azorense, the fastest CA known, is highly activated by amino acids and amines. |
AID1815475 | Activation of human carbonic anhydrase 2 by stopped flow assay | 2021 | European journal of medicinal chemistry, Dec-15, Volume: 226 | Binding site comparison for coumarin inhibitors and amine/amino acid activators of human carbonic anhydrases. |
AID1397319 | Activation of human CA1 by stopped-flow CO2 hydration assay | | | |
AID1398360 | Cis-inhibition of human LAT1 expressed in TREx HEK293 cells at 200 uM assessed as inhibition of [3H]-gabapentin uptake at 200 uM preincubated for 3 mins at 37 degC followed by washing with choline buffer and measured after 3 hrs by scintillation counting | 2018 | Journal of medicinal chemistry, 08-23, Volume: 61, Issue:16
| Reevaluating the Substrate Specificity of the L-Type Amino Acid Transporter (LAT1). |
AID691715 | Activity of Sulfurihydrogenibium yellowstonense YO3AOP1 recombinant CA expressed in Escherichia coli BL21(DE3) after 15 mins by phenol red staining based stopped flow CO2 hydration assay | 2012 | Bioorganic & medicinal chemistry letters, Oct-15, Volume: 22, Issue:20
| The first activation study of a bacterial carbonic anhydrase (CA). The thermostable α-CA from Sulfurihydrogenibium yellowstonense YO3AOP1 is highly activated by amino acids and amines. |
AID365578 | Activity of human recombinant CA3 at 10 uM stopped-flow CO2 hydration method | 2008 | Bioorganic & medicinal chemistry letters, Aug-01, Volume: 18, Issue:15
| Carbonic anhydrase activators: Activation of the human cytosolic isozyme III and membrane-associated isoform IV with amino acids and amines. |
AID365576 | Activity of human recombinant CA1 at 10 uM by stopped-flow CO2 hydration method | 2008 | Bioorganic & medicinal chemistry letters, Aug-01, Volume: 18, Issue:15
| Carbonic anhydrase activators: Activation of the human cytosolic isozyme III and membrane-associated isoform IV with amino acids and amines. |
AID458784 | Activation of Candida albicans beta-carbonic anhydrase Nce103 by stopped flow CO2 hydration assay | 2010 | Bioorganic & medicinal chemistry, Feb, Volume: 18, Issue:3
| Carbonic anhydrase activators: activation of the beta-carbonic anhydrases from the pathogenic fungi Candida albicans and Cryptococcus neoformans with amines and amino acids. |
AID291067 | Activation of of human recombinant CA14 by CO2 hydrase assay | 2007 | Bioorganic & medicinal chemistry letters, Aug-01, Volume: 17, Issue:15
| Carbonic anhydrase activators: activation of the human isoforms VII (cytosolic) and XIV (transmembrane) with amino acids and amines. |
AID365828 | Activation of human recombinant CA2 at 10 uM by stopped-flow CO2 hydration method | 2008 | Bioorganic & medicinal chemistry letters, Aug-01, Volume: 18, Issue:15
| Carbonic anhydrase activators: Activation of the human cytosolic isozyme III and membrane-associated isoform IV with amino acids and amines. |
AID409992 | Activation of Methanosarcina thermophila cobalt(2)-derived gamma-class CA by stopped-flow CO2 hydrase assay | 2008 | Bioorganic & medicinal chemistry letters, Dec-01, Volume: 18, Issue:23
| Carbonic anhydrase activators: activation of the archaeal beta-class (Cab) and gamma-class (Cam) carbonic anhydrases with amino acids and amines. |
AID318343 | Activation of human recombinant CA1 by stopped-flow CO2 hydration method | 2008 | Bioorganic & medicinal chemistry, Apr-01, Volume: 16, Issue:7
| Carbonic anhydrase activators: activation of the human tumor-associated isozymes IX and XII with amino acids and amines. |
