| Assay ID | Title | Year | Journal | Article |
|---|
| AID73730 | Effective concentration for stimulation of [3H]phosphoinositide formation in guinea pig synaptoneurosomes expressing alpha-1 receptor | 1993 | Journal of medicinal chemistry, Nov-26, Volume: 36, Issue:24
| Syntheses of 2,5- and 2,6-difluoronorepinephrine, 2,5-difluoroepinephrine, and 2,6-difluorophenylephrine: effect of disubstitution with fluorine on adrenergic activity. |
| AID32954 | Displacement of [3H]WB-4101 from adrenergic alpha 1 receptor of rat cerebral cortical membranes | 1993 | Journal of medicinal chemistry, Nov-26, Volume: 36, Issue:24
| Syntheses of 2,5- and 2,6-difluoronorepinephrine, 2,5-difluoroepinephrine, and 2,6-difluorophenylephrine: effect of disubstitution with fluorine on adrenergic activity. |
| AID40408 | Binding of [3H]dihydroalprenolol to beta-1 adrenergic receptor of rat cerebral cortical membranes | 2000 | Journal of medicinal chemistry, Apr-20, Volume: 43, Issue:8
| Syntheses of (R)- and (S)-2- and 6-fluoronorepinephrine and (R)- and (S)-2- and 6-fluoroepinephrine: effect of stereochemistry on fluorine-induced adrenergic selectivities. |
| AID42050 | Beta-1 adrenergic receptor agonist activity by stimulation of contraction rate of isolated guinea pig atrial preparations | 1988 | Journal of medicinal chemistry, Oct, Volume: 31, Issue:10
| Syntheses and adrenergic activities of ring-fluorinated epinephrines. |
| AID35430 | Binding affinity against alpha-1 adrenergic receptor in rat using [3H]prazosin as radioligand | 1985 | Journal of medicinal chemistry, Oct, Volume: 28, Issue:10
| Conformationally defined adrenergic agents. 1. Design and synthesis of novel alpha 2 selective adrenergic agents: electrostatic repulsion based conformational prototypes. |
| AID32977 | Binding affinity against alpha 2-Adrenergic receptor in guinea pig cerebral cortical membranes by displacement of [3H]clonidine | 1988 | Journal of medicinal chemistry, Oct, Volume: 31, Issue:10
| Syntheses and adrenergic activities of ring-fluorinated epinephrines. |
| AID33078 | Displacement of [3H]dihydroalprenolol from adrenergic beta 1 receptor of rat cerebral cortical membranes | 1993 | Journal of medicinal chemistry, Nov-26, Volume: 36, Issue:24
| Syntheses of 2,5- and 2,6-difluoronorepinephrine, 2,5-difluoroepinephrine, and 2,6-difluorophenylephrine: effect of disubstitution with fluorine on adrenergic activity. |
| AID32956 | Displacement of [3H]clonidine from adrenergic alpha 2 receptor of rat cerebral cortical membranes | 1993 | Journal of medicinal chemistry, Nov-26, Volume: 36, Issue:24
| Syntheses of 2,5- and 2,6-difluoronorepinephrine, 2,5-difluoroepinephrine, and 2,6-difluorophenylephrine: effect of disubstitution with fluorine on adrenergic activity. |
| AID44627 | Stimulation of cyclic AMP accumulation in C6 glioma cells expressing adrenergic beta receptor | 1993 | Journal of medicinal chemistry, Nov-26, Volume: 36, Issue:24
| Syntheses of 2,5- and 2,6-difluoronorepinephrine, 2,5-difluoroepinephrine, and 2,6-difluorophenylephrine: effect of disubstitution with fluorine on adrenergic activity. |
| AID36103 | Binding affinity against alpha-1 adrenergic receptor in guinea pig cerebral cortical membranes by displacement of [3H]- WB-4101 | 1988 | Journal of medicinal chemistry, Oct, Volume: 31, Issue:10
| Syntheses and adrenergic activities of ring-fluorinated epinephrines. |
| AID41478 | Binding of [3H]dihydroalprenolol to beta-2 adrenergic receptor of rat cerebral cortical membranes | 2000 | Journal of medicinal chemistry, Apr-20, Volume: 43, Issue:8
| Syntheses of (R)- and (S)-2- and 6-fluoronorepinephrine and (R)- and (S)-2- and 6-fluoroepinephrine: effect of stereochemistry on fluorine-induced adrenergic selectivities. |
| AID219797 | Binding of [3H]clonidine to alpha-2-adrenergic receptor of rat cerebral cortical membranes | 2000 | Journal of medicinal chemistry, Apr-20, Volume: 43, Issue:8
| Syntheses of (R)- and (S)-2- and 6-fluoronorepinephrine and (R)- and (S)-2- and 6-fluoroepinephrine: effect of stereochemistry on fluorine-induced adrenergic selectivities. |
| AID35192 | Binding affinity towards alpha-2 adrenergic receptor in rat using [3H]rauwolscine as radioligand | 1985 | Journal of medicinal chemistry, Oct, Volume: 28, Issue:10
| Conformationally defined adrenergic agents. 1. Design and synthesis of novel alpha 2 selective adrenergic agents: electrostatic repulsion based conformational prototypes. |
| AID231532 | Ratio of binding affinity towards alpha1 to alpha-2 receptor | 1988 | Journal of medicinal chemistry, Oct, Volume: 31, Issue:10
| Syntheses and adrenergic activities of ring-fluorinated epinephrines. |
| AID42193 | Binding affinity against beta-1 adrenergic receptor in guinea pig cerebral cortical membranes by displacement of Dihydro-[3H]-alprenolol | 1988 | Journal of medicinal chemistry, Oct, Volume: 31, Issue:10
| Syntheses and adrenergic activities of ring-fluorinated epinephrines. |
| AID35994 | Agonistic potency at alpha-1 adrenergic receptor for the amine-induced increase of phosphatidylinositol breakdown in synaptoneurosomes from guinea pig cerebral cortex | 1988 | Journal of medicinal chemistry, Oct, Volume: 31, Issue:10
| Syntheses and adrenergic activities of ring-fluorinated epinephrines. |
| AID33079 | Binding affinity against adrenergic beta 2 receptor versus 1 nM [3H]dihydroalprenolol in rat cerebral cerebellar membranes | 1993 | Journal of medicinal chemistry, Nov-26, Volume: 36, Issue:24
| Syntheses of 2,5- and 2,6-difluoronorepinephrine, 2,5-difluoroepinephrine, and 2,6-difluorophenylephrine: effect of disubstitution with fluorine on adrenergic activity. |
| AID37459 | Binding of [3H]prazosin to alpha-1 adrenergic receptor of rat cerebral cortical membranes | 2000 | Journal of medicinal chemistry, Apr-20, Volume: 43, Issue:8
| Syntheses of (R)- and (S)-2- and 6-fluoronorepinephrine and (R)- and (S)-2- and 6-fluoroepinephrine: effect of stereochemistry on fluorine-induced adrenergic selectivities. |
| [information is prepared from bioassay data collected from National Library of Medicine (NLM), extracted Dec-2023] |