Page last updated: 2024-08-05 15:03:14

orphan drug

Any drug that has been developed specifically for treatment of a rare medical condition, the condition itself being known as an orphan disease.

ChEBI ID: 71031

Members (13)

MemberDefinitionClass
4-aminopyridineAn aromatic amine that is pyridine bearing a single amino substituent at position 4. An orphan drug in the US, it is used to improve walking in adults with multiple sclerosis.4-aminopyridine
4-phenylbutyric acid, sodium saltThe organic sodium salt of 4-phenylbutyric acid. A prodrug for phenylacetate, it is used to treat urea cycle disorders.sodium phenylbutyrate
carglumic acidA urea that is the N-carbamoyl derivative of L-glutamic acid. An orphan drug used to treat a deficiency in the enzyme N-acetylglutamate synthase, which leads to acute hyperammonaemia.carglumic acid
isavuconazoleA 1,3-thiazole that is butan-2-ol which is substituted at positions 1, 2, and 3 by 1,2,4-triazol-1-yl, 2,5-difluorophenyl, and 4-(p-cyanophenyl)-1,3-thiazol-2-yl groups, respectively. It is an antifungal drug used for the treatment of invasive aspergillosis and invasive mucormycosis.isavuconazole
ixazomibA glycine derivative that is the amide obtained by formal condensation of the carboxy group of N-(2,5-dichlorobenzoyl)glycine with the amino group of [(1R)-1-amino-3-methylbutyl]boronic acid. The active metabolite of ixazomib citrate, it is used in combination therapy for treatment of multiple myeloma.ixazomib
lenvatinibA member of the class of quinolines that is the carboxamide of 4-{3-chloro-4-[(cyclopropylcarbamoyl)amino]phenoxy}-7-methoxyquinoline-6-carboxylic acid. A multi-kinase inhibitor and orphan drug used (as its mesylate salt) for the treatment of various types of thyroid cancer that do not respond to radioiodine.lenvatinib
lumacaftorAn aromatic amide obtained by formal condensation of the carboxy group of 1-(2,2-difluoro-1,3-benzodioxol-5-yl)cyclopropane-1-carboxylic acid with the aromatic amino group of 3-(6-amino-3-methylpyridin-2-yl)benzoic acid. Used for the treatment of cystic fibrosis.lumacaftor
macitentanA member of the class of sulfamides in which the two amino groups of sulfonamide are substituted by 5-(4-bromophenyl)-6-{2-[(5-bromopyrimidin-2-yl)oxy]ethoxy}pyrimidin-4-yl and propyl groups. An orphan drug used for the treatment of pulmonary arterial hypertension.macitentan
mre 269A member of the class of pyrazines that is {4-[(propan-2-yl)(pyrazin-2-yl)amino]butoxy}acetic acid carrying two additional phenyl substituents at positions 5 and 6 on the pyrazine ring. The active metabolite of selexipag, an orphan drug used for the treatment of pulmonary arterial hypertension.ACT-333679
pn 401An acetate ester that is uracil in which the three hydroxy hydrogens are replaced by acetate group. A prodrug for uridine, it is used for the treatment of hereditary orotic aciduria and for management of fluorouracil toxicity.uridine triacetate
rifaximinA semisynthetic member of the class of rifamycins and non-systemic gastrointestinal site-specific broad spectrum antibiotic. Used in the treatment of traveller's diarrhoea, hepatic encephalopathy and irritable bowel syndrome.rifaximin
selexipagA member of the class of pyrazines that is N-(methanesulfonyl)-2-{4-[(propan-2-yl)(pyrazin-2-yl)amino]butoxy}acetamide carrying two additional phenyl substituents at positions 5 and 6 on the pyrazine ring. An orphan drug used for the treatment of pulmonary arterial hypertension. It is a prodrug for ACT-333679 (the free carboxylic acid).selexipag
vx-770An aromatic amide obtained by formal condensation of the carboxy group of 4-oxo-1,4-dihydroquinoline-3-carboxylic acid with the amino group of 5-amino-2,4-di-tert-butylphenol. Used for the treatment of cystic fibrosis.ivacaftor

Research

Studies (6,975)

TimeframeStudies, Drugs with This Role(%)All Drugs %
pre-1990708 (10.15)18.7374
1990's1,320 (18.92)18.2507
2000's1,183 (16.96)29.6817
2010's2,217 (31.78)24.3611
2020's1,547 (22.18)2.80

Study Types

Publication TypeStudies, Drugs with this Role (%)All Drugs (%)
Trials527 (7.11%)5.53%
Reviews638 (8.60%)6.00%
Case Studies483 (6.51%)4.05%
Observational95 (1.28%)0.25%
Other5,674 (76.50%)84.16%

Protein Targets (399)

