| Member | Definition | Class |
|---|
| (E,E)-1-bromo-2,5-bis-(4-hydroxystyryl)benzene | An organobromine compound that is bromobenzene in which the hydrogens at positions 2 and 5 are replaced by 4-hydroxystyryl groups. | (E,E)-1-bromo-2,5-bis-(4-hydroxystyryl)benzene |
| aminacrine | An aminoacridine that is acridine in which the hydrogen at position 9 is replaced by an amino group. A fluorescent dyd and topical antiseptic agent, it is used (usually as the hydrochloride salt) in eye drops for the treatment of superficial eye infections. | 9-aminoacridine |
| coumarin | A chromenone having the keto group located at the 2-position. | coumarin |
| eosine i bluish | An organic sodium salt which is the disodium salt of eosin b diphenol. | eosin b |
| fluorescein | A xanthene dye that is highly fluorescent, detectable even when present in minute quantities. Used forensically to detect traces of blood, in analytical chemistry as an indicator in silver nitrate titrations and in microscopy. | fluorescein (lactone form) |
| fluorescite | A xanthene dye that is highly fluorescent and commonly used as a fluorescent tracer. | fluorescein (acid form) |
| n-(4-(7-diethylamino-4-methylcoumarin-3-yl)phenyl)maleimide | A member of the class of coumarins that is 2H-chromen-2-one substituted by 4-(2,5-dioxo-2,5-dihydro-1H-pyrrol-1-yl)phenyl, methyl, and diethylamino groups at positions 3, 4 and 7, respectively. It is a thiol-reactive fluorescent dye. | 7-diethylamino-3-(4-maleimidophenyl)-4-methylcoumarin |
| picogreen | A cyanine dye that is 1-phenylquinoline which is substituted at position 2 by a bis[3-(dimethylamino)propyl]amino group and at position 4 by a (3-methyl-1,3-benzothiazol-3-ium-2-yl)methylene group. The counter ion is not stated. A fluorochrome that selectively binds double-stranded DNA and has characteristics similar to that of SYBR-Green I. | PicoGreen |
| sybr green i | A benzothiazolium ion resulting from the methylation of the nitrogen of the benzothiazole group of N-[4-(1,3-benzothiazol-2-ylmethylene)-1-phenyl-1,4-dihydroquinolin-2-yl]-N',N'-dimethyl-N-propylpropane-1,3-diamine. A cationic unsymmetrical cyanine dye that binds to double-stranded DNA and is used as a nucleic acid stain in molecular biology. | SYBR Green I |
| Protein | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Drugs |
|---|
| 15-hydroxyprostaglandin dehydrogenase [NAD(+)] isoform 1 | Homo sapiens (human) | Potency | 22.0164 | 1 | 2 |
| 67.9K protein | Vaccinia virus | Potency | 28.1838 | 2 | 2 |
| acetylcholinesterase | Homo sapiens (human) | Potency | 0.5638 | 1 | 1 |
| activating transcription factor 6 | Homo sapiens (human) | Potency | 41.2434 | 2 | 2 |
| aldehyde dehydrogenase 1 family, member A1 | Homo sapiens (human) | Potency | 28.1838 | 1 | 1 |
| alpha-galactosidase | Homo sapiens (human) | Potency | 40.0748 | 2 | 2 |
| Amyloid-beta precursor protein | Homo sapiens (human) | Potency | 29.0929 | 1 | 1 |
| AR protein | Homo sapiens (human) | Potency | 109.1875 | 7 | 11 |
