Protein | Potency Measurements | Inhibition Measurements | Activation Measurements | Drugs |
GLI family zinc finger 3 | 2 | 0 | 0 | 2 |
cytochrome P450 family 3 subfamily A polypeptide 4 | 3 | 0 | 0 | 3 |
estrogen-related nuclear receptor alpha | 2 | 0 | 0 | 2 |
estrogen nuclear receptor alpha | 2 | 0 | 0 | 2 |
thyroid hormone receptor beta isoform 2 | 2 | 0 | 0 | 2 |
importin subunit beta-1 isoform 1 | 1 | 0 | 0 | 1 |
mitogen-activated protein kinase 1 | 1 | 0 | 0 | 1 |
snurportin-1 | 1 | 0 | 0 | 1 |
GTP-binding nuclear protein Ran isoform 1 | 1 | 0 | 0 | 1 |
urokinase-type plasminogen activator precursor | 1 | 0 | 0 | 1 |
plasminogen precursor | 1 | 0 | 0 | 1 |
urokinase plasminogen activator surface receptor precursor | 1 | 0 | 0 | 1 |
geminin | 3 | 0 | 0 | 3 |
streptokinase A precursor | 0 | 0 | 3 | 3 |
ATP-binding cassette sub-family C member 3 | 0 | 4 | 0 | 4 |
Multidrug resistance-associated protein 4 | 0 | 4 | 0 | 4 |
Bile salt export pump | 0 | 5 | 0 | 5 |
ATP-dependent translocase ABCB1 | 0 | 1 | 0 | 2 |
Cytochrome P450 3A4 | 0 | 4 | 0 | 4 |
Potassium voltage-gated channel subfamily H member 2 | 0 | 5 | 0 | 6 |
Canalicular multispecific organic anion transporter 1 | 0 | 4 | 0 | 4 |
Solute carrier organic anion transporter family member 1B3 | 0 | 1 | 0 | 1 |
Solute carrier organic anion transporter family member 1B1 | 0 | 1 | 0 | 1 |
Chain A, JmjC domain-containing histone demethylation protein 3A | 1 | 0 | 0 | 1 |
Chain A, 2-oxoglutarate Oxygenase | 1 | 0 | 0 | 1 |
thioredoxin reductase | 1 | 0 | 0 | 1 |
TDP1 protein | 2 | 0 | 0 | 2 |
EWS/FLI fusion protein | 3 | 0 | 0 | 3 |
euchromatic histone-lysine N-methyltransferase 2 | 1 | 0 | 0 | 1 |
Replicase polyprotein 1ab | 0 | 1 | 0 | 1 |
CAAX prenyl protease 2 isoform 2 | 0 | 0 | 0 | 1 |
DNA polymerase beta | 1 | 0 | 0 | 1 |
histone acetyltransferase KAT2A isoform 1 | 1 | 0 | 0 | 1 |
Bile salt export pump | 0 | 1 | 0 | 1 |
Tubulin beta-4A chain | 0 | 1 | 0 | 1 |
Tubulin beta chain | 0 | 1 | 0 | 1 |
Tubulin alpha-3C chain | 0 | 1 | 0 | 1 |
Spike glycoprotein | 2 | 0 | 0 | 2 |
Tubulin alpha-1B chain | 0 | 1 | 0 | 1 |
Tubulin alpha-4A chain | 0 | 1 | 0 | 1 |
Tubulin beta-4B chain | 0 | 1 | 0 | 1 |
Fatty-acid amide hydrolase 1 | 0 | 1 | 0 | 1 |
DNA gyrase subunit A | 0 | 2 | 0 | 3 |
DNA primase | 0 | 1 | 0 | 1 |
Tubulin beta-3 chain | 0 | 1 | 0 | 1 |
Tubulin beta-2A chain | 0 | 1 | 0 | 1 |
Tubulin beta-8 chain | 0 | 1 | 0 | 1 |
Tubulin alpha-3E chain | 0 | 1 | 0 | 1 |
Tubulin alpha-1A chain | 0 | 1 | 0 | 1 |
Multidrug and toxin extrusion protein 1 | 0 | 1 | 0 | 1 |
Tubulin alpha-1C chain | 0 | 1 | 0 | 1 |
Tubulin beta-6 chain | 0 | 1 | 0 | 1 |
