| Assay ID | Title | Year | Journal | Article |
|---|
| AID156630 | In vitro binding affinity for human PPAR delta in SPA | 2003 | Bioorganic & medicinal chemistry letters, Apr-07, Volume: 13, Issue:7
| Phenylacetic acid derivatives as hPPAR agonists. |
| AID665204 | Agonist activity at PPARdelta | 2012 | Bioorganic & medicinal chemistry, Jun-01, Volume: 20, Issue:11
| Activity landscape modeling of PPAR ligands with dual-activity difference maps. |
| AID175938 | In vivo plasma triglyceride in Zucker diabetic fatty rat after 11 days at 10 mg/kg/day | 2003 | Bioorganic & medicinal chemistry letters, Apr-07, Volume: 13, Issue:7
| Phenylacetic acid derivatives as hPPAR agonists. |
| AID174361 | In vivo plasma glucose in Zucker diabetic fatty rat after 11 days at 30 mg/kg/day | 2003 | Bioorganic & medicinal chemistry letters, Apr-07, Volume: 13, Issue:7
| Phenylacetic acid derivatives as hPPAR agonists. |
| AID156281 | In vitro binding affinity for human PPAR alpha in SPA | 2003 | Bioorganic & medicinal chemistry letters, Apr-07, Volume: 13, Issue:7
| Phenylacetic acid derivatives as hPPAR agonists. |
| AID12364 | Dose-normalized AUC was determined by po administration (10 mg/kg) in fasted male Sprague-Dawley rats | 2003 | Bioorganic & medicinal chemistry letters, Apr-07, Volume: 13, Issue:7
| Phenylacetic acid derivatives as hPPAR agonists. |
| AID665203 | Agonist activity at PPARalpha | 2012 | Bioorganic & medicinal chemistry, Jun-01, Volume: 20, Issue:11
| Activity landscape modeling of PPAR ligands with dual-activity difference maps. |
| AID175789 | In vivo plasma free fatty acid in Zucker diabetic fatty rat after 11 days at 10 mg/kg/day | 2003 | Bioorganic & medicinal chemistry letters, Apr-07, Volume: 13, Issue:7
| Phenylacetic acid derivatives as hPPAR agonists. |
| AID220378 | In vivo plasma glucose in db/db mouse after 11 days at 10 mg/kg/day | 2003 | Bioorganic & medicinal chemistry letters, Apr-07, Volume: 13, Issue:7
| Phenylacetic acid derivatives as hPPAR agonists. |
| AID156955 | In vitro binding affinity for human PPAR gamma in SPA | 2003 | Bioorganic & medicinal chemistry letters, Apr-07, Volume: 13, Issue:7
| Phenylacetic acid derivatives as hPPAR agonists. |
| AID220383 | In vivo plasma triglyceride in db/db mouse after 11 days at 10 mg/kg/day | 2003 | Bioorganic & medicinal chemistry letters, Apr-07, Volume: 13, Issue:7
| Phenylacetic acid derivatives as hPPAR agonists. |
| AID175939 | In vivo plasma triglyceride in Zucker diabetic fatty rat after 11 days at 30 mg/kg/day | 2003 | Bioorganic & medicinal chemistry letters, Apr-07, Volume: 13, Issue:7
| Phenylacetic acid derivatives as hPPAR agonists. |
| AID663659 | Binding affinity at human GST-tagged PPARdelta ligand binding domain after 1 hr by time-resolved FRET analysis | 2012 | European journal of medicinal chemistry, Jul, Volume: 53 | Discovery, design and synthesis of Y-shaped peroxisome proliferator-activated receptor δ agonists as potent anti-obesity agents in vivo. |
| AID141908 | Agonist activity for murine PPAR delta receptor in transcriptional activation assay | 2000 | Journal of medicinal chemistry, Feb-24, Volume: 43, Issue:4
| The PPARs: from orphan receptors to drug discovery. |
| AID141903 | Agonist activity for murine PPAR alpha receptor in transcriptional activation assay | 2000 | Journal of medicinal chemistry, Feb-24, Volume: 43, Issue:4
| The PPARs: from orphan receptors to drug discovery. |
| AID91237 | Agonist activity for Human PPAR alpha receptor in transcriptional activation assay | 2000 | Journal of medicinal chemistry, Feb-24, Volume: 43, Issue:4
| The PPARs: from orphan receptors to drug discovery. |
| AID220384 | In vivo plasma triglyceride in db/db mouse after 11 days at 30 mg/kg/day | 2003 | Bioorganic & medicinal chemistry letters, Apr-07, Volume: 13, Issue:7
| Phenylacetic acid derivatives as hPPAR agonists. |
| AID600728 | Displacement of radio-labeled full agonist from PPARgamma receptor | 2011 | European journal of medicinal chemistry, Jun, Volume: 46, Issue:6