Potency Measurements

ProteinTaxonomyMeasurementAverage (mM)Bioassay(s)Drugs
aldehyde dehydrogenase 1 family, member A1Homo sapiens (human)Potency44.668411
ATP-dependent phosphofructokinaseTrypanosoma brucei brucei TREU927Potency0.756911
Cellular tumor antigen p53Homo sapiens (human)Potency13.333211
Chain A, CruzipainTrypanosoma cruziPotency3.355222
Chain A, MAJOR APURINIC/APYRIMIDINIC ENDONUCLEASEHomo sapiens (human)Potency1,995.260011
chromobox protein homolog 1Homo sapiens (human)Potency68.842922
cytochrome P450 2C9, partialHomo sapiens (human)Potency16.458214
cytochrome P450 2D6Homo sapiens (human)Potency26.689714
cytochrome P450 2D6 isoform 1Homo sapiens (human)Potency0.063111
cytochrome P450 family 3 subfamily A polypeptide 4Homo sapiens (human)Potency15.914816
estrogen receptor 2 (ER beta)Homo sapiens (human)Potency61.628211
euchromatic histone-lysine N-methyltransferase 2Homo sapiens (human)Potency0.022411
EWS/FLI fusion proteinHomo sapiens (human)Potency0.4001412
Fumarate hydrataseHomo sapiens (human)Potency18.724314
GVesicular stomatitis virusPotency16.458214
GALC proteinHomo sapiens (human)Potency0.631011
gemininHomo sapiens (human)Potency6.309611
GLI family zinc finger 3Homo sapiens (human)Potency13.333211
glucocerebrosidaseHomo sapiens (human)Potency0.631011
glucocorticoid receptor [Homo sapiens]Homo sapiens (human)Potency7.079511
HLA class I histocompatibility antigen, B alpha chain Homo sapiens (human)Potency16.458214
IDH1Homo sapiens (human)Potency29.092911
Inositol hexakisphosphate kinase 1Homo sapiens (human)Potency16.458218
Interferon betaHomo sapiens (human)Potency13.5110213
lamin isoform A-delta10Homo sapiens (human)Potency0.891311
lethal factor (plasmid)Bacillus anthracis str. A2012Potency7.943311
Microtubule-associated protein tauHomo sapiens (human)Potency8.912511
mitogen-activated protein kinase 1Homo sapiens (human)Potency10.000011
nuclear factor of kappa light polypeptide gene enhancer in B-cells 1 (p105), isoform CRA_aHomo sapiens (human)Potency49.397911
peripheral myelin protein 22Rattus norvegicus (Norway rat)Potency25.099911
polyproteinZika virusPotency18.724314
PPM1D proteinHomo sapiens (human)Potency12.201116
Rap guanine nucleotide exchange factor 3Homo sapiens (human)Potency28.183811
RAR-related orphan receptor gammaMus musculus (house mouse)Potency17.051524
Spike glycoproteinSevere acute respiratory syndrome-related coronavirusPotency19.959928
survival motor neuron protein isoform dHomo sapiens (human)Potency1.000012
thioredoxin reductaseRattus norvegicus (Norway rat)Potency89.125122
thyroid hormone receptor beta isoform 2Rattus norvegicus (Norway rat)Potency77.585411
thyroid stimulating hormone receptorHomo sapiens (human)Potency0.125911
transcriptional regulator ERG isoform 3Homo sapiens (human)Potency2.818411
tyrosine-protein kinase YesHomo sapiens (human)Potency3.449911
USP1 protein, partialHomo sapiens (human)Potency14.125411