Tubulin beta-2B chain | 0 | 1 | 0 | 1 |
Tubulin beta-1 chain | 0 | 1 | 0 | 1 |
PPM1D protein | 2 | 0 | 0 | 2 |
G | 1 | 0 | 0 | 1 |
cytochrome P450 2D6 | 1 | 0 | 0 | 1 |
Histone deacetylase 3 | 0 | 2 | 0 | 2 |
Nuclear receptor corepressor 1 | 0 | 1 | 0 | 1 |
Interferon beta | 2 | 0 | 0 | 2 |
HLA class I histocompatibility antigen, B alpha chain | 1 | 0 | 0 | 1 |
Integrin beta-1 | 0 | 1 | 0 | 1 |
Leukotriene A-4 hydrolase | 0 | 1 | 0 | 1 |
Cytochrome P450 2D6 | 0 | 1 | 0 | 1 |
Integrin alpha-4 | 0 | 1 | 0 | 1 |
Cytochrome P450 2C19 | 0 | 1 | 0 | 1 |
Histone deacetylase 4 | 0 | 1 | 0 | 1 |
Histone deacetylase 1 | 0 | 2 | 0 | 2 |
Histone deacetylase 7 | 0 | 1 | 0 | 1 |
Inositol hexakisphosphate kinase 1 | 1 | 0 | 0 | 1 |
Histone deacetylase 2 | 0 | 2 | 0 | 2 |
Histone deacetylase 11 | 0 | 1 | 0 | 1 |
Histone deacetylase 8 | 0 | 1 | 0 | 1 |
Histone deacetylase 6 | 0 | 1 | 0 | 1 |
Histone deacetylase 5 | 0 | 1 | 0 | 1 |
Nuclear receptor corepressor 2 | 0 | 1 | 0 | 1 |
cytochrome P450 2C9, partial | 1 | 0 | 0 | 1 |
Voltage-dependent L-type calcium channel subunit alpha-1C | 0 | 1 | 0 | 1 |
Voltage-dependent L-type calcium channel subunit alpha-1F | 0 | 1 | 0 | 1 |
DNA gyrase subunit B | 0 | 1 | 0 | 1 |
DNA gyrase subunit A | 0 | 1 | 0 | 2 |
DNA gyrase subunit B | 0 | 1 | 0 | 2 |
DNA topoisomerase 4 subunit A | 0 | 1 | 0 | 1 |
DNA gyrase subunit B | 0 | 1 | 0 | 1 |
Replicase polyprotein 1ab | 0 | 1 | 0 | 1 |
Replicase polyprotein 1ab | 0 | 1 | 0 | 1 |
DNA topoisomerase 2-alpha | 0 | 0 | 0 | 1 |
Potassium voltage-gated channel subfamily E member 1 | 0 | 1 | 0 | 1 |
DNA gyrase subunit A | 0 | 1 | 0 | 1 |
Voltage-dependent L-type calcium channel subunit alpha-1C | 0 | 1 | 0 | 1 |
Potassium voltage-gated channel subfamily KQT member 1 | 0 | 1 | 0 | 1 |
DNA gyrase subunit B | 0 | 1 | 0 | 2 |
Voltage-dependent L-type calcium channel subunit alpha-1D | 0 | 1 | 0 | 1 |
Voltage-dependent L-type calcium channel subunit alpha-1S | 0 | 1 | 0 | 1 |
Voltage-dependent L-type calcium channel subunit alpha-1C | 0 | 1 | 0 | 1 |
Sodium channel protein type 5 subunit alpha | 0 | 1 | 0 | 1 |
Sphingosine kinase 2 | 0 | 2 | 0 | 2 |
Sphingosine kinase 1 | 0 | 1 | 0 | 1 |
90-kda heat shock protein beta HSP90 beta, partial | 0 | 1 | 0 | 1 |
glucocorticoid receptor [Homo sapiens] | 1 | 0 | 0 | 1 |
peroxisome proliferator activated receptor gamma | 1 | 0 | 0 | 1 |
Histone H2A.x | 1 | 0 | 0 | 1 |
estrogen receptor beta isoform 1 | 0 | 1 | 0 | 1 |
heat shock protein HSP 90-alpha isoform 2 | 0 | 1 | 0 | 1 |
tyrosine-protein phosphatase non-receptor type 7 isoform 2 | 0 | 1 | 0 | 1 |
Dihydroxyacetone phosphate acyltransferase | 0 | 0 | 0 | 1 |
