Proteins > ATP-dependent Clp protease proteolytic subunit
Page last updated: 2024-08-07 23:54:26
ATP-dependent Clp protease proteolytic subunit
An ATP-dependent Clp protease proteolytic subunit that is encoded in the genome of Staphylococcus aureus subsp. aureus NCTC 8325. [OMA:Q2G036, PRO:DNx]
Synonyms
EC 3.4.21.92;
Endopeptidase Clp
Research
Bioassay Publications (1)
Timeframe | Studies on this Protein(%) | All Drugs % |
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 0 (0.00) | 18.2507 |
2000's | 0 (0.00) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 1 (100.00) | 2.80 |
Compounds (3)
Drugs with Inhibition Measurements
Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
bortezomib | Staphylococcus aureus subsp. aureus NCTC 8325 | IC50 | 5.3000 | 1 | 1 |
ixazomib | Staphylococcus aureus subsp. aureus NCTC 8325 | IC50 | 5.3000 | 1 | 1 |
Drugs with Activation Measurements
Drug | Taxonomy | Measurement | Average (mM) | Bioassay(s) | Publication(s) |
bortezomib | Staphylococcus aureus subsp. aureus NCTC 8325 | EC50 | 23.5000 | 1 | 1 |
ixazomib | Staphylococcus aureus subsp. aureus NCTC 8325 | EC50 | 3.6000 | 1 | 1 |
mln 9708 | Staphylococcus aureus subsp. aureus NCTC 8325 | EC50 | 19.9000 | 1 | 1 |
mln 9708 | Staphylococcus aureus subsp. aureus NCTC 8325 | Kd | 7.3000 | 1 | 1 |