| aryl hydrocarbon receptor | Homo sapiens (human) | Potency | 21.6899 | 1 | 1 |
| arylsulfatase A | Homo sapiens (human) | Potency | 19.0115 | 1 | 1 |
| Ataxin-2 | Homo sapiens (human) | Potency | 28.1838 | 1 | 1 |
| ATP-dependent phosphofructokinase | Trypanosoma brucei brucei TREU927 | Potency | 33.8078 | 1 | 1 |
| atrial natriuretic peptide receptor 1 precursor | Homo sapiens (human) | Potency | 8.4921 | 1 | 1 |
| Bloom syndrome protein isoform 1 | Homo sapiens (human) | Potency | 29.8304 | 1 | 3 |
| caspase-1 isoform alpha precursor | Homo sapiens (human) | Potency | 15.8489 | 1 | 1 |
| Caspase-7 | Homo sapiens (human) | Potency | 12.5893 | 1 | 1 |
| Cellular tumor antigen p53 | Homo sapiens (human) | Potency | 38.1818 | 2 | 3 |
| Chain A, 2-oxoglutarate Oxygenase | Homo sapiens (human) | Potency | 31.6228 | 1 | 1 |
| Chain A, ATP-DEPENDENT DNA HELICASE Q1 | Homo sapiens (human) | Potency | 54.5326 | 3 | 5 |
| Chain A, Beta-lactamase | Escherichia coli K-12 | Potency | 112.2020 | 1 | 1 |
| Chain A, Cruzipain | Trypanosoma cruzi | Potency | 11.2202 | 1 | 1 |
| Chain A, Ferritin light chain | Equus caballus (horse) | Potency | 34.5167 | 1 | 4 |
| Chain A, HADH2 protein | Homo sapiens (human) | Potency | 31.6228 | 1 | 1 |
| Chain A, MAJOR APURINIC/APYRIMIDINIC ENDONUCLEASE | Homo sapiens (human) | Potency | 29.9033 | 1 | 2 |
| Chain A, TYROSYL-DNA PHOSPHODIESTERASE | Homo sapiens (human) | Potency | 17.1269 | 1 | 5 |
| Chain B, HADH2 protein | Homo sapiens (human) | Potency | 31.6228 | 1 | 1 |
| chromobox protein homolog 1 | Homo sapiens (human) | Potency | 79.4328 | 1 | 1 |
| DNA polymerase iota isoform a (long) | Homo sapiens (human) | Potency | 0.6310 | 1 | 1 |
| DNA polymerase kappa isoform 1 | Homo sapiens (human) | Potency | 29.9650 | 1 | 4 |
| estrogen nuclear receptor alpha | Homo sapiens (human) | Potency | 133.3995 | 5 | 10 |
| estrogen receptor 2 (ER beta) | Homo sapiens (human) | Potency | 54.4827 | 2 | 2 |
| estrogen-related nuclear receptor alpha | Homo sapiens (human) | Potency | 12.2910 | 5 | 5 |
| euchromatic histone-lysine N-methyltransferase 2 | Homo sapiens (human) | Potency | 15.5962 | 1 | 2 |
| farnesoid X nuclear receptor | Homo sapiens (human) | Potency | 177.0229 | 4 | 4 |
| GALC protein | Homo sapiens (human) | Potency | 0.6310 | 1 | 2 |
| GLS protein | Homo sapiens (human) | Potency | 7.0795 | 1 | 1 |
| glucocorticoid receptor [Homo sapiens] | Homo sapiens (human) | Potency | 25.9743 | 4 | 7 |
| heat shock 70kDa protein 5 (glucose-regulated protein, 78kDa) | Homo sapiens (human) | Potency | 23.3383 | 1 | 2 |
| heat shock protein beta-1 | Homo sapiens (human) | Potency | 29.9758 | 2 | 2 |
| Histamine H2 receptor | Cavia porcellus (domestic guinea pig) | Potency | 28.1838 | 1 | 2 |
| histone acetyltransferase KAT2A isoform 1 | Homo sapiens (human) | Potency | 30.4765 | 1 | 3 |
| histone-lysine N-methyltransferase 2A isoform 2 precursor | Homo sapiens (human) | Potency | 79.4328 | 1 | 1 |
| huntingtin isoform 2 | Homo sapiens (human) | Potency | 0.0316 | 1 | 1 |