AID725226 | Activation of Sulfurihydrogenibium azorense recombinant alpha carbonic anhydrase by stopped flow CO2 hydrase method | 2013 | Bioorganic & medicinal chemistry letters, Feb-15, Volume: 23, Issue:4
| The extremo-α-carbonic anhydrase (CA) from Sulfurihydrogenibium azorense, the fastest CA known, is highly activated by amino acids and amines. |
AID307897 | Activation of human recombinant CA2 by stopped flow CO2 hydrase method | 2007 | Bioorganic & medicinal chemistry, Aug-01, Volume: 15, Issue:15
| Carbonic anhydrase activators: the first activation study of the human secretory isoform VI with amino acids and amines. |
AID1815478 | Activation of human carbonic anhydrase 5A by stopped flow assay | 2021 | European journal of medicinal chemistry, Dec-15, Volume: 226 | Binding site comparison for coumarin inhibitors and amine/amino acid activators of human carbonic anhydrases. |
AID1398361 | Trans-stimulation of human LAT1 expressed in TREx HEK293 cells assessed as induction of [3H]-gabapentin efflux at 200 uM after 3 mins by scintillation counting analysis relative to L-phenylalanine | 2018 | Journal of medicinal chemistry, 08-23, Volume: 61, Issue:16
| Reevaluating the Substrate Specificity of the L-Type Amino Acid Transporter (LAT1). |
AID414330 | Activation of Methanothermobacter thermautotrophicus recombinant Cab by stopped-flow CO2 hydrase method | 2009 | Bioorganic & medicinal chemistry letters, Mar-15, Volume: 19, Issue:6
| Carbonic anhydrase activators: activation of the beta-carbonic anhydrase Nce103 from the yeast Saccharomyces cerevisiae with amines and amino acids. |
AID1397320 | Activation of human CA2 by stopped-flow CO2 hydration assay | | | |
AID462832 | Activation of Stylophora pistillata carbonic anhydrase STPCA by stopped flow CO2 hydration assay | 2010 | Bioorganic & medicinal chemistry, Mar-15, Volume: 18, Issue:6
| Carbonic anhydrase activators. The first activation study of a coral secretory isoform with amino acids and amines. |
AID198301 | Cleavage rate against hairpin ribozyme at 2 mM, in presence of 0.5 uM magnesium ions | 2001 | Bioorganic & medicinal chemistry letters, Dec-03, Volume: 11, Issue:23
| Novel spermine-amino acid conjugates and basic tripeptides enhance cleavage of the hairpin ribozyme at low magnesium ion concentration. |
AID375785 | Activity of membrane associated mouse recombinant carbonic anhydrase 15 isoform | 2009 | Bioorganic & medicinal chemistry letters, Jul-01, Volume: 19, Issue:13
| Carbonic anhydrase activators. Activation of the membrane-associated isoform XV with amino acids and amines. |
AID462831 | Activation of human full length CA6 by stopped flow CO2 hydration assay | 2010 | Bioorganic & medicinal chemistry, Mar-15, Volume: 18, Issue:6
| Carbonic anhydrase activators. The first activation study of a coral secretory isoform with amino acids and amines. |
AID1331206 | Activation of Burkholderia pseudomallei gamma carbonic anhydrase at 10 uM incubated for 15 mins prior to testing by stopped flow CO2 hydration assay | 2017 | Bioorganic & medicinal chemistry letters, 01-01, Volume: 27, Issue:1
| Burkholderia pseudomallei γ-carbonic anhydrase is strongly activated by amino acids and amines. |
AID1281543 | Activation of Malassezia globosa beta-carbonic anhydrase incubated for 15 mins prior to testing by stopped flow CO2 hydrase method | 2016 | Bioorganic & medicinal chemistry letters, Mar-01, Volume: 26, Issue:5
| Carbonic anhydrase activators: Activation of the β-carbonic anhydrase from Malassezia globosa with amines and amino acids. |
AID375786 | Activation of human recombinant carbonic anhydrase 4 lacking 20 amino terminal residues by stopped-flow CO2 hydrase method | 2009 | Bioorganic & medicinal chemistry letters, Jul-01, Volume: 19, Issue:13