Inhibition Measurements

ProteinTaxonomyMeasurementAverage (mM)Bioassay(s)Drugs
AcetylcholinesteraseRattus norvegicus (Norway rat)IC50500.000012
ATP-binding cassette sub-family C member 3Homo sapiens (human)IC5065.000011
ATP-dependent Clp protease proteolytic subunitStaphylococcus aureus subsp. aureus NCTC 8325IC505.300011
Bile salt export pumpHomo sapiens (human)IC5042.000011
Broad substrate specificity ATP-binding cassette transporter ABCG2Homo sapiens (human)IC5011.000011
Canalicular multispecific organic anion transporter 1Homo sapiens (human)IC5015.400011
Carbonic anhydrase 1Homo sapiens (human)Ki10.000011
Carbonic anhydrase 2Homo sapiens (human)Ki10.000011
Carbonic anhydrase 5A, mitochondrialHomo sapiens (human)Ki0.132711
Coiled-coil domain-containing protein 6Homo sapiens (human)IC500.010011
Cytochrome P450 1A2Homo sapiens (human)IC5020.000011
Cytochrome P450 2C19Homo sapiens (human)IC5020.000011
Cytochrome P450 2C8Homo sapiens (human)IC5012.000011
Cytochrome P450 2C9 Homo sapiens (human)IC5026.000022
Cytochrome P450 2D6Homo sapiens (human)IC5020.000022
Cytochrome P450 2E1Homo sapiens (human)IC5020.000011
Cytochrome P450 3A4Homo sapiens (human)IC5020.000011
Endothelin receptor type BHomo sapiens (human)IC500.589733
Endothelin receptor type BRattus norvegicus (Norway rat)IC500.391011
Endothelin-1 receptorHomo sapiens (human)IC500.001533
Histone deacetylase 1Homo sapiens (human)IC50162.000011
Histone deacetylase 1Homo sapiens (human)Ki6.340011
Histone deacetylase 11 Homo sapiens (human)Ki6.340011
Histone deacetylase 2Homo sapiens (human)Ki6.340011
Histone deacetylase 3Homo sapiens (human)Ki6.340011
Histone deacetylase 4Homo sapiens (human)Ki6.340011
Histone deacetylase 5Homo sapiens (human)Ki6.340011
Histone deacetylase 6Homo sapiens (human)Ki6.340011
Histone deacetylase 7Homo sapiens (human)Ki6.340011
Histone deacetylase 8Homo sapiens (human)Ki6.340011
Histone deacetylase 9Homo sapiens (human)Ki6.340011
Kinesin-1 heavy chainHomo sapiens (human)IC500.010011
Multidrug resistance-associated protein 4Homo sapiens (human)IC5030.200011
NACHT, LRR and PYD domains-containing protein 3 Mus musculus (house mouse)IC500.199511
Nuclear receptor coactivator 4Homo sapiens (human)IC500.010011
Platelet-derived growth factor receptor alphaHomo sapiens (human)IC500.051011
Platelet-derived growth factor receptor betaHomo sapiens (human)IC500.039011
Polyamine deacetylase HDAC10Homo sapiens (human)Ki6.340011
Potassium voltage-gated channel subfamily A member 1Homo sapiens (human)IC5089.000011
Potassium voltage-gated channel subfamily H member 2Homo sapiens (human)IC504,382.580022
Prostacyclin receptorHomo sapiens (human)IC500.175012
Proteasome subunit alpha type-1Homo sapiens (human)IC500.015011
Proteasome subunit alpha type-2Homo sapiens (human)IC500.015011
Proteasome subunit alpha type-3Homo sapiens (human)IC500.015011
Proteasome subunit alpha type-4Homo sapiens (human)IC500.015011
Proteasome subunit alpha type-5Homo sapiens (human)IC500.015011
Proteasome subunit alpha type-6Homo sapiens (human)IC500.015011
Proteasome subunit alpha type-7Homo sapiens (human)IC500.015011
Proteasome subunit alpha-type 8Homo sapiens (human)IC500.015011
Proteasome subunit beta type-1Homo sapiens (human)IC500.016333
Proteasome subunit beta type-10Homo sapiens (human)IC500.015011
Proteasome subunit beta type-11Homo sapiens (human)IC500.015011
Proteasome subunit beta type-2Homo sapiens (human)IC501.181733
Proteasome subunit beta type-3Homo sapiens (human)IC500.015011
Proteasome subunit beta type-4Homo sapiens (human)IC500.015011
Proteasome subunit beta type-5Homo sapiens (human)IC500.006555
Proteasome subunit beta type-6Homo sapiens (human)IC500.015011
Proteasome subunit beta type-7Homo sapiens (human)IC500.015011
Proteasome subunit beta type-8Homo sapiens (human)IC500.015011
Proteasome subunit beta type-9Homo sapiens (human)IC500.015011
Proto-oncogene tyrosine-protein kinase receptor RetHomo sapiens (human)IC500.016244
Proto-oncogene tyrosine-protein kinase receptor RetHomo sapiens (human)Ki0.001511
Pteridine reductase 1Leishmania majorIC501,900.000011
Replicase polyprotein 1abSevere acute respiratory syndrome coronavirus 2IC506.570011
Sodium/bile acid cotransporterHomo sapiens (human)IC5010,000.000011
Vascular endothelial growth factor receptor 1 Homo sapiens (human)IC500.022033
Vascular endothelial growth factor receptor 2Homo sapiens (human)IC500.003577
Vascular endothelial growth factor receptor 3Homo sapiens (human)IC500.005244