| hypoxia-inducible factor 1 alpha subunit | Homo sapiens (human) | Potency | 43.6465 | 1 | 1 |
| lamin isoform A-delta10 | Homo sapiens (human) | Potency | 0.7943 | 1 | 1 |
| Microtubule-associated protein tau | Homo sapiens (human) | Potency | 0.4929 | 1 | 2 |
| muscleblind-like protein 1 isoform 1 | Homo sapiens (human) | Potency | 1.0000 | 1 | 1 |
| NPC intracellular cholesterol transporter 1 precursor | Homo sapiens (human) | Potency | 3.6626 | 1 | 1 |
| nuclear factor erythroid 2-related factor 2 isoform 1 | Homo sapiens (human) | Potency | 373.1428 | 4 | 5 |
| nuclear factor of kappa light polypeptide gene enhancer in B-cells 1 (p105), isoform CRA_a | Homo sapiens (human) | Potency | 48.9722 | 1 | 1 |
| nuclear receptor ROR-gamma isoform 1 | Mus musculus (house mouse) | Potency | 11.2202 | 1 | 1 |
| nuclear receptor subfamily 1, group I, member 2 | Rattus norvegicus (Norway rat) | Potency | 35.4813 | 1 | 1 |
| Parkin | Homo sapiens (human) | Potency | 23.7246 | 2 | 2 |
| peripheral myelin protein 22 | Rattus norvegicus (Norway rat) | Potency | 11.2079 | 2 | 2 |
| peroxisome proliferator activated receptor gamma | Homo sapiens (human) | Potency | 25.9850 | 3 | 5 |
| peroxisome proliferator-activated receptor delta | Homo sapiens (human) | Potency | 26.1014 | 3 | 3 |
| Polyunsaturated fatty acid lipoxygenase ALOX15B | Homo sapiens (human) | Potency | 28.1838 | 1 | 1 |
| pregnane X nuclear receptor | Homo sapiens (human) | Potency | 640.3100 | 2 | 2 |
| pregnane X receptor | Rattus norvegicus (Norway rat) | Potency | 1,412.5400 | 1 | 1 |
| progesterone receptor | Homo sapiens (human) | Potency | 54.4827 | 2 | 2 |
| regulator of G-protein signaling 4 | Homo sapiens (human) | Potency | 21.1923 | 1 | 1 |
| retinoic acid nuclear receptor alpha variant 1 | Homo sapiens (human) | Potency | 76.9588 | 1 | 1 |
| retinoid X nuclear receptor alpha | Homo sapiens (human) | Potency | 20.0731 | 2 | 3 |
| serine/threonine-protein kinase mTOR isoform 1 | Homo sapiens (human) | Potency | 18.4927 | 1 | 1 |
| SMAD family member 2 | Homo sapiens (human) | Potency | 35.5964 | 3 | 3 |
| SMAD family member 3 | Homo sapiens (human) | Potency | 35.5964 | 3 | 3 |
| survival motor neuron protein isoform d | Homo sapiens (human) | Potency | 35.4813 | 1 | 1 |
| TDP1 protein | Homo sapiens (human) | Potency | 3.4634 | 2 | 2 |
| thioredoxin reductase | Rattus norvegicus (Norway rat) | Potency | 19.7119 | 4 | 4 |
| thyroid hormone receptor beta isoform 2 | Rattus norvegicus (Norway rat) | Potency | 51.0530 | 2 | 2 |
| thyroid hormone receptor beta isoform a | Homo sapiens (human) | Potency | 0.0089 | 1 | 1 |
| thyrotropin-releasing hormone receptor | Homo sapiens (human) | Potency | 0.3455 | 2 | 2 |
| USP1 protein, partial | Homo sapiens (human) | Potency | 52.4870 | 2 | 2 |
| v-jun sarcoma virus 17 oncogene homolog (avian) | Homo sapiens (human) | Potency | 34.0954 | 2 | 2 |
| vitamin D (1,25- dihydroxyvitamin D3) receptor | Homo sapiens (human) | Potency | 26.9577 | 3 | 4 |