30S ribosomal protein S6 | 0 | 2 | 0 | 2 |
30S ribosomal protein S7 | 0 | 2 | 0 | 2 |
50S ribosomal protein L15 | 0 | 2 | 0 | 2 |
Tetracycline resistance protein, class B | 0 | 0 | 0 | 1 |
Muscarinic acetylcholine receptor M2 | 0 | 1 | 0 | 1 |
72 kDa type IV collagenase | 0 | 1 | 0 | 1 |
Stromelysin-1 | 0 | 1 | 0 | 1 |
50S ribosomal protein L10 | 0 | 2 | 0 | 2 |
50S ribosomal protein L11 | 0 | 2 | 0 | 2 |
50S ribosomal protein L7/L12 | 0 | 2 | 0 | 2 |
50S ribosomal protein L19 | 0 | 2 | 0 | 2 |
50S ribosomal protein L1 | 0 | 2 | 0 | 2 |
50S ribosomal protein L20 | 0 | 2 | 0 | 2 |
50S ribosomal protein L27 | 0 | 2 | 0 | 2 |
50S ribosomal protein L28 | 0 | 2 | 0 | 2 |
50S ribosomal protein L29 | 0 | 2 | 0 | 2 |
50S ribosomal protein L31 | 0 | 2 | 0 | 2 |
50S ribosomal protein L31 type B | 0 | 2 | 0 | 2 |
50S ribosomal protein L32 | 0 | 2 | 0 | 2 |
50S ribosomal protein L33 | 0 | 2 | 0 | 2 |
50S ribosomal protein L34 | 0 | 2 | 0 | 2 |
50S ribosomal protein L35 | 0 | 2 | 0 | 2 |
50S ribosomal protein L36 | 0 | 2 | 0 | 2 |
30S ribosomal protein S10 | 0 | 2 | 0 | 2 |
30S ribosomal protein S11 | 0 | 2 | 0 | 2 |
30S ribosomal protein S12 | 0 | 2 | 0 | 2 |
30S ribosomal protein S13 | 0 | 2 | 0 | 2 |
30S ribosomal protein S16 | 0 | 2 | 0 | 2 |
30S ribosomal protein S18 | 0 | 2 | 0 | 2 |
30S ribosomal protein S19 | 0 | 2 | 0 | 2 |
30S ribosomal protein S20 | 0 | 2 | 0 | 2 |
30S ribosomal protein S2 | 0 | 2 | 0 | 2 |
30S ribosomal protein S3 | 0 | 2 | 0 | 2 |
30S ribosomal protein S4 | 0 | 2 | 0 | 2 |
30S ribosomal protein S5 | 0 | 2 | 0 | 2 |
30S ribosomal protein S8 | 0 | 2 | 0 | 2 |
30S ribosomal protein S9 | 0 | 2 | 0 | 2 |
50S ribosomal protein L13 | 0 | 2 | 0 | 2 |
50S ribosomal protein L14 | 0 | 2 | 0 | 2 |
50S ribosomal protein L16 | 0 | 2 | 0 | 2 |
50S ribosomal protein L23 | 0 | 2 | 0 | 2 |
30S ribosomal protein S15 | 0 | 2 | 0 | 2 |
Multidrug transporter MdfA | 0 | 1 | 0 | 1 |
50S ribosomal protein L17 | 0 | 2 | 0 | 2 |
50S ribosomal protein L21 | 0 | 2 | 0 | 2 |
50S ribosomal protein L30 | 0 | 2 | 0 | 2 |
50S ribosomal protein L6 | 0 | 2 | 0 | 2 |
30S ribosomal protein S14 | 0 | 2 | 0 | 2 |
30S ribosomal protein S17 | 0 | 2 | 0 | 2 |
30S ribosomal protein S1 | 0 | 2 | 0 | 2 |
50S ribosomal protein L18 | 0 | 2 | 0 | 2 |
Alpha-1B adrenergic receptor | 0 | 1 | 0 | 1 |
Neutrophil collagenase | 0 | 1 | 0 | 1 |
Alpha-1D adrenergic receptor | 0 | 1 | 0 | 1 |
Alpha-synuclein | 0 | 1 | 0 | 1 |
Alpha-1A adrenergic receptor | 0 | 1 | 0 | 1 |
Collagenase 3 | 0 | 1 | 0 | 1 |
Cannabinoid receptor 1 | 0 | 1 | 0 | 1 |
50S ribosomal protein L2 | 0 | 2 | 0 | 2 |
50S ribosomal protein L3 | 0 | 2 | 0 | 2 |