| Carbonic anhydrase activators. Activation of the membrane-associated isoform XV with amino acids and amines. |
AID307896 | Activation of human recombinant CA1 by stopped flow CO2 hydrase method | 2007 | Bioorganic & medicinal chemistry, Aug-01, Volume: 15, Issue:15
| Carbonic anhydrase activators: the first activation study of the human secretory isoform VI with amino acids and amines. |
AID464319 | Activation of human recombinant carbonic anhydrase isoenzyme 2 by stopped flow CO2 hydration method | 2010 | Bioorganic & medicinal chemistry letters, Mar-01, Volume: 20, Issue:5
| Carbonic anhydrase activators: Activation of the beta-carbonic anhydrase from the pathogenic yeast Candida glabrata with amines and amino acids. |
AID414331 | Activation of yeast recombinant CA by stopped-flow CO2 hydrase method | 2009 | Bioorganic & medicinal chemistry letters, Mar-15, Volume: 19, Issue:6
| Carbonic anhydrase activators: activation of the beta-carbonic anhydrase Nce103 from the yeast Saccharomyces cerevisiae with amines and amino acids. |
AID409984 | Activation of human recombinant CA1 by stopped-flow CO2 hydrase assay | 2008 | Bioorganic & medicinal chemistry letters, Dec-01, Volume: 18, Issue:23
| Carbonic anhydrase activators: activation of the archaeal beta-class (Cab) and gamma-class (Cam) carbonic anhydrases with amino acids and amines. |
AID1397321 | Activation of Leishmania donovani chagasi CA preincubated for 15 mins followed by CO2 addition by stopped-flow assay | | | |
AID305777 | Activation of human recombinant carbonic anhydrase 5B by stopped-flow CO2 hydrase method | 2007 | Bioorganic & medicinal chemistry letters, Mar-01, Volume: 17, Issue:5
| Carbonic anhydrase activators: an activation study of the human mitochondrial isoforms VA and VB with amino acids and amines. |
AID1815477 | Activation of human carbonic anhydrase 4 by stopped flow assay | 2021 | European journal of medicinal chemistry, Dec-15, Volume: 226 | Binding site comparison for coumarin inhibitors and amine/amino acid activators of human carbonic anhydrases. |
AID365830 | Activation of human recombinant truncated CA4 at 10 uM by stopped-flow CO2 hydration method | 2008 | Bioorganic & medicinal chemistry letters, Aug-01, Volume: 18, Issue:15
| Carbonic anhydrase activators: Activation of the human cytosolic isozyme III and membrane-associated isoform IV with amino acids and amines. |
AID268622 | Activation of mouse recombinant CA13 by CO2 hydrase method | 2006 | Bioorganic & medicinal chemistry letters, Aug-01, Volume: 16, Issue:15
| Carbonic anhydrase activators: activation of isozyme XIII with amino acids and amines. |
AID409990 | Activation of Methanosarcina thermophila Zinc(2)-derived gamma-class CA by stopped-flow CO2 hydrase assay | 2008 | Bioorganic & medicinal chemistry letters, Dec-01, Volume: 18, Issue:23
| Carbonic anhydrase activators: activation of the archaeal beta-class (Cab) and gamma-class (Cam) carbonic anhydrases with amino acids and amines. |
AID318346 | Activation of human recombinant CA12 catalytic domain by stopped-flow CO2 hydration method | 2008 | Bioorganic & medicinal chemistry, Apr-01, Volume: 16, Issue:7
| Carbonic anhydrase activators: activation of the human tumor-associated isozymes IX and XII with amino acids and amines. |
AID365826 | Activity of human recombinant truncated CA4 at 10 uM stopped-flow CO2 hydration method | 2008 | Bioorganic & medicinal chemistry letters, Aug-01, Volume: 18, Issue:15
| Carbonic anhydrase activators: Activation of the human cytosolic isozyme III and membrane-associated isoform IV with amino acids and amines. |