Activation Measurements

ProteinTaxonomyMeasurementAverage (mM)Bioassay(s)Drugs
26S proteasome regulatory subunit 6BHomo sapiens (human)Kd30.000011
5'-AMP-activated protein kinase catalytic subunit alpha-1Homo sapiens (human)Kd30.000011
5'-AMP-activated protein kinase subunit gamma-1Homo sapiens (human)Kd30.000011
5'-AMP-activated protein kinase subunit gamma-2Homo sapiens (human)Kd30.000011
AarF domain-containing protein kinase 1Homo sapiens (human)Kd30.000011
Actin-related protein 2Homo sapiens (human)Kd30.000011
Actin-related protein 3Homo sapiens (human)Kd30.000011
Activated CDC42 kinase 1Homo sapiens (human)Kd30.000011
Activin receptor type-1Homo sapiens (human)Kd30.000011
Activin receptor type-1BHomo sapiens (human)Kd30.000011
Activin receptor type-2BHomo sapiens (human)Kd30.000011
Acyl-CoA dehydrogenase family member 10Homo sapiens (human)Kd30.000011
Acyl-CoA dehydrogenase family member 11Homo sapiens (human)Kd30.000011
Adenine phosphoribosyltransferaseHomo sapiens (human)Kd30.000011
Adenosine kinaseHomo sapiens (human)Kd30.000011
Adenylate kinase 2, mitochondrialHomo sapiens (human)Kd30.000011
ADP/ATP translocase 2Homo sapiens (human)Kd30.000011
ADP/ATP translocase 3Homo sapiens (human)Kd30.000011
AP2-associated protein kinase 1Homo sapiens (human)Kd30.000011
ATP-dependent 6-phosphofructokinase, platelet typeHomo sapiens (human)Kd30.000011
ATP-dependent Clp protease proteolytic subunitStaphylococcus aureus subsp. aureus NCTC 8325EC503.600011
ATP-dependent RNA helicase DDX1Homo sapiens (human)Kd30.000011
ATP-dependent RNA helicase DDX3XHomo sapiens (human)Kd30.000012
ATP-dependent RNA helicase DDX42Homo sapiens (human)Kd30.000011
Atypical kinase COQ8A, mitochondrialHomo sapiens (human)Kd30.000011
Aurora kinase AHomo sapiens (human)Kd30.000011
Aurora kinase BHomo sapiens (human)Kd1.781011
Beta-adrenergic receptor kinase 1Homo sapiens (human)Kd30.000011
BMP-2-inducible protein kinaseHomo sapiens (human)Kd30.000011
Bone morphogenetic protein receptor type-1AHomo sapiens (human)Kd30.000011
Bone morphogenetic protein receptor type-1BHomo sapiens (human)Kd30.000011
Bone morphogenetic protein receptor type-2Homo sapiens (human)Kd30.000011
Breakpoint cluster region proteinHomo sapiens (human)Kd4.113011
Calcium/calmodulin-dependent protein kinase kinase 2Homo sapiens (human)Kd30.000011
Calcium/calmodulin-dependent protein kinase type II subunit deltaHomo sapiens (human)Kd30.000011
Calcium/calmodulin-dependent protein kinase type II subunit gammaHomo sapiens (human)Kd30.000011
Calcium/calmodulin-dependent protein kinase type IVHomo sapiens (human)Kd30.000011
cAMP-dependent protein kinase catalytic subunit alphaHomo sapiens (human)Kd30.000011
cAMP-dependent protein kinase catalytic subunit betaHomo sapiens (human)Kd30.000011
cAMP-dependent protein kinase catalytic subunit gammaHomo sapiens (human)Kd30.000011
cAMP-dependent protein kinase type II-alpha regulatory subunitHomo sapiens (human)Kd30.000011
Casein kinase I isoform alphaHomo sapiens (human)Kd30.000011
Casein kinase I isoform deltaHomo sapiens (human)Kd30.000011
Casein kinase I isoform epsilonHomo sapiens (human)Kd30.000011
Casein kinase I isoform gamma-1Homo sapiens (human)Kd30.000011
Casein kinase I isoform gamma-3Homo sapiens (human)Kd30.000011
Casein kinase II subunit alpha'Homo sapiens (human)Kd30.000011
cGMP-dependent protein kinase 1 Homo sapiens (human)Kd30.000011
Chromodomain-helicase-DNA-binding protein 4Homo sapiens (human)Kd30.000011
Citron Rho-interacting kinaseHomo sapiens (human)Kd30.000011
Cyclin-dependent kinase 1Homo sapiens (human)Kd30.000011
Cyclin-dependent kinase 12Homo sapiens (human)Kd30.000011
Cyclin-dependent kinase 13Homo sapiens (human)Kd30.000011
Cyclin-dependent kinase 16Homo sapiens (human)Kd30.000011
Cyclin-dependent kinase 17Homo sapiens (human)Kd30.000011
Cyclin-dependent kinase 2Homo sapiens (human)Kd30.000011
Cyclin-dependent kinase 4Homo sapiens (human)Kd30.000011
Cyclin-dependent kinase 6Homo sapiens (human)Kd30.000011
Cyclin-dependent kinase 7Homo sapiens (human)Kd30.000011
Cyclin-dependent kinase 9Homo sapiens (human)Kd30.000011
