| Assay ID | Title | Year | Journal | Article |
|---|
| AID277673 | Displacement of [3H]spiperone from human dopamine D3 expressed in CHO cell membrane | 2007 | Journal of medicinal chemistry, Feb-08, Volume: 50, Issue:3
| Structure-selectivity investigations of D2-like receptor ligands by CoMFA and CoMSIA guiding the discovery of D3 selective PET radioligands. |
| AID1152406 | Displacement of [3H]N-methylspiperone from rat dopamine D4 receptor by PDSP assay | 2014 | Bioorganic & medicinal chemistry, Jun-15, Volume: 22, Issue:12
| Identification of a new selective dopamine D4 receptor ligand. |
| AID61806 | Intrinsic activity as rate of incorporation of [3H]thymidine in human D4.2 receptor established in mitogenesis assay relative to quinpirole | 2002 | Bioorganic & medicinal chemistry letters, Feb-25, Volume: 12, Issue:4
| Di- and trisubstituted pyrazolo[1,5-a]pyridine derivatives: synthesis, dopamine receptor binding and ligand efficacy. |
| AID3968 | Ability to displace [3H]8-OH-DPAT radioligand from porcine 5-hydroxytryptamine 1A receptor; ND denotes not determined | 2002 | Bioorganic & medicinal chemistry letters, Aug-05, Volume: 12, Issue:15
| 2,4-Disubstituted pyrroles: synthesis, traceless linking and pharmacological investigations leading to the dopamine D4 receptor partial agonist FAUC 356. |
| AID1456729 | Inhibition of human dopamine D3 receptor | 2017 | Journal of medicinal chemistry, 09-14, Volume: 60, Issue:17
| Return of D |
| AID266772 | Displacement of [3H]SCH 23990 from dopamine receptor D1 in porcine striatal membrane | 2006 | Journal of medicinal chemistry, Jun-29, Volume: 49, Issue:13
| 2-[(4-phenylpiperazin-1-yl)methyl]imidazo(di)azines as selective D4-ligands. Induction of penile erection by 2-[4-(2-methoxyphenyl)piperazin-1-ylmethyl]imidazo[1,2-a]pyridine (PIP3EA), a potent and selective D4 partial agonist. |
| AID62901 | Ability to displace [3H]SCH-23390 radioligand from cloned human Dopamine receptor D2 in CHO cells | 2002 | Bioorganic & medicinal chemistry letters, Aug-05, Volume: 12, Issue:15
| 2,4-Disubstituted pyrroles: synthesis, traceless linking and pharmacological investigations leading to the dopamine D4 receptor partial agonist FAUC 356. |
| AID226202 | Intrinsic activity which is established by measuring the stimulation of mitogenesis | 2001 | Journal of medicinal chemistry, Aug-16, Volume: 44, Issue:17
| Rationally based efficacy tuning of selective dopamine d4 receptor ligands leading to the complete antagonist 2-[4-(4-chlorophenyl)piperazin-1-ylmethyl]pyrazolo[1,5-a]pyridine (FAUC 213). |
| AID1152403 | Displacement of [3H]SCH23390 from human dopamine D1 receptor by PDSP assay | 2014 | Bioorganic & medicinal chemistry, Jun-15, Volume: 22, Issue:12
| Identification of a new selective dopamine D4 receptor ligand. |
| AID242944 | Ratio of dopamine receptor D2 long and D3 ki values | 2005 | Journal of medicinal chemistry, Feb-10, Volume: 48, Issue:3
| Modeling the similarity and divergence of dopamine D2-like receptors and identification of validated ligand-receptor complexes. |
| AID319914 | Agonist activity at rat dopamine D4.2 receptor expressed in CHO10001A cells assessed as incorporation of [3H]thymidine relative to quinpirole | 2008 | Journal of medicinal chemistry, Mar-27, Volume: 51, Issue:6
| Synthesis, radiofluorination, and in vitro evaluation of pyrazolo[1,5-a]pyridine-based dopamine D4 receptor ligands: discovery of an inverse agonist radioligand for PET. |
| AID62928 | In vitro binding affinity at human cloned dopamine receptor D2 (long) stably expressed in CHO cells by [3H]-Spiperone displacement. | 2002 | Bioorganic & medicinal chemistry letters, Feb-25, Volume: 12, Issue:4
| Di- and trisubstituted pyrazolo[1,5-a]pyridine derivatives: synthesis, dopamine receptor binding and ligand efficacy. |
