Page last updated: 2024-08-07 13:17:51
Prostacyclin receptor
A prostacyclin receptor that is encoded in the genome of rat. [OMA:P43253, PRO:DNx]
Synonyms
Prostaglandin I2 receptor;
PGI receptor;
PGI2 receptor;
Prostanoid IP receptor
Research
Bioassay Publications (2)
Timeframe | Studies on this Protein(%) | All Drugs % |
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 0 (0.00) | 18.2507 |
2000's | 1 (50.00) | 29.6817 |
2010's | 1 (50.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Compounds (3)
Drugs with Inhibition Measurements
Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
iloprost | Rattus norvegicus (Norway rat) | Ki | 0.0010 | 1 | 1 |
fr181157 | Rattus norvegicus (Norway rat) | IC50 | 1.2000 | 1 | 1 |
Drugs with Activation Measurements
Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
iloprost | Rattus norvegicus (Norway rat) | EC50 | 0.0007 | 1 | 1 |
selexipag | Rattus norvegicus (Norway rat) | EC50 | 0.2000 | 1 | 1 |