AID268620 | Activation of human recombinant CA1 by CO2 hydrase assay | 2006 | Bioorganic & medicinal chemistry letters, Aug-01, Volume: 16, Issue:15
| Carbonic anhydrase activators: activation of isozyme XIII with amino acids and amines. |
AID464322 | Activation of Candida glabrata recombinant carbonic anhydrase by stopped flow CO2 hydration method | 2010 | Bioorganic & medicinal chemistry letters, Mar-01, Volume: 20, Issue:5
| Carbonic anhydrase activators: Activation of the beta-carbonic anhydrase from the pathogenic yeast Candida glabrata with amines and amino acids. |
AID1331203 | Activation of recombinant human carbonic anhydrase 1 at 10 uM incubated for 15 mins prior to testing by stopped flow CO2 hydration assay | 2017 | Bioorganic & medicinal chemistry letters, 01-01, Volume: 27, Issue:1
| Burkholderia pseudomallei γ-carbonic anhydrase is strongly activated by amino acids and amines. |
AID1815481 | Activation of human carbonic anhydrase 7 by stopped flow assay | 2021 | European journal of medicinal chemistry, Dec-15, Volume: 226 | Binding site comparison for coumarin inhibitors and amine/amino acid activators of human carbonic anhydrases. |
AID464321 | Activation of Saccharomyces cerevisiae recombinant Nce103p by stopped flow CO2 hydration method | 2010 | Bioorganic & medicinal chemistry letters, Mar-01, Volume: 20, Issue:5
| Carbonic anhydrase activators: Activation of the beta-carbonic anhydrase from the pathogenic yeast Candida glabrata with amines and amino acids. |
AID691714 | Activity of human recombinant CA2 cytosolic isoform after 15 mins by phenol red staining based stopped flow CO2 hydration assay | 2012 | Bioorganic & medicinal chemistry letters, Oct-15, Volume: 22, Issue:20
| The first activation study of a bacterial carbonic anhydrase (CA). The thermostable α-CA from Sulfurihydrogenibium yellowstonense YO3AOP1 is highly activated by amino acids and amines. |
AID1815476 | Activation of human carbonic anhydrase 3 by stopped flow assay | 2021 | European journal of medicinal chemistry, Dec-15, Volume: 226 | Binding site comparison for coumarin inhibitors and amine/amino acid activators of human carbonic anhydrases. |
AID409988 | Activation of Methanobacterium thermoautotrophicum beta-class CA by stopped-flow CO2 hydrase assay | 2008 | Bioorganic & medicinal chemistry letters, Dec-01, Volume: 18, Issue:23
| Carbonic anhydrase activators: activation of the archaeal beta-class (Cab) and gamma-class (Cam) carbonic anhydrases with amino acids and amines. |
AID307898 | Activation of human recombinant CA6 by stopped flow CO2 hydrase method | 2007 | Bioorganic & medicinal chemistry, Aug-01, Volume: 15, Issue:15
| Carbonic anhydrase activators: the first activation study of the human secretory isoform VI with amino acids and amines. |
AID291063 | Activation of human recombinant CA2 by CO2 hydrase assay | 2007 | Bioorganic & medicinal chemistry letters, Aug-01, Volume: 17, Issue:15
| Carbonic anhydrase activators: activation of the human isoforms VII (cytosolic) and XIV (transmembrane) with amino acids and amines. |
AID291061 | Activation of human recombinant CA1 by CO2 hydrase assay | 2007 | Bioorganic & medicinal chemistry letters, Aug-01, Volume: 17, Issue:15
| Carbonic anhydrase activators: activation of the human isoforms VII (cytosolic) and XIV (transmembrane) with amino acids and amines. |
AID291065 | Activation of human recombinant CA7 by CO2 hydrase assay | 2007 | Bioorganic & medicinal chemistry letters, Aug-01, Volume: 17, Issue:15