50S ribosomal protein L24 | 0 | 2 | 0 | 2 |
50S ribosomal protein L4 | 0 | 2 | 0 | 2 |
50S ribosomal protein L22 | 0 | 2 | 0 | 2 |
50S ribosomal protein L5 | 0 | 2 | 0 | 2 |
30S ribosomal protein S21 | 0 | 2 | 0 | 2 |
50S ribosomal protein L25 | 0 | 2 | 0 | 2 |
50S ribosomal protein L36 2 | 0 | 2 | 0 | 2 |
Integrase | 0 | 1 | 0 | 1 |
Solute carrier family 22 member 8 | 0 | 0 | 0 | 1 |
P2Y purinoceptor 12 | 0 | 1 | 0 | 1 |
Solute carrier family 22 member 11 | 0 | 0 | 0 | 1 |
Protein-arginine deiminase type-4 | 0 | 2 | 0 | 2 |
Solute carrier family 22 member 7 | 0 | 0 | 0 | 1 |
retinoic acid nuclear receptor alpha variant 1 | 2 | 0 | 0 | 2 |
activating transcription factor 6 | 1 | 0 | 0 | 1 |
interleukin 8 | 1 | 0 | 0 | 1 |
glp-1 receptor, partial | 1 | 0 | 0 | 1 |
thyroid stimulating hormone receptor | 1 | 0 | 0 | 1 |
retinoid X nuclear receptor alpha | 1 | 0 | 0 | 1 |
peroxisome proliferator-activated receptor delta | 1 | 0 | 0 | 1 |
IDH1 | 1 | 0 | 0 | 1 |
thyroid stimulating hormone receptor | 1 | 0 | 0 | 1 |
nuclear receptor subfamily 1, group I, member 2 | 1 | 0 | 0 | 1 |
chromobox protein homolog 1 | 1 | 0 | 0 | 1 |
nuclear factor erythroid 2-related factor 2 isoform 1 | 1 | 0 | 0 | 1 |
cytochrome P450 3A4 isoform 1 | 1 | 0 | 0 | 1 |
twin arginine protein translocation system - TatA protein | 0 | 0 | 0 | 1 |
lamin isoform A-delta10 | 1 | 0 | 0 | 1 |
Gamma-aminobutyric acid receptor subunit pi | 1 | 0 | 0 | 1 |
Gamma-aminobutyric acid receptor subunit beta-1 | 1 | 0 | 0 | 1 |
Gamma-aminobutyric acid receptor subunit delta | 1 | 0 | 0 | 1 |
Gamma-aminobutyric acid receptor subunit gamma-2 | 1 | 0 | 0 | 1 |
Gamma-aminobutyric acid receptor subunit alpha-5 | 1 | 0 | 0 | 1 |
Gamma-aminobutyric acid receptor subunit alpha-3 | 1 | 0 | 0 | 1 |
Gamma-aminobutyric acid receptor subunit gamma-1 | 1 | 0 | 0 | 1 |
Gamma-aminobutyric acid receptor subunit alpha-2 | 1 | 0 | 0 | 1 |
Gamma-aminobutyric acid receptor subunit alpha-4 | 1 | 0 | 0 | 1 |
Gamma-aminobutyric acid receptor subunit gamma-3 | 1 | 0 | 0 | 1 |
Gamma-aminobutyric acid receptor subunit alpha-6 | 1 | 0 | 0 | 1 |
Nuclear receptor ROR-gamma | 1 | 0 | 0 | 1 |
Gamma-aminobutyric acid receptor subunit alpha-1 | 1 | 0 | 0 | 1 |
Gamma-aminobutyric acid receptor subunit beta-3 | 1 | 0 | 0 | 1 |
Gamma-aminobutyric acid receptor subunit beta-2 | 1 | 0 | 0 | 1 |
TAR DNA-binding protein 43 | 1 | 0 | 0 | 1 |
GABA theta subunit | 1 | 0 | 0 | 1 |
Gamma-aminobutyric acid receptor subunit epsilon | 1 | 0 | 0 | 1 |
[prepared from compound, protein, and bioassay information from National Library of Medicine (NLM), extracted Dec-2023] |