Cyclin-dependent-like kinase 5 Homo sapiens (human)Kd30.000011
Cyclin-G-associated kinaseHomo sapiens (human)Kd30.000011
Cysteine--tRNA ligase, cytoplasmicHomo sapiens (human)Kd30.000011
Cystic fibrosis transmembrane conductance regulatorHomo sapiens (human)EC500.74471717
Cystic fibrosis transmembrane conductance regulatorHomo sapiens (human)Kd60.300022
Cytochrome c1, heme protein, mitochondrialHomo sapiens (human)Kd30.000011
dCTP pyrophosphatase 1Homo sapiens (human)Kd30.000011
Delta(24)-sterol reductaseHomo sapiens (human)Kd30.000011
Deoxycytidine kinaseHomo sapiens (human)Kd30.000011
Discoidin domain-containing receptor 2Homo sapiens (human)Kd0.218011
DNA replication licensing factor MCM4Homo sapiens (human)Kd30.000011
DNA topoisomerase 2-alphaHomo sapiens (human)Kd30.000011
DNA topoisomerase 2-betaHomo sapiens (human)Kd30.000011
DnaJ homolog subfamily A member 1Homo sapiens (human)Kd30.000011
Dual specificity mitogen-activated protein kinase kinase 1Homo sapiens (human)Kd30.000011
Dual specificity mitogen-activated protein kinase kinase 2Homo sapiens (human)Kd30.000011
Dual specificity mitogen-activated protein kinase kinase 3Homo sapiens (human)Kd30.000011
Dual specificity mitogen-activated protein kinase kinase 5Homo sapiens (human)Kd2.910011
Dual specificity mitogen-activated protein kinase kinase 6Homo sapiens (human)Kd30.000011
Dual specificity protein kinase CLK1Homo sapiens (human)Kd30.000011
Dual specificity protein kinase CLK2Homo sapiens (human)Kd30.000012
Dual specificity protein kinase CLK3Homo sapiens (human)Kd30.000011
Dual specificity protein kinase CLK4Homo sapiens (human)Kd30.000011
Dual specificity testis-specific protein kinase 1Homo sapiens (human)Kd30.000011
Dual specificity tyrosine-phosphorylation-regulated kinase 1AHomo sapiens (human)Kd30.000011
Dynamin-like 120 kDa protein, mitochondrialHomo sapiens (human)Kd30.000011
EKC/KEOPS complex subunit TP53RKHomo sapiens (human)Kd30.000011
Electron transfer flavoprotein subunit betaHomo sapiens (human)Kd30.000012
Elongation factor Tu, mitochondrialHomo sapiens (human)Kd30.000011
Ephrin type-A receptor 1Homo sapiens (human)Kd30.000011
Ephrin type-A receptor 2Homo sapiens (human)Kd30.000011
Ephrin type-A receptor 4Homo sapiens (human)Kd30.000011
Ephrin type-A receptor 5Homo sapiens (human)Kd30.000011
Ephrin type-B receptor 2Homo sapiens (human)Kd30.000011
Ephrin type-B receptor 3Homo sapiens (human)Kd30.000011
Ephrin type-B receptor 4Homo sapiens (human)Kd30.000011
Ephrin type-B receptor 6Homo sapiens (human)Kd30.000011
Epidermal growth factor receptorHomo sapiens (human)Kd30.000011
Epithelial discoidin domain-containing receptor 1Homo sapiens (human)Kd0.046011
Eukaryotic translation initiation factor 2-alpha kinase 1Homo sapiens (human)Kd30.000011
Eukaryotic translation initiation factor 5BHomo sapiens (human)Kd30.000011
Exosome RNA helicase MTR4Homo sapiens (human)Kd30.000011
Ferrochelatase, mitochondrialHomo sapiens (human)Kd2.953022
Fibroblast growth factor receptor 1Homo sapiens (human)Kd30.000011
Focal adhesion kinase 1Homo sapiens (human)Kd30.000011
G protein-coupled receptor kinase 6Homo sapiens (human)Kd30.000011
General transcription and DNA repair factor IIH helicase subunit XPDHomo sapiens (human)Kd30.000011
Glycine--tRNA ligaseHomo sapiens (human)Kd30.000012
Glycogen phosphorylase, brain formHomo sapiens (human)Kd30.000011
Glycogen phosphorylase, liver formHomo sapiens (human)Kd30.000011
Glycogen synthase kinase-3 alphaHomo sapiens (human)Kd30.000011
Glycogen synthase kinase-3 betaHomo sapiens (human)Kd30.000011
GTP-binding nuclear protein RanHomo sapiens (human)Kd30.000011
Guanine nucleotide-binding protein G(i) subunit alpha-2Homo sapiens (human)Kd30.000011
Heme oxygenase 2Homo sapiens (human)Kd30.000011
Hepatocyte growth factor receptorHomo sapiens (human)Kd30.000011
Inhibitor of nuclear factor kappa-B kinase subunit epsilonHomo sapiens (human)Kd30.000011
Inosine-5'-monophosphate dehydrogenase 2Homo sapiens (human)Kd30.000011
Insulin receptorHomo sapiens (human)Kd30.000011