| AID1456758 | Inhibition of human dopamine D2 (short) receptor | 2017 | Journal of medicinal chemistry, 09-14, Volume: 60, Issue:17
| Return of D |
| AID242945 | Ratio of dopamine receptor D2 long and D4 ki values | 2005 | Journal of medicinal chemistry, Feb-10, Volume: 48, Issue:3
| Modeling the similarity and divergence of dopamine D2-like receptors and identification of validated ligand-receptor complexes. |
| AID277668 | Selectivity for dopamine D3 over dopamine D2 | 2007 | Journal of medicinal chemistry, Feb-08, Volume: 50, Issue:3
| Structure-selectivity investigations of D2-like receptor ligands by CoMFA and CoMSIA guiding the discovery of D3 selective PET radioligands. |
| AID238699 | Binding affinity for human dopamine receptor D2 long | 2005 | Journal of medicinal chemistry, Feb-10, Volume: 48, Issue:3
| Modeling the similarity and divergence of dopamine D2-like receptors and identification of validated ligand-receptor complexes. |
| AID266775 | Displacement of [3H]spiperone from human dopamine receptor D3 in CHO cell membrane | 2006 | Journal of medicinal chemistry, Jun-29, Volume: 49, Issue:13
| 2-[(4-phenylpiperazin-1-yl)methyl]imidazo(di)azines as selective D4-ligands. Induction of penile erection by 2-[4-(2-methoxyphenyl)piperazin-1-ylmethyl]imidazo[1,2-a]pyridine (PIP3EA), a potent and selective D4 partial agonist. |
| AID226201 | Rate of incorporation of [3H]thymidine as evidence of mitogenetic activity | 2001 | Journal of medicinal chemistry, Aug-16, Volume: 44, Issue:17
| Rationally based efficacy tuning of selective dopamine d4 receptor ligands leading to the complete antagonist 2-[4-(4-chlorophenyl)piperazin-1-ylmethyl]pyrazolo[1,5-a]pyridine (FAUC 213). |
| AID319909 | Displacement of [3H]ketanserin from 5HT2 receptor in pig cortical membranes | 2008 | Journal of medicinal chemistry, Mar-27, Volume: 51, Issue:6
| Synthesis, radiofluorination, and in vitro evaluation of pyrazolo[1,5-a]pyridine-based dopamine D4 receptor ligands: discovery of an inverse agonist radioligand for PET. |
| AID266779 | Displacement of [3H]prazosin from porcine Adrenergic alpha-1 receptor in porcine brain | 2006 | Journal of medicinal chemistry, Jun-29, Volume: 49, Issue:13
| 2-[(4-phenylpiperazin-1-yl)methyl]imidazo(di)azines as selective D4-ligands. Induction of penile erection by 2-[4-(2-methoxyphenyl)piperazin-1-ylmethyl]imidazo[1,2-a]pyridine (PIP3EA), a potent and selective D4 partial agonist. |
| AID266773 | Displacement of [3H]spiperone from human dopamine receptor D2(long) in CHO cell membrane | 2006 | Journal of medicinal chemistry, Jun-29, Volume: 49, Issue:13
| 2-[(4-phenylpiperazin-1-yl)methyl]imidazo(di)azines as selective D4-ligands. Induction of penile erection by 2-[4-(2-methoxyphenyl)piperazin-1-ylmethyl]imidazo[1,2-a]pyridine (PIP3EA), a potent and selective D4 partial agonist. |
| AID319906 | Displacement of [3H]spiperone from cloned human dopamine D4.4 receptor expressed in CHO cells | 2008 | Journal of medicinal chemistry, Mar-27, Volume: 51, Issue:6
| Synthesis, radiofluorination, and in vitro evaluation of pyrazolo[1,5-a]pyridine-based dopamine D4 receptor ligands: discovery of an inverse agonist radioligand for PET. |
| AID62903 | Ability to displace [3H]spiperone radioligand from cloned human Dopamine receptor D2 in CHO cells | 2002 | Bioorganic & medicinal chemistry letters, Aug-05, Volume: 12, Issue:15
| 2,4-Disubstituted pyrroles: synthesis, traceless linking and pharmacological investigations leading to the dopamine D4 receptor partial agonist FAUC 356. |
| AID319907 | Displacement of [3H]SCH23990 from dopamine D1 receptor in pig striatal membrane | 2008 | Journal of medicinal chemistry, Mar-27, Volume: 51, Issue:6
| Synthesis, radiofluorination, and in vitro evaluation of pyrazolo[1,5-a]pyridine-based dopamine D4 receptor ligands: discovery of an inverse agonist radioligand for PET. |
