| Assay ID | Title | Year | Journal | Article |
|---|
| AID1456746 | Inhibition of histamine H1 receptor (unknown origin) | 2017 | Journal of medicinal chemistry, 09-14, Volume: 60, Issue:17
| Return of D |
| AID63537 | Binding affinity towards human dopamine receptor D4 | 2001 | Journal of medicinal chemistry, Feb-15, Volume: 44, Issue:4
| Current and novel approaches to the drug treatment of schizophrenia. |
| AID1456756 | Inhibition of human dopamine D4.2 receptor | 2017 | Journal of medicinal chemistry, 09-14, Volume: 60, Issue:17
| Return of D |
| AID1456728 | Inhibition of human dopamine D2 receptor | 2017 | Journal of medicinal chemistry, 09-14, Volume: 60, Issue:17
| Return of D |
| AID1456732 | Inhibition of serotonin 5-HT2 receptor (unknown origin) | 2017 | Journal of medicinal chemistry, 09-14, Volume: 60, Issue:17
| Return of D |
| AID1456778 | Inhibition of dopamine D5 receptor (unknown origin) at 10 uM | 2017 | Journal of medicinal chemistry, 09-14, Volume: 60, Issue:17
| Return of D |
| AID1456752 | Inhibition of NPY2 receptor (unknown origin) | 2017 | Journal of medicinal chemistry, 09-14, Volume: 60, Issue:17
| Return of D |
| AID1456753 | Inhibition of beta-adrenergic receptor (unknown origin) | 2017 | Journal of medicinal chemistry, 09-14, Volume: 60, Issue:17
| Return of D |
| AID1456734 | Inhibition of serotonin 5-HT2C receptor (unknown origin) | 2017 | Journal of medicinal chemistry, 09-14, Volume: 60, Issue:17
| Return of D |
| AID1456751 | Inhibition of NPY1 receptor (unknown origin) | 2017 | Journal of medicinal chemistry, 09-14, Volume: 60, Issue:17
| Return of D |
| AID63534 | Binding affinity on human Dopamine receptor D4 expressed in CHO cells using radioligand [3H]-YM 09151 | 1997 | Journal of medicinal chemistry, Jan-03, Volume: 40, Issue:1
| 2-Phenyl-4(5)-[[4-(pyrimidin-2-yl)piperazin-1-yl]methyl]imidazole. A highly selective antagonist at cloned human D4 receptors. |
| AID63064 | Binding affinity on human Dopamine receptor D2 expressed in CHO cells using radioligand [3H]-YM 09151 | 1997 | Journal of medicinal chemistry, Jan-03, Volume: 40, Issue:1
| 2-Phenyl-4(5)-[[4-(pyrimidin-2-yl)piperazin-1-yl]methyl]imidazole. A highly selective antagonist at cloned human D4 receptors. |
| AID3797 | Binding affinity against 5-hydroxytryptamine 1A receptor | 1997 | Journal of medicinal chemistry, Jan-03, Volume: 40, Issue:1
| 2-Phenyl-4(5)-[[4-(pyrimidin-2-yl)piperazin-1-yl]methyl]imidazole. A highly selective antagonist at cloned human D4 receptors. |
| AID65119 | Binding affinity on human Dopamine receptor D3 expressed in CHO cells using radioligand [3H]-YM 09151 | 1997 | Journal of medicinal chemistry, Jan-03, Volume: 40, Issue:1
| 2-Phenyl-4(5)-[[4-(pyrimidin-2-yl)piperazin-1-yl]methyl]imidazole. A highly selective antagonist at cloned human D4 receptors. |
| AID1456750 | Inhibition of NMDA receptor (unknown origin) | 2017 | Journal of medicinal chemistry, 09-14, Volume: 60, Issue:17
| Return of D |
| AID1456747 | Inhibition of alpha1 adrenergic receptor (unknown origin) | 2017 | Journal of medicinal chemistry, 09-14, Volume: 60, Issue:17
| Return of D |
| AID1456731 | Inhibition of serotonin 5-HT1A receptor (unknown origin) | 2017 | Journal of medicinal chemistry, 09-14, Volume: 60, Issue:17
| Return of D |
| AID1456754 | Inhibition of histamine H3 receptor (unknown origin) | 2017 | Journal of medicinal chemistry, 09-14, Volume: 60, Issue:17