Insulin-like growth factor 1 receptorHomo sapiens (human)Kd30.000011
Integrin-linked protein kinaseHomo sapiens (human)Kd30.000011
Interleukin-1 receptor-associated kinase 1Homo sapiens (human)Kd30.000011
Interleukin-1 receptor-associated kinase 3Homo sapiens (human)Kd30.000011
Interleukin-1 receptor-associated kinase 4Homo sapiens (human)Kd30.000011
Isoleucine--tRNA ligase, mitochondrialHomo sapiens (human)Kd30.000011
LIM domain kinase 1Homo sapiens (human)Kd30.000011
LIM domain kinase 2Homo sapiens (human)Kd30.000011
Long-chain-fatty-acid--CoA ligase 5Homo sapiens (human)Kd30.000011
Macrophage-stimulating protein receptorHomo sapiens (human)Kd30.000011
MAP kinase-activated protein kinase 2Homo sapiens (human)Kd0.063011
MAP kinase-activated protein kinase 3Homo sapiens (human)Kd30.000011
MAP kinase-activated protein kinase 5Homo sapiens (human)Kd30.000011
MAP/microtubule affinity-regulating kinase 3Homo sapiens (human)Kd30.000011
MAP/microtubule affinity-regulating kinase 4Homo sapiens (human)Kd30.000011
Maternal embryonic leucine zipper kinaseHomo sapiens (human)Kd30.000011
Membrane-associated progesterone receptor component 1Homo sapiens (human)Kd30.000011
Membrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinaseHomo sapiens (human)Kd30.000011
MidasinHomo sapiens (human)Kd30.000011
Misshapen-like kinase 1Homo sapiens (human)Kd30.000011
Mitogen-activated protein kinase 1Homo sapiens (human)Kd30.000011
Mitogen-activated protein kinase 10Homo sapiens (human)Kd30.000011
Mitogen-activated protein kinase 11Homo sapiens (human)Kd30.000011
Mitogen-activated protein kinase 14Homo sapiens (human)Kd0.217011
Mitogen-activated protein kinase 15Homo sapiens (human)Kd30.000011
Mitogen-activated protein kinase 3 Homo sapiens (human)Kd30.000011
Mitogen-activated protein kinase 7Homo sapiens (human)Kd30.000011
Mitogen-activated protein kinase 8Homo sapiens (human)Kd30.000011
Mitogen-activated protein kinase 9Homo sapiens (human)Kd30.000012
Mitogen-activated protein kinase kinase kinase 1Homo sapiens (human)Kd30.000011
Mitogen-activated protein kinase kinase kinase 11Homo sapiens (human)Kd30.000011
Mitogen-activated protein kinase kinase kinase 2Homo sapiens (human)Kd30.000011
Mitogen-activated protein kinase kinase kinase 20Homo sapiens (human)Kd30.000011
Mitogen-activated protein kinase kinase kinase 3Homo sapiens (human)Kd30.000011
Mitogen-activated protein kinase kinase kinase 4Homo sapiens (human)Kd30.000011
Mitogen-activated protein kinase kinase kinase 5Homo sapiens (human)Kd30.000011
Mitogen-activated protein kinase kinase kinase 6Homo sapiens (human)Kd1.575011
Mitogen-activated protein kinase kinase kinase kinase 1Homo sapiens (human)Kd30.000011
Mitogen-activated protein kinase kinase kinase kinase 2Homo sapiens (human)Kd0.578011
Mitogen-activated protein kinase kinase kinase kinase 3Homo sapiens (human)Kd30.000011
Mitogen-activated protein kinase kinase kinase kinase 4Homo sapiens (human)Kd30.000011
Mitogen-activated protein kinase kinase kinase kinase 5Homo sapiens (human)Kd3.117011
Mitotic checkpoint serine/threonine-protein kinase BUB1Homo sapiens (human)Kd30.000011
Multifunctional protein ADE2Homo sapiens (human)Kd30.000011
Myosin light chain kinase 3Homo sapiens (human)Kd30.000011
Myosin light chain kinase, smooth muscleHomo sapiens (human)Kd30.000011
Myosin-10Homo sapiens (human)Kd30.000011
Myosin-14Homo sapiens (human)Kd30.000011
NADH dehydrogenase [ubiquinone] 1 alpha subcomplex subunit 13Homo sapiens (human)Kd30.000011
Non-receptor tyrosine-protein kinase TNK1Homo sapiens (human)Kd30.000011
Non-receptor tyrosine-protein kinase TYK2Homo sapiens (human)Kd30.000011
NUAK family SNF1-like kinase 2Homo sapiens (human)Kd30.000011
Nuclear receptor subfamily 1 group I member 2Homo sapiens (human)EC509.120055
Nucleolar GTP-binding protein 1Homo sapiens (human)Kd30.000011
Obg-like ATPase 1Homo sapiens (human)Kd30.000011
PAS domain-containing serine/threonine-protein kinaseHomo sapiens (human)Kd30.000011
Peroxisomal acyl-coenzyme A oxidase 1Homo sapiens (human)Kd30.000011
Peroxisomal acyl-coenzyme A oxidase 3Homo sapiens (human)Kd30.000011