| AID63188 | In vitro binding affinity at human cloned dopamine receptor D1 stably expressed in CHO cells by [3H]-SCH- 23390 displacement. | 2002 | Bioorganic & medicinal chemistry letters, Feb-25, Volume: 12, Issue:4
| Di- and trisubstituted pyrazolo[1,5-a]pyridine derivatives: synthesis, dopamine receptor binding and ligand efficacy. |
| AID61803 | Tested for the effective concentration against CHO 10001 cells in human D4.2 receptor established in mitogenesis assay | 2002 | Bioorganic & medicinal chemistry letters, Feb-25, Volume: 12, Issue:4
| Di- and trisubstituted pyrazolo[1,5-a]pyridine derivatives: synthesis, dopamine receptor binding and ligand efficacy. |
| AID633277 | Binding affinity to dopamine D4 receptor in Wistar rat brain slices | 2011 | Journal of medicinal chemistry, Dec-22, Volume: 54, Issue:24
| Evaluation of 18F-labeled benzodioxine piperazine-based dopamine D4 receptor ligands: lipophilicity as a determinate of nonspecific binding. |
| AID63189 | Binding affinity was evaluated for the displacement of [3H]-SCH- 23390 against bovine Dopamine receptor D1 | 1999 | Bioorganic & medicinal chemistry letters, Jan-04, Volume: 9, Issue:1
| Azaindole derivatives with high affinity for the dopamine D4 receptor: synthesis, ligand binding studies and comparison of molecular electrostatic potential maps. |
| AID319910 | Displacement of [3H]prazosin from adrenergic alpha1 receptor in pig cortical membranes | 2008 | Journal of medicinal chemistry, Mar-27, Volume: 51, Issue:6
| Synthesis, radiofluorination, and in vitro evaluation of pyrazolo[1,5-a]pyridine-based dopamine D4 receptor ligands: discovery of an inverse agonist radioligand for PET. |
| AID266776 | Displacement of [3H]spiperone from human dopamine receptor D4.4 in CHO cell membrane | 2006 | Journal of medicinal chemistry, Jun-29, Volume: 49, Issue:13
| 2-[(4-phenylpiperazin-1-yl)methyl]imidazo(di)azines as selective D4-ligands. Induction of penile erection by 2-[4-(2-methoxyphenyl)piperazin-1-ylmethyl]imidazo[1,2-a]pyridine (PIP3EA), a potent and selective D4 partial agonist. |
| AID319904 | Displacement of [3H]spiperone from cloned human dopamine D2S receptor expressed in CHO cells | 2008 | Journal of medicinal chemistry, Mar-27, Volume: 51, Issue:6
| Synthesis, radiofluorination, and in vitro evaluation of pyrazolo[1,5-a]pyridine-based dopamine D4 receptor ligands: discovery of an inverse agonist radioligand for PET. |
| AID238613 | Binding affinity for human dopamine receptor D3 | 2005 | Journal of medicinal chemistry, Feb-10, Volume: 48, Issue:3
| Modeling the similarity and divergence of dopamine D2-like receptors and identification of validated ligand-receptor complexes. |
| AID319915 | Agonist activity at rat dopamine D4.2 receptor expressed in CHO10001A cells assessed as incorporation of [3H]thymidine | 2008 | Journal of medicinal chemistry, Mar-27, Volume: 51, Issue:6
| Synthesis, radiofluorination, and in vitro evaluation of pyrazolo[1,5-a]pyridine-based dopamine D4 receptor ligands: discovery of an inverse agonist radioligand for PET. |
| AID64179 | Ability to displace [3H]spiperone from dopamine receptor D4.4 expressed in CHO-K1 cells | 2001 | Journal of medicinal chemistry, Apr-12, Volume: 44, Issue:8
| Comparative molecular field analysis of dopamine D4 receptor antagonists including 3-[4-(4-chlorophenyl)piperazin-1-ylmethyl]pyrazolo[1,5-a]pyridine (FAUC 113), 3-[4-(4-chlorophenyl)piperazin-1-ylmethyl]-1H-pyrrolo-[2,3-b]pyridine (L-745,870), and clozapi |
| AID266777 | Displacement of [3H]8-OH-DPAT from 5HT1A receptor in porcine cortical membrane | 2006 | Journal of medicinal chemistry, Jun-29, Volume: 49, Issue:13
| 2-[(4-phenylpiperazin-1-yl)methyl]imidazo(di)azines as selective D4-ligands. Induction of penile erection by 2-[4-(2-methoxyphenyl)piperazin-1-ylmethyl]imidazo[1,2-a]pyridine (PIP3EA), a potent and selective D4 partial agonist. |