| Carbonic anhydrase activators: activation of the human isoforms VII (cytosolic) and XIV (transmembrane) with amino acids and amines. |
AID268621 | Activation of human recombinant CA2 by CO2 hydrase assay | 2006 | Bioorganic & medicinal chemistry letters, Aug-01, Volume: 16, Issue:15
| Carbonic anhydrase activators: activation of isozyme XIII with amino acids and amines. |
AID725229 | Activation of human recombinant CA2 by stopped flow CO2 hydrase method | 2013 | Bioorganic & medicinal chemistry letters, Feb-15, Volume: 23, Issue:4
| The extremo-α-carbonic anhydrase (CA) from Sulfurihydrogenibium azorense, the fastest CA known, is highly activated by amino acids and amines. |
AID725228 | Activation of human recombinant CA1 by stopped flow CO2 hydrase method | 2013 | Bioorganic & medicinal chemistry letters, Feb-15, Volume: 23, Issue:4
| The extremo-α-carbonic anhydrase (CA) from Sulfurihydrogenibium azorense, the fastest CA known, is highly activated by amino acids and amines. |
AID1331205 | Activation of recombinant Methanosarcina thermophila gamma carbonic anhydrase at 10 uM incubated for 15 mins prior to testing by stopped flow CO2 hydration assay | 2017 | Bioorganic & medicinal chemistry letters, 01-01, Volume: 27, Issue:1
| Burkholderia pseudomallei γ-carbonic anhydrase is strongly activated by amino acids and amines. |
AID462830 | Activation of human recombinant CA2by stopped flow CO2 hydration assay | 2010 | Bioorganic & medicinal chemistry, Mar-15, Volume: 18, Issue:6
| Carbonic anhydrase activators. The first activation study of a coral secretory isoform with amino acids and amines. |
AID1398359 | Cis-inhibition of human LAT1 expressed in TREx HEK293 cells at 200 uM assessed as inhibition of [3H]-gabapentin uptake preincubated for 3 mins at 37 degC followed by washing with choline buffer and measured after 3 hrs by scintillation counting analysis r | 2018 | Journal of medicinal chemistry, 08-23, Volume: 61, Issue:16
| Reevaluating the Substrate Specificity of the L-Type Amino Acid Transporter (LAT1). |
AID375784 | Activity of human recombinant carbonic anhydrase 4 lacking 20 amino terminal residues | 2009 | Bioorganic & medicinal chemistry letters, Jul-01, Volume: 19, Issue:13
| Carbonic anhydrase activators. Activation of the membrane-associated isoform XV with amino acids and amines. |
AID462829 | Activation of human recombinant CA1 by stopped flow CO2 hydration assay | 2010 | Bioorganic & medicinal chemistry, Mar-15, Volume: 18, Issue:6
| Carbonic anhydrase activators. The first activation study of a coral secretory isoform with amino acids and amines. |
AID305776 | Activation of human recombinant carbonic anhydrase 5A by stopped-flow CO2 hydrase method | 2007 | Bioorganic & medicinal chemistry letters, Mar-01, Volume: 17, Issue:5
| Carbonic anhydrase activators: an activation study of the human mitochondrial isoforms VA and VB with amino acids and amines. |
AID1815482 | Activation of human carbonic anhydrase 9 by stopped flow assay | 2021 | European journal of medicinal chemistry, Dec-15, Volume: 226 | Binding site comparison for coumarin inhibitors and amine/amino acid activators of human carbonic anhydrases. |
AID1331210 | Activation of Burkholderia pseudomallei gamma carbonic anhydrase assessed as Kcat at 10 uM incubated for 15 mins prior to testing by stopped flow CO2 hydration assay | 2017 | Bioorganic & medicinal chemistry letters, 01-01, Volume: 27, Issue:1
| Burkholderia pseudomallei γ-carbonic anhydrase is strongly activated by amino acids and amines. |
AID409986 | Activation of human recombinant CA2 by stopped-flow CO2 hydrase assay | 2008 | Bioorganic & medicinal chemistry letters, Dec-01, Volume: 18, Issue:23