Phenylalanine--tRNA ligase beta subunitHomo sapiens (human)Kd30.000011
Phosphatidylethanolamine-binding protein 1Homo sapiens (human)Kd30.000011
Phosphatidylinositol 5-phosphate 4-kinase type-2 alphaHomo sapiens (human)Kd30.000011
Phosphatidylinositol 5-phosphate 4-kinase type-2 gammaHomo sapiens (human)Kd30.000011
Phosphorylase b kinase gamma catalytic chain, liver/testis isoformHomo sapiens (human)Kd30.000011
Platelet-derived growth factor receptor betaHomo sapiens (human)Kd0.316011
Potassium channel subfamily K member 2Homo sapiens (human)EC502,750.000011
Potassium voltage-gated channel subfamily A member 3Homo sapiens (human)Kd195.000011
Probable ATP-dependent RNA helicase DDX6Homo sapiens (human)Kd30.000011
Prostacyclin receptorHomo sapiens (human)EC500.014012
Prostacyclin receptorRattus norvegicus (Norway rat)EC500.200011
Prostaglandin D2 receptorHomo sapiens (human)EC500.127012
Protein kinase C alpha typeHomo sapiens (human)Kd30.000011
Protein kinase C beta typeHomo sapiens (human)Kd30.000011
Protein kinase C delta typeHomo sapiens (human)Kd30.000012
Protein kinase C iota typeHomo sapiens (human)Kd30.000011
Protein kinase C theta typeHomo sapiens (human)Kd30.000011
Protein-tyrosine kinase 2-betaHomo sapiens (human)Kd30.000011
Protein-tyrosine kinase 6Homo sapiens (human)Kd0.173011
Proto-oncogene tyrosine-protein kinase receptor RetHomo sapiens (human)Kd0.009011
Proto-oncogene tyrosine-protein kinase SrcHomo sapiens (human)Kd30.000011
Putative heat shock protein HSP 90-beta 2Homo sapiens (human)Kd30.000012
Pyridoxal kinaseHomo sapiens (human)Kd30.000011
Rab-like protein 3Homo sapiens (human)Kd30.000011
RAC-alpha serine/threonine-protein kinaseHomo sapiens (human)Kd30.000011
RAC-beta serine/threonine-protein kinaseHomo sapiens (human)Kd30.000011
RAC-gamma serine/threonine-protein kinaseHomo sapiens (human)Kd30.000011
Ras-related protein Rab-10Homo sapiens (human)Kd30.000011
Ras-related protein Rab-27AHomo sapiens (human)Kd30.000011
Ras-related protein Rab-6AHomo sapiens (human)Kd30.000011
Receptor-interacting serine/threonine-protein kinase 2Homo sapiens (human)Kd0.011011
Receptor-interacting serine/threonine-protein kinase 3Homo sapiens (human)Kd0.316011
Receptor-type tyrosine-protein kinase FLT3Homo sapiens (human)Kd30.000011
Rho-associated protein kinase 1Homo sapiens (human)Kd30.000011
Rho-associated protein kinase 2Homo sapiens (human)Kd30.000011
Ribosomal protein S6 kinase alpha-1Homo sapiens (human)Kd30.000011
Ribosomal protein S6 kinase alpha-3Homo sapiens (human)Kd30.000011
Ribosomal protein S6 kinase alpha-4Homo sapiens (human)Kd30.000011
Ribosomal protein S6 kinase alpha-5Homo sapiens (human)Kd30.000011
Ribosomal protein S6 kinase alpha-6Homo sapiens (human)Kd30.000011
Ribosyldihydronicotinamide dehydrogenase [quinone]Homo sapiens (human)Kd1.523011
RNA cytidine acetyltransferaseHomo sapiens (human)Kd30.000011
S-adenosylmethionine synthase isoform type-2Homo sapiens (human)Kd30.000011
Septin-9Homo sapiens (human)Kd30.000011
Serine/threonine-protein kinase 10Homo sapiens (human)Kd0.793011
Serine/threonine-protein kinase 16Homo sapiens (human)Kd30.000011
Serine/threonine-protein kinase 24Homo sapiens (human)Kd30.000011
Serine/threonine-protein kinase 26Homo sapiens (human)Kd30.000011
Serine/threonine-protein kinase 3Homo sapiens (human)Kd30.000011
Serine/threonine-protein kinase 38-likeHomo sapiens (human)Kd30.000011
Serine/threonine-protein kinase 4Homo sapiens (human)Kd30.000011
Serine/threonine-protein kinase A-RafHomo sapiens (human)Kd30.000011
Serine/threonine-protein kinase B-rafHomo sapiens (human)Kd30.000012
Serine/threonine-protein kinase Chk1Homo sapiens (human)Kd30.000011
Serine/threonine-protein kinase D2Homo sapiens (human)Kd30.000011
Serine/threonine-protein kinase D3Homo sapiens (human)Kd30.000011
Serine/threonine-protein kinase ICKHomo sapiens (human)Kd30.000011
Serine/threonine-protein kinase LATS1Homo sapiens (human)Kd30.000011
Serine/threonine-protein kinase MARK2Homo sapiens (human)Kd30.000011
Serine/threonine-protein kinase MRCK alphaHomo sapiens (human)Kd30.000011