| AID1456726 | Inhibition of human dopamine D4.4 receptor | 2017 | Journal of medicinal chemistry, 09-14, Volume: 60, Issue:17
| Return of D |
| AID64980 | Binding affinity evaluated for the displacement of [3H]-spiperone against human dopamine receptor D3 | 1999 | Bioorganic & medicinal chemistry letters, Jan-04, Volume: 9, Issue:1
| Azaindole derivatives with high affinity for the dopamine D4 receptor: synthesis, ligand binding studies and comparison of molecular electrostatic potential maps. |
| AID277677 | Binding affinity to dopamine D2 | 2007 | Journal of medicinal chemistry, Feb-08, Volume: 50, Issue:3
| Structure-selectivity investigations of D2-like receptor ligands by CoMFA and CoMSIA guiding the discovery of D3 selective PET radioligands. |
| AID64976 | Binding affinity against dopamine receptor D3 using radioligand [3H]spiperone | 2001 | Journal of medicinal chemistry, Aug-16, Volume: 44, Issue:17
| Rationally based efficacy tuning of selective dopamine d4 receptor ligands leading to the complete antagonist 2-[4-(4-chlorophenyl)piperazin-1-ylmethyl]pyrazolo[1,5-a]pyridine (FAUC 213). |
| AID1456727 | Inhibition of human dopamine D1 receptor | 2017 | Journal of medicinal chemistry, 09-14, Volume: 60, Issue:17
| Return of D |
| AID277674 | Displacement of [3H]spiperone from human dopamine D4.4 expressed in CHO cell membrane | 2007 | Journal of medicinal chemistry, Feb-08, Volume: 50, Issue:3
| Structure-selectivity investigations of D2-like receptor ligands by CoMFA and CoMSIA guiding the discovery of D3 selective PET radioligands. |
| AID63519 | Binding affinity evaluated for the displacement of [3H]spiperone against human dopamine receptor D4 | 1999 | Bioorganic & medicinal chemistry letters, Jan-04, Volume: 9, Issue:1
| Azaindole derivatives with high affinity for the dopamine D4 receptor: synthesis, ligand binding studies and comparison of molecular electrostatic potential maps. |
| AID1152404 | Displacement of [3H]N-methylspiperone from human dopamine D2 receptor by PDSP assay | 2014 | Bioorganic & medicinal chemistry, Jun-15, Volume: 22, Issue:12
| Identification of a new selective dopamine D4 receptor ligand. |
| AID319905 | Displacement of [3H]spiperone from cloned human dopamine D3 receptor expressed in CHO cells | 2008 | Journal of medicinal chemistry, Mar-27, Volume: 51, Issue:6
| Synthesis, radiofluorination, and in vitro evaluation of pyrazolo[1,5-a]pyridine-based dopamine D4 receptor ligands: discovery of an inverse agonist radioligand for PET. |
| AID1152405 | Displacement of [3H]N-methylspiperone from human dopamine D3 receptor by PDSP assay | 2014 | Bioorganic & medicinal chemistry, Jun-15, Volume: 22, Issue:12
| Identification of a new selective dopamine D4 receptor ligand. |
| AID242943 | Ratio of dopamine receptor D3 and D4 ki values | 2005 | Journal of medicinal chemistry, Feb-10, Volume: 48, Issue:3
| Modeling the similarity and divergence of dopamine D2-like receptors and identification of validated ligand-receptor complexes. |
| AID319903 | Displacement of [3H]spiperone from cloned human dopamine D2L receptor expressed in CHO cells | 2008 | Journal of medicinal chemistry, Mar-27, Volume: 51, Issue:6
| Synthesis, radiofluorination, and in vitro evaluation of pyrazolo[1,5-a]pyridine-based dopamine D4 receptor ligands: discovery of an inverse agonist radioligand for PET. |
| AID63527 | In vitro binding affinity at human cloned dopamine receptor D4 stably expressed in CHO cells by [3H]spiperone displacement. | 2002 | Bioorganic & medicinal chemistry letters, Feb-25, Volume: 12, Issue:4
| Di- and trisubstituted pyrazolo[1,5-a]pyridine derivatives: synthesis, dopamine receptor binding and ligand efficacy. |