| Discovery of new nanomolar peroxisome proliferator-activated receptor γ activators via elaborate ligand-based modeling. |
| AID141913 | Agonist activity for murine PPAR gamma receptor in transcriptional activation assay | 2000 | Journal of medicinal chemistry, Feb-24, Volume: 43, Issue:4
| The PPARs: from orphan receptors to drug discovery. |
| AID13633 | Oral bioavailability in rat (Sprague-Dawley) (fasted male) (dose 10 mg/kg) | 2003 | Bioorganic & medicinal chemistry letters, Apr-07, Volume: 13, Issue:7
| Phenylacetic acid derivatives as hPPAR agonists. |
| AID156132 | Transcriptional activation by human PPAR alpha | 2003 | Bioorganic & medicinal chemistry letters, Apr-07, Volume: 13, Issue:7
| Phenylacetic acid derivatives as hPPAR agonists. |
| AID12877 | Half-life was determined by iv administration (1.5 mg/kg) in fasted male Sprague-Dawley rats | 2003 | Bioorganic & medicinal chemistry letters, Apr-07, Volume: 13, Issue:7
| Phenylacetic acid derivatives as hPPAR agonists. |
| AID665205 | Agonist activity at PPARgamma | 2012 | Bioorganic & medicinal chemistry, Jun-01, Volume: 20, Issue:11
| Activity landscape modeling of PPAR ligands with dual-activity difference maps. |
| AID156607 | Transcriptional activation by human PPAR delta | 2003 | Bioorganic & medicinal chemistry letters, Apr-07, Volume: 13, Issue:7
| Phenylacetic acid derivatives as hPPAR agonists. |
| AID175790 | In vivo plasma free fatty acid in Zucker diabetic fatty rat after 11 days at 30 mg/kg/day | 2003 | Bioorganic & medicinal chemistry letters, Apr-07, Volume: 13, Issue:7
| Phenylacetic acid derivatives as hPPAR agonists. |
| AID174360 | In vivo plasma glucose in Zucker diabetic fatty rat after 11 days at 10 mg/kg/day | 2003 | Bioorganic & medicinal chemistry letters, Apr-07, Volume: 13, Issue:7
| Phenylacetic acid derivatives as hPPAR agonists. |
| AID220379 | In vivo plasma glucose in db/db mouse after 11 days at 30 mg/kg/day | 2003 | Bioorganic & medicinal chemistry letters, Apr-07, Volume: 13, Issue:7
| Phenylacetic acid derivatives as hPPAR agonists. |
| AID91246 | Agonist activity for Human PPAR gamma receptor in transcriptional activation assay | 2000 | Journal of medicinal chemistry, Feb-24, Volume: 43, Issue:4
| The PPARs: from orphan receptors to drug discovery. |
| AID91241 | Agonist activity for Human PPAR delta receptor in transcriptional activation assay | 2000 | Journal of medicinal chemistry, Feb-24, Volume: 43, Issue:4
| The PPARs: from orphan receptors to drug discovery. |
| AID156933 | Transcriptional activation by human PPAR gamma | 2003 | Bioorganic & medicinal chemistry letters, Apr-07, Volume: 13, Issue:7
| Phenylacetic acid derivatives as hPPAR agonists. |
| AID173095 | In vivo plasma triglyceride in db/db mouse after 11 days at 10 mg/kg/day | 2003 | Bioorganic & medicinal chemistry letters, Apr-07, Volume: 13, Issue:7
| Phenylacetic acid derivatives as hPPAR agonists. |
| AID1346790 | Human Peroxisome proliferator-activated receptor-beta/delta (1C. Peroxisome proliferator-activated receptors) | 2004 | Journal of medicinal chemistry, Aug-12, Volume: 47, Issue:17
| Peroxisome proliferator-activated receptor alpha/gamma dual agonists for the treatment of type 2 diabetes. |
| AID1346800 | Human Peroxisome proliferator-activated receptor-gamma (1C. Peroxisome proliferator-activated receptors) | 1999 | The Journal of biological chemistry, Mar-05, Volume: 274, Issue:10
| Novel peroxisome proliferator-activated receptor (PPAR) gamma and PPARdelta ligands produce distinct biological effects. |
| AID1346790 | Human Peroxisome proliferator-activated receptor-beta/delta (1C. Peroxisome proliferator-activated receptors) | 1999 | The Journal of biological chemistry, Mar-05, Volume: 274, Issue:10
| Novel peroxisome proliferator-activated receptor (PPAR) gamma and PPARdelta ligands produce distinct biological effects. |
| [information is prepared from bioassay data collected from National Library of Medicine (NLM), extracted Dec-2023] |