Serine/threonine-protein kinase MRCK betaHomo sapiens (human)Kd30.000011
Serine/threonine-protein kinase MRCK gammaHomo sapiens (human)Kd30.000011
Serine/threonine-protein kinase N1Homo sapiens (human)Kd30.000011
Serine/threonine-protein kinase N2Homo sapiens (human)Kd30.000011
Serine/threonine-protein kinase N3Homo sapiens (human)Kd30.000011
Serine/threonine-protein kinase Nek1Homo sapiens (human)Kd30.000011
Serine/threonine-protein kinase Nek2Homo sapiens (human)Kd30.000011
Serine/threonine-protein kinase Nek3Homo sapiens (human)Kd30.000011
Serine/threonine-protein kinase Nek7Homo sapiens (human)Kd30.000012
Serine/threonine-protein kinase Nek9Homo sapiens (human)Kd30.000011
Serine/threonine-protein kinase NLKHomo sapiens (human)Kd30.000011
Serine/threonine-protein kinase PAK 2Homo sapiens (human)Kd30.000011
Serine/threonine-protein kinase PAK 4Homo sapiens (human)Kd30.000011
Serine/threonine-protein kinase pim-1Homo sapiens (human)Kd30.000011
Serine/threonine-protein kinase PLK4Homo sapiens (human)Kd30.000011
Serine/threonine-protein kinase SIK2Homo sapiens (human)Kd30.000011
Serine/threonine-protein kinase SIK3Homo sapiens (human)Kd30.000011
Serine/threonine-protein kinase STK11Homo sapiens (human)Kd30.000011
Serine/threonine-protein kinase TAO1Homo sapiens (human)Kd30.000011
Serine/threonine-protein kinase TAO2Homo sapiens (human)Kd30.000011
Serine/threonine-protein kinase TAO3Homo sapiens (human)Kd30.000011
Serine/threonine-protein kinase TBK1Homo sapiens (human)Kd30.000011
Serine/threonine-protein kinase ULK1Homo sapiens (human)Kd30.000012
Serine/threonine-protein kinase ULK3Homo sapiens (human)Kd30.000011
Serine/threonine-protein kinase/endoribonuclease IRE1Homo sapiens (human)Kd2.242011
Serine/threonine-protein kinase/endoribonuclease IRE2Homo sapiens (human)Kd30.000011
Signal recognition particle receptor subunit alphaHomo sapiens (human)Kd30.000011
STE20-like serine/threonine-protein kinase Homo sapiens (human)Kd3.851011
STE20-related kinase adapter protein alphaHomo sapiens (human)Kd30.000011
Structural maintenance of chromosomes protein 1AHomo sapiens (human)Kd30.000011
Structural maintenance of chromosomes protein 2Homo sapiens (human)Kd30.000011
Succinate--CoA ligase [ADP-forming] subunit beta, mitochondrialHomo sapiens (human)Kd30.000011
TGF-beta receptor type-1Homo sapiens (human)Kd30.000011
TGF-beta receptor type-2Homo sapiens (human)Kd30.000011
Thyroid hormone receptor-associated protein 3Homo sapiens (human)Kd30.000011
TRAF2 and NCK-interacting protein kinaseHomo sapiens (human)Kd0.565011
Tyrosine--tRNA ligase, cytoplasmicHomo sapiens (human)Kd30.000011
Tyrosine-protein kinase ABL1Homo sapiens (human)Kd3.771011
Tyrosine-protein kinase ABL2Homo sapiens (human)Kd30.000011
Tyrosine-protein kinase BTKHomo sapiens (human)Kd30.000011
Tyrosine-protein kinase CSKHomo sapiens (human)Kd30.000011
Tyrosine-protein kinase FerHomo sapiens (human)Kd30.000011
Tyrosine-protein kinase Fes/FpsHomo sapiens (human)Kd30.000011
Tyrosine-protein kinase FRKHomo sapiens (human)Kd30.000011
Tyrosine-protein kinase FynHomo sapiens (human)Kd30.000011
Tyrosine-protein kinase HCKHomo sapiens (human)Kd30.000011
Tyrosine-protein kinase JAK1Homo sapiens (human)Kd30.000011
Tyrosine-protein kinase JAK2Homo sapiens (human)Kd30.000011
Tyrosine-protein kinase LckHomo sapiens (human)Kd30.000011
Tyrosine-protein kinase LynHomo sapiens (human)Kd30.000012
Tyrosine-protein kinase SYKHomo sapiens (human)Kd30.000011
Tyrosine-protein kinase TecHomo sapiens (human)Kd30.000011
Tyrosine-protein kinase YesHomo sapiens (human)Kd30.000011
U5 small nuclear ribonucleoprotein 200 kDa helicaseHomo sapiens (human)Kd30.000011
UMP-CMP kinase Homo sapiens (human)Kd30.000012
Uncharacterized aarF domain-containing protein kinase 5Homo sapiens (human)Kd30.000011
Uncharacterized protein FLJ45252Homo sapiens (human)Kd30.000011
Vascular endothelial growth factor receptor 2Homo sapiens (human)Kd0.002111
Very long-chain specific acyl-CoA dehydrogenase, mitochondrialHomo sapiens (human)Kd30.000011
Wee1-like protein kinaseHomo sapiens (human)Kd30.000011