| Carbonic anhydrase activators: activation of the archaeal beta-class (Cab) and gamma-class (Cam) carbonic anhydrases with amino acids and amines. |
AID464320 | Activation of archaea Methanobacterium thermoautotrophicum recombinant carbonic anhydrase by stopped flow CO2 hydration method | 2010 | Bioorganic & medicinal chemistry letters, Mar-01, Volume: 20, Issue:5
| Carbonic anhydrase activators: Activation of the beta-carbonic anhydrase from the pathogenic yeast Candida glabrata with amines and amino acids. |
AID365827 | Activation of human recombinant CA1 at 10 uM by stopped-flow CO2 hydration method | 2008 | Bioorganic & medicinal chemistry letters, Aug-01, Volume: 18, Issue:15
| Carbonic anhydrase activators: Activation of the human cytosolic isozyme III and membrane-associated isoform IV with amino acids and amines. |
AID318344 | Activation of human recombinant CA2 by stopped-flow CO2 hydration method | 2008 | Bioorganic & medicinal chemistry, Apr-01, Volume: 16, Issue:7
| Carbonic anhydrase activators: activation of the human tumor-associated isozymes IX and XII with amino acids and amines. |
AID375787 | Activation of membrane associated mouse recombinant carbonic anhydrase 15 isoform by stopped-flow CO2 hydrase method | 2009 | Bioorganic & medicinal chemistry letters, Jul-01, Volume: 19, Issue:13
| Carbonic anhydrase activators. Activation of the membrane-associated isoform XV with amino acids and amines. |
AID409993 | Activation of human recombinant CA3 by stopped-flow CO2 hydrase assay | 2008 | Bioorganic & medicinal chemistry letters, Dec-01, Volume: 18, Issue:23
| Carbonic anhydrase activators: activation of the archaeal beta-class (Cab) and gamma-class (Cam) carbonic anhydrases with amino acids and amines. |
AID414329 | Activation of human recombinant CA2 by stopped-flow CO2 hydrase method | 2009 | Bioorganic & medicinal chemistry letters, Mar-15, Volume: 19, Issue:6
| Carbonic anhydrase activators: activation of the beta-carbonic anhydrase Nce103 from the yeast Saccharomyces cerevisiae with amines and amino acids. |
AID1815480 | Activation of human carbonic anhydrase 6 by stopped flow assay | 2021 | European journal of medicinal chemistry, Dec-15, Volume: 226 | Binding site comparison for coumarin inhibitors and amine/amino acid activators of human carbonic anhydrases. |
AID198302 | Cleavage rate against hairpin ribozyme at 5 mM with 0.5 uM magnesium ions | 2001 | Bioorganic & medicinal chemistry letters, Dec-03, Volume: 11, Issue:23
| Novel spermine-amino acid conjugates and basic tripeptides enhance cleavage of the hairpin ribozyme at low magnesium ion concentration. |
AID977611 | Experimentally measured binding affinity data (Kd) for protein-ligand complexes derived from PDB | 2006 | Chemistry (Weinheim an der Bergstrasse, Germany), Sep-18, Volume: 12, Issue:27
| Carbonic anhydrase activators. Activation of isozymes I, II, IV, VA, VII, and XIV with l- and d-histidine and crystallographic analysis of their adducts with isoform II: engineering proton-transfer processes within the active site of an enzyme. |
AID1811 | Experimentally measured binding affinity data derived from PDB | 2006 | Chemistry (Weinheim an der Bergstrasse, Germany), Sep-18, Volume: 12, Issue:27
| Carbonic anhydrase activators. Activation of isozymes I, II, IV, VA, VII, and XIV with l- and d-histidine and crystallographic analysis of their adducts with isoform II: engineering proton-transfer processes within the active site of an enzyme. |
[information is prepared from bioassay data collected from National Library of Medicine (NLM), extracted Dec-2023] |