| AID266778 | Displacement of [3H]ketanserin from 5HT2 receptor in porcine cortical membrane | 2006 | Journal of medicinal chemistry, Jun-29, Volume: 49, Issue:13
| 2-[(4-phenylpiperazin-1-yl)methyl]imidazo(di)azines as selective D4-ligands. Induction of penile erection by 2-[4-(2-methoxyphenyl)piperazin-1-ylmethyl]imidazo[1,2-a]pyridine (PIP3EA), a potent and selective D4 partial agonist. |
| AID1456759 | Inhibition of human dopamine D2 (long) receptor (unknown origin) | 2017 | Journal of medicinal chemistry, 09-14, Volume: 60, Issue:17
| Return of D |
| AID64991 | In vitro binding affinity at human cloned dopamine receptor D3 stably expressed in CHO cells by [3H]spiperone displacement. | 2002 | Bioorganic & medicinal chemistry letters, Feb-25, Volume: 12, Issue:4
| Di- and trisubstituted pyrazolo[1,5-a]pyridine derivatives: synthesis, dopamine receptor binding and ligand efficacy. |
| AID319912 | Selectivity for human dopamine D4.4 receptor over human dopamine D2S receptor | 2008 | Journal of medicinal chemistry, Mar-27, Volume: 51, Issue:6
| Synthesis, radiofluorination, and in vitro evaluation of pyrazolo[1,5-a]pyridine-based dopamine D4 receptor ligands: discovery of an inverse agonist radioligand for PET. |
| AID63856 | Intrinsic activity at human Dopamine D4.2 receptor as stimulation of mitogenesis | 2002 | Bioorganic & medicinal chemistry letters, Aug-05, Volume: 12, Issue:15
| 2,4-Disubstituted pyrroles: synthesis, traceless linking and pharmacological investigations leading to the dopamine D4 receptor partial agonist FAUC 356. |
| AID63047 | Ability to displace [3H]SCH-23,390 radioligand from bovine Dopamine receptor D1 | 2002 | Bioorganic & medicinal chemistry letters, Aug-05, Volume: 12, Issue:15
| 2,4-Disubstituted pyrroles: synthesis, traceless linking and pharmacological investigations leading to the dopamine D4 receptor partial agonist FAUC 356. |
| AID63182 | Binding affinity against dopamine receptor D1 using radioligand [3H]-SCH- 23390 | 2001 | Journal of medicinal chemistry, Aug-16, Volume: 44, Issue:17
| Rationally based efficacy tuning of selective dopamine d4 receptor ligands leading to the complete antagonist 2-[4-(4-chlorophenyl)piperazin-1-ylmethyl]pyrazolo[1,5-a]pyridine (FAUC 213). |
| AID277669 | Selectivity for dopamine D3 over dopamine D4 | 2007 | Journal of medicinal chemistry, Feb-08, Volume: 50, Issue:3
| Structure-selectivity investigations of D2-like receptor ligands by CoMFA and CoMSIA guiding the discovery of D3 selective PET radioligands. |
| AID64661 | Binding affinity against dopamine receptor D2S using radioligand [3H]spiperone | 2001 | Journal of medicinal chemistry, Aug-16, Volume: 44, Issue:17
| Rationally based efficacy tuning of selective dopamine d4 receptor ligands leading to the complete antagonist 2-[4-(4-chlorophenyl)piperazin-1-ylmethyl]pyrazolo[1,5-a]pyridine (FAUC 213). |
| AID62331 | Binding affinity was evaluated for the displacement of [3H]spiperone against bovine Dopamine receptor D2 | 1999 | Bioorganic & medicinal chemistry letters, Jan-04, Volume: 9, Issue:1
| Azaindole derivatives with high affinity for the dopamine D4 receptor: synthesis, ligand binding studies and comparison of molecular electrostatic potential maps. |
| AID62929 | In vitro binding affinity at human cloned dopamine receptor D2 (short) stably expressed in CHO cells by [3H]spiperone displacement. | 2002 | Bioorganic & medicinal chemistry letters, Feb-25, Volume: 12, Issue:4
| Di- and trisubstituted pyrazolo[1,5-a]pyridine derivatives: synthesis, dopamine receptor binding and ligand efficacy. |
| AID1152407 | Displacement of [3H]SCH23390 from human dopamine D5 receptor by PDSP assay | 2014 | Bioorganic & medicinal chemistry, Jun-15, Volume: 22, Issue:12
| Identification of a new selective dopamine D4 receptor ligand. |