| Return of D |
| AID1456777 | Inhibition of dopamine D3 receptor (unknown origin) at 10 uM | 2017 | Journal of medicinal chemistry, 09-14, Volume: 60, Issue:17
| Return of D |
| AID1456737 | Inhibition of serotonin 5-HT3 receptor (unknown origin) | 2017 | Journal of medicinal chemistry, 09-14, Volume: 60, Issue:17
| Return of D |
| AID1456757 | Inhibition of human dopamine D4.7 receptor | 2017 | Journal of medicinal chemistry, 09-14, Volume: 60, Issue:17
| Return of D |
| AID1456776 | Inhibition of dopamine D1 receptor (unknown origin) at 10 uM | 2017 | Journal of medicinal chemistry, 09-14, Volume: 60, Issue:17
| Return of D |
| AID1456726 | Inhibition of human dopamine D4.4 receptor | 2017 | Journal of medicinal chemistry, 09-14, Volume: 60, Issue:17
| Return of D |
| AID1456749 | Inhibition of alpha2 adrenergic receptor (unknown origin) | 2017 | Journal of medicinal chemistry, 09-14, Volume: 60, Issue:17
| Return of D |
| AID1347160 | Primary screen NINDS Rhodamine qHTS for Zika virus inhibitors | 2020 | Proceedings of the National Academy of Sciences of the United States of America, 12-08, Volume: 117, Issue:49
| Therapeutic candidates for the Zika virus identified by a high-throughput screen for Zika protease inhibitors. |
| AID1296008 | Cytotoxic Profiling of Annotated Libraries Using Quantitative High-Throughput Screening | 2020 | SLAS discovery : advancing life sciences R & D, 01, Volume: 25, Issue:1
| Cytotoxic Profiling of Annotated and Diverse Chemical Libraries Using Quantitative High-Throughput Screening. |
| AID1346986 | P-glycoprotein substrates identified in KB-3-1 adenocarcinoma cell line, qHTS therapeutic library screen | 2019 | Molecular pharmacology, 11, Volume: 96, Issue:5
| A High-Throughput Screen of a Library of Therapeutics Identifies Cytotoxic Substrates of P-glycoprotein. |
| AID1346987 | P-glycoprotein substrates identified in KB-8-5-11 adenocarcinoma cell line, qHTS therapeutic library screen | 2019 | Molecular pharmacology, 11, Volume: 96, Issue:5
| A High-Throughput Screen of a Library of Therapeutics Identifies Cytotoxic Substrates of P-glycoprotein. |
| AID1347159 | Primary screen GU Rhodamine qHTS for Zika virus inhibitors: Unlinked NS2B-NS3 protease assay | 2020 | Proceedings of the National Academy of Sciences of the United States of America, 12-08, Volume: 117, Issue:49
| Therapeutic candidates for the Zika virus identified by a high-throughput screen for Zika protease inhibitors. |
| AID1347024 | Rat D4 receptor (Dopamine receptors) | 2004 | Molecular pharmacology, Dec, Volume: 66, Issue:6
| Certain 1,4-disubstituted aromatic piperidines and piperazines with extreme selectivity for the dopamine D4 receptor interact with a common receptor microdomain. |
| AID1345814 | Human D4 receptor (Dopamine receptors) | 1997 | The Journal of pharmacology and experimental therapeutics, Aug, Volume: 282, Issue:2
| II. Localization and characterization of dopamine D4 binding sites in rat and human brain by use of the novel, D4 receptor-selective ligand [3H]NGD 94-1. |
| AID493017 | Wombat Data for BeliefDocking | 1999 | Journal of medicinal chemistry, Aug-12, Volume: 42, Issue:16
| Chiral resolution and stereospecificity of 6-phenyl-4-phenylethynyl- 1,4-dihydropyridines as selective A(3) adenosine receptor antagonists. |
| [information is prepared from bioassay data collected from National Library of Medicine (NLM), extracted Dec-2023] |