| AID319913 | Selectivity for human dopamine D4.4 receptor over human dopamine D3 receptor | 2008 | Journal of medicinal chemistry, Mar-27, Volume: 51, Issue:6
| Synthesis, radiofluorination, and in vitro evaluation of pyrazolo[1,5-a]pyridine-based dopamine D4 receptor ligands: discovery of an inverse agonist radioligand for PET. |
| AID64958 | Ability to displace [3H]spiperone radioligand from cloned human Dopamine receptor D3 in CHO cells | 2002 | Bioorganic & medicinal chemistry letters, Aug-05, Volume: 12, Issue:15
| 2,4-Disubstituted pyrroles: synthesis, traceless linking and pharmacological investigations leading to the dopamine D4 receptor partial agonist FAUC 356. |
| AID266774 | Displacement of [3H]spiperone from human dopamine receptor D2(short) in CHO cell membrane | 2006 | Journal of medicinal chemistry, Jun-29, Volume: 49, Issue:13
| 2-[(4-phenylpiperazin-1-yl)methyl]imidazo(di)azines as selective D4-ligands. Induction of penile erection by 2-[4-(2-methoxyphenyl)piperazin-1-ylmethyl]imidazo[1,2-a]pyridine (PIP3EA), a potent and selective D4 partial agonist. |
| AID63859 | Effective concentration of compound required against human Dopamine D4.2 receptor | 2002 | Bioorganic & medicinal chemistry letters, Aug-05, Volume: 12, Issue:15
| 2,4-Disubstituted pyrroles: synthesis, traceless linking and pharmacological investigations leading to the dopamine D4 receptor partial agonist FAUC 356. |
| AID65946 | Ability to displace [3H]spiperone radioligand from cloned human Dopamine receptor D4 in CHO cells | 2002 | Bioorganic & medicinal chemistry letters, Aug-05, Volume: 12, Issue:15
| 2,4-Disubstituted pyrroles: synthesis, traceless linking and pharmacological investigations leading to the dopamine D4 receptor partial agonist FAUC 356. |
| AID64031 | Binding affinity against human dopamine receptor D4.4 using radioligand [3H]spiperone | 2001 | Journal of medicinal chemistry, Aug-16, Volume: 44, Issue:17
| Rationally based efficacy tuning of selective dopamine d4 receptor ligands leading to the complete antagonist 2-[4-(4-chlorophenyl)piperazin-1-ylmethyl]pyrazolo[1,5-a]pyridine (FAUC 213). |
| AID238274 | Binding affinity for Dopamine receptor D4 | 2005 | Journal of medicinal chemistry, Feb-10, Volume: 48, Issue:3
| Modeling the similarity and divergence of dopamine D2-like receptors and identification of validated ligand-receptor complexes. |
| AID5447 | Ability to displace [3H]ketanserin radioligand from porcine 5-hydroxytryptamine 2A receptor; ND denotes not determined | 2002 | Bioorganic & medicinal chemistry letters, Aug-05, Volume: 12, Issue:15
| 2,4-Disubstituted pyrroles: synthesis, traceless linking and pharmacological investigations leading to the dopamine D4 receptor partial agonist FAUC 356. |
| AID64333 | Binding affinity against dopamine receptor D2L using radioligand [3H]-spiperone | 2001 | Journal of medicinal chemistry, Aug-16, Volume: 44, Issue:17
| Rationally based efficacy tuning of selective dopamine d4 receptor ligands leading to the complete antagonist 2-[4-(4-chlorophenyl)piperazin-1-ylmethyl]pyrazolo[1,5-a]pyridine (FAUC 213). |
| AID319908 | Displacement of [3H]8-OH-DPAT from 5HT1A receptor in pig cortical membranes | 2008 | Journal of medicinal chemistry, Mar-27, Volume: 51, Issue:6
| Synthesis, radiofluorination, and in vitro evaluation of pyrazolo[1,5-a]pyridine-based dopamine D4 receptor ligands: discovery of an inverse agonist radioligand for PET. |
| AID319911 | Selectivity for human dopamine D4.4 receptor over human dopamine D2L receptor | 2008 | Journal of medicinal chemistry, Mar-27, Volume: 51, Issue:6
| Synthesis, radiofluorination, and in vitro evaluation of pyrazolo[1,5-a]pyridine-based dopamine D4 receptor ligands: discovery of an inverse agonist radioligand for PET. |
| [information is prepared from bioassay data collected from National Library of Medicine (NLM), extracted